首页 工具
登录
购物车

搜索结果

Search Results for " gli "
Targets Recommended: Hedgehog/Smoothened

226

抑制剂 & 化合物

17

天然产物

1

化合物库

12

重组蛋白

26

同位素标记化合物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name
L7840 高溶解性卤化片段化合物库

796 compounds
高溶解性卤化片段库包含796 个卤化片段化合物。

化合物库

高溶解性卤化片段化合物库
Cat.No: L7840
Compounds: 796
Cat. No. Product Name Target Signaling Pathways
T22089 HPI 1

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
HPI 1 是一种刺猬 (Hh) 信号抑制剂。在 Shh-LIGHT2 细胞中抑制 Sonic Hedgehog (Shh)-、SAG- 和 Gli 诱导的 Hh 通路激活(Shh-、SAG-、Gli2- 和 Gli1 诱导的激活的 IC50 值为 1.5、1.5、4 和 6 μM) .
T24159 IHR-1

IHR 1

Smo Stem Cells
IHR-1 是一种Smo 拮抗剂,不能透过细胞膜。
T15370 GANT 58

4,44乔,4乔(2,3,4,5-Thiophentetrayl)tetrakis-pyridine,NSC 75503

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
GANT 58 (NSC-75503) 是GLI 拮抗剂,能够抑制 GLI1 诱导的转录,其IC50=5 μM。
T3070 GANT 61

NSC 136476,GANT61

Hedgehog/Smoothened; Autophagy Autophagy; GPCR/G Protein; Stem Cells
GANT 61 (GANT61) 是一种Gli1和Gli2抑制剂,靶向Hedgehog/GLi 通路。
T6203 Saxagliptin

BMS-477118,沙克列汀,Onglyza,沙格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin (BMS-477118) 是一种选择性,可逆性,竞争性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin 能够用于 2 型糖尿病的研究。
T12710 Retagliptin Phosphate

SP 2086,瑞格列汀磷酸盐

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Retagliptin Phosphate (SP 2086) 是一种选择性、竞争性、口服活性的二肽基肽酶 4 (DPP-4) 抑制剂。Retagliptin phosphate 能够用于 2 型糖尿病 (T2DM) 的研究。
T64332 Glimepiride sulfonamide

Immunology/Inflammation related Immunology/Inflammation
Glimepiride sulfonamide 是一种抗炎活性化合物。
T28757 Sergliflozin etabonate

GW-869682,GW-869682X,KGT-1251,GW869682X,GW869682,KGT1251

SGLT GPCR/G Protein
Sergliflozin etabonate (KGT-1251) 是一种 SGLT-2 抑制剂,可用于 2 型糖尿病和肥胖症的研究。
T34286 Remogliflozin etabonate

GSK189075,GSK 189075,GSK-189075A,GSK189075A,GSK-189075,GSK 189075A

SGLT GPCR/G Protein
Remogliflozin etabonate (GSK189075A) 是 regaliflozin 的前药和 SGLT2 抑制剂,对 hSGLT2、rSGLT2、rSGLT1 和 hSGLT1 的 Ki 值分别为 1.95、2.14、8.57 和 43.1μM。
T2385 Ipragliflozin

伊格列净,ASP1941

SGLT GPCR/G Protein
Ipragliflozin (ASP1941) 是一种口服有效的,选择性的 SGLT2抑制剂,对人 SGLT2 和 SGLT1,大鼠 SGLT2 和 SGLT1,小鼠 SGLT2 和 SGLT1 的 IC50分别为 7.38 和 1876 nM,6.73 和 1166 nM,5.64 和 1380 nM。Ipragliflozin 具有抗糖尿病活性。
T0191 Linagliptin

BI 1356,利格列汀,利拉利汀

Ferroptosis; Proteasome; DPP-4; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
Linagliptin (BI 1356) 是一种有效的、可口服的、基于二氢嘌呤二酮的二肽基肽酶 4 抑制剂,具有降血糖活性。
T1502 Vildagliptin

维达列汀,NVP-LAF 237,维格列汀,LAF237

Apoptosis; Ferroptosis; Proteasome; DPP-4 Apoptosis; Proteases/Proteasome; Ubiquitination
Vildagliptin (LAF237) 是一种选择性二肽基肽酶IV (DPP-IV) 抑制剂,在人 Caco-2 细胞中抑制 DPP-IV 的IC50为 3.5 nM。它具有出色的口服生物利用度和降血糖活性。
T0242L Sitagliptin phosphate monohydrate

MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物

Proteasome; DPP-4; Autophagy Autophagy; Proteases/Proteasome; Ubiquitination
Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) 是一种有效的 DPP-IV 抑制剂,在 Caco-2 细胞提取物中的 IC50 为 19 nM。
T12835 Saroglitazar

Lipaglyn

PPAR DNA Damage/DNA Repair; Metabolism
Saroglitazar (Lipaglyn) 是 PPAR 的激动剂,对 PPARα 和 PPARγ 的 EC50 值为 0.65 pM 和 3 nM。
T10998 Deriglidole

SL 86-0715

Adrenergic Receptor GPCR/G Protein; Neuroscience
Deriglidole (SL 86-0715) 是一种外周肾上腺素能受体拮抗剂,是一种具有选择性的α2受体抑制剂。 Deriglidole 对可乐定和 Idazoxan 有抑制作用而对哌唑嗪与大鼠皮质和人血小板α2-肾上腺素能受体不显示活性。
T1634 Glibenclamide

格列本脲,Glyburide

Potassium Channel; Mitochondrial Metabolism; CFTR; P-gp; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
Glibenclamide (Glyburide) 是一种具有口服活性的 ATP 敏感的 K+通道抑制剂,可研究糖尿病和肥胖。它抑制 P-糖蛋白,可直接结合并阻断 KATP 的 SUR1亚基并抑制囊性纤维化跨膜传导调节蛋白。它通过诱导膜离子通透性干扰线粒体生物能,可诱导自噬。
T19710 Ciglitazone

Ciglitazona,U 63287,ADD3878,ADD-3878,U-63287,ADD 3878

Apoptosis; p38 MAPK; PPAR Apoptosis; DNA Damage/DNA Repair; MAPK; Metabolism
Ciglitazone (ADD 3878) 是一种强效和选择性的PPARγ激动剂(EC50:3μM)和口服降糖药。Ciglitazone 抑制th17细胞的增殖和分化,降低胰岛素水平、血管内皮生长因子的产生和血压,诱导胃癌细胞的细胞周期停止。Ciglitazone 能诱导负鼠肾上皮细胞的凋亡,激活p38 MAPK 和凋亡诱导因子(AIF)的核转位。 Ciglitazone 在肥胖症和高血糖症的动物模型中表现出降血糖活性。
T4639 Azemiglitazone

MSDC 0602

Mitochondrial Metabolism; mTOR Metabolism; PI3K/Akt/mTOR signaling
Azemiglitazone (MSDC 0602) 是一种 PPARγ 保留的噻唑烷二酮类药物 (TZD),与能够线粒体丙酮酸载体 (MPC) 相互作用并抑制其活性,降低 pparγ 介导的副作用的风险,有用于 2 型糖尿病研究的潜能。
T0214 Pioglitazone

U 72107,吡格列酮,匹格列酮

Ferroptosis; PPAR Apoptosis; DNA Damage/DNA Repair; Metabolism
Pioglitazone (U 72107) 是一种胰岛素增敏剂和噻唑烷二酮,适用于治疗 2 型糖尿病。它是一种选择性PPARγ激动剂,高亲和力结合到 PPARγ 配体结合域,作用于人和鼠 PPARγ的EC50分别为 0.93 和 0.99 μM。
T3104 Globalagliatin

LY2608204

Glucokinase Metabolism
Globalagliatin (LY2608204) 是一种葡萄糖激酶 (GK) 活化剂,EC50=42 nM。
T26986 Cevoglitazar

LBM-642,LBM 642,LBM642

PPAR DNA Damage/DNA Repair; Metabolism
Cevoglitazar (LBM-642) 是一种 PPARɑ 激动剂和 PPARγ激动剂。Cevoglitazar 能有效减少肥胖小鼠和猴的食物摄入量和体重。
T16009L Managlinat dialanetil

MB06322,MB 6322,CS-917

Phosphatase Metabolism
Managlinat dialanetil (MB06322) 是一种可口服且具有有效性的 fructose 1,6-bisphosphatase (FBPase) 抑制剂,具有降糖活性,可用于研究 2 型糖尿病。
T6237 Trelagliptin

SYR-472,曲格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Trelagliptin (SYR-472) 是一种有效的,具有口服活性的DPP-4抑制剂,IC50=4 nM。它可以改善体内血糖控制,能够用于2 型糖尿病 (T2DM) 的研究。
T22708 Darglitazone

CP-86325

PPAR DNA Damage/DNA Repair; Metabolism
Darglitazone (CP-86325) 是一种噻唑烷二酮,是口服有效的PPAR-γ选择性激动剂。Darglitazone 可以有效控制血糖和脂质代谢,在 II 型糖尿病中有研究价值。
T1622 Rosiglitazone maleate

BRL 49653C,BRL 49653,马来酸罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone maleate (BRL 49653) 是一种选择性PPARγ激活剂,具有抗糖尿病特性和潜在抗肿瘤活性。它也是TRP 通道调节剂,可抑制 TRPM2、TRPM3 的活性,激活 TRPC5。
T15575 Indeglitazar

PPM 204

PPAR DNA Damage/DNA Repair; Metabolism
Indeglitazar (PPM 204) 是 PPAR 的泛激动剂,包括亚型 alpha (α)、delta (δ) 和 gamma (γ)。
T28501 Ragaglitazar

NNC61-0029,NN-622,(-)-DRF-2725,NNC-61-0029,NN 622,NNC 61-0029

PPAR DNA Damage/DNA Repair; Metabolism
Ragaglitazar(NNC-61-0029) 是一种有效的 PPARα和 PPARγ双重激动剂,在动物模型中显示出有效的降脂和胰岛素增敏作用。Ragaglitazar 可用于研究 2 型糖尿病。
T16083 Mizagliflozin

GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base

SGLT GPCR/G Protein
Mizagliflozin (GSK-1614235 free base) 是口服有效的、选择性的 SGLT1抑制剂,对人 SGLT1 的 Ki 值为 27 nM。Mizagliflozin 对 SGLT1 的选择性是 SGLT2的303 倍。它是抗糖尿病药物,可以改善餐后血糖波动。它在改善慢性便秘方面具有潜在的作用。
T7486 Imeglimin hydrochloride

EMD 387008 hydrochloride,(6R)-1,6-二氢-N2,N2,6-三甲基-1,3,5-三嗪-2,4-二胺盐酸盐

Reactive Oxygen Species; Mitochondrial Metabolism Immunology/Inflammation; Metabolism; NF-κB
Imeglimin hydrochloride (EMD 387008 hydrochloride) 是一种口服降糖剂。Imeglimin 可改善胰岛素敏感性,能够抑制活性氧的产生、增加线粒体 DNA、改善线粒体功能。
T1674 Nateglinide

那格列奈,A4166,Senaglinide

Potassium Channel; Proteasome; PPAR DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome; Ubiquitination
Nateglinide (Senaglinide) 是 D-苯丙氨酸的一种衍生物,是口服有效的、短效促胰岛素释放化合物,也是 DPP IV 抑制剂。 Nateglinide 抑制胰岛 β 细胞中 ATP 敏感的 K+通道。Nateglinide 在 2 型糖尿病中具有研究价值。
T7133 Anagliptin

SK-0403,阿拉格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Anagliptin (SK-0403) 是一种选择性的二肽酰肽酶 4 抑制剂,IC50=3.8 nM,对 DPP-8/9 的选择性相对较弱,IC50分别为 68 和 60 nM。
T0334 Rosiglitazone

BRL49653,罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone (BRL49653) 是一种 PPARγ 激动剂、TRPC5 激活剂和 TRPM3 抑制剂,具有口服活性。Rosiglitazone 也是一种降糖剂,是噻唑烷二酮类胰岛素增敏剂。
T0178 Saxagliptin hydrate

沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin hydrate (Onglyza hydrate) 是一种选择性,竞争性,可逆性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin hydrate 能够用于 2 型糖尿病的研究。
T4460 Dapagliflozin ((2S)-1,2-propanediol, hydrate)

BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate

SGLT GPCR/G Protein
Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) 是 Dapagliflozin 1,2-propanediol, hydrate 的 S 型异构体,是竞争性葡萄糖协同转运蛋白2 抑制剂,可促进尿液中葡萄糖的排泄,可用于糖尿病的研究。它诱导 HIF1表达并减轻肾脏 IR 损伤。
T28743 Seglitide acetate

MK 678,MK678,MK-678

Somatostatin GPCR/G Protein
Seglitide acetate (MK-678) 是一种选择性的 sst2生长抑素受体激动剂。
T23358 Sitagliptin phosphate

磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)

DPP-4; Autophagy Autophagy; Proteases/Proteasome
Sitagliptin phosphate (MK-0431 phosphate) 是一种二肽基肽酶 4 (DPP4) 抑制剂,在 Caco-2 细胞中,IC50值为 19 nM。
T2401 Alogliptin Benzoate

苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate

Ferroptosis; Proteasome; DPP-4 Apoptosis; Proteases/Proteasome; Ubiquitination
Alogliptin Benzoate (SYR 322) 是一种有效且特异性的 DPP-4 抑制剂 ,IC50值小于 10 nM,其选择性比 DPP-8/9 高 10,000 倍以上,可用于研究 2 型糖尿病。
T27841 Lobeglitazone Sulfate

CKD501 Sulfate,CKD501,CKD-501 Sulfate,CKD 501 Sulfate,CKD 501,CKD-501,Lobeglitazone Sulfate. trade name Duvie, Chong Kun Dang

NOD Immunology/Inflammation; NF-κB
Lobeglitazone Sulfate(CKD-501 Sulfate) 是一种新型噻唑烷二酮,具有抗炎活性,抑制LPS诱导的NLRP3炎症小体活化和肝脏炎症,可用于研究 2 型糖尿病 (T2DM)。
T14176 Aleglitazar

RO0728804,R1439

PPAR DNA Damage/DNA Repair; Metabolism
Aleglitazar (R1439) 是一种高效的 PPARα/γ 双重激动剂,对人 PPARα 和 PPARγ 作用的 IC50 分别为 38 nM 和 19 nM。Aleglitazar 可用于 II 型糖尿病的研究。
T1875 Atglistatin

Lipase Metabolism
Atglistatin 是脂肪甘油三酯脂酶的选择性抑制剂(IC50:0.7 μM),在体外具有抑制脂解的功能。
T68053 Denagliptin

GW823093

DPP-4 Proteases/Proteasome
Denagliptin是一种小分子二肽基肽酶IV(DPP-4)抑制剂,可用于治疗内分泌于代谢疾病,可用于研究2型糖尿病。
T17044 Tesaglitazar

PPAR DNA Damage/DNA Repair; Metabolism
Tesaglitazar 是一种有效且具有选择性的过氧化物 PPAR α / γ受体双重激动剂,对 PPARγ的亲和力比 PPARα更有效,对大鼠PPARα和人PPARα的EC50分别为13.4 μM 和3.6 μM,对大鼠PPARγ和人类 PPARγ的EC50都是0.2 μM。Tesaglitazar 诱导大鼠皮下组织间质间充质细胞DNA 合成和纤维肉瘤形成。
T2389 Dapagliflozin

达格列净,BMS-512148

SGLT; HIF Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein
Dapagliflozin (BMS-512148) 是一种葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可与靶点竞争性结合。Dapagliflozin 可用于 2 型糖尿病的治疗,可以减少肾脏的葡萄糖重吸收,增加尿液中葡萄糖的排泄,从而降低血浆葡萄糖水平。
T22860 Imeglimin

EMD 387008,EMD-387008,RVT-1501,PXL 008

ROS; Mitochondrial Metabolism Immunology/Inflammation; Metabolism
Imeglimin (EMD 387008) 是一种可口服的抗糖尿病化合物,可增强线粒体功能、增强胰岛素分泌、促进β细胞增殖并改善小鼠胰岛β细胞存活率。
T1782 Canagliflozin

卡格列净,JNJ 24831754ZAE,JNJ 28431754AAA,TA 7284,JNJ 28431754

SGLT GPCR/G Protein
Canagliflozin (JNJ 28431754AAA) 是SGLT2的选择性抑制剂,在表达 mSGLT2,rSGLT2 和 hSGLT2 的 CHO 细胞上,IC50分别为 2 nM,3.7 nM 和 4.4 nM。
T0127 Glimepiride

Glimperide,HOE-490,格列美脲

Potassium Channel Membrane transporter/Ion channel
Glimepiride (HOE-490) 是一种中长效的磺酰脲类抗糖尿病化合物,其 ED50=182 μg/k。
T7217 Bexagliflozin

THR-1442,EGT1442,EGT0001442

SGLT GPCR/G Protein
Bexagliflozin (EGT1442) 是一种选择性的,口服有效的钠葡萄糖协同转运蛋白-2 (SGLT2) 抑制剂,对人 SGLT2 和 SGLT1 作用的 IC50值分别为 2 nM 和 5.6 μM。EGT1442在 2 型糖尿病中有研究价值。
T7369L Gemigliptin Tartrate(911637-19-9 free base)

吉格列汀酒石酸盐,LC15-0444 tartrate

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Gemigliptin Tartrate (LC15-0444 tartrate) 是一种选择性的,可逆的,竞争性的二肽基肽酶 4 (DPP-4) 抑制剂,对于人重组 DPP-4 的IC50=10.3 nM。Gemigliptin tartrate 具有很强的抗糖基化活性,能够用于晚期糖基化终产物相关的糖尿病并发症的研究。
T6999 Teneligliptin hydrobromide

Teneligliptin hydrobromide anhydrous,MP-513 (hydrobromide)

Others; Proteasome; DPP-4 Others; Proteases/Proteasome; Ubiquitination
Teneligliptin hydrobromide (MP-513(hydrobromide)) 是β2肾上腺素能受体 (β2AR) 阻滞剂,具有抗高血压、抗氧化、清除自由基的活性。
T7369 Gemigliptin

吉格列汀酒石酸盐,LC15-0444

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Gemigliptin (LC15-0444) 是一种选择性的,可逆的,竞争性的二肽基肽酶 4 (DPP-4) 抑制剂,对人重组 DPP-4 的 IC50=10.3 nM。Gemigliptin 具有很强的抗糖基化活性,能够用于晚期糖基化终产物相关的糖尿病并发症的研究。

化合物

HPI 1
Cat.No: T22089
Synonym:
Target: Hedgehog/Smoothened
IHR-1
Cat.No: T24159
Synonym: IHR 1
Target: Smo
GANT 58
Cat.No: T15370
Synonym: 4,44乔,4乔(2,3,4,5-Thiophentetrayl)tetrakis-pyridine,NSC 75503
Target: Hedgehog/Smoothened
GANT 61
Cat.No: T3070
Synonym: NSC 136476,GANT61
Target: Hedgehog/Smoothened, Autophagy
Saxagliptin
Cat.No: T6203
Synonym: BMS-477118,沙克列汀,Onglyza,沙格列汀
Target: Proteasome, DPP-4
Retagliptin Phosphate
Cat.No: T12710
Synonym: SP 2086,瑞格列汀磷酸盐
Target: Proteasome, DPP-4
Glimepiride sulfonamide
Cat.No: T64332
Synonym:
Target: Immunology/Inflammation related
Sergliflozin etabonate
Cat.No: T28757
Synonym: GW-869682,GW-869682X,KGT-1251,GW869682X,GW869682,KGT1251
Target: SGLT
Remogliflozin etabonate
Cat.No: T34286
Synonym: GSK189075,GSK 189075,GSK-189075A,GSK189075A,GSK-189075,GSK 189075A
Target: SGLT
Ipragliflozin
Cat.No: T2385
Synonym: 伊格列净,ASP1941
Target: SGLT
Linagliptin
Cat.No: T0191
Synonym: BI 1356,利格列汀,利拉利汀
Target: Ferroptosis, Proteasome, DPP-4, Autophagy
Vildagliptin
Cat.No: T1502
Synonym: 维达列汀,NVP-LAF 237,维格列汀,LAF237
Target: Apoptosis, Ferroptosis, Proteasome, DPP-4
Sitagliptin phosphate monohydrate
Cat.No: T0242L
Synonym: MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物
Target: Proteasome, DPP-4, Autophagy
Saroglitazar
Cat.No: T12835
Synonym: Lipaglyn
Target: PPAR
Deriglidole
Cat.No: T10998
Synonym: SL 86-0715
Target: Adrenergic Receptor
Glibenclamide
Cat.No: T1634
Synonym: 格列本脲,Glyburide
Target: Potassium Channel, Mitochondrial Metabolism, CFTR, P-gp, Autophagy
Ciglitazone
Cat.No: T19710
Synonym: Ciglitazona,U 63287,ADD3878,ADD-3878,U-63287,ADD 3878
Target: Apoptosis, p38 MAPK, PPAR
Azemiglitazone
Cat.No: T4639
Synonym: MSDC 0602
Target: Mitochondrial Metabolism, mTOR
Pioglitazone
Cat.No: T0214
Synonym: U 72107,吡格列酮,匹格列酮
Target: Ferroptosis, PPAR
Globalagliatin
Cat.No: T3104
Synonym: LY2608204
Target: Glucokinase
Cevoglitazar
Cat.No: T26986
Synonym: LBM-642,LBM 642,LBM642
Target: PPAR
Managlinat dialanetil
Cat.No: T16009L
Synonym: MB06322,MB 6322,CS-917
Target: Phosphatase
Trelagliptin
Cat.No: T6237
Synonym: SYR-472,曲格列汀
Target: Proteasome, DPP-4
Darglitazone
Cat.No: T22708
Synonym: CP-86325
Target: PPAR
Rosiglitazone maleate
Cat.No: T1622
Synonym: BRL 49653C,BRL 49653,马来酸罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Indeglitazar
Cat.No: T15575
Synonym: PPM 204
Target: PPAR
Ragaglitazar
Cat.No: T28501
Synonym: NNC61-0029,NN-622,(-)-DRF-2725,NNC-61-0029,NN 622,NNC 61-0029
Target: PPAR
Mizagliflozin
Cat.No: T16083
Synonym: GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base
Target: SGLT
Imeglimin hydrochloride
Cat.No: T7486
Synonym: EMD 387008 hydrochloride,(6R)-1,6-二氢-N2,N2,6-三甲基-1,3,5-三嗪-2,4-二胺盐酸盐
Target: Reactive Oxygen Species, Mitochondrial Metabolism
Nateglinide
Cat.No: T1674
Synonym: 那格列奈,A4166,Senaglinide
Target: Potassium Channel, Proteasome, PPAR
Anagliptin
Cat.No: T7133
Synonym: SK-0403,阿拉格列汀
Target: Proteasome, DPP-4
Rosiglitazone
Cat.No: T0334
Synonym: BRL49653,罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Saxagliptin hydrate
Cat.No: T0178
Synonym: 沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate
Target: Proteasome, DPP-4
Dapagliflozin ((2S)-1,2-propanediol, hydrate)
Cat.No: T4460
Synonym: BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate
Target: SGLT
Seglitide acetate
Cat.No: T28743
Synonym: MK 678,MK678,MK-678
Target: Somatostatin
Sitagliptin phosphate
Cat.No: T23358
Synonym: 磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)
Target: DPP-4, Autophagy
Alogliptin Benzoate
Cat.No: T2401
Synonym: 苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate
Target: Ferroptosis, Proteasome, DPP-4
Lobeglitazone Sulfate
Cat.No: T27841
Synonym: CKD501 Sulfate,CKD501,CKD-501 Sulfate,CKD 501 Sulfate,CKD 501,CKD-501,Lobeglitazone Sulfate. trade name Duvie, Chong Kun Dang
Target: NOD
Aleglitazar
Cat.No: T14176
Synonym: RO0728804,R1439
Target: PPAR
Atglistatin
Cat.No: T1875
Synonym:
Target: Lipase
Denagliptin
Cat.No: T68053
Synonym: GW823093
Target: DPP-4
Tesaglitazar
Cat.No: T17044
Synonym:
Target: PPAR
Dapagliflozin
Cat.No: T2389
Synonym: 达格列净,BMS-512148
Target: SGLT, HIF
Imeglimin
Cat.No: T22860
Synonym: EMD 387008,EMD-387008,RVT-1501,PXL 008
Target: ROS, Mitochondrial Metabolism
Canagliflozin
Cat.No: T1782
Synonym: 卡格列净,JNJ 24831754ZAE,JNJ 28431754AAA,TA 7284,JNJ 28431754
Target: SGLT
Glimepiride
Cat.No: T0127
Synonym: Glimperide,HOE-490,格列美脲
Target: Potassium Channel
Bexagliflozin
Cat.No: T7217
Synonym: THR-1442,EGT1442,EGT0001442
Target: SGLT
Gemigliptin Tartrate(911637-19-9 free base)
Cat.No: T7369L
Synonym: 吉格列汀酒石酸盐,LC15-0444 tartrate
Target: Proteasome, DPP-4
Teneligliptin hydrobromide
Cat.No: T6999
Synonym: Teneligliptin hydrobromide anhydrous,MP-513 (hydrobromide)
Target: Others, Proteasome, DPP-4
Gemigliptin
Cat.No: T7369
Synonym: 吉格列汀酒石酸盐,LC15-0444
Target: Proteasome, DPP-4
Cat. No. Product Name Target Signaling Pathways
T6723 Voglibose

AO 128,伏格列波糖,Glustat,Basen

Glucosidase Metabolism
Voglibose (Glustat) 是一种 valiolamine 的衍生物,可抑制α-葡萄糖苷酶活性,可作用于高血糖症等。
T5542 Tiglic acid

惕格酸,Sabadillic acid,Tiglinic acid,巴豆酸,Cevadic acid

Endogenous Metabolite; HSV Metabolism; Microbiology/Virology
Tiglic acid 是一种存在于巴豆油和其他几种天然产物中的单羧酸不饱和有机酸。它具有植物代谢物的作用。
T1529 Miglitol

BAY1099,米格列醇,BAY-m1099

Others Others
Miglitol (BAY1099) 是一种口服抗糖尿病化合物,能够抑制糖复合体分解为葡萄糖。
TN3520 Bisdethiobis(methylthio)gliotoxin

PAFR GPCR/G Protein
Bisdethiobis(methylthio)gliotoxin is a platelet activating factor (PAF) antagonist.
TN6086 Machigline

Machigline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6086,CAS号为 87264-30-0。
TN4137 Glicoricone

MAO Metabolism; Neuroscience
Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M.
TN3362 Aglinin A

Others Others
Aglinin A displays moderate cytotoxicity against all the three cancer cell lines((NCI-H187), epidermoid carcinoma (KB) and breast cancer (BC) cell lines).
T41304 Hydroaurantiogliocladin

Hydroaurantiogliocladin 在生命科学相关研究中具有广泛的应用。
T82341 Ganglioside GM1

Ganglioside GM1,一种神经节苷脂家族成员,用于神经系统疾病研究。同时,它作为霍乱毒素 1 的功能性组织受体。
T35741 Gliovirin

Others Others
Gliovirin is a fungal metabolite that has been found inT. harzianumand has fungicidal, antimicrobial and anti-inflammatory activities.1It is active against the plant pathogenic fungusP. ultimum(MIC = 60 ng/ml) and the parasiteT. brucei brucei(IC50= 90 ng/ml), but has no effect on the plant pathogenic fungiR. solani,P. omnivorum,T. basicola,R. arrhizus, andV. dahliaeor the bacteriaB. thuringiensis,P. fluorescens, andX. malvacearumwhen used at concentrations up to 1,000 ng/ml.2,3Gliovirin decrease...
T31935 Gliorosein

Others Others
Gliorosein is a biohcemical.
TN5409 Maglifloenone

Denudatone

Maglifloenone是一种天然产物,属于木兰科木兰属,其产品编号为 TN5409,CAS号为 82427-77-8。Maglifloenone可用作对照参考。
T74200 Glicophenone

Others Others
Glicophenone 作为一种抗细菌(antibacterial)剂,对MRSA OM481、MRSA OM505、MRSA OM584、MRSA OM623 以及MSSA 209P的MIC值均为32 μg/mL。
T82277 GM1a Ganglioside oligosaccharide

GM1a Ganglioside oligosaccharide为ganglioside GM1的半合成形式,后者作为霍乱毒素的天然受体,在生长调节及激素诱导反应的耦合中具有关键功能。
T82339 Gangliotetraose

Gg4

Gangliotetraose(Gg4)是一种含有GM1及其唾液酸化衍生物的四糖。它能促进分化神经元核内Ca2+的外流,进而降低核内Ca2+浓度。Gg4参与调节神经元的可塑性、修复过程以及大脑中神经营养素的释放。
TN1694 Gliotoxin

Apoptosis; NF-κB; Wnt/beta-catenin; COX; PKA; Antibacterial; Antifection Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Gliotoxin 是一种次生代谢产物,由A. fumigatus 分泌,可以抑制巨噬细胞的吞噬作用和其他免疫细胞的免疫功能。它通过阻止 IκB 降解来抑制诱导型NF-κB 活性,从而诱导宿主细胞凋亡。它可以激活PKA 并增加细胞内 cAMP 浓度,调节肌动蛋白细胞骨架重排以促进A. fumigatus 内化到肺上皮细胞。
TN1379 Alphitolic acid

麦珠子酸

NF-κB; Akt; p53 Apoptosis; Cytoskeletal Signaling; NF-κB; PI3K/Akt/mTOR signaling
Alphitolic acid is a potent Hh/GLI signaling inhibitor, it shows an important relationship between Hh/GLI signaling inhibition, the decrease of BCL2, and cytotoxicity against cancer cells.

天然产物

Voglibose
Cat.No: T6723
Synonym: AO 128,伏格列波糖,Glustat,Basen
Target: Glucosidase
Tiglic acid
Cat.No: T5542
Synonym: 惕格酸,Sabadillic acid,Tiglinic acid,巴豆酸,Cevadic acid
Target: Endogenous Metabolite, HSV
Miglitol
Cat.No: T1529
Synonym: BAY1099,米格列醇,BAY-m1099
Target: Others
Bisdethiobis(methylthio)gliotoxin
Cat.No: TN3520
Synonym:
Target: PAFR
Machigline
Cat.No: TN6086
Synonym:
Target:
Glicoricone
Cat.No: TN4137
Synonym:
Target: MAO
Aglinin A
Cat.No: TN3362
Synonym:
Target: Others
Hydroaurantiogliocladin
Cat.No: T41304
Synonym:
Target:
Ganglioside GM1
Cat.No: T82341
Synonym:
Target:
Gliovirin
Cat.No: T35741
Synonym:
Target: Others
Gliorosein
Cat.No: T31935
Synonym:
Target: Others
Maglifloenone
Cat.No: TN5409
Synonym: Denudatone
Target:
Glicophenone
Cat.No: T74200
Synonym:
Target: Others
GM1a Ganglioside oligosaccharide
Cat.No: T82277
Synonym:
Target:
Gangliotetraose
Cat.No: T82339
Synonym: Gg4
Target:
Gliotoxin
Cat.No: TN1694
Synonym:
Target: Apoptosis, NF-κB, Wnt/beta-catenin, COX, PKA, Antibacterial, Antifection
Alphitolic acid
Cat.No: TN1379
Synonym: 麦珠子酸
Target: NF-κB, Akt, p53
Cat. No. Product Name Species Expression System
TMPH-02321 GLI1 Protein, Human, Recombinant (His)

Zinc finger protein GLI1,Glioma-associated...

Human E. coli
Acts as a transcriptional activator. Binds to the DNA consensus sequence 5'-GACCACCCA-3'. Regulates the transcription of specific genes during normal development. Plays a role in craniofacial development and digital development, as well as development of the central nervous system and gastrointestinal tract. Mediates SHH signaling. Plays a role in cell proliferation and differentiation via its role in SHH signaling.; Acts as a transcriptional activator, but activates a different set of genes tha...
TMPY-01457 GLIPR1 Protein, Human, Recombinant (His)

RTVP1,GLI pathogenesis-related 1,CRISP7,GLI

Human HEK293 Cells
GLIPR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.7 kDa and the accession number is P48060-1.
TMPY-03940 GLIPR1 Protein, Mouse, Recombinant (His)

RTVP-1,2410114O14Rik,mRTVP-1,GLI pathogenesis-relat...

Mouse HEK293 Cells
GLIPR1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.1 kDa and the accession number is Q4QQK5.
TMPY-01384 Endoglin/CD105 Protein, Human, Recombinant (His)

endoglin,HHT1,END,ORW1

Human HEK293 Cells
Endoglin/CD105 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 62.3 kDa and the accession number is A0A024R878.
TMPY-00783 Endoglin/CD105 Protein, Human, Recombinant (hFc)

END,HHT1,ORW1,endoglin

Human HEK293 Cells
Endoglin/CD105 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 87.5 kDa and the accession number is A0A024R878.
TMPH-03646 Omega-gliadin Protein, Triticum monococcum, Recombinant (E. coli, GST)

Omega-gliadin

Triticum monococcum E. coli
N/A. Omega-gliadin Protein, Triticum monococcum, Recombinant (E. coli, GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 30.3 kDa and the accession number is P02865.
TMPY-04227 Gliomedin Protein, Human, Recombinant (hFc)

COLM,CRGL2,UNC-112,gliomedin,CRG-L2,CLOM

Human HEK293 Cells
Gliomedin Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 74.3 kDa and the accession number is AAQ88511.1.
TMPY-06725 Jug r 1 Protein, English walnut, Recombinant

English walnut E. coli
Jug r 1 Protein, English walnut, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.3 kDa.
TMPY-01615 Endoglin/CD105 Protein, Mouse, Recombinant (His)

Endo,CD105,S-endoglin,AI528660,endoglin,AI...

Mouse HEK293 Cells
Endoglin/CD105 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 61.2 kDa and the accession number is Q63961.
TMPH-03647 Omega-gliadin Protein, Triticum monococcum, Recombinant (GST)

Omega-gliadin

Triticum monococcum P. pastoris (Yeast)
N/A. Omega-gliadin Protein, Triticum monococcum, Recombinant (GST) is expressed in yeast with N-GST tag. The predicted molecular weight is 30.3 kDa and the accession number is P02865.
TMPK-00359 Endoglin/CD105 Protein, Human, Recombinant (His & Avi)

CD105,ORW,ORW1,ENG,END,Endoglin,HHT1

Human HEK293 Cells
Endoglin (CD105) is a 90 kDa type I transmembrane glycoprotein of the zona pellucida (ZP) family of proteins. Endoglin is a vascular endothelium glycoprotein that plays an important role in the regulation of angiogenesis. Required for normal structure and integrity of adult vasculature (PubMed:7894484). Regulates the migration of vascular endothelial cells. Required for normal extraembryonic angiogenesis and for embryonic heart development. May regulate endothelial cell shape changes in response...
TMPJ-00361 Endoglin Protein, Human, Recombinant (Trx & His)

CD105,END,Endoglin,ENG

Human E. coli
Endoglin is a single-pass type I membrane protein which restricted to endothelial cells in all tissues except bone marrow. Endoglin as major glycoprotein of vascular endothelium, it has been found on endothelial cells, activated macrophages, fibroblasts, and smooth muscle cells. Furthermore, Homodimer forms a heteromeric complex with the signaling receptors for transforming growth factor-beta: TGFBR1 and/or TGFBR2. It may have an important role in the binding of endothelial cells to integrins an...

重组蛋白

GLI1 Protein, Human, Recombinant (His)
Cat.No: TMPH-02321
Species: Human
Expression System: E. coli
GLIPR1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01457
Species: Human
Expression System: HEK293 Cells
GLIPR1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-03940
Species: Mouse
Expression System: HEK293 Cells
Endoglin/CD105 Protein, Human, Recombinant (His)
Cat.No: TMPY-01384
Species: Human
Expression System: HEK293 Cells
Endoglin/CD105 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00783
Species: Human
Expression System: HEK293 Cells
Omega-gliadin Protein, Triticum monococcum, Recombinant (E. coli, GST)
Cat.No: TMPH-03646
Species: Triticum monococcum
Expression System: E. coli
Gliomedin Protein, Human, Recombinant (hFc)
Cat.No: TMPY-04227
Species: Human
Expression System: HEK293 Cells
Jug r 1 Protein, English walnut, Recombinant
Cat.No: TMPY-06725
Species: English walnut
Expression System: E. coli
Endoglin/CD105 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01615
Species: Mouse
Expression System: HEK293 Cells
Omega-gliadin Protein, Triticum monococcum, Recombinant (GST)
Cat.No: TMPH-03647
Species: Triticum monococcum
Expression System: P. pastoris (Yeast)
Endoglin/CD105 Protein, Human, Recombinant (His & Avi)
Cat.No: TMPK-00359
Species: Human
Expression System: HEK293 Cells
Endoglin Protein, Human, Recombinant (Trx & His)
Cat.No: TMPJ-00361
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMIH-0517 Saroglitazar oxide-d4

Saroglitazar oxide-d4 是 Saroglitazar oxide 的氘代化合物。Saroglitazar oxide 的 CAS 号为 495399-09-2。Saroglitazar 是 PPAR 的激动剂,对 PPARα 和 PPARγ 的 EC50 值为 0.65 pM 和 3 nM。
TMIH-0253 Gliclazide-d7

Gliclazide-d7 是 Gliclazide 的氘代化合物。Gliclazide 的 CAS 号为 21187-98-4。Gliclazide 是一种有效的全细胞的 β 细胞 ATP 敏感型钾流阻断剂,IC50为 184 nM,用作降糖药。
TMIH-0516 Saroglitazar-d4

Saroglitazar-d4 是 Saroglitazar 的氘代化合物。Saroglitazar 的 CAS 号为 495399-09-2。Saroglitazar 是 PPAR 的激动剂,对 PPARα 和 PPARγ 的 EC50 值为 0.65 pM 和 3 nM。
T10669 Canagliflozin-d4

Canagliflozin D4

Others Others
Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.
TMIJ-0142 Vildagliptin-d7

Vildagliptin-d7 是 Vildagliptin 的氘代化合物。Vildagliptin 的 CAS 号为 274901-16-5。Vildagliptin 是一种选择性二肽基肽酶IV (DPP-IV) 抑制剂,在人 Caco-2 细胞中抑制 DPP-IV 的IC50为 3.5 nM。它具有出色的口服生物利用度和降血糖活性。
TMIJ-0126 5-Hydroxy Saxagliptin-13C-d2 HCl

5-Hydroxy Saxagliptin-13C-d2 HCl 是 5-Hydroxy Saxagliptin HCl 的 13C 和氘代化合物。5-Hydroxy Saxagliptin HCl 的 CAS 号为 841302-24-7。
T19548 Repaglinide D5

AG-EE 623ZW D5,瑞格列奈 D5

Others Others
Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.
TMIH-0302 Linagliptin-d4

Linagliptin-d4 是 Linagliptin 的氘代化合物。Linagliptin 的 CAS 号为 668270-12-0。Linagliptin 是一种有效的、可口服的、基于二氢嘌呤二酮的二肽基肽酶 4 抑制剂,具有降血糖活性。
TMIH-0013 (S)-Empagliflozin-d4

(S)-Empagliflozin-d4 是 (S)-Empagliflozin 的氘代化合物。(S)-Empagliflozin 的 CAS 号为 864070-44-0。Empagliflozin 是有效的、选择性的钠葡萄糖协同转运蛋白-2 (SGLT-2) 抑制剂,对人 SGLT-2 的IC50为 3.1 nM。
TMIJ-0153 Dapagliflozin-13C6 (glucitol-13C6)

Dapagliflozin-13C6 (glucitol-13C6) 是 Dapagliflozin 的 13C 的标记化合物。Dapagliflozin 的 CAS 号为 461432-26-8。Dapagliflozin竞争性的葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可促进尿液中葡萄糖的排泄,在糖尿病 (DM) 研究中具有价值。Dapagliflozin 诱导HIF1表达并减轻肾脏 IR 损伤。
T10288 Alogliptin (13CD3)

SYR-322 (13CD3)

Others Others
Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.
TMIH-0010 (S)-Alogliptin Benzoate Salt-13C-d3

(S)-Alogliptin Benzoate Salt-13C-d3 是 (S)-Alogliptin Benzoate Salt 的 13C 和氘代化合物。
TMIH-0045 3-Hydroxy Repaglinide-d5

3-Hydroxy Repaglinide-d5 是 3-Hydroxy Repaglinide 的氘代化合物。
TMIJ-0133 Empagliflozin-d4

Empagliflozin-d4 是 Empagliflozin 的氘代化合物。Empagliflozin 的 CAS 号为 864070-44-0。Empagliflozin 是有效的、选择性的钠葡萄糖协同转运蛋白-2 (SGLT-2) 抑制剂,对人 SGLT-2 的IC50为 3.1 nM。
TMIJ-0156 rac-Sitagliptin-d4 HCl

rac-Sitagliptin-d4 HCl 是 rac-Sitagliptin HCl 的氘代化合物。
TMIJ-0143 Linagliptin-13C-d3

Linagliptin-13C-d3 是 Linagliptin 的 13C 和氘代化合物。Linagliptin 的 CAS 号为 668270-12-0。Linagliptin 是一种有效的、可口服的、基于二氢嘌呤二酮的二肽基肽酶 4 抑制剂,具有降血糖活性。
T71981 Gliclazide-d4

Gliclazide-d4 is intended for use as an internal standard for the quantification of gliclazide by GC- or LC-MS. Gliclazide is a sulfonylurea and an inhibitor of pancreatic β-cell ATP-sensitive potassium (KATP) channels. It is selective for pancreatic β-cell over cardiac and arterial smooth muscle cell KATP channels. Gliclazide (5 μM) increases insulin-induced glucose uptake and glucose transporter 4 (GLUT4) translocation to the plasma membrane in a differentiated 3T3L1 adipocyte model of insulin...
TMIH-0267 Hydroxy Pioglitazone M-IV-d4

Hydroxy Pioglitazone M-IV-d4 是 Hydroxy Pioglitazone M-IV 的氘代化合物。
T12178 Nateglinide D5

Senaglinide D5,A4166 D5

Others Others
Nateglinide D5 is a deuterium labeled Nateglinide.
T12479 Pioglitazone-d4

U 72107 D4

Others Others
Pioglitazone D4 is a deuterium labeled Pioglitazone. Pioglitazone is a agonist of PPARγ .
TMIH-0583 Trelagliptin-13C-d3

Trelagliptin-13C-d3 是 Trelagliptin 的 13C 和氘代化合物。Trelagliptin 的 CAS 号为 865759-25-7。Trelagliptin 是一种有效的,具有口服活性的DPP-4抑制剂,IC50=4 nM。它可以改善体内血糖控制,能够用于2 型糖尿病 (T2DM) 的研究。
T10958 Dapagliflozin-d5

BMS-512148 D5

Others Others
Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.
T13121 Teneligliptin D8

MP-513 D8

Others Others
Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.
TMIJ-0093 Keto Pioglitazone-d4

Keto Pioglitazone-d4 是 Keto Pioglitazone 的氘代化合物。Keto Pioglitazone 的 CAS 号为 146062-45-5。
TMID-0267 Glipizide-d11

Glipizide-d11 是 Glipizide 的氘代化合物。Glipizide 的 CAS 号为 29094-61-9。Glipizide 是一种有效的、具有口服活性的磺酰脲类抗糖尿病试剂 (anti-diabetic agent),在 2 型糖尿病的研究中具有价值,但不适用于1 型糖尿病。Glipizide 是通过部分阻断郎格汉斯胰岛细胞中 ATP 敏感钾通道 (KATP)发挥活性 。
TMIJ-0523 Gliquidone-d6

Gliquidone-d6 是 Gliquidone 的氘代化合物。Gliquidone 的 CAS 号为 33342-05-1。Gliquidone 是一种磺酰脲类的抗糖尿病药物,可用于2型糖尿病的研究。

同位素标记化合物

Saroglitazar oxide-d4
Cat.No: TMIH-0517
Synonym:
Target:
Gliclazide-d7
Cat.No: TMIH-0253
Synonym:
Target:
Saroglitazar-d4
Cat.No: TMIH-0516
Synonym:
Target:
Canagliflozin-d4
Cat.No: T10669
Synonym: Canagliflozin D4
Target: Others
Vildagliptin-d7
Cat.No: TMIJ-0142
Synonym:
Target:
5-Hydroxy Saxagliptin-13C-d2 HCl
Cat.No: TMIJ-0126
Synonym:
Target:
Repaglinide D5
Cat.No: T19548
Synonym: AG-EE 623ZW D5,瑞格列奈 D5
Target: Others
Linagliptin-d4
Cat.No: TMIH-0302
Synonym:
Target:
(S)-Empagliflozin-d4
Cat.No: TMIH-0013
Synonym:
Target:
Dapagliflozin-13C6 (glucitol-13C6)
Cat.No: TMIJ-0153
Synonym:
Target:
Alogliptin (13CD3)
Cat.No: T10288
Synonym: SYR-322 (13CD3)
Target: Others
(S)-Alogliptin Benzoate Salt-13C-d3
Cat.No: TMIH-0010
Synonym:
Target:
3-Hydroxy Repaglinide-d5
Cat.No: TMIH-0045
Synonym:
Target:
Empagliflozin-d4
Cat.No: TMIJ-0133
Synonym:
Target:
rac-Sitagliptin-d4 HCl
Cat.No: TMIJ-0156
Synonym:
Target:
Linagliptin-13C-d3
Cat.No: TMIJ-0143
Synonym:
Target:
Gliclazide-d4
Cat.No: T71981
Synonym:
Target:
Hydroxy Pioglitazone M-IV-d4
Cat.No: TMIH-0267
Synonym:
Target:
Nateglinide D5
Cat.No: T12178
Synonym: Senaglinide D5,A4166 D5
Target: Others
Pioglitazone-d4
Cat.No: T12479
Synonym: U 72107 D4
Target: Others
Trelagliptin-13C-d3
Cat.No: TMIH-0583
Synonym:
Target:
Dapagliflozin-d5
Cat.No: T10958
Synonym: BMS-512148 D5
Target: Others
Teneligliptin D8
Cat.No: T13121
Synonym: MP-513 D8
Target: Others
Keto Pioglitazone-d4
Cat.No: TMIJ-0093
Synonym:
Target:
Glipizide-d11
Cat.No: TMID-0267
Synonym:
Target:
Gliquidone-d6
Cat.No: TMIJ-0523
Synonym:
Target:
共226条,每页50条 1 2 3 4 5
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼