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ART-IN-1 (compound 7) 是一种 PARP 的选择性抑制剂,对 PARP2, TNKS2, PARP10, PARP14, PARP15 的 IC50值分别为 19, 22, 2.4, >100, 1.1 μM。
ART-IN-1 (compound 7) 是一种 PARP 的选择性抑制剂,对 PARP2, TNKS2, PARP10, PARP14, PARP15 的 IC50值分别为 19, 22, 2.4, >100, 1.1 μM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 10,600 | 6-8周 | |
50 mg | ¥ 13,800 | 6-8周 | |
100 mg | ¥ 17,500 | 6-8周 |
产品描述 | ART-IN-1 (compound 7) is a selective inhibitor of PARP with IC 50 s of 19, 22, 2.4, >100, 1.1 μM for PARP2, TNKS2, PARP10, PARP14, PARP15, respectively [1]. |
体外活性 | ART-IN-1 (compound 7) (0-100 μM) is an analog of TIQ-A which shows inhibition of PARP2, TNKS2, PARP10, PARP14, PARP15 with IC 50 s of 19, 22, 2.4, >100, 1.1 μM, respectively [1]. |
分子量 | 259.32 |
分子式 | C14H13NO2S |
CAS No. | 2418014-98-7 |
存储 | Shipping with blue ice. |
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