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Search Results for " glutamate "
Targets Recommended: Others

425

抑制剂 & 化合物

70

天然产物

3

化合物库

53

重组蛋白

8

同位素标记化合物

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Cat. No. Product Name
L2550 谷氨酰胺代谢化合物库

565 compounds
565 种谷氨酰胺代谢相关的分子,可以用于高通量和高内涵筛选;
L2610 神经递质受体化合物库

1513 compounds
1513 种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
L9830 抗帕金森病化合物库

857 compounds
857 种帕金森病相关的化合物集合,可用于高通量和高内涵筛选;

化合物库

谷氨酰胺代谢化合物库
Cat.No: L2550
Compounds: 565
神经递质受体化合物库
Cat.No: L2610
Compounds: 1513
抗帕金森病化合物库
Cat.No: L9830
Compounds: 857
Cat. No. Product Name Target Signaling Pathways
T20365 Monopotassium glutamate

L-谷氨酸钾盐,Potassium glutamate,Potassium L-glutamate

Others Others
Monopotassium glutamate (Potassium glutamate) 可在食品中用作增味剂。
T20266 Tetrasodium glutamate diacetate

Glutamate diacetate tetrasodium,GLDA

Others Others
Tetrasodium glutamate diacetate (Glutamate diacetate tetrasodium) 是一种可降解螯合剂,可用作膳食成分,可从废活性污泥 (WAS) 絮凝体中提取多价金属离子,可增强废活性污泥中挥发性脂肪酸的产生。
T7658 Dimethyl DL-Glutamate (hydrochloride)

Others Others
Dimethyl DL-Glutamate (hydrochloride) 是一种细胞渗透性谷氨酸衍生物,可在孤立的胰岛和糖尿病动物模型中增强胰岛素释放以响应葡萄糖。
T20331 Sodium lauroyl glutamate

Hostapon CLG,Amisoft LS 11,Sodium N-lauroylglutamate,月桂酰谷氨酸钠,Acylglutamate LS-11

Others Others
Sodium lauroyl glutamate (Acylglutamate LS-11) 是一种氨基酸去污剂,可增加长链没食子酸烷基酯(如没食子酸烷基酯)的溶解度。
T72460 Dimethyl L-glutamate

Dimethyl glutamate

Dimethyl L-glutamate (Dimethyl glutamate), 一种可透膜的谷氨酸类似物,可刺激葡萄糖诱导的胰岛素 (insulin) 释放。Dimethyl L-glutamate 抑制KATP 通道的活性。Dimethyl L-glutamate 抑制E. gracilis 生长并导致细胞异常分裂。Dimethyl L-glutamate 可用于糖尿病、葡萄糖转运、磷酸化和进一步代谢的研究。
T40973 MDNI-caged-L-glutamate

MDNI-caged-L-glutamate,MDNI-glu

Others Others
MDNI-glu is a photosensitive derivative of L-glutamate, a major excitatory amino acid, that is biologically inert. It demonstrates improved utilization of incident light.
T35369 L(+)-Monosodium glutamate monohydrate

L(+)-Monosodium glutamate monohydrate,MSG monohydrate,L-Glutamic acid monosodium salt monohydrate,Monosodium L-glutamate monohydrate

Others Others
L(+)-Monosodium glutamate monohydrate (MSG monohydrate, L-Glutamic acid monosodium salt monohydrate, Monosodium L-glutamate monohydrate, Monosodium L-glutamate monohydrate)是一种广泛使用的营养添加剂和调味剂。L(+)-Monosodium glutamate monohydrate 可导致氧化应激介导的 DNA 损伤和细胞凋亡。
T34938 Triethanolamine linoleoyl glutamate

TEA-linoleoyl glutamate

Others Others
Triethanolamine linoleoyl glutamate is a bioactive chemical.
T34677 Sodium palmitoyl glutamate

Sodium N-palmitoyl-L-glutamate,Monosodium N-palmitoyl-L-glutamate

Others Others
Sodium palmitoyl glutamate is a amino acid.
T73616 Glutamate dehydrogenase (NAD(P))

GLDH

Mitochondrial Metabolism Metabolism
Glutamate dehydrogenase NAD(P) (GLDH)是一种线粒体酶,广泛存在于生物体内,催化谷氨酸可逆的氧化脱氨生成 α-酮戊二酸 (α-KG),可用于研究谷氨酸代谢异常引起的疾病。
T23278 RuBi-Glutamate

Others Others
Ruthenium-bipyridine-trimethylphosphine caged glutamate
T31266 Deanol glutamate

Others Others
Deanol glutamate is a central stimulant.
T31941 Glutamate cobalt

Others Others
Glutamate cobalt is a bioactive chemical.
T33724 Norfloxacin glutamate

Others Others
Norfloxacin glutamate is a bioactive chemical.
T34937 Triethanolamine glutamate

Others Others
Triethanolamine glutamate is a bioactive chemical.
T24043 Erythromycin glutamate

Others Others
Erythromycin glutamate is a macrolide bacteriostatic antibiotic. This antibiotic is metabolized through the liver and inhibits cytochrome enzyme P450A 3A41.
T34675 Sodium linoleoyl glutamate

Others Others
Sodium linoleoyl glutamate is salt obtained from linoleoyl glutamate.
T33326 Methotrexate-alpha glutamate

Meapa-glu-glu

Others Others
Methotrexate-alpha glutamate is a chemotherapy agent and immune system suppressant. It is used to treat cancer, autoimmune diseases, ectopic pregnancy, and medical abortions.
T31518 Dipinacoline glutamate

L-Glutamic acid dipinacoline ester,DiPG

Others Others
Dipinacoline glutamate is a bioactive chemical.
T31497 Dineopentyl glutamate

L-Glutamic acid bis(2,2-dimethylpropyl) ester,DNPE

Others Others
Dineopentyl glutamate is a bioactive chemical.
T33911 PENB-L-Glutamate

Others Others
PENB-L-Glutamate is a caged glutamate.
T31709 Ethyl glutamate

NSC-156977,NSC156977,Alpha-ethylglutamic acid,gamma-Ethylglutamate,NSC 156977

Others Others
Ethyl glutamate 可用于生命科学领域的相关研究。其产品编号为 T31709,CAS号为 1119-33-1。
TP2397 Ornithine glutamate dipeptide

Orn-glu

Ornithine glutamate dipeptide is a amino acid.
T21053 L-Lysine L-glutamate

Others Others
L-Lysine L-glutamate is a bioactive chemical.
T23013 MNI-caged-L-glutamate

Others Others
rapidly and efficiently releases glutamate
T20362 Glutamyl-glutamic acid

Glu-glu,Dipotassium glutamyl-glutamate,N-L-alpha-Glutamyl-L-glutamic acid

Amino Acids and Derivatives Metabolism
Glutamyl-glutamic acid (Glu-glu) 是一些微球菌和节杆菌属菌的胞壁中的肽桥。
T34676 Sodium oleoyl glutamate

N-Oleoyl-L-glutamic acid monosodium salt,Acylglutamate OS-11

Others Others
Sodium oleoyl glutamate is a sodium salt oleoyl glutamate.
T20264L Alanine glutamate acetate(13187-90-1 Free base)

Alanine glutamate acetate(13187-90-1 Free base) 是一种二肽,在生命科学相关研究中具有广泛的应用。
T78350 Glutamate dehydrogenase

Others Others
Glutamate dehydrogenase为存在于原核生物与真核生物线粒体中的酶类,适用于氨、α-酮戊二酸、L-谷氨酸及脲酶的酶促反应检测。
T2A2497L Glutamic acid diethyl ester

L-Glutamate diethylester,Diethyl glutamate,Glutamyl diethyl ester

Others Others
Glutamic acid diethyl ester is a glutamic acid antagonist.
T66113 1-Methyl L-Glutamate

1-Methyl L-Glutamate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66113,CAS号为 6384-08-3。
T60645 Glutamate-5-kinase-IN-2

Others Others
Glutamate-5-kinase-IN-2 (compound 54) 通过促进 L-谷氨酸结合位点的构象变化,从而抑制 G5K 活性,它是谷氨酸 5-激酶 (G5K)的有效抑制剂,MIC 为 4.2 μM。Glutamate-5-kinase-IN-2 具有用于抗结核药物研究的潜力。
T60693 Glutamate-5-kinase-IN-1

Others Others
Glutamate-5-kinase-IN-1 (compound 50) 是谷氨酸-5-激酶 (G5K)的有效抑制剂 ,它通过改变 ATP 结合位点构象发挥抑制作用,其抑制浓度为 4.1 μM。Glutamate-5-kinase-IN-1 具有研究抗结核的潜力
T84390 MNI-caged-L-glutamate TFA

Others Others
MNI-caged-L-glutamate, a derivative of glutamate conjugated with a 4-methoxy-7-nitroindolinyl (MNI) photoprotective group, remains pharmacologically inactive at neuronal glutamate receptors at concentrations up to mM. Upon light exposure (300 - 380 nm excitation), it rapidly releases L-glutamate by cleaving the MNI group within submicroseconds. This characteristic enables the investigation of fast synaptic glutamate receptor mechanisms in situ.
T22641 CDPPB

GluR Neuroscience
CDPPB 是选择性和脑渗透性的代谢型谷氨酸受体亚型5 (mGluR5) 阳性变构的调节剂,在表达人类 mGluR5 的中国仓鼠卵巢细胞中的 EC50值为 27 nM。它为开发抗精神病药提供了一种可能性。
T21747 VU0483605

GluR Neuroscience
VU0483605 是一种有效的特异性 mGluR1 正变构调节剂,对人和大鼠的 EC50 分别为 390 和 356 nM。
T14971 CIQ

NMDAR Neuroscience
CIQ 是亚基选择性NMDA 受体增强剂,可作用于NR2C 或NR2D 亚基。
T3482 CFMTI

GluR Neuroscience
CFMTI 是选择性代谢型谷氨酸受体 1 变构拮抗剂,IC50为2.6 nM。它对 mGluR1 的选择性比 mGluR5 高 2000 倍。
T6598 MPEP

GluR Neuroscience
MPEP 是一种选择性 mGlu5 受体拮抗剂,IC50 为 36 nM,有抗焦虑和抗抑郁活性。
T3483 FTIDC

GluR Neuroscience
FTIDC 是非竞争性和选择性的口服变构代谢型谷氨酸受体 1 拮抗剂,对人 mGluR1a 的IC50为 5.8 nM。
T8779 HBT1

GluR Neuroscience
HBT1 是一种 AMPA 受体增强剂,可诱导脑源性神经营养因子 (BDNF) 的产生,并且在原代神经元中几乎没有激动作用。 HBT1 以谷氨酸依赖的方式与 AMPA-R 的配体结合结构域结合。
T12406 PEPA

iGluR Membrane transporter/Ion channel; Neuroscience
PEPA 是一种变构 AMPA 受体调节剂,可与 GluA2o 和 GluA3o LBD 结合,可用作 AMPA 受体异质性的指标。
T35319 Zy 15109

N-Acetyl-aspartyl magnesium glutamate,Zy15109,Magnesium N-acetyl-aspartylglutamate

Others Others
Zy 15109 can be used as inhaled mast cell stabilizer.
T60112 H-Glu(OEt)-OEt.HCl

Diethyl L-glutamate hydrochloride,(S)-Diethyl 2-aminopentanedioate hydrochloride,L-谷氨酸二乙酯盐酸盐,Diethyl glutamate hydrochloride

Amino Acids and Derivatives Metabolism
H-Glu(OEt)-OEt.HCl (Diethyl L-glutamate hydrochloride) 是一种谷氨酸衍生物。
T16402 Org-26576

GluR; iGluR Membrane transporter/Ion channel; Neuroscience
Org-26576 是 AMPA 受体的一种正变构调节剂。
T6022 LY404039

pomaglumetad

Glucocorticoid Receptor; GluR Endocrinology/Hormones; Neuroscience
LY404039 (pomaglumetad) 是可口服的mGluR2和mGluR3选择性激动剂,有抗精神病和抗焦虑的作用。它对重组人mGluR2和mGluR3的Ki 分别为 149 和 92 nM,比对其他受体/转运蛋白的抑制性高 100 倍以上。
T3477 E4CPG

GluR Neuroscience
E4CPG 是一种 I/II 组代谢型谷氨酸受体的拮抗剂,可抑制单突触后机制中突触后电流 (IPSC) 增强的成对脉冲比。
T3464 PHCCC

(-) PHCCC

GluR Neuroscience
PHCCC ((-) PHCCC) 是 I 组代谢型谷氨酸受体拮抗剂和 mGluR4 的正变构调节剂。 它对 mGluR2 和 mGluR8 也有很强的拮抗作用,具有抗帕金森病作用。
T20264 Ala-Glu-OH

L-Glutamic acid, N-L-alanyl-,Alanine glutamate,Alanylglutamic acid

Alanine glutamate is an agent of the dipeptide.
T9133 Caroverine hydrochloride

Caroverine HCL

GluR; NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Caroverine hydrochloride (Caroverine HCL) 是竞争性可逆的NMDA 和AMPA 谷氨酸受体拮抗剂。它也是抗氧化和钙阻滞剂,具有血管舒张作用,可用于内耳耳鸣的研究。

化合物

Monopotassium glutamate
Cat.No: T20365
Synonym: L-谷氨酸钾盐,Potassium glutamate,Potassium L-glutamate
Target: Others
Tetrasodium glutamate diacetate
Cat.No: T20266
Synonym: Glutamate diacetate tetrasodium,GLDA
Target: Others
Dimethyl DL-Glutamate (hydrochloride)
Cat.No: T7658
Synonym:
Target: Others
Sodium lauroyl glutamate
Cat.No: T20331
Synonym: Hostapon CLG,Amisoft LS 11,Sodium N-lauroylglutamate,月桂酰谷氨酸钠,Acylglutamate LS-11
Target: Others
Dimethyl L-glutamate
Cat.No: T72460
Synonym: Dimethyl glutamate
Target:
MDNI-caged-L-glutamate
Cat.No: T40973
Synonym: MDNI-caged-L-glutamate,MDNI-glu
Target: Others
L(+)-Monosodium glutamate monohydrate
Cat.No: T35369
Synonym: L(+)-Monosodium glutamate monohydrate,MSG monohydrate,L-Glutamic acid monosodium salt monohydrate,Monosodium L-glutamate monohydrate
Target: Others
Triethanolamine linoleoyl glutamate
Cat.No: T34938
Synonym: TEA-linoleoyl glutamate
Target: Others
Sodium palmitoyl glutamate
Cat.No: T34677
Synonym: Sodium N-palmitoyl-L-glutamate,Monosodium N-palmitoyl-L-glutamate
Target: Others
Glutamate dehydrogenase (NAD(P))
Cat.No: T73616
Synonym: GLDH
Target: Mitochondrial Metabolism
RuBi-Glutamate
Cat.No: T23278
Synonym:
Target: Others
Deanol glutamate
Cat.No: T31266
Synonym:
Target: Others
Glutamate cobalt
Cat.No: T31941
Synonym:
Target: Others
Norfloxacin glutamate
Cat.No: T33724
Synonym:
Target: Others
Triethanolamine glutamate
Cat.No: T34937
Synonym:
Target: Others
Erythromycin glutamate
Cat.No: T24043
Synonym:
Target: Others
Sodium linoleoyl glutamate
Cat.No: T34675
Synonym:
Target: Others
Methotrexate-alpha glutamate
Cat.No: T33326
Synonym: Meapa-glu-glu
Target: Others
Dipinacoline glutamate
Cat.No: T31518
Synonym: L-Glutamic acid dipinacoline ester,DiPG
Target: Others
Dineopentyl glutamate
Cat.No: T31497
Synonym: L-Glutamic acid bis(2,2-dimethylpropyl) ester,DNPE
Target: Others
PENB-L-Glutamate
Cat.No: T33911
Synonym:
Target: Others
Ethyl glutamate
Cat.No: T31709
Synonym: NSC-156977,NSC156977,Alpha-ethylglutamic acid,gamma-Ethylglutamate,NSC 156977
Target: Others
Ornithine glutamate dipeptide
Cat.No: TP2397
Synonym: Orn-glu
Target:
L-Lysine L-glutamate
Cat.No: T21053
Synonym:
Target: Others
MNI-caged-L-glutamate
Cat.No: T23013
Synonym:
Target: Others
Glutamyl-glutamic acid
Cat.No: T20362
Synonym: Glu-glu,Dipotassium glutamyl-glutamate,N-L-alpha-Glutamyl-L-glutamic acid
Target: Amino Acids and Derivatives
Sodium oleoyl glutamate
Cat.No: T34676
Synonym: N-Oleoyl-L-glutamic acid monosodium salt,Acylglutamate OS-11
Target: Others
Alanine glutamate acetate(13187-90-1 Free base)
Cat.No: T20264L
Synonym:
Target:
Glutamate dehydrogenase
Cat.No: T78350
Synonym:
Target: Others
Glutamic acid diethyl ester
Cat.No: T2A2497L
Synonym: L-Glutamate diethylester,Diethyl glutamate,Glutamyl diethyl ester
Target: Others
1-Methyl L-Glutamate
Cat.No: T66113
Synonym:
Target:
Glutamate-5-kinase-IN-2
Cat.No: T60645
Synonym:
Target: Others
Glutamate-5-kinase-IN-1
Cat.No: T60693
Synonym:
Target: Others
MNI-caged-L-glutamate TFA
Cat.No: T84390
Synonym:
Target: Others
CDPPB
Cat.No: T22641
Synonym:
Target: GluR
VU0483605
Cat.No: T21747
Synonym:
Target: GluR
CIQ
Cat.No: T14971
Synonym:
Target: NMDAR
CFMTI
Cat.No: T3482
Synonym:
Target: GluR
MPEP
Cat.No: T6598
Synonym:
Target: GluR
FTIDC
Cat.No: T3483
Synonym:
Target: GluR
HBT1
Cat.No: T8779
Synonym:
Target: GluR
PEPA
Cat.No: T12406
Synonym:
Target: iGluR
Zy 15109
Cat.No: T35319
Synonym: N-Acetyl-aspartyl magnesium glutamate,Zy15109,Magnesium N-acetyl-aspartylglutamate
Target: Others
H-Glu(OEt)-OEt.HCl
Cat.No: T60112
Synonym: Diethyl L-glutamate hydrochloride,(S)-Diethyl 2-aminopentanedioate hydrochloride,L-谷氨酸二乙酯盐酸盐,Diethyl glutamate hydrochloride
Target: Amino Acids and Derivatives
Org-26576
Cat.No: T16402
Synonym:
Target: GluR, iGluR
LY404039
Cat.No: T6022
Synonym: pomaglumetad
Target: Glucocorticoid Receptor, GluR
E4CPG
Cat.No: T3477
Synonym:
Target: GluR
PHCCC
Cat.No: T3464
Synonym: (-) PHCCC
Target: GluR
Ala-Glu-OH
Cat.No: T20264
Synonym: L-Glutamic acid, N-L-alanyl-,Alanine glutamate,Alanylglutamic acid
Target:
Caroverine hydrochloride
Cat.No: T9133
Synonym: Caroverine HCL
Target: GluR, NMDAR, iGluR
Cat. No. Product Name Target Signaling Pathways
T20262 Arginine glutamate

Modumate,NSC-122009,NSC 122009,NSC122009,NCI-C02120,Argimate

Others Others
Arginine glutamate is an agent of ammonia Detoxicant.
T6871 L-Glutamic acid monosodium salt

Monosodium glutamate,谷氨酸单钠盐,Glutacyl,Glutavene,L-谷氨酸单钠盐,Ajinomoto,MSG

Apoptosis; Ferroptosis; GluR; iGluR Apoptosis; Membrane transporter/Ion channel; Neuroscience
L-Glutamic acid monosodium salt (MSG) 作为兴奋性氨基酸神经递质,是谷氨酸盐受体所有亚型的激动剂,对多巴胺从神经末梢释放的过程有激动作用。
T3379 Decanoic Acid

Decoic acid,CAPRIC ACID,Caprynic acid,癸酸

GluR; iGluR Membrane transporter/Ion channel; Neuroscience
Decanoic Acid (Caprynic acid) 是中链甘油三酯中的成分,是非竞争性和可透过血脑屏障的 AMPA 受体抑制剂,具有抗癫痫作用。
T1186 Ifenprodil Tartrate

Potassium Channel; NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Ifenprodil tartrate 是典型的非竞争性 NMDA 受体拮抗剂,抑制 GIRK (Kir3),通过基底 GIRK 活性减少内向电流,有用做脑血管舒张试剂的潜力。它对 NR1A/NR2B 受体亲和力是 NR1A/NR2A 受体的 400 倍。
T2S2264 Linalool

Linalol,(±)-Linalool,Phantol,沉香醇

Apoptosis; IL Receptor; TNF; Endogenous Metabolite; iGluR Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Linalool (Linalol) 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA 受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。
T8394 D-Serine

(R)-Serine,D-丝氨酸

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
D-Serine ((R)-Serine) 是一种具有独特的神经递质特性的神经胶质-突触相互作用中涉及的内源性氨基酸,是 NMDA 谷氨酸受体的有效共激动剂。D-Serine 在主要的 NMDAR 依赖性过程中具有主要的调节作用,包括 NMDAR 介导的神经传递,神经毒性,突触可塑性和细胞迁移。
T6S1653 Albiflorin

Alibiflorin,芍药内酯苷

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分,是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。
T20191 (-)-Camphoric acid

(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

GluR Neuroscience
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。
T6608 NMDA

N-甲基-D-天冬氨酸,N-Methyl-D-aspartic acid

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
NMDA (N-Methyl-D-aspartic acid) 是一种氨基酸,作为 D-异构体,是谷氨酸受体的 NMDA 受体亚型的定义激动剂。
TQ0027 Transcrocetinate disodium

Disodium trans-crocetinate,藏红花,藏红花酸二钠盐

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Transcrocetinate disodium (Disodium trans-crocetinate) 从藏红花中提取的一种天然产物,是高亲和力NMDA 受体拮抗剂。
T4096 Quinolinic acid

喹啉酸,pyridine-2,3-dicarboxylic acid,QUIN

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
Quinolinic acid (QUIN) 是一种内源性 N-甲基-D-天冬氨酸 (NMDA) 受体激动剂,由 L-色氨酸通过犬尿氨酸途径合成,具有调节 NMDA 神经元损伤和功能障碍的潜力。
T1589 D-Cycloserine

RO-1-9213,D-环丝氨酸

Others; Antibacterial; Antibiotic; iGluR Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Others
D-Cycloserine (RO-1-9213) 是一种抗生素,靶向细菌细胞壁肽聚糖生物合成酶。它是一种NMDA 部分激动剂,可以改善认知功能,可研究耐多药结核病。
T4S0171 Transcrocetin

trans-Crocetin,藏红花酸,藏红花,8,8'-Diapocarotenedioic Acid,Crocetin

Others; Endogenous Metabolite; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Transcrocetin (8,8'-Diapocarotenedioic Acid) 是来源于藏红花 (Crocus sativus L.) 的活性化合物,是一种能够透过血脑屏障的,高亲和力的NMDA 受体拮抗剂。
T2O2728 glycine

2-Aminoacetic acid,Glycolixir,Aminoacetic acid,Glycosthene,Glycocoll,甘氨酸

MT Receptor; Endogenous Metabolite; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
glycine (2-Aminoacetic acid) 是中枢神经系统的抑制性神经递质,也是谷氨酸的联合激动剂,有促进谷氨酸能NMDA 受体兴奋的潜力。它主要存在于明胶和丝素蛋白中,并在治疗上用作营养物质。
T3010 Xanthurenic Acid

8-Hydroxykynurenic acid,黄尿酸,4,8-Dihydroxyquinaldic acid,xanthurenate

Apoptosis; Endogenous Metabolite; GluR Apoptosis; Metabolism; Neuroscience
Xanthurenic Acid (8-Hydroxykynurenic acid) 是通过 3-羟基犬尿氨酸转氨而由色氨酸代谢产生的分子,可激活 mGlu2/3 代谢型谷氨酸受体。在下丘脑的感觉传输过程中,它被认为是Group II 代谢型谷氨酸受体的激动剂。
T0326L L-Glutamine

L-Glutamic acid 5-amide,L-谷氨酰胺

Ferroptosis; Endogenous Metabolite; GluR Apoptosis; Metabolism; Neuroscience
L-Glutamine (L-Glutamic acid 5-amide) 是在人体中大量存在的一种非必需氨基酸,由谷氨酸和氨合成。它为某些细胞中的氧化提供了碳源。
T3026 (-)-Huperzine A

HupA,石杉碱,Huperzine A,石杉碱甲

Apoptosis; AChR; AChE; iGluR Apoptosis; Membrane transporter/Ion channel; Neuroscience
(-)-Huperzine A (HupA) 是从中国梅花苔中分离得到的一种生物碱,具有神经保护活性。它是高特异性可逆的,具有血脑屏障渗透性的一种乙酰胆碱酯酶抑制剂, 其IC50值为 82 nM。 它也是 N-甲基-D-天冬氨酸受体的非竞争性拮抗剂,可研究神经退行性疾病,如阿尔茨海默病。
T1324 O-Phospho-L-serine

L-Serine O-phosphate,磷酸化丝氨酸,Phosphoserine,Dexfosfoserine,L-SOP

Amino Acids and Derivatives; Endogenous Metabolite; GluR; NMDAR Metabolism; Neuroscience
O-Phospho-L-serine (Phosphoserine) 是 L-serine 合成过程中的直接前体物质,是 mGluR 激动剂。
T2A2497 L-Glutamic acid

谷氨酸,(S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,L-谷氨酸,glutacid,Glutaminol

Apoptosis; Ferroptosis; Endogenous Metabolite; iGluR Apoptosis; Membrane transporter/Ion channel; Metabolism; Neuroscience
L-Glutamic acid (Glutaminol) 作为一种兴奋性氨基酸神经递质,为谷氨酸盐受体所有亚型的激动剂,对多巴胺从神经末梢释放的过程有激动作用。
T4885 (-)-Aspartic acid

(R)-Aspartic acid,Asp,D-(-)-Aspartic acid,D-天门冬氨酸,Aminosuccinic acid,asparagic acid,L-Homoproline,D-Aspartic acid

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
(-)-Aspartic acid (L-Homoproline) 是一种存在于无脊椎动物和脊椎动物中的内源性氨基酸,是 NMDA 受体激动剂,可调节睾酮合成。
T0948L Corticosterone

皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Corticosterone (Kendall's compound B) 是一种肾上腺皮质类固醇,有盐皮质激素和糖皮质激素的活性,具有口服活性。Corticosterone 参与体内能量、免疫反应和应激反应的调节。
T3377 L-Phenylalanine

L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine

Calcium Channel; Endogenous Metabolite; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
L-Phenylalanine (3-Phenyl-L-alanine) 是分离自大肠杆菌的必需氨基酸,是 NMDARs(KB573 μM) 和非 NMDARs 的甘氨酸和谷氨酸结合位点的竞争性拮抗剂,用于食品香料和药品的生产中。它是一种电压依赖性 α2δ 亚基 Ca2+通道拮抗剂,Ki 为 980 nM。
T12016 Methyl L-pyroglutamate

L-Pyroglutamic acid methyl ester,L-焦谷氨酸甲酯,(S)-Methyl 5-oxopyrrolidine-2-carboxylate

Others Others
Methyl L-pyroglutamate (L-Pyroglutamic acid methyl ester) 分离自甘蓝中分离,显示出抗炎活性。
T4920 2-Ketoglutaric acid Sodium

Oxoglutaric acid,AKG,2-oxoglutarate monobasic,LPHA-酮戊二酸钠,α-Ketoglutaric acid sodium salt

Tyrosinase; Endogenous Metabolite Metabolism; Proteases/Proteasome
2-Ketoglutaric acid Sodium (AKG) 是一种三羧酸循环的中间产物,它可以由谷氨酸通过谷氨酸脱氢酶氧化脱氨产生,也可以作为磷酸吡哆醛依赖的转氨化反应的产物(由支链氨基酸转氨酶介导),其中谷氨酸是常见的氨基供体。
T4913 Maleic acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
Maleic Acid 是大肠杆菌和单核细胞增生李斯特菌的谷氨酸脱羧酶抑制剂。
T4752 1-Aminocyclopropane-1-carboxylic acid

1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC

Endogenous Metabolite; NMDAR Metabolism; Neuroscience
1-Aminocyclopropane-1-carboxylic acid (ACC) 是内源性代谢产物的一种。
T10191L 7-Chlorokynurenic acid

7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA

GluR; NMDAR Neuroscience
7-Chlorokynurenic acid (7-chloro-4-hydroxy-2-carboxyquinoline) 是一种有效的选择性 NMDA 受体拮抗剂,对甘氨酸 B 激动剂位点的 IC50 为 0.56 μM。 7-Chlorokynurenic acid 抑制谷氨酸再摄取到突触小泡中,Ki 为 0.59 μM,并在神经轴输送后显示出镇痛作用。
T65135 Kynurenic acid

Fibrostop 2,Quinurenic acid

GPR; GluR; NMDAR Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Kynurenic acid (Quinurenic acid) 是一种内源性色氨酸活性代谢物,是一种 NMDA, glutamate, α7 nicotinic acetylcholine receptor 三重拮抗剂,也是 GPR35/CXCR8 激动剂,具有神经保护和抗惊厥特性,可用于研究神经分裂和与代谢相关的疾病。
T7060 Amantadine

1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine

Others Others
Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
T4813 L-Citrulline

Endogenous Metabolite Metabolism
L-Citrulline 是一种氨基酸,源自于精氨酸-瓜氨酸途径获得的 l-精氨酸,或脯氨酸、谷氨酰胺和谷氨酸盐的分解代谢过程中产生的鸟氨酸。
T6S0659 Rhynchophylline

钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin

Calcium Channel; NF-κB Membrane transporter/Ion channel; Metabolism; NF-κB
Rhynchophylline (Mitrinermine) 是一种生物碱类化合物,从钩藤中分离得到,具有很高的生物活性,被广泛用于抗炎、神经保护等方面的研究。
T5267 N-Acetyl-L-glutamic acid

Ac-L-Glu-OH,N-乙酰-L-谷氨酰胺,N-Acetylglutamic acid

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-glutamic acid (Ac-L-Glu-OH) 是一种 N-Acyl-L-氨基酸,是动物细胞培养基的组成成分,是一种酿酒酵母和人类的代谢物。
T6S0654 Isocorynoxeine

7-Isocorynoxeine,异去氢钩藤碱

5-HT Receptor GPCR/G Protein; Neuroscience
Isocorynoxeine (7-Isocorynoxeine) 是钩藤中的一种生物碱,剂量依赖性抑制5-HT2A 受体介导的电流反应,IC50为 72.4 μM。
TN1449 Brandioside

2'-O-Acetylpoliumoside,2'-Acetylpoliumoside

Antioxidant oxidation-reduction
Brandioside (2'-Acetylpoliumoside) 是可从马鞭草科植物 Callicarpa dichotoma Raeuschel  提取得到的苯丙素类糖苷,具有抗氧化活性,可削弱谷氨酸诱导的神经毒性,可用于研究糖尿病。
T5692 Pyrroloquinoline quinone

Others; Endogenous Metabolite Metabolism; Others
Pyrroloquinoline quinone 是氧化还原辅助因子,一种阴离子型氧化还原循环原醌。它是哺乳动物的必需营养素,对免疫功能很重要。它是从嗜甲基细菌的培养物中分离的,也存在于哺乳动物的组织。
T1131 Ivermectin

MK-933,伊维菌素

Mitophagy; GluCls; P2X Receptor; SARS-CoV; HIV Protease; Antibiotic; Parasite; Autophagy; HSV Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ivermectin (MK-933) 是谷氨酸门控氯离子通道激活剂,具有抗寄生虫活性。它特异性抑制Impα/β1 介导的核导入,还抑制牛疱疹病毒 1 复制并抑制BoHV-1DNA 聚合酶的核输入。它具有很强的抗病毒活性。它也是P2X4和 α7nAChRs 的正异构效应物。
T2596 N-Acetyl-β-Asp-Glu

Others Others
N-Acetyl-β-Asp-Glu 是一种肽类神经递质,是哺乳动物神经系统中第三常见的神经递质。 NAAG 由通过肽键偶联的 N-乙酰天冬氨酸 (NAA) 和谷氨酸组成。
TN1196 17-Hydroxyisolathyrol

Others Others
17-Hydroxyisolathyrol 是一种大环千金子二萜醇衍生物,分离自Euphorbla luthyrrs种子。17-Hydroxyisolathyrol 抑制蛋白质-蛋白质相互作用。
TN1677 Gartanin

1,3,5,8-四羟基-2,4-双(3-甲基-2-丁烯基)-9H-氧杂蒽-9-酮,藤黄苷

BCL; Caspase; JNK Apoptosis; MAPK; Proteases/Proteasome
Gartanin 是山竹果中的一种天然黄酮,具有抗氧化、抗真菌、抗炎、神经保护和抗肿瘤活性。它能够诱导人脑胶质瘤细胞的细胞周期阻滞和自噬,抑制其迁移。
TN1905 Magnolioside

七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷

Antifection Microbiology/Virology
Magnolioside 是分离自Angelica gigas Nakai(Umbelliferae) 中,对谷氨酸诱导的毒性有显著的神经保护作用。 它显示出对金黄色葡萄球菌 CIP 53.154 的中等抗菌活性。它具有抗疟原虫活性,对氯喹敏感的恶性疟原虫菌株具有强烈的生长抑制作用。
T6102 2'-acetylacteoside

Antioxidant; Reductase Endocrinology/Hormones; Metabolism; oxidation-reduction
2'-Acetylacteoside 是一种苯乙醇苷类化合物,分离自来江藤中,可抑制自由基诱导的红细胞溶血,具有清除自由基的作用。
T5558 Chelidonic acid

Jervaic acid,Jerva acid,白屈菜酸,γ-Pyrone-2,6-dicarboxylic acid

NF-κB; Caspase Apoptosis; NF-κB; Proteases/Proteasome
Chelidonic acid (Jervaic acid) 是从白屈菜中分到的酸类物质,用作温和的镇痛剂、抗菌剂和中枢神经系统镇静剂。它是谷氨酸脱羧酶抑制剂,Ki 值为 1.2 μM。它可能通过抑制 NF-κB 和caspase-1来降低 IL-6 的产生抗炎作用。
T5083 L-Cysteic acid monohydrate

L-磺基丙氨酸 一水合物,3-Sulfo-L-alanine Monohydrate

Endogenous Metabolite; GluR Metabolism; Neuroscience
L-Cysteic acid monohydrate (3-Sulfo-L-alanine Monohydrate) 是内源性代谢产物的一种。
T3578 Pyridoxal phosphate

PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate

Reverse Transcriptase; Endogenous Metabolite Metabolism; Microbiology/Virology
Pyridoxal phosphate (Vitamin B6 phosphate) 是维生素 B6 的活性形式,可抑制逆转录酶活性,用于研究迟发性运动障碍症。
T4705 Aminoadipic acid

DL-2-Aminoadipic acid,DL-2-氨基己二酸

Others; Endogenous Metabolite Metabolism; Others
Aminoadipic acid (DL-2-Aminoadipic acid) 是赖氨酸主要生化途径中的代谢物。 它是赖氨酸和糖碱代谢的中间体。 它拮抗由谷氨酸受体 N-甲基-D-天冬氨酸调节的神经兴奋特性。
TN3808 Dehydroheliobuphthalmin

Others Others
Dehydroheliobuphthalmin has significant neuroprotective activities against glutamate- induced neurotoxicity.
TN1581 Dihydroguaiaretic acid

二氢愈创木酸

COX; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Neuroscience
Dihydroguaiaretic acid has antioxidative activity, can significantly protect primary cultured neuronal cells against glutamate-induced oxidative stress.
T38054 Avenaciolide

Others Others
Avenaciolide is a water-insoluble fungal metabolite originally isolated from A. avenaceus. It inhibits glutamate transport in isolated rat liver mitochondria (Ki = 8 μM).
TN5169 Traxillaside

香榧

Others Others
Traxillaside has significant neuroprotective activities against glutamate-induced toxicity in primary cultures of rat cortical cells .
TN3473 Axillarin

Axillarin has antioxidant activity, it shows xanthine oxidase inhibitory activity ( IC(50) :36.0 uM). Axillarin can strongly protect primary cultured neurons against glutamate-induced oxidative stress.
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天然产物

Arginine glutamate
Cat.No: T20262
Synonym: Modumate,NSC-122009,NSC 122009,NSC122009,NCI-C02120,Argimate
Target: Others
L-Glutamic acid monosodium salt
Cat.No: T6871
Synonym: Monosodium glutamate,谷氨酸单钠盐,Glutacyl,Glutavene,L-谷氨酸单钠盐,Ajinomoto,MSG
Target: Apoptosis, Ferroptosis, GluR, iGluR
Decanoic Acid
Cat.No: T3379
Synonym: Decoic acid,CAPRIC ACID,Caprynic acid,癸酸
Target: GluR, iGluR
Ifenprodil Tartrate
Cat.No: T1186
Synonym:
Target: Potassium Channel, NMDAR, iGluR
Linalool
Cat.No: T2S2264
Synonym: Linalol,(±)-Linalool,Phantol,沉香醇
Target: Apoptosis, IL Receptor, TNF, Endogenous Metabolite, iGluR
D-Serine
Cat.No: T8394
Synonym: (R)-Serine,D-丝氨酸
Target: Endogenous Metabolite, NMDAR, iGluR
Albiflorin
Cat.No: T6S1653
Synonym: Alibiflorin,芍药内酯苷
Target: Reactive Oxygen Species
(-)-Camphoric acid
Cat.No: T20191
Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-
Target: GluR
NMDA
Cat.No: T6608
Synonym: N-甲基-D-天冬氨酸,N-Methyl-D-aspartic acid
Target: Endogenous Metabolite, NMDAR, iGluR
Transcrocetinate disodium
Cat.No: TQ0027
Synonym: Disodium trans-crocetinate,藏红花,藏红花酸二钠盐
Target: NMDAR, iGluR
Quinolinic acid
Cat.No: T4096
Synonym: 喹啉酸,pyridine-2,3-dicarboxylic acid,QUIN
Target: Endogenous Metabolite, NMDAR, iGluR
D-Cycloserine
Cat.No: T1589
Synonym: RO-1-9213,D-环丝氨酸
Target: Others, Antibacterial, Antibiotic, iGluR
Transcrocetin
Cat.No: T4S0171
Synonym: trans-Crocetin,藏红花酸,藏红花,8,8'-Diapocarotenedioic Acid,Crocetin
Target: Others, Endogenous Metabolite, iGluR
glycine
Cat.No: T2O2728
Synonym: 2-Aminoacetic acid,Glycolixir,Aminoacetic acid,Glycosthene,Glycocoll,甘氨酸
Target: MT Receptor, Endogenous Metabolite, iGluR
Xanthurenic Acid
Cat.No: T3010
Synonym: 8-Hydroxykynurenic acid,黄尿酸,4,8-Dihydroxyquinaldic acid,xanthurenate
Target: Apoptosis, Endogenous Metabolite, GluR
L-Glutamine
Cat.No: T0326L
Synonym: L-Glutamic acid 5-amide,L-谷氨酰胺
Target: Ferroptosis, Endogenous Metabolite, GluR
(-)-Huperzine A
Cat.No: T3026
Synonym: HupA,石杉碱,Huperzine A,石杉碱甲
Target: Apoptosis, AChR, AChE, iGluR
O-Phospho-L-serine
Cat.No: T1324
Synonym: L-Serine O-phosphate,磷酸化丝氨酸,Phosphoserine,Dexfosfoserine,L-SOP
Target: Amino Acids and Derivatives, Endogenous Metabolite, GluR, NMDAR
L-Glutamic acid
Cat.No: T2A2497
Synonym: 谷氨酸,(S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,L-谷氨酸,glutacid,Glutaminol
Target: Apoptosis, Ferroptosis, Endogenous Metabolite, iGluR
(-)-Aspartic acid
Cat.No: T4885
Synonym: (R)-Aspartic acid,Asp,D-(-)-Aspartic acid,D-天门冬氨酸,Aminosuccinic acid,asparagic acid,L-Homoproline,D-Aspartic acid
Target: Endogenous Metabolite, NMDAR, iGluR
Corticosterone
Cat.No: T0948L
Synonym: 皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
L-Phenylalanine
Cat.No: T3377
Synonym: L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine
Target: Calcium Channel, Endogenous Metabolite, iGluR
Methyl L-pyroglutamate
Cat.No: T12016
Synonym: L-Pyroglutamic acid methyl ester,L-焦谷氨酸甲酯,(S)-Methyl 5-oxopyrrolidine-2-carboxylate
Target: Others
2-Ketoglutaric acid Sodium
Cat.No: T4920
Synonym: Oxoglutaric acid,AKG,2-oxoglutarate monobasic,LPHA-酮戊二酸钠,α-Ketoglutaric acid sodium salt
Target: Tyrosinase, Endogenous Metabolite
Maleic acid
Cat.No: T4913
Synonym:
Target: Endogenous Metabolite, Antibacterial
1-Aminocyclopropane-1-carboxylic acid
Cat.No: T4752
Synonym: 1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC
Target: Endogenous Metabolite, NMDAR
7-Chlorokynurenic acid
Cat.No: T10191L
Synonym: 7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA
Target: GluR, NMDAR
Kynurenic acid
Cat.No: T65135
Synonym: Fibrostop 2,Quinurenic acid
Target: GPR, GluR, NMDAR
Amantadine
Cat.No: T7060
Synonym: 1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine
Target: Others
L-Citrulline
Cat.No: T4813
Synonym:
Target: Endogenous Metabolite
Rhynchophylline
Cat.No: T6S0659
Synonym: 钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
N-Acetyl-L-glutamic acid
Cat.No: T5267
Synonym: Ac-L-Glu-OH,N-乙酰-L-谷氨酰胺,N-Acetylglutamic acid
Target: Others, Endogenous Metabolite
Isocorynoxeine
Cat.No: T6S0654
Synonym: 7-Isocorynoxeine,异去氢钩藤碱
Target: 5-HT Receptor
Brandioside
Cat.No: TN1449
Synonym: 2'-O-Acetylpoliumoside,2'-Acetylpoliumoside
Target: Antioxidant
Pyrroloquinoline quinone
Cat.No: T5692
Synonym:
Target: Others, Endogenous Metabolite
Ivermectin
Cat.No: T1131
Synonym: MK-933,伊维菌素
Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV
N-Acetyl-β-Asp-Glu
Cat.No: T2596
Synonym:
Target: Others
17-Hydroxyisolathyrol
Cat.No: TN1196
Synonym:
Target: Others
Gartanin
Cat.No: TN1677
Synonym: 1,3,5,8-四羟基-2,4-双(3-甲基-2-丁烯基)-9H-氧杂蒽-9-酮,藤黄苷
Target: BCL, Caspase, JNK
Magnolioside
Cat.No: TN1905
Synonym: 七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷
Target: Antifection
2'-acetylacteoside
Cat.No: T6102
Synonym:
Target: Antioxidant, Reductase
Chelidonic acid
Cat.No: T5558
Synonym: Jervaic acid,Jerva acid,白屈菜酸,γ-Pyrone-2,6-dicarboxylic acid
Target: NF-κB, Caspase
L-Cysteic acid monohydrate
Cat.No: T5083
Synonym: L-磺基丙氨酸 一水合物,3-Sulfo-L-alanine Monohydrate
Target: Endogenous Metabolite, GluR
Pyridoxal phosphate
Cat.No: T3578
Synonym: PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate
Target: Reverse Transcriptase, Endogenous Metabolite
Aminoadipic acid
Cat.No: T4705
Synonym: DL-2-Aminoadipic acid,DL-2-氨基己二酸
Target: Others, Endogenous Metabolite
Dehydroheliobuphthalmin
Cat.No: TN3808
Synonym:
Target: Others
Dihydroguaiaretic acid
Cat.No: TN1581
Synonym: 二氢愈创木酸
Target: COX, DNA/RNA Synthesis
Avenaciolide
Cat.No: T38054
Synonym:
Target: Others
Traxillaside
Cat.No: TN5169
Synonym: 香榧
Target: Others
Axillarin
Cat.No: TN3473
Synonym:
Target:
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Cat. No. Product Name Species Expression System
TMPH-00795 Glutamate racemase Protein, Helicobacter pylori, Recombinant (His & Myc)

murI,Glutamate racemase

Helicobacter pylori E. coli
Provides the (R)-glutamate required for cell wall biosynthesis. Glutamate racemase Protein, Helicobacter pylori, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 35.9 kDa and the accession number is B5Z6S2.
TMPY-04699 GAD65 Protein, Human, Recombinant (GST)

glutamate decarboxylase 2 (pancreatic islets and br...

Human Baculovirus Insect Cells
GAD65 Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 92.6 kDa and the accession number is Q05329.
TMPJ-00855 GLUL Protein, Human, Recombinant (His)

GLUL,GS,Glutamine Synthetase,Glutamate-Ammonia Liga...

Human E. coli
Glutamine Synthetase reglutes intracellular concentration of glutamate. Glutamine Synthetase catalyzes the synthesis of glutamine from glutamate and ammonia. Glutamine is an important source of energy and that takes part in cell prolifetation, inhibition of apoptosis, and cell signaling. Glutamine Synthetase is expressed during early fetal stages, and has a role in maintaining body PH by removing ammonia from circulation. Mutations in the GLUL gene are related to congenital glutamine deficiency.
TMPH-00627 GAD-alpha Protein, E. coli, Recombinant (His)

Glutamate decarboxylase alpha,gadA

E. coli E. coli
Converts glutamate to gamma-aminobutyrate (GABA), consuming one intracellular proton in the reaction. The gad system helps to maintain a near-neutral intracellular pH when cells are exposed to extremely acidic conditions. The ability to survive transit through the acidic conditions of the stomach is essential for successful colonization of the mammalian host by commensal and pathogenic bacteria.
TMPH-01392 GRIA2 Protein, Human, Recombinant (His & Myc)

GRIA2,Glutamate receptor ionotropic, AMPA 2,Glu...

Human E. coli
GRIA2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 63.3 kDa and the accession number is P42262.
TMPH-01393 GRIA3 Protein, Human, Recombinant (His & SUMO)

AMPA-selective glutamate receptor 3,GRIA3,Gluta...

Human E. coli
GRIA3 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 28.0 kDa and the accession number is P42263.
TMPH-00416 NAD-GDH Protein, Clostridium difficile, Recombinant (His)

gluD,NAD-specific glutamate dehydrogenase

Peptoclostridium difficile E. coli
NAD-GDH Protein, Clostridium difficile, Recombinant (His) is expressed in E. coli.
TMPH-01663 GRM5 Protein, Human, Recombinant (His & Myc)

Metabotropic glutamate receptor 5,GRM5

Human E. coli
G-protein coupled receptor for glutamate. Ligand binding causes a conformation change that triggers signaling via guanine nucleotide-binding proteins (G proteins) and modulates the activity of down-stream effectors. Signaling activates a phosphatidylinositol-calcium second messenger system and generates a calcium-activated chloride current. Plays an important role in the regulation of synaptic plasticity and the modulation of the neural network activity.
TMPH-00438 GLUL Protein, Cricetulus griseus, Recombinant (His)

Glutamine synthetase,GLUL,Glutamate--ammonia ligase...

Chinese hamster E. coli
GLUL Protein, Cricetulus griseus, Recombinant (His) is expressed in E. coli.
TMPH-00628 GltI/YbeJ Protein, E. coli, Recombinant (His & SUMO)

gltI,Glutamate/aspartate import solute-binding prot...

E. coli E. coli
Part of the ABC transporter complex GltIJKL involved in glutamate and aspartate uptake. Binds to both glutamate and aspartate. GltI/YbeJ Protein, E. coli, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 47.2 kDa and the accession number is P37902.
TMPH-01394 GRIN1 Protein, Human, Recombinant (His)

N-methyl-D-aspartate receptor subunit NR1,Glutamate...

Human E. coli
Component of NMDA receptor complexes that function as heterotetrameric, ligand-gated ion channels with high calcium permeability and voltage-dependent sensitivity to magnesium. Channel activation requires binding of the neurotransmitter glutamate to the epsilon subunit, glycine binding to the zeta subunit, plus membrane depolarization to eliminate channel inhibition by Mg(2+). Sensitivity to glutamate and channel kinetics depend on the subunit composition. GRIN1 Protein, Human, Recombinant (His)...
TMPY-02091 GAD67 Protein, Human, Recombinant (His)

SCP,CPSQ1,glutamate decarboxylase 1 (brain, 67kDa),...

Human Baculovirus Insect Cells
Glutamate decarboxylase 1, also known as 67 kDa glutamic acid decarboxylase, Glutamate decarboxylase 67 kDa isoform and GAD1, is a member of thegroup II decarboxylase family. GAD1 is expressed in benign and malignant prostatic tissue and may serve as a highly prostate-specific tissue biomarker. GAD1 isoform3 is expressed in pancreatic islets, testis, adrenal cortex, and perhaps other endocrine tissues, but not in brain. Tissue-specific markers are useful for identification of tumour type ...
TMPH-03304 GRIN1 Protein, Rat, Recombinant (His)

Glutamate [NMDA] receptor subunit zeta-1,Glutam...

Rat E. coli
GRIN1 Protein, Rat, Recombinant (His) is expressed in E. coli.
TMPH-00629 Gamma-GCS Protein, E. coli, Recombinant (His & SUMO)

Glutamate--cysteine ligase,Gamma-ECS,gshA,Gamma-glu...

E. coli E. coli
N/A. Gamma-GCS Protein, E. coli, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 74.3 kDa and the accession number is P0A6W9.
TMPH-00796 gltX1 Protein, Helicobacter pylori, Recombinant (His)

Glutamyl-tRNA synthetase 1,gltX1,Glutamate--tRNA li...

Helicobacter pylori P. pastoris (Yeast)
Catalyzes the attachment of glutamate to tRNA(Glu) in a two-step reaction: glutamate is first activated by ATP to form Glu-AMP and then transferred to the acceptor end of tRNA(Glu).
TMPJ-01393 Carboxypeptidase Q Protein, Mouse, Recombinant (His)

Plasma glutamate carboxypeptidase,Hls2,Hematopoieti...

Mouse HEK293 Cells
Carboxypeptidase Q (Cpq) is a member of the peptidase M28 family. PGCP is involved in a number of fundamental biological processes such as the hydrolysis of circulating peptides, catalyzing the hydrolysis of dipeptides with unsubstituted terminals into amino acids. Carboxypeptidase may play an important role in the liberation of thyroxine hormone from its thyroglobulin (Tg) precursor. The monomeric form is inactive while the homodimer is active.
TMPH-00626 GPR Protein, E. coli, Recombinant (His)

proA,Glutamyl-gamma-semialdehyde dehydrogenase,Gamma-glutamy...

E. coli E. coli
Catalyzes the NADPH-dependent reduction of L-glutamate 5-phosphate into L-glutamate 5-semialdehyde and phosphate. The product spontaneously undergoes cyclization to form 1-pyrroline-5-carboxylate. GPR Protein, E. coli, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 48.7 kDa and the accession number is P07004.
TMPY-04318 GRIK2 Protein, Human, Recombinant (hFc)

GLUR6,EAA4,MRT6,GLR6,glutamate receptor, ionotropic...

Human HEK293 Cells
GRIK2 (Glutamate Ionotropic Receptor Kainate Type Subunit 2, also known as GluR6) is a Protein Coding gene. The GRIK2 (one of the kainate receptors) gene resides in a genetic linkage region (6q21) associated with bipolar disorder (BPD). The gene coding for GRIK2 has been suggested as a candidate gene for autism based on its localization in the autism-specific region on chromosome 6q21 and the involvement of receptor protein in cognitive functions like learning and memory. GRIK2 belongs to the gl...
TMPY-01590 GAD65 Protein, Mouse, Recombinant (His & GST)

glutamate decarboxylase 2 (pancreatic islets and br...

Mouse Baculovirus Insect Cells
GAD65 Protein, Mouse, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 93 kDa and the accession number is P48320.
TMPY-03515 GAD65 Protein, Mouse, Recombinant

glutamate decarboxylase 2 (pancreatic islets and br...

Mouse Baculovirus Insect Cells
GAD65 Protein, Mouse, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 65.4 kDa and the accession number is P48320.
TMPH-03190 CPG2 Protein, Pseudomonas sp., Recombinant (GST)

Folate hydrolase G2,Pteroylmonoglutamic acid hydrolase G2,

Pseudomonas E. coli
Catalyzes the hydrolysis of reduced and non-reduced folates to pteroates and L-glutamate. This enzyme has a broad specificity. CPG2 Protein, Pseudomonas sp., Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 68.7 kDa and the accession number is P06621.
TMPH-00911 GPT Protein, Human, Recombinant (His)

Glutamic--alanine transaminase 1,Glutamate pyruvate...

Human E. coli
Catalyzes the reversible transamination between alanine and 2-oxoglutarate to form pyruvate and glutamate. Participates in cellular nitrogen metabolism and also in liver gluconeogenesis starting with precursors transported from skeletal muscles. GPT Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 58.5 kDa and the accession number is P24298.
TMPH-03750 SLC7A11 Protein, Human, Recombinant (His)

SLC7A11,Calcium channel blocker resistance protein CCBR1,Sol...

Human E. coli
Sodium-independent, high-affinity exchange of anionic amino acids with high specificity for anionic form of cystine and glutamate.
TMPH-03400 SLC17A6 Protein, Rat, Recombinant (His)

Slc17a6,Vesicular glutamate transporter 2,Solute ca...

Rat P. pastoris (Yeast)
Mediates the uptake of glutamate into synaptic vesicles at presynaptic nerve terminals of excitatory neural cells. May also mediate the transport of inorganic phosphate. Involved in the regulation of retinal hyaloid vessel regression during postnatal development. May also play a role in the endocrine glutamatergic system of other tissues such as pineal gland and pancreas. SLC17A6 Protein, Rat, Recombinant (His) is expressed in yeast with C-6xHis tag. The predicted molecular weight is 11.1 kDa an...
TMPH-01314 SLC1A3 Protein, Human, Recombinant (His & KSI)

Excitatory amino acid transporter 1,Solute carrier family 1 ...

Human E. coli
SLC1A3 Protein, Human, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 25.5 kDa and the accession number is P43003.
TMPH-01199 CNDP2 Protein, Human, Recombinant (E. coli, His)

HEL-S-13,CPGL,Threonyl dipeptidase,PEPA,CNDP dipeptidase 2,C...

Human E. coli
CNDP2 Protein, Human, Recombinant (E. coli, His) is expressed in E. coli.
TMPH-02807 NPTXR Protein, Mouse, Recombinant (His & Myc)

Neuronal pentraxin receptor,Nptxr

Mouse Baculovirus Insect Cells
May be involved in mediating uptake of synaptic material during synapse remodeling or in mediating the synaptic clustering of AMPA glutamate receptors at a subset of excitatory synapses.
TMPK-00798 IGSF11 Protein, Mouse, Recombinant (His)

Bt-IGSF,BtIGSF,IgSF11,VSIG3,Bt IGSF,CXADRL1,CT119

Mouse HEK293 Cells
Immunoglobulin superfamily member 11 (IgSF11), a homophilic adhesion molecule that preferentially expressed in the brain, is a dual-binding partner of the postsynaptic scaffolding protein PSD-95 and AMPA glutamate receptors (AMPARs).
TMPH-02808 NPTX1 Protein, Mouse, Recombinant (His)

Nptx1,Neuronal pentraxin-1,Neuronal pentraxin I

Mouse E. coli
May be involved in mediating uptake of synaptic material during synapse remodeling or in mediating the synaptic clustering of AMPA glutamate receptors at a subset of excitatory synapses.
TMPH-02882 NQO2 Protein, Mouse, Recombinant (His)

Ribosyldihydronicotinamide dehydrogenase [quinone],Quinone r...

Mouse P. pastoris (Yeast)
The enzyme apparently serves as a quinone reductase in connection with conjugation reactions of hydroquinones involved in detoxification pathways as well as in biosynthetic processes such as the vitamin K-dependent gamma-carboxylation of glutamate residues in prothrombin synthesis.
TMPH-01862 PFAS Protein, Human, Recombinant (His & Myc & SUMO)

Phosphoribosylformylglycinamidine synthase,Formylglycinamide...

Human E. coli
Phosphoribosylformylglycinamidine synthase involved in the purines biosynthetic pathway. Catalyzes the ATP-dependent conversion of formylglycinamide ribonucleotide (FGAR) and glutamine to yield formylglycinamidine ribonucleotide (FGAM) and glutamate. PFAS Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 45.4 kDa and the accession number is O15067.
TMPH-02616 CSAD Protein, Mouse, Recombinant (His & SUMO)

Csad,Cysteine sulfinic acid decarboxylase,Cysteine-sulfinate...

Mouse E. coli
Catalyzes the decarboxylation of L-aspartate, 3-sulfino-L-alanine (cysteine sulfinic acid), and L-cysteate to beta-alanine, hypotaurine and taurine, respectively. The preferred substrate is 3-sulfino-L-alanine. Does not exhibit any decarboxylation activity toward glutamate.
TMPH-02797 NQO1 Protein, Mouse, Recombinant (His)

Quinone reductase 1,NAD(P)H dehydrogenase [quinone] 1,NAD(P)...

Mouse P. pastoris (Yeast)
The enzyme apparently serves as a quinone reductase in connection with conjugation reactions of hydroquinons involved in detoxification pathways as well as in biosynthetic processes such as the vitamin K-dependent gamma-carboxylation of glutamate residues in prothrombin synthesis. NQO1 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 32.8 kDa and the accession number is Q64669.
TMPH-03604 Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)

Phosphinothricin-resistance protein,Phosphinothricin N-acety...

Streptomyces hygroscopicus E. coli
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. Can also acetylate demethylphosphinothricin but not PTT or glutamate. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 24.6 kDa and the accession number is P16426.
TMPH-00863 5-oxoprolinase/OPLAH Protein, Human, Recombinant (His & Myc)

5-oxo-L-prolinase,5-OPase,Pyroglutamase,OPLAH

Human E. coli
Catalyzes the cleavage of 5-oxo-L-proline to form L-glutamate coupled to the hydrolysis of ATP to ADP and inorganic phosphate. 5-oxoprolinase/OPLAH Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.4 kDa and the accession number is O14841.
TMPH-01596 AADAT Protein, Human, Recombinant (His & SUMO)

2-aminoadipate transaminase,Glycine transaminase AADAT,Alpha...

Human E. coli
Transaminase with broad substrate specificity. Has transaminase activity towards aminoadipate, kynurenine, methionine and glutamate. Shows activity also towards tryptophan, aspartate and hydroxykynurenine. Accepts a variety of oxo-acids as amino-group acceptors, with a preference for 2-oxoglutarate, 2-oxocaproic acid, phenylpyruvate and alpha-oxo-gamma-methiol butyric acid. Can also use glyoxylate as amino-group acceptor (in vitro).
TMPJ-00489 NTAQ1 Protein, Human, Recombinant (GST)

Nt(Q)-amidase,C8orf32,NTAQ1,Protein NH2-terminal glutamine d...

Human E. coli
Human protein N-terminal glutamine amidohydrolase (WDYHV1) is an enzyme that in humans is encoded by the WDYHV1 gene, belongs to the NTAQ1 family.WDYHV1 mediates the side-chain deamidation of N-terminal glutamine residues to glutamate, which is an important step in N-end rule pathway of protein degradation. Conversion of the resulting N-terminal glutamine to glutamate renders the protein susceptible to arginylation, polyubiquitination and degradation as specified by the N-end rule. However,it do...
TMPY-01100 GPT2 Protein, Rat, Recombinant (His)

glutamic pyruvate transaminase (alanine aminotransferase) 2

Rat Baculovirus Insect Cells
Alanine aminotransferase (ALT), also known as glutamate pyruvate transaminase (Gpt), is a pyridoxal enzyme that catalyzes the reversible interconversion of L-alanine and 2-oxoglutalate to pyruvate and L-glutamate and plays a key role in the intermediary metabolism of glucose and amino acids. As a key enzyme for gluconeogenesis, Gpt is a widely-used serum marker for liver injury. Two ALT isoenzymes have been identified, ALT1 and ALT2 (GPT1 and GPT2), which are encoded by separate genes and share ...
TMPH-01609 LGI1 Protein, Human, Recombinant (His & Myc)

Leucine-rich glioma-inactivated protein 1,Epitempin-1,LGI1

Human E. coli
Regulates voltage-gated potassium channels assembled from KCNA1, KCNA4 and KCNAB1. It slows down channel inactivation by precluding channel closure mediated by the KCNAB1 subunit. Ligand for ADAM22 that positively regulates synaptic transmission mediated by AMPA-type glutamate receptors. Plays a role in suppressing the production of MMP1/3 through the phosphatidylinositol 3-kinase/ERK pathway. May play a role in the control of neuroblastoma cell survival.
TMPY-03257 Calumenin Protein, Human, Recombinant (His)

calumenin

Human HEK293 Cells
Calumenin belongs to the CREC family. It contains 6 EF-hand domains. Calumenin is expressed in skeletal muscle (at protein level). Calumenin interacts with GGCX and RYR1 in the presence of calcium ions, but not in the presence of EDTA. Calumenin is Involved in regulation of vitamin K-dependent carboxylation of multiple N-terminal glutamate residues. It seems to inhibit gamma-carboxylase GGCX. Calumenin also binds 7 calcium ions with a low affinity and may modulate calcium release from the sarcop...
TMPH-02716 HADH Protein, Mouse, Recombinant (His & SUMO)

Short-chain 3-hydroxyacyl-CoA dehydrogenase,Hydroxyacyl-coen...

Mouse E. coli
Mitochondrial fatty acid beta-oxidation enzyme that catalyzes the third step of the beta-oxidation cycle for medium and short-chain 3-hydroxy fatty acyl-CoAs (C4 to C10). Plays a role in the control of insulin secretion by inhibiting the activation of glutamate dehydrogenase 1 (GLUD1), an enzyme that has an important role in regulating amino acid-induced insulin secretion. HADH Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted...
TMPY-01099 GPT Protein, Rat, Recombinant (His)

Gpt1,ALAT,glutamic-pyruvate transaminase (alanine aminotrans...

Rat Baculovirus Insect Cells
Alanine aminotransferase (ALT), also known as glutamate pyruvate transaminase (GPT), is a pyridoxal enzyme that belongs to the class-I pyridoxal-phosphate-dependent aminotransferase family, Alanine aminotransferase subfamily. Gpt / Gpt1 / ALT catalyzes the reversible interconversion of L-alanine and 2-oxoglutalate to pyruvate and L-glutamate and plays a key role in the intermediary metabolism of glucose and amino acids. Gpt / Gpt1 / ALT is expressed in the liver, kidney, heart, and skeletal musc...
TMPK-00370 PSMA Protein, Human, Recombinant (hFc)

NAALAdase,FOLH1,FOLHNAALADase I,FGCP,mGCP,PSMAFGCP,NAALADase...

Human HEK293 Cells
Prostate-specific membrane antigen (PSMA) is an enzyme that in humans is encoded by the FOLH1 (folate hydrolase 1) gene, also known as Glutamate carboxypeptidase II (GCPII). Human PSMA is highly expressed in the prostate, roughly a hundred times greater than in most other tissues. In some prostate cancers, PSMA is the second-most upregulated gene product, with an 8- to 12-fold increase over levels in noncancerous prostate cells. PSMA Protein, Human, Recombinant (hFc) is expressed in HEK293 mamma...
TMPK-00521 PSMA Protein, Cynomolgus, Recombinant (His)

PSMA,FOLHNAALADase I,FGCP,GCPII,PSMAFGCP,NAALADase I,PSM,NAA...

Cynomolgus HEK293 Cells
Prostate-specific membrane antigen (PSMA) is an enzyme that in humans is encoded by the FOLH1 (folate hydrolase 1) gene, also known as Glutamate carboxypeptidase II (GCPII). Human PSMA is highly expressed in the prostate, roughly a hundred times greater than in most other tissues. In some prostate cancers, PSMA is the second-most upregulated gene product, with an 8- to 12-fold increase over levels in noncancerous prostate cells. PSMA Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 ...
TMPK-00522 PSMA Protein (Primary Amine Labeling), Cynomolgus, Recombinant (His), Biotinylated

PSMAFGCP,PSM,NAALAdase,NAALADase I,FOLHNAALADase I,GCPIImGCP...

Cynomolgus HEK293 Cells
Prostate-specific membrane antigen (PSMA) is an enzyme that in humans is encoded by the FOLH1 (folate hydrolase 1) gene, also known as Glutamate carboxypeptidase II (GCPII). Human PSMA is highly expressed in the prostate, roughly a hundred times greater than in most other tissues. In some prostate cancers, PSMA is the second-most upregulated gene product, with an 8- to 12-fold increase over levels in noncancerous prostate cells. PSMA Protein (Primary Amine Labeling), Cynomolgus, Recombinant (His...
TMPK-00371 PSMA Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated

NAALADase I,FOLH1,GCPIImGCP,FGCP,GCP2,PSM,mGCP,NAALAdase,FOL...

Mouse HEK293 Cells
Prostate-specific membrane antigen (PSMA) is an enzyme that in humans is encoded by the FOLH1 (folate hydrolase 1) gene, also known as Glutamate carboxypeptidase II (GCPII). Human PSMA is highly expressed in the prostate, roughly a hundred times greater than in most other tissues. In some prostate cancers, PSMA is the second-most upregulated gene product, with an 8- to 12-fold increase over levels in noncancerous prostate cells. PSMA Protein (Primary Amine Labeling), Mouse, Recombinant (His), Bi...
TMPJ-00871 BAR Protein, S. hygroscopicus, Recombinant

bar,PPT N-acetyltransferase,Phosphinothricin-resistance prot...

Streptomyces hygroscopicus E. coli
Phosphinothricin N-acetyltransferase (PAT) is an enzyme that acetylates the free NH2 group of L-phosphinothricin (L-PPT) in the presence of acetyl-CoA as a co-substrate. It is highly specific for L-PPT and does not acetylate other L-amino acids or structurally similar molecules. L-PPT is a glutamate analog that can inhibit glutamine synthetase activity in plants, resulting in the accumulation of ammonia to toxic levels and impairment of photosynthesis. The introduction of a PAT gene into a plant...
TMPJ-01130 NPTX1 Protein, Human, Recombinant (His)

Neuronal pentraxin-1,NPTX1,NP1

Human HEK293 Cells
Neuronal Pentraxin (NPTX1, NP1) is a secreted glycoprotein within the Pentraxin family. NPTX1 is co‑expressed and forms heteromultimers with the related secreted protein, NPTX2/NARP, NPTXR (Neuronal Pentraxin Receptor) at excitatory synapses. Mature human NPTX1 shares 97% aa sequence identity with mouse, and rat NPTX1. It is produced by hippocampal, cerebral and cerebellar neurons, retinal ganglia and the inner nuclear layer of the retina. It is enriched on presynaptic axonal membranes where it ...
TMPY-00286 Neuropeptide Y Protein, Human, Recombinant (hFc)

PYY4,neuropeptide Y

Human HEK293 Cells
NPY (Neuropeptide Y) is a Protein Coding gene. This gene encodes a neuropeptide that is widely expressed in the central nervous system and influences many physiological processes, including cortical excitability, stress response, food intake, circadian rhythms, and cardiovascular function. NPY is a neuromodulator that is widely expressed throughout the central nervous system (CNS) and is consecrated with classic neurotransmitters including GABA and glutamate. NPY/Agouti-related protein (AgRP) ne...
TMPY-03445 Aspartate Aminotransferase Protein, Human, Recombinant (His)

ASTQTL1,glutamic-oxaloacetic transaminase 1, soluble,cCAT,cA...

Human E. coli
GOT1 (Glutamic-Oxaloacetic Transaminase 1) is a Protein Coding gene. GOT1 belongs to the class-I pyridoxal-phosphate-dependent aminotransferase family. Glutamic-oxaloacetic transaminase is a pyridoxal phosphate-dependent enzyme that exists in cytoplasmic and mitochondrial forms, GOT1 and GOT2, respectively. GOT plays a role in amino acid metabolism and the urea and tricarboxylic acid cycles. The two enzymes are homodimeric and show close homology. GOT1 is an important regulator of levels of glut...
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重组蛋白

Glutamate racemase Protein, Helicobacter pylori, Recombinant (His & Myc)
Cat.No: TMPH-00795
Species: Helicobacter pylori
Expression System: E. coli
GAD65 Protein, Human, Recombinant (GST)
Cat.No: TMPY-04699
Species: Human
Expression System: Baculovirus Insect Cells
GLUL Protein, Human, Recombinant (His)
Cat.No: TMPJ-00855
Species: Human
Expression System: E. coli
GAD-alpha Protein, E. coli, Recombinant (His)
Cat.No: TMPH-00627
Species: E. coli
Expression System: E. coli
GRIA2 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01392
Species: Human
Expression System: E. coli
GRIA3 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01393
Species: Human
Expression System: E. coli
NAD-GDH Protein, Clostridium difficile, Recombinant (His)
Cat.No: TMPH-00416
Species: Peptoclostridium difficile
Expression System: E. coli
GRM5 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01663
Species: Human
Expression System: E. coli
GLUL Protein, Cricetulus griseus, Recombinant (His)
Cat.No: TMPH-00438
Species: Chinese hamster
Expression System: E. coli
GltI/YbeJ Protein, E. coli, Recombinant (His & SUMO)
Cat.No: TMPH-00628
Species: E. coli
Expression System: E. coli
GRIN1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01394
Species: Human
Expression System: E. coli
GAD67 Protein, Human, Recombinant (His)
Cat.No: TMPY-02091
Species: Human
Expression System: Baculovirus Insect Cells
GRIN1 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03304
Species: Rat
Expression System: E. coli
Gamma-GCS Protein, E. coli, Recombinant (His & SUMO)
Cat.No: TMPH-00629
Species: E. coli
Expression System: E. coli
gltX1 Protein, Helicobacter pylori, Recombinant (His)
Cat.No: TMPH-00796
Species: Helicobacter pylori
Expression System: P. pastoris (Yeast)
Carboxypeptidase Q Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-01393
Species: Mouse
Expression System: HEK293 Cells
GPR Protein, E. coli, Recombinant (His)
Cat.No: TMPH-00626
Species: E. coli
Expression System: E. coli
GRIK2 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-04318
Species: Human
Expression System: HEK293 Cells
GAD65 Protein, Mouse, Recombinant (His & GST)
Cat.No: TMPY-01590
Species: Mouse
Expression System: Baculovirus Insect Cells
GAD65 Protein, Mouse, Recombinant
Cat.No: TMPY-03515
Species: Mouse
Expression System: Baculovirus Insect Cells
CPG2 Protein, Pseudomonas sp., Recombinant (GST)
Cat.No: TMPH-03190
Species: Pseudomonas
Expression System: E. coli
GPT Protein, Human, Recombinant (His)
Cat.No: TMPH-00911
Species: Human
Expression System: E. coli
SLC7A11 Protein, Human, Recombinant (His)
Cat.No: TMPH-03750
Species: Human
Expression System: E. coli
SLC17A6 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03400
Species: Rat
Expression System: P. pastoris (Yeast)
SLC1A3 Protein, Human, Recombinant (His & KSI)
Cat.No: TMPH-01314
Species: Human
Expression System: E. coli
CNDP2 Protein, Human, Recombinant (E. coli, His)
Cat.No: TMPH-01199
Species: Human
Expression System: E. coli
NPTXR Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02807
Species: Mouse
Expression System: Baculovirus Insect Cells
IGSF11 Protein, Mouse, Recombinant (His)
Cat.No: TMPK-00798
Species: Mouse
Expression System: HEK293 Cells
NPTX1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02808
Species: Mouse
Expression System: E. coli
NQO2 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02882
Species: Mouse
Expression System: P. pastoris (Yeast)
PFAS Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-01862
Species: Human
Expression System: E. coli
CSAD Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02616
Species: Mouse
Expression System: E. coli
NQO1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02797
Species: Mouse
Expression System: P. pastoris (Yeast)
Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)
Cat.No: TMPH-03604
Species: Streptomyces hygroscopicus
Expression System: E. coli
5-oxoprolinase/OPLAH Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00863
Species: Human
Expression System: E. coli
AADAT Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01596
Species: Human
Expression System: E. coli
NTAQ1 Protein, Human, Recombinant (GST)
Cat.No: TMPJ-00489
Species: Human
Expression System: E. coli
GPT2 Protein, Rat, Recombinant (His)
Cat.No: TMPY-01100
Species: Rat
Expression System: Baculovirus Insect Cells
LGI1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01609
Species: Human
Expression System: E. coli
Calumenin Protein, Human, Recombinant (His)
Cat.No: TMPY-03257
Species: Human
Expression System: HEK293 Cells
HADH Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02716
Species: Mouse
Expression System: E. coli
GPT Protein, Rat, Recombinant (His)
Cat.No: TMPY-01099
Species: Rat
Expression System: Baculovirus Insect Cells
PSMA Protein, Human, Recombinant (hFc)
Cat.No: TMPK-00370
Species: Human
Expression System: HEK293 Cells
PSMA Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPK-00521
Species: Cynomolgus
Expression System: HEK293 Cells
PSMA Protein (Primary Amine Labeling), Cynomolgus, Recombinant (His), Biotinylated
Cat.No: TMPK-00522
Species: Cynomolgus
Expression System: HEK293 Cells
PSMA Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated
Cat.No: TMPK-00371
Species: Mouse
Expression System: HEK293 Cells
BAR Protein, S. hygroscopicus, Recombinant
Cat.No: TMPJ-00871
Species: Streptomyces hygroscopicus
Expression System: E. coli
NPTX1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01130
Species: Human
Expression System: HEK293 Cells
Neuropeptide Y Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00286
Species: Human
Expression System: HEK293 Cells
Aspartate Aminotransferase Protein, Human, Recombinant (His)
Cat.No: TMPY-03445
Species: Human
Expression System: E. coli
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Cat. No. Product Name Target Signaling Pathways
T40376 L-Phenylalanine-15N

L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N

Calcium Channel Membrane transporter/Ion channel; Metabolism
L-Phenylalanine-15N ((S)-2-Amino-3-phenylpropionic acid-15N) 是 15N 标记的 L-Phenylalanine。L-Phenylalanine 是从大肠杆菌中分离出来的一种必需氨基酸。 L-Phenylalanine 广泛用于食品香精和药物的生产。
T37608 Riluzole-13C,15N2

Riluzole-13C,15N2

Riluzole-13C,15N2 is intended for use as an internal standard for the quantification of riluzole by GC- or LC-MS. Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM). Riluzole suppresses glutamate-induced seizures in rats at an ED50 value of 3.2 mg/kg and displays neuroprotective effects in hypoxic animals a...
T39565 L-Glutamic acid-15N

L-Glutamic acid-15N is the 15N-labeled version of L-Glutamic acid, an excitatory neurotransmitter and an agonist at metabotropic, kainate, NMDA, and AMPA glutamate receptor subtypes. It directly activates the release of dopamine (DA) from dopaminergic terminals.
TMIJ-0160 Dextrorphan-d3 Tartrate

Dextromethorphan EP Impurity B-d3 Tartrate

Dextrorphan-d3 Tartrate 是 Dextrorphan Tartrate 的氘代化合物。Dextrorphan Tartrate 的 CAS 号为 77-07-6。Dextrorphan tartrate 是一种非竞争性 NMDA 谷氨酸受体拮抗剂。
T71305 Clofibric Acid-d4

Clofibric acid-d4 is intended for use as an internal standard for the quantification of clofibric acid by GC- or LC-MS. Clofibric acid is a peroxisome proliferator-activated receptor α (PPARα) agonist (EC50 = 50 µM in a transactivation assay) and the active metabolite of clofibrate. It is formed from clofibrate by tissue and serum esterases. Dietary administration of clofibric acid (0.067-0.22%) reduces serum cholesterol, phospholipid, and triglyceride levels in rats. It decreases glutamate oxal...
TMIJ-0030 1-Aminoadamantane-d15

1-Aminoadamantane-d15 是 1-Aminoadamantane 的氘代化合物。1-Aminoadamantane 的 CAS 号为 768-94-5。Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
TMIJ-0019 Amantadine-d6

Amantadine-d6 是 Amantadine 的氘代化合物。Amantadine 的 CAS 号为 768-94-5。Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
TMID-0299 Zonisamide-d4

Zonisamide-d4 是 Zonisamide 的氘代化合物。Zonisamide 的 CAS 号为 68291-97-4。Zonisamide 是锌酶碳酸酐酶 (carbonic anhydrase) 的有效抑制剂,对人类线粒体同工酶 hCA II 和 hCA V 作用的Ki值分别为 35.2 nM 和 20.6 nM。Zonisamide 具有抗癫痫活性,在癫痫、癫痫发作和帕金森病的研究中具有价值。

同位素标记化合物

L-Phenylalanine-15N
Cat.No: T40376
Synonym: L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N
Target: Calcium Channel
Riluzole-13C,15N2
Cat.No: T37608
Synonym: Riluzole-13C,15N2
Target:
L-Glutamic acid-15N
Cat.No: T39565
Synonym:
Target:
Dextrorphan-d3 Tartrate
Cat.No: TMIJ-0160
Synonym: Dextromethorphan EP Impurity B-d3 Tartrate
Target:
Clofibric Acid-d4
Cat.No: T71305
Synonym:
Target:
1-Aminoadamantane-d15
Cat.No: TMIJ-0030
Synonym:
Target:
Amantadine-d6
Cat.No: TMIJ-0019
Synonym:
Target:
Zonisamide-d4
Cat.No: TMID-0299
Synonym:
Target:
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