89
270
3
4
4
Cat. No. | Product Name | ||
---|---|---|---|
L2900 | 氧化还原化合物库 | 1264 compounds | |
1264 个活性化合物,已经验证具有一定的抗氧化活性,包括 ROS 清除剂、iNOS、eNOS、及抗氧化的天然产物,是研究疾病机理以及药物研究的优良载体 | |||
L6120 | 黄酮类天然产物库 | 514 compounds | |
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L6820 | 烟草单体化合物库 | 747 compounds | |
747种烟草单体化合物的独特集合,可用于高通量筛选和高内涵筛选 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2333 |
cyclo(L-Pro-L-Tyr)
|
Others | Others |
cyclo(L-Pro-L-Tyr) 是真菌和细菌的次生代谢产物。 | |||
T7644 |
DPN
Diarylpropionitrile,2,3-双(4-羟苯基)丙腈 |
Apoptosis; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Autophagy | Apoptosis; Autophagy; Endocrinology/Hormones |
DPN (Diarylpropionitrile) 是一种非甾体雌激素受体 ERβ选择性配体,其 EC50值为 0.85 nM。DPN 在许多神经系统疾病具有神经保护作用。 | |||
T21233 |
Dihydrolipoic acid
Reduced thioctic acid,Reduced lipoic acid,DHLA,USAF XR-12,6,8-Dihydrothioctic acid,二氢硫辛酸 |
Antioxidant | oxidation-reduction |
Dihydrolipoic acid (USAF XR-12) 是高效的抗氧化剂,对所有以氧为中心的自由基都有很强的清除能力。它在多种疾病中表现出抗炎特性。在 LPS 诱导的疾病行为大鼠中,它通过 ERK/Nrf2/HO-1/ROS/NLRP3 通路发挥预防作用。它还可以可用于抑郁症的研究。 | |||
T25985 |
Prifelone
R-830,R830,S-16820,S 16820,R 830 |
Others | Others |
Prifelone (R 830) 是一种非甾体抗炎化合物,具有抗氧化活性。 | |||
T37890L |
GLP-1(28-36)amide acetate
GLP-1(28-36)amide acetate(1225021-13-5 Free base) |
Antioxidant; Glucagon Receptor | GPCR/G Protein; oxidation-reduction |
GLP-1(28-36)amide acetate 抑制线粒体通透性转变,具有抗氧化、抗糖尿病和心脏保护活性。 | |||
T10063 |
LDL-IN-3
|
Antioxidant | oxidation-reduction |
LDL-IN-3 具有抗动脉粥样硬化和抗氧化活性。 | |||
T17111 |
Todralazine hydrochloride
Ecarazine hydrochloride,盐酸托屈嗪 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Todralazine hydrochloride (Ecarazine hydrochloride) 是一种 β2AR 阻滞剂,具有抗氧化和自由基清除活性。 Todralazine hydrochloride 可用于抗高血压的研究。 | |||
T39527 |
Se-DMC
|
Antioxidant | oxidation-reduction |
Se-DMC 具有抗氧化、抗伤害和抗水肿作用,可用于研究与代谢和炎症相关的疾病。 | |||
T23040 |
N-Arachidonylglycine
NA-Gly,N-Arachidonyl Glycine |
Antioxidant | oxidation-reduction |
N-Arachidonylglycine (NA-Gly)是一种具有生物活性的脂质分子,是一种热态依赖性循环代谢物,具有抗炎、抗癌、抗糖尿病和抗氧化活性,可调节人 CD4T 细胞反应性+,可用于研究与代谢疾病相关的营养水平依赖性炎症。 | |||
T4287 |
Succinobucol
Probucol monosuccinate,AGI-1067 |
Antioxidant; Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
Succinobucol (Probucol monosuccinate) 是酚类抗氧化剂,具有抗炎、抗血小板聚集活性。 | |||
T4510 |
Polaprezinc
Zinc L-carnosine,聚普瑞锌,L-肌肽锌 |
Others | Others |
Polaprezinc是一种含有锌和L-carnosine的生物可用螯合物,以其胃肠保护性能、抗溃疡、抗氧化和抗炎效果而闻名。 | |||
T78650 |
Nrf2 activator-3
|
Antioxidant; Nrf2 | Immunology/Inflammation; oxidation-reduction |
Nrf2 activator-3为一种高效 Nrf2 激活剂,具有潜在的抗炎抗氧化抗肿瘤活性,可用于研究神经系统疾病和免疫相关疾病。 | |||
T38041 |
(R)-3-hydroxy Myristic Acid
|
Antioxidant; Serine Protease; Antifungal | Microbiology/Virology; oxidation-reduction; Proteases/Proteasome |
(R)-3-hydroxy Myristic Acid 是一种来自植物乳杆菌MiLAB 14的抗真菌化合物,具有抗氧化、抗弹性蛋白酶和抗脲酶活性,可用于研究真菌感染。 | |||
T8368 |
Geranylacetone(Z/E)
6,10-二甲基-5,9-十一双烯-2-酮,Dihydropseudoionone |
Others | Others |
Geranylacetone(Z/E) (Dihydropseudoionone) 是一种天然存在的化合物,存在于许多植物的精油中,包括迷迭香、薰衣草和茉莉花。它具有抗氧化、抗炎和抗微生物的特性。 | |||
T38343 |
Quercetin pentaacetate
Pentaacetylquercetin |
RSV | Microbiology/Virology |
Quercetin pentaacetate (Pentaacetylquercetin) 具有多种生物活性,包括抗氧化、抗炎和抗癌特性。 Quercetin pentaacetate 与 RSV 相互作用并抑制病毒在细胞表面的粘附。 | |||
T41345 |
AFMK
Formyl-N-acetyl-5-methoxykynurenamine,Acetyl-N-formyl-5-methoxykynurenamine |
Apoptosis; Free radical scavengers; Antioxidant; Endogenous Metabolite | Apoptosis; Metabolism; oxidation-reduction |
AFMK (Formyl-N-acetyl-5-methoxykynurenamine) 是褪黑激素的活性代谢物,具有抗氧化和自由基清除活性。 AFMK 是一种凋亡调节剂,可提高吉西他滨在 PANC-1 细胞中的抗肿瘤作用。 | |||
T26091 |
Riparin III
Riparin |
Antioxidant; Calcium Channel | Membrane transporter/Ion channel; Metabolism; oxidation-reduction |
Riparin III (Riparin) 是一种平滑肌松弛剂,抑制 CaCl2 诱导的收缩。Riparin III 具有潜在的抗氧化、抗炎和抗抑郁,可逆转皮质酮诱导的异常行为和神经化学改变。 | |||
T126022 |
beta-Glucogallin
1-O-Galloyl-β-D-glucose,β-Glucogallin |
Reductase | Endocrinology/Hormones; Metabolism |
beta-Glucogallin (beta-Glucogallin) 是选择性醛糖还原酶 (AKR1B1) 抑制剂,具有抗氧化抗糖化和抗炎特性。beta-Glucogallin 是从余甘子 (Emblica officinalis) 中提取得到的天然化合物,可用于研究糖尿病。 | |||
TP2279L |
Obestatin (rat) acetate
|
GHSR | GPCR/G Protein |
Obestatin (rat) acetate 是 G 蛋白偶联受体 39 (GPR39) 的内源性配体。它具有抗炎、抗心肌梗塞和抗氧化特性。 它抑制食物摄入,抑制空肠收缩,并减少体重增加。 | |||
T83628 |
TNF/IFNγ-IN-1
|
Antioxidant; TNF; COX | Apoptosis; Immunology/Inflammation; Neuroscience; oxidation-reduction |
TNF/IFNγ-IN-1(TGA) 是 TNF 和 IFN-γ 的双重抑制剂。TNF/IFNγ-IN-1 具有潜在的抗氧化和抗炎活性,可用于类似阿尔茨海默等的神经退行性疾病。 | |||
T31615 |
Elsibucol
AGI-1096,UNII-O7T92N1Y8T,AGI 1096 |
Antioxidant | oxidation-reduction |
Elsibucol (AGI 1096) 是一种VCAM1抑制剂,可用于研究器官移植排斥。Elsibucol 是一种代谢稳定的丙醇衍生物,具有抗氧化、抗炎和抗增殖的特性。它能降低血液中的胆固醇水平,减少受伤动脉中的氧化应激和炎症反应,从而抑制动脉粥样硬化,保护动脉损伤后的内皮愈合。 | |||
T4184 |
NSC 409012
5-(4-iodobenzylidene)rhodanine,5-(4-碘苯亚甲基)罗丹宁 |
Others | Others |
NSC-409012 (5-(4-iodobenzylidene)rhodanine) 是一种活性化合物,已被发现具有多种生化和生理作用,包括调节基因表达、细胞增殖和凋亡。它还具有抗炎、抗肿瘤、抗氧化和抗真菌活性。 | |||
T32098L |
Homocarnosine acetate
|
GABA Receptor; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Homocarnosine acetate 是大脑特有的二肽,由 γ-氨基丁酸 (GABA) 和组氨酸组成。它具有抗氧化和抗炎作用、预防 DNA 损伤和抑制晚期糖基化终产物形成 | |||
T125575 |
Isourolithin A
|
Others | Others |
Isourolithin A 是一种天然存在的化合物,存在于各种植物中,包括欧芹、芹菜和洋甘菊。Isourolithin A 是类黄酮家族的一员,以其抗氧化和抗炎特性而闻名。 | |||
T15044 |
D609
|
Apoptosis; Antioxidant | Apoptosis; oxidation-reduction |
D609 (Tricyclodecan-9-yl-Xanthogenate) 具有广泛的生物活性,包括抗氧化、抗凋亡、抗胆碱能、抗肿瘤、抗炎、抗病毒、抗增殖和神经保护活性。D609 通过引起磷脂酰胆碱 (PC) 特异性磷脂酶 C (PC-PLC) 和鞘磷脂合酶 (SMS) 的竞争性抑制来发挥作用。 | |||
T65167 |
EDTA copper(II) disodium salt
|
Antibiotic | Microbiology/Virology |
EDTA copper(II) disodium salt 是一种金属螯合剂,具有抗菌、抗炎、抗氧化活性,可减缓金属离子造成的损伤,可维持蛋白纯化过程中的渗透压,可用于研究神经系统疾病。 | |||
T50003 |
Debrisoquin hydriodide
1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide |
Others | Others |
Debrisoquin hydriodide (1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide) 具有抗氧化、抗炎和神经保护特性,也被发现可以调节某些神经递质的活性,包括多巴胺和血清素,使其成为治疗帕金森病和抑郁症等神经疾病的有前途的候选药物。 | |||
T4632 |
NSC 6038
4-chloro-N,N-dipropylbenzamide,4-Chloro-N,N-di-n-propylbenzaMide,4-氯-N,N-二-N-丙基苯甲酰胺 |
Others | Others |
NSC-6038 (4-chloro-N,N-dipropylbenzamide) 是一种苯甲酰胺类生物活性化合物,具有广泛的生物活性,已被证明具有抗炎、抗氧化和抗血管生成的活性,也被证明能有效治疗多种疾病,如癌症、糖尿病和心血管疾病。 | |||
T7911 |
Arbidol
Umifenovir |
Antiviral; SARS-CoV | Immunology/Inflammation; Microbiology/Virology |
Arbidol (Umifenovir) 是一种具有口服活性广谱抗病毒化合物,属于融合抑制剂,可与 SARS-CoV-2 刺突蛋白相互作用。Arbidol 对多种冠状病毒显示出抑制活性。Arbidol 具有抗炎抗氧化活性,可用于研究浓度感染。 | |||
T5509 |
FPTQ
|
GluR | Neuroscience |
FPTQ,一种mGluR 1的高效拮抗剂,在人类和小鼠mGluR1上展示出6 nM和1.4 nM的IC50值[1]。除了其强大的抑制特性外,FPTQ在体外和体内实验中均表现出显著的抗氧化和抗炎效应[2]。 | |||
T50071 |
Xanthine dehydrogenase Inhibitor 1
|
Others | Others |
5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile 是一种用作分子结构单元的化合物,被认为是 COX-2、5-LOX 等酶的抑制剂,具有多种生化和生理作用,包括抗肿瘤活性、抗炎作用和抗氧化活性。 | |||
T50069 |
1-pentyl-1H-indole-3-carboxylic acid
|
Others | Others |
1-pentyl-1H-indole-3-carboxylic acid 是一种天然存在的吲哚生物碱类化合物,具有多种生物活性,包括抗炎、镇痛、抗氧化和抗真菌、抗肿瘤活性等;它通过结合体内的各种受体和酶发挥作用,包括血清素受体、大麻素受体、PPARγ受体和PDE4酶。 | |||
T32535 |
Ladostigil
TV-3326,Ladostigil,TV 3326,TV3326,Ladostigil free base |
Antioxidant; MAO; AChE | Metabolism; Neuroscience; oxidation-reduction |
Ladostigil (Ladostigil free base) 是一种具有口服活性的胆碱酯酶和脑选择性单胺氧化酶(MAO)双重抑制剂,对 MAO-B 和 AChE 具有抑制作用,IC50值分别为37.1和31.8μM。Ladostigil 具有抗炎、抗氧化和神经保护活性,可用于研究抑郁症和阿尔茨海默病。 | |||
T38164 |
MnTBAP chloride
Mn(III)TBAP |
Others | Others |
MnTBAP chloride (Mn(III)TBAP) 是一种具有细胞渗透性的超氧化物歧化酶 (SOD) 模拟物和过氧亚硝酸盐清除剂,能使SOD-大肠杆菌的加倍时间减少了2倍。 MnTBAP chloride 通过上调 BMPR-II 和抑制 NFκB 信号传导展现抗炎作用。MnTBAP chloride 是一种锰卟啉配合物,具有抗氧化性能,具有用于研究慢性肾脏疾病 (CKDs) 纤维化反应的潜力。 | |||
T28222 |
5-Hydroxy-1-methylhydantoin
HD-003,HD003,5-羟基-1-甲基咪唑啉-2,4-二酮,NZ419,NZ-419,HD 003,NZ 419 |
Bradykinin Receptor | GPCR/G Protein |
5-Hydroxy-1-methylhydantoin (HD-003) 是一种可能用于治疗肾衰竭的抗氧化剂。它是肌酐代谢物,是一种羟基自由基清除剂,此前已显示通过抑制大鼠慢性肾病的进展来提供肾脏保护。 它是一种新型抗氧化药物,可完全抑制 B2-激肽受体(B2KR) 对 VSMC 中高葡萄糖 (25 mM) 刺激的反应,并且还显示可减弱 BK 对 VSMC 重塑的影响。它抑制 BK 诱导的 MAPK 磷酸化增加并减弱 VSMC 中结缔组织生长因子 (CTGF) 蛋白水平的增加。这些研究结果表明,它可能通过其抗氧化特性赋予血管保护免受高葡萄糖浓度和 BK 刺激以改善血管损伤和重塑。 | |||
T36674 |
DMU-212
|
Apoptosis; ERK | Apoptosis; MAPK |
DMU-212 是具有口服活性的白藜芦醇的甲基化衍生物,表现出抗分裂、抗增殖、抗氧化和促进细胞凋亡的活性。它通过诱导凋亡和激活ERK1/2蛋白阻止有丝分裂。 | |||
T27901 |
LY 221068
LY221068,LY-221068 |
Others | Others |
LY 221068 is a potent antioxidant with anti-inflammatory activity. | |||
T25735 |
Linearol
|
Others | Others |
Linearol is a diterpene found in Sideritis L. spp. (Lamiaceae) with a broad range of demonstrated properties including antioxidant, anti-inflammatory, and anti-apoptotic activities. | |||
T83030 |
Antioxidant agent-11
|
Others | Others |
Antioxidant agent-11 (compound 3d) 是具备抗氧化以及轻度抗癌活性的化学化合物。 | |||
T24261 |
KHG26693
KHG-26693,KHG 26693 |
Others | Others |
KHG26693 is an anti-inflammatory and antioxidant agent that acts by significantly decreasing blood glucose, triglycerides, cholesterol and increased insulin. | |||
T14861 |
Camobucol
AGIX 4207 |
Others | Others |
Camobucol is an orally active, anti-inflammatory compound. It also is a phenolic antioxidant with antirheumatic properties. | |||
T27908 |
LY 269415
LY269415,LY-269415 |
Others | Others |
LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis. | |||
T17112 |
Todralazine
Ecarazine |
Others | Others |
Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity. | |||
T23697 |
AL-8417
J1.090.276B,AL8417,(2R)-AL-5898 |
Others | Others |
AL-8417 is an enzyme inhibitor. It acting as an antioxidant, anti-inflammatory, and cytostatic agent. It also has the ability to suppress vitrectomy-induced posterior lens fiber changes. | |||
T37252 |
Chitoheptaose heptahydrochloride
|
Others | Others |
Chitoheptaose heptahydrochloride is a chitosan oligosaccharide with antioxidant, anti-inflammatory, antiapoptotic, and cardioprotective properties. It effectively promotes the growth and photosynthesis parameters of wheat seedlings[1][2]. | |||
T13773 |
Mito-apocynin (C11)
|
Others | Others |
Mito-apocynin (C11)是一种线粒体靶向抗氧化剂,通过靶向和中和细胞呼吸过程中产生的活性氧(ROS)发挥作用。三苯基溴化鏻已被发现能有效预防线粒体功能障碍,线粒体功能障碍是衰老过程和各种疾病的主要原因。它具有抗炎、抗凋亡和抗氧化活性。 | |||
T36178 |
Aspalatone
|
Others | Others |
Aspalatone is an anti-platelet aggregator (IC50 = 180 μM, in vitro) that prolongs bleeding time significantly in a rodent model of thromboembolism. Additionally at a minimal effective dose of 24 mg/kg, aspalatone generates antioxidant and neuroprotective effects against kainic acid-induced epilepsy in rat hippocampus. | |||
T67870 |
DKI5
(E)-N'-benzylidenehydrazinecarbothiohydrazide |
Lipoxygenase | Metabolism |
DKI5 ((E)-N'-benzylidenehydrazinecarbothiohydrazide) 是一种 LOX-1 抑制剂,IC50 值为 22.5 μM。DKI5 可能具有抗炎和抗氧化活性,在体外生物测定中显示出抗脂质过氧化活性。 | |||
T83048 |
Anti-inflammatory agent 64
|
ROS Kinase | Tyrosine Kinase/Adaptors |
Anti-inflammatory agent 64(compound 4b)能抑制IL-6和TNF-α的分泌,具备抗氧化及抗炎活性,无论在体内外均有效,能显著减轻足跖水肿。 | |||
T79538 |
PDE4-IN-13
|
Others | Others |
PDE4-IN-13 is a phosphodiesterase 4 inhibitor with an IC50 value of 1.56 μM, exhibiting anti-inflammatory and antioxidative properties. It is utilized in the study of chronic obstructive pulmonary disease (COPD). |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5660 |
Menthone
|
IL Receptor; TNF; NF-κB; Parasite | Apoptosis; Immunology/Inflammation; Microbiology/Virology; NF-κB |
Menthone 是一种从植物和薄荷油中提取的单萜,是精油的主要挥发性成分,具有抗炎和抗氧化特性。 | |||
T5712 |
zerumbone
花薑酮,球姜酮 |
Antioxidant; HSV | Microbiology/Virology; oxidation-reduction |
Zerumbone 是从Zingiber zerumbetSmith 的根茎中分离的一种单环倍半萜烯,可有效抑制Epstein-Barr 病毒的激活,IC50为 0.14 mM,具有抗癌、抗炎、抗氧化和抗增殖的作用。 | |||
TN1990 |
Norathyriol
芒果苷元 |
Akt; DNA/RNA Synthesis; AMPK; PPAR | Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling |
Norathyriol 是来自芒果的芒果苷代谢物,具有抗氧化、抗癌、抗菌和抗炎活性。它以非竞争性方式抑制 α-葡萄糖苷酶,IC50为 3.12 μM。它还抑制PPARα、PPARβ和PPARγ,IC50分别为 92.8、102.4 和 153.5 µM。 | |||
TN1686 |
Ginsenoside Rg4
人参皂苷 RG4 |
Antibacterial | Microbiology/Virology |
Ginsenoside Rg4 是分离自Panax ginsengC. A. Meyer 叶子中的一种人参三醇型人参皂苷。人参三醇型人参皂苷具有多种生物活性,包括防腐,抗糖尿病,伤口愈合,免疫刺激和抗氧化活性等。 | |||
T4518 |
Licochalcone D
|
ERK; NF-κB | MAPK; NF-κB |
Licochalcone D 是一种 NF-κB p65的有效抑制剂,是一种存在于 Glycyrrhiza inflate 中的黄酮类化合物,具有抗氧化、抗炎、抗癌等作用。 | |||
T9135 |
Epirosmanol
|
Others | Others |
Epirosmanol 是含有内酯部分的二萜类化合物。 Epirosmanol 是一种极弱碱性(基本中性)的化合物(基于其 pKa)。 | |||
T5814 |
Aurantiamide
TMC-58B,橙黄胡椒酰胺 |
p38 MAPK; NF-κB | MAPK; NF-κB |
Aurantiamide 是马齿苋的活性成分,具有多种生物活性(如抗氧化、抗血小板、抗炎、抗肿瘤活性等),具有口服活性。 | |||
T6917 |
Oleuropein
洋橄榄苦甙,橄榄苦苷 |
Apoptosis; Aromatase; ROS; PPAR | Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism |
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。 | |||
TN5634 |
Aureusidin
Auresudidin,金鱼草素,Auresidin |
Antioxidant; Reactive Oxygen Species; Lipoxygenase | Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。 | |||
T6S1572 |
Sauchinone
|
ERK; p38 MAPK; NF-κB | MAPK; NF-κB |
Sauchinone 是一种从Saururus chinensis 中获得的非对映异构的木脂素。它通过抑制I-κBα磷酸化和p65核易位来抑制 LPS 诱导的 iNOS,TNF-α 和 COX-2 表达。它具有抗炎和抗氧化活性。 | |||
T11685 |
Isolongifolene
异长叶烯,(-)-Isolongifolene |
Apoptosis; Others | Apoptosis; Others |
Isolongifolene ((-)-Isolongifolene) 是一种从调料九里香中分离的三环倍半萜烯,具有抗氧化,抗炎,抗癌和神经保护的特性。它通过调节 PI3K/AKT/GSK-3β 信号通路来减轻鱼藤酮诱导的氧化应激,线粒体功能障碍和细胞凋亡。 | |||
TN2883 |
3',4'-Dimethoxyflavone
|
Others; PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair; Others |
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。 | |||
T2899 |
Liquiritin
Liquiritigenin-4'-O-glucoside,Liquiritoside,甘草苷 |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Liquiritin (Liquiritigenin-4'-O-glucoside) 是一种从甘草中分离出的类黄酮,是一种竞争性的 AKR1C1 抑制剂,对 AKR1C1,AKR1C2 和 AKR1C3 的 IC50分别为 0.62 μM,0.61 μM 和 3.72 μM,在体内有效抑制 AKR1C1 介导的孕酮代谢。它是一种抗氧化剂,具有神经保护、抗癌、抗炎的活性。 | |||
T3921 |
Punicalagin
安石榴甙,安石榴苷 |
SARS-CoV; HBV | Microbiology/Virology |
Punicalagin 是一种在石榴中发现的主要鞣花单宁,是可逆且非竞争性的 3CLpro 抑制剂。Punicalagin 具有抗氧化、抗炎和抗肿瘤活性。 | |||
T6569 |
Mimosine
Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine |
Others | Others |
Mimosine (Leucenol) 是一种酪氨酸类似物,具有抗癌和抗炎等活性。它可通过其强大的铁结合活性作为抗氧化剂,是一种 Fe(III) 螯合剂。它作用于人类白血病细胞,通过金属离子螯合、线粒体激活和诱导活性氧产生来诱导细胞凋亡。 | |||
T6S1653 |
Albiflorin
Alibiflorin,芍药内酯苷 |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分,是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。 | |||
T8733 |
Antrodin A
(2-氯苯基)二苯基甲醇,camphorataanhydride A |
Others | Others |
Antrodin A (camphorataanhydride A) 是固体发酵樟脑菌菌丝体的一种主要活性成分。它能够增强肝脏的抗炎及抗氧化能力,维持肠道菌群的稳定,避免酒精对肝脏的损伤。 | |||
T2957 |
Arctigenin
牛蒡苷元,牛蒡子苷元,(-)-Arctigenin |
Apoptosis; MMP; Influenza Virus; Autophagy | Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome |
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。 | |||
TN1237 |
3-O-Methylgallic acid
3,4-Dihydroxy-5-methoxybenzoic acid,3-O-甲基没食子酸 |
Apoptosis; NF-κB; OCT; DNA/RNA Synthesis; STAT | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; JAK/STAT signaling; Membrane transporter/Ion channel; NF-κB; Stem Cells |
3-O-Methylgallic acid (3,4-Dihydroxy-5-methoxybenzoic acid) 是一种花青素代谢产物,具有强大的抗氧化能力。它还诱导细胞凋亡并具有抗癌作用,可抑制 Caco-2 细胞增殖,IC50值为 24.1 μM。 | |||
T3416 |
Aucubin
Aucuboside,桃叶珊瑚苷,Rhinanthin |
IL Receptor; NF-κB; Antibacterial | Immunology/Inflammation; Microbiology/Virology; NF-κB |
Aucubin (Rhinanthin) 是一种可从许多传统的草药中提取的环烯醚萜苷,有许多生物学活性。 | |||
T8516 |
Levomenol
没药醇,(-)-α-BISABOLOL,(-)-α-红没药醇 |
Others | Others |
Levomenol ((-)-α-BISABOLOL) 是一种单环倍半萜醇,具有有神经保护、抗氧化、抗炎和抗凋亡的作用。它可减轻三叉神经性疼痛啮齿动物模型的伤害性行为和中枢敏感性。它通过减少小鼠永久性局灶性脑缺血诱导的促炎标志物,防止神经元损伤和记忆缺陷。 | |||
T2950 |
Schisandrin
Wuweizi alcohol-A,Wuweizichun-A,Schizandrol-A,Schizandrol,五味子醇甲 |
Autophagy | Autophagy |
Schisandrin (Wuweizi alcohol-A) 是一种从五味子中分离出来的联苯环辛烯类木脂素,可逆转大鼠的记忆障碍,具有保肝、抗氧化、抗哮喘、抗癌和抗炎作用。 | |||
T0795 |
Rutin
Quercetin 3-O-rutinoside,芦丁,Rutoside |
Beta Amyloid; Prostaglandin Receptor; Autophagy | Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Rutin (Quercetin 3-O-rutinoside) 属于黄酮类天然产物,具有血脑屏障渗透性。Rutin 具有广泛的生物活性,包括抗氧化、抗炎、抗肿瘤、降血糖、神经保护、抗菌、抗衰老等等。 | |||
T3363 |
Jervine
蒜黎芦碱,Iervin,11-Ketocyclopamine,Jerwiny |
Hedgehog/Smoothened; Smo | GPCR/G Protein; Stem Cells |
Jervine (Jerwiny) 是一种有效的刺猬 (Hh) 抑制剂(IC50:500-700 nM)。它是一种天然致畸性甾体生物碱,来自于 Veratrumalbum 的根茎,具有抗炎和抗氧化作用。 | |||
T5S1923 |
Schisandrin C
五味子丙素,Schizandrin-C,Wuweizisu-C |
Apoptosis; Others; Virus Protease | Apoptosis; Microbiology/Virology; Others |
Schisandrin C (Wuweizisu-C) 是从五味子中分离得到的一种植物化学木脂素。它具有抗癌、抗炎和抗氧化等多种生物活性,可研究癌症、阿尔茨海默病、肝病。 | |||
T0492 |
Dimethyl fumarate
富马酸二甲酯,DMF |
Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy | Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome |
Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂,可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物,可作抗炎和免疫调节剂,可研究多发性硬化症。 | |||
T26288 |
Clovamide
trans-Clovamide,N-trans-Caffeoy-L-dopa |
Apoptosis; Influenza Virus; ROS; Antibacterial | Apoptosis; Immunology/Inflammation; Microbiology/Virology |
Clovamide (trans-Clovamide) 是一种天然存在的咖啡酰结合物,具有抗菌、抗炎、抗氧化和神经保护作用。它是一种极好的活性氧和氧自由基清除剂。 | |||
T5728 |
OsMundacetone
4-(3,4-Dihydroxyphenyl)-3-buten-2-one |
Apoptosis; Reactive Oxygen Species | Apoptosis; Immunology/Inflammation; Metabolism; NF-κB |
OsMundacetone (4-(3,4-Dihydroxyphenyl)-3-buten-2-one) 是从白桦茸中分离出的一种天然产物,具有抗凋亡作用。它具有DPPH 清除活性,保护神经细胞免受氧化应激,可研究神经退行性疾病。 | |||
TN4893 |
Rapanone
拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌 |
Apoptosis; Phospholipase; Antibacterial; Parasite | Apoptosis; Metabolism; Microbiology/Virology |
Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) 是一种具有广泛生物活性的天然苯醌,如抗肿瘤、抗氧化、抗炎、抗菌和抗寄生虫活性。它还是选择性人滑膜 PLA2抑制剂,IC50值为 2.6 μM。 | |||
TL0006 |
Cichoric Acid
菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid |
Reactive Oxygen Species; HIV Protease | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome |
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。 | |||
T22417 |
Rutin hydrate
芦丁,Rutoside,Sophorin,Quercetin-3-O-rutinoside |
Beta Amyloid; Others; Autophagy | Autophagy; Neuroscience; Others |
Rutin hydrate (Sophorin) 是一种广泛存在于多种植物中的黄酮类天然产物,具有降糖、抗炎、抗氧化、神经保护、肾脏保护、肝脏保护和降低 Aβ 低聚物活性等多种生物活性。它能穿过血脑屏障,通过抑制细胞凋亡、线粒体功能紊乱和氧化应激抑制万古霉素诱导的肾小管细胞凋亡。 | |||
TN1238 |
3,4-O-Isopropylidene-shikimic acid
3,4-O-异亚丙基莽草酸,3,4-O-Isopropylidene shikimic acid |
NOS; NO Synthase | Immunology/Inflammation |
3,4-O-Isopropylidene-shikimic acid (3,4-O-Isopropylidene shikimic acid) 是一种从Hypericum wightianum 中提取得到的天然产物。它具有抗炎症和抗氧化作用。 | |||
T2S1158 |
4,5-Dicaffeoylquinic acid
3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C |
Others; HBV; Endogenous Metabolite | Metabolism; Microbiology/Virology; Others |
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。 | |||
TN1353 |
N-Benzyllinoleamide
(9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺 |
Others | Others |
N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) 是一种分离自 Lepidium meyeniiWalp,能够抗运动性疲劳的药物。 | |||
T4S1659 |
Xanthotoxol
8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene |
Reactive Oxygen Species; 5-HT Receptor; Endogenous Metabolite | GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
Xanthotoxol (Psoralen) 是一种具有生物活性的线性呋喃香豆素,具有很强的抗炎、抗氧化、5-HT 拮抗和神经保护作用等药理活性。 | |||
T6S1917 |
Schisandrol B
Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B |
P450; Reactive Oxygen Species; Autophagy | Autophagy; Immunology/Inflammation; Metabolism; NF-κB |
Schisandrol B (Besigomsin) 是华中五味子的主要活性成分,具有保肝、抗炎、抗糖尿病和抗氧化的作用。它抑制活性氧的产生,也抑制 P-糖蛋白和CYP3A 的活性。 | |||
TN6732 |
Oenothein B
|
Apoptosis; HCV Protease; Antibacterial; Antifungal | Apoptosis; Microbiology/Virology; Proteases/Proteasome |
Oenothein B 是一种聚(ADP-核糖)糖水解酶的特异性抑制剂。 Oenothein B 具有抗氧化、抗炎、抗真菌、抗 HCV 和抗肿瘤特性。 | |||
T5145 |
Oxytocin acetate
Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素 |
Oxytocin Receptor | Endocrinology/Hormones; GPCR/G Protein |
Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。 | |||
T6S1101 |
Astragalin
Kaempferol 3-D-glucoside,Kaempferol 3-O-glucoside,kaempferol-3-glucoside,3-Glucosylkaempferol,Astragaline,紫云英苷,Kaempferol 3-β-D-glucopyranoside |
Apoptosis; NF-κB | Apoptosis; NF-κB |
Astragalin (Kaempferol 3-O-glucoside) 是一种具有生物活性的天然黄酮类化合物。 它具有多种药理特性,包括抗氧化、抗炎、抗癌、神经保护和心脏保护特性。 | |||
T2S2104 |
Sinigrin hydrate
黑芥子苷,Sinigrin monohydrate,芥子甙单水合物,Allylglucosinolate monohydrate |
Antibacterial | Microbiology/Virology |
Sinigrin hydrate (Allylglucosinolate monohydrate) 是一种天然脂肪族芥子油苷,存在于十字花科植物中。它具有消炎、抗癌、抗真菌、抗菌、抗氧化作用。 | |||
T3376 |
Cynaroside
朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside |
Others; Influenza Virus; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。 | |||
TQ0188 |
Miquelianin
槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide |
stilbene oxidase; Endogenous Metabolite | Metabolism |
Miquelianin (Quercetin 3-glucuronide) 是槲皮素的代谢产物,属于类黄酮化合物。 | |||
TN2233 |
Spathulenol
|
Antioxidant; Antifungal | Microbiology/Virology; oxidation-reduction |
Spathulenol 是一种来自 Aristolochia yunnanensis 的天然成分,具有抗炎、抗氧化、抗增殖、抗溃疡和抗分枝杆菌活性。 Spathulenol 在 DPPH 系统中显示出显著的抗氧化活性,IC50 为 85.60 μg/mL。 | |||
TN1599 |
Eburicoic acid
Eburicoicacid,MFCD00238594,ZINC4655149,齿孔菌酸 |
Antioxidant; TNF; NOS; NO Synthase; CCR; Immunology/Inflammation related | Apoptosis; Immunology/Inflammation; Microbiology/Virology; oxidation-reduction |
Eburicoic acid (ZINC4655149) 具有抗炎和抗氧化活性,从而保护肝脏免受 CCl4 引起的肝损伤,可用于抗肝癌研究。 | |||
TN1438 |
beta-Amyrin acetate
beta-香树脂醇乙酸酯 |
Antioxidant; HMG-CoA Reductase; Epoxide Hydrolase; Antifungal | Metabolism; Microbiology/Virology; oxidation-reduction |
beta-Amyrin acetate 抑制 HMG-CoA 还原酶 (HMGCR) 和 sEH 活性,IC50 为 3.4 μM。 beta-Amyrin acetate 具有抗炎、抗真菌、抗氧化和抗高血脂活性。 | |||
T2837 |
Chrysin
5, 7-Dihydroxyflavone,NSC 407436,白杨素,5,7-Dihydroxyflavone |
Estrogen Receptor/ERR; Antioxidant | Endocrinology/Hormones; oxidation-reduction |
Chrysin (5,7-Dihydroxyflavone) 是一种雌激素阻断剂。 | |||
T5098 |
Isochlorogenic acid A
3,5-CQA,异绿原酸 A,3,5-Dicaffeoylquinic acid,金银花 |
Reactive Oxygen Species; HBV; Endogenous Metabolite | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Isochlorogenic acid A (3,5-Dicaffeoylquinic acid) 是一种天然酚酸,具有抗氧化和抗炎活性。 | |||
TN1432 |
Bacopasaponin C
(-)-假马齿苋皂苷 C,假马齿苋皂苷C |
Anti-infection; GABA Receptor; NMDAR | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷,具有抗肿瘤和抗利什曼原虫作用。 | |||
T2912 |
Ergosterol
麦角固醇,Provitamin D,Ergosterin,Provitamin D2 |
Others; Antioxidant; Endogenous Metabolite | Metabolism; Others; oxidation-reduction |
Ergosterol 是真菌中的主要固醇类,具有抗炎,抗氧化和抗增殖的作用。 | |||
T1368 |
Methyl 3,4-dihydroxybenzoate
3,4-Dihydroxybenzoic acid methyl ester,Methyl protocatechuate,原儿茶酸甲酯,3,4-二羟基苯甲酸甲酯,Protocatechuic acid methyl ester |
Apoptosis; Antioxidant; Nrf2 | Apoptosis; Immunology/Inflammation; oxidation-reduction |
Methyl 3,4-dihydroxybenzoate (Protocatechuic acid methyl ester) 是绿茶中发现的主要代谢产物,是一种多酚,有抗氧化和抗炎作用。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-02084 |
Thioredoxin 2/TRX2 Protein, Human, Recombinant (His)
MT-TRX,RP5-1119A7. 13-005,TRX2,MTRX,thioredoxin 2 |
Human | E. coli |
Thioredoxin-2, also known as TXN2, MTRX and TRX2, is a member of the thioredoxin family. Tryparedoxins (TXN) are thioredoxin-related proteins which, as trypanothione:peroxiredoxin oxidoreductases, constitute the trypanothione-dependent antioxidant defense and may also serve as substrates for ribonucleotide reductase in trypanosomatids. Thioredoxin-2 / TXN2 contains one thioredoxin domain. It is widely expressed in adult (at protein level) and fetal tissues. Human Thioredoxin-2 / TXN2 is a small ... | |||
TMPY-04122 |
ATOX1 Protein, Human, Recombinant (His)
HAH1,ATX1,antioxidant 1 copper chaperone |
Human | E. coli |
ATOX1 is a cytoplasmic copper chaperone that interacts with the copper-binding domain of the membrane copper transporters ATP7A and ATP7B. ATOX1 has also been suggested to have a potential anti-oxidant activity. As the trace element copper is essential, but extremely toxic in high concentrations, intracellular copper concentrations are tightly controlled. Once in the cell, copper is distributed by metallochaperones, including the small cytoplasmic protein ATOX1. ATOX1 plays an important role in ... | |||
TMPJ-01106 |
NAD(P) transhydrogenase/NNT Protein, Human, Recombinant (His)
NAD(P) transhydrogenase,NNT |
Human | E. coli |
NAD(P)+transhydrogenase (NNT) is located in the inner mitochondrial membrane and catalyzes a reversible hydride transfer between NAD(H) and NADP(H) that is coupled to proton translocation between the intermembrane space and mitochondrial matrix. NNT activity has an essential role in maintaining the NADPH supply for antioxidant defense and biosynthetic pathways. Structurally, NNT is composed of three domains; domains I and III are hydrophilic and have binding sites for NAD and NADP, respectively,... | |||
TMPY-00186 |
GHRH Protein, Human, Recombinant (hFc)
GRF,INN,growth hormone releasing hormone,GHRF |
Human | HEK293 Cells |
The role of hypothalamic growth hormone-releasing hormone (GHRH) in the release of growth hormone (GH) from the pituitary is well established. Extra-hypothalamic growth hormone-releasing hormone (GHRH) plays an important role in infertility. Growth hormone releasing hormone (GHRH) has recently been shown to increase the level of gamma-aminobutyric acid (GABA) and activate GABA receptors (GABARs) in the cerebral cortex. GABA is an inhibitory neurotransmitter that can inhibit seizures. GHRH may pl... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10901 |
Curcumin-d6
Turmeric yellow D6,Natural Yellow 3 D6,Curcumin D6,Diferuloylmethane D6 |
Others | Others |
Curcumin D6 (difluoroformylmethane D6) is deuterium-labeled curcumin (Turmeric yellow). Curcumin (Turmeric yellow) is a natural phenolic compound with various pharmacological effects, including anti-inflammatory, antioxidant, anti-proliferative and anti-a | |||
TMIH-0181 |
Demethoxy Curcumin-d4
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Demethoxy Curcumin-d4 是 Demethoxy Curcumin 的氘代化合物。Demethoxy Curcumin 的 CAS 号为 22608-11-3。Demethoxycurcumin是姜黄素的主要活性成分,有抗炎和抗癌作用。 | |||
TMIJ-0194 |
Tetramethylpyrazine-d12
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Tetramethylpyrazine-d12 是 Tetramethylpyrazine 的氘代化合物。Tetramethylpyrazine 的 CAS 号为 1124-11-4。Tetramethylpyrazine 是从Ligusticum wallichii中提取的一种烷基吡嗪,常在薯条、面包、茶、乳制品、豆制品等食物中作为香精。它对大鼠具有潜在的抗神经和抗炎活性。 | |||
TMID-0254 |
Linalool-d3
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Linalool-d3 是 Linalool 的氘代化合物。Linalool 的 CAS 号为 78-70-6。Linalool 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。 |