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Search Results for " anti-antioxidant "
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抑制剂 & 化合物

270

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同位素标记化合物

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Cat. No. Product Name
L2900 氧化还原化合物库

1264 compounds
1264 个活性化合物,已经验证具有一定的抗氧化活性,包括 ROS 清除剂、iNOS、eNOS、及抗氧化的天然产物,是研究疾病机理以及药物研究的优良载体
L6120 黄酮类天然产物库

514 compounds
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L6820 烟草单体化合物库

747 compounds
747种烟草单体化合物的独特集合,可用于高通量筛选和高内涵筛选

化合物库

氧化还原化合物库
Cat.No: L2900
Compounds: 1264
黄酮类天然产物库
Cat.No: L6120
Compounds: 514
烟草单体化合物库
Cat.No: L6820
Compounds: 747
Cat. No. Product Name Target Signaling Pathways
TP2333 cyclo(L-Pro-L-Tyr)

Others Others
cyclo(L-Pro-L-Tyr) 是真菌和细菌的次生代谢产物。
T7644 DPN

Diarylpropionitrile,2,3-双(4-羟苯基)丙腈

Apoptosis; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones
DPN (Diarylpropionitrile) 是一种非甾体雌激素受体 ERβ选择性配体,其 EC50值为 0.85 nM。DPN 在许多神经系统疾病具有神经保护作用。
T21233 Dihydrolipoic acid

Reduced thioctic acid,Reduced lipoic acid,DHLA,USAF XR-12,6,8-Dihydrothioctic acid,二氢硫辛酸

Antioxidant oxidation-reduction
Dihydrolipoic acid (USAF XR-12) 是高效的抗氧化剂,对所有以氧为中心的自由基都有很强的清除能力。它在多种疾病中表现出抗炎特性。在 LPS 诱导的疾病行为大鼠中,它通过 ERK/Nrf2/HO-1/ROS/NLRP3 通路发挥预防作用。它还可以可用于抑郁症的研究。
T25985 Prifelone

R-830,R830,S-16820,S 16820,R 830

Others Others
Prifelone (R 830) 是一种非甾体抗炎化合物,具有抗氧化活性。
T37890L GLP-1(28-36)amide acetate

GLP-1(28-36)amide acetate(1225021-13-5 Free base)

Antioxidant; Glucagon Receptor GPCR/G Protein; oxidation-reduction
GLP-1(28-36)amide acetate 抑制线粒体通透性转变,具有抗氧化、抗糖尿病和心脏保护活性。
T10063 LDL-IN-3

Antioxidant oxidation-reduction
LDL-IN-3 具有抗动脉粥样硬化和抗氧化活性。
T17111 Todralazine hydrochloride

Ecarazine hydrochloride,盐酸托屈嗪

Adrenergic Receptor GPCR/G Protein; Neuroscience
Todralazine hydrochloride (Ecarazine hydrochloride) 是一种 β2AR 阻滞剂,具有抗氧化和自由基清除活性。 Todralazine hydrochloride 可用于抗高血压的研究。
T39527 Se-DMC

Antioxidant oxidation-reduction
Se-DMC 具有抗氧化、抗伤害和抗水肿作用,可用于研究与代谢和炎症相关的疾病。
T23040 N-Arachidonylglycine

NA-Gly,N-Arachidonyl Glycine

Antioxidant oxidation-reduction
N-Arachidonylglycine (NA-Gly)是一种具有生物活性的脂质分子,是一种热态依赖性循环代谢物,具有抗炎、抗癌、抗糖尿病和抗氧化活性,可调节人 CD4T 细胞反应性+,可用于研究与代谢疾病相关的营养水平依赖性炎症。
T4287 Succinobucol

Probucol monosuccinate,AGI-1067

Antioxidant; Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Succinobucol (Probucol monosuccinate) 是酚类抗氧化剂,具有抗炎、抗血小板聚集活性。
T4510 Polaprezinc

Zinc L-carnosine,聚普瑞锌,L-肌肽锌

Others Others
Polaprezinc是一种含有锌和L-carnosine的生物可用螯合物,以其胃肠保护性能、抗溃疡、抗氧化和抗炎效果而闻名。
T78650 Nrf2 activator-3

Antioxidant; Nrf2 Immunology/Inflammation; oxidation-reduction
Nrf2 activator-3为一种高效 Nrf2 激活剂,具有潜在的抗炎抗氧化抗肿瘤活性,可用于研究神经系统疾病和免疫相关疾病。
T38041 (R)-3-hydroxy Myristic Acid

Antioxidant; Serine Protease; Antifungal Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
(R)-3-hydroxy Myristic Acid 是一种来自植物乳杆菌MiLAB 14的抗真菌化合物,具有抗氧化、抗弹性蛋白酶和抗脲酶活性,可用于研究真菌感染。
T8368 Geranylacetone(Z/E)

6,10-二甲基-5,9-十一双烯-2-酮,Dihydropseudoionone

Others Others
Geranylacetone(Z/E) (Dihydropseudoionone) 是一种天然存在的化合物,存在于许多植物的精油中,包括迷迭香、薰衣草和茉莉花。它具有抗氧化、抗炎和抗微生物的特性。
T38343 Quercetin pentaacetate

Pentaacetylquercetin

RSV Microbiology/Virology
Quercetin pentaacetate (Pentaacetylquercetin) 具有多种生物活性,包括抗氧化、抗炎和抗癌特性。 Quercetin pentaacetate 与 RSV 相互作用并抑制病毒在细胞表面的粘附。
T41345 AFMK

Formyl-N-acetyl-5-methoxykynurenamine,Acetyl-N-formyl-5-methoxykynurenamine

Apoptosis; Free radical scavengers; Antioxidant; Endogenous Metabolite Apoptosis; Metabolism; oxidation-reduction
AFMK (Formyl-N-acetyl-5-methoxykynurenamine) 是褪黑激素的活性代谢物,具有抗氧化和自由基清除活性。 AFMK 是一种凋亡调节剂,可提高吉西他滨在 PANC-1 细胞中的抗肿瘤作用。
T26091 Riparin III

Riparin

Antioxidant; Calcium Channel Membrane transporter/Ion channel; Metabolism; oxidation-reduction
Riparin III (Riparin) 是一种平滑肌松弛剂,抑制 CaCl2 诱导的收缩。Riparin III 具有潜在的抗氧化、抗炎和抗抑郁,可逆转皮质酮诱导的异常行为和神经化学改变。
T126022 beta-Glucogallin

1-O-Galloyl-β-D-glucose,β-Glucogallin

Reductase Endocrinology/Hormones; Metabolism
beta-Glucogallin (beta-Glucogallin) 是选择性醛糖还原酶 (AKR1B1) 抑制剂,具有抗氧化抗糖化和抗炎特性。beta-Glucogallin 是从余甘子 (Emblica officinalis) 中提取得到的天然化合物,可用于研究糖尿病。
TP2279L Obestatin (rat) acetate

GHSR GPCR/G Protein
Obestatin (rat) acetate 是 G 蛋白偶联受体 39 (GPR39) 的内源性配体。它具有抗炎、抗心肌梗塞和抗氧化特性。 它抑制食物摄入,抑制空肠收缩,并减少体重增加。
T83628 TNF/IFNγ-IN-1

Antioxidant; TNF; COX Apoptosis; Immunology/Inflammation; Neuroscience; oxidation-reduction
TNF/IFNγ-IN-1(TGA) 是 TNF 和 IFN-γ 的双重抑制剂。TNF/IFNγ-IN-1 具有潜在的抗氧化和抗炎活性,可用于类似阿尔茨海默等的神经退行性疾病。
T31615 Elsibucol

AGI-1096,UNII-O7T92N1Y8T,AGI 1096

Antioxidant oxidation-reduction
Elsibucol (AGI 1096) 是一种VCAM1抑制剂,可用于研究器官移植排斥。Elsibucol 是一种代谢稳定的丙醇衍生物,具有抗氧化、抗炎和抗增殖的特性。它能降低血液中的胆固醇水平,减少受伤动脉中的氧化应激和炎症反应,从而抑制动脉粥样硬化,保护动脉损伤后的内皮愈合。
T4184 NSC 409012

5-(4-iodobenzylidene)rhodanine,5-(4-碘苯亚甲基)罗丹宁

Others Others
NSC-409012 (5-(4-iodobenzylidene)rhodanine) 是一种活性化合物,已被发现具有多种生化和生理作用,包括调节基因表达、细胞增殖和凋亡。它还具有抗炎、抗肿瘤、抗氧化和抗真菌活性。
T32098L Homocarnosine acetate

GABA Receptor; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
Homocarnosine acetate 是大脑特有的二肽,由 γ-氨基丁酸 (GABA) 和组氨酸组成。它具有抗氧化和抗炎作用、预防 DNA 损伤和抑制晚期糖基化终产物形成
T125575 Isourolithin A

Others Others
Isourolithin A 是一种天然存在的化合物,存在于各种植物中,包括欧芹、芹菜和洋甘菊。Isourolithin A 是类黄酮家族的一员,以其抗氧化和抗炎特性而闻名。
T15044 D609

Apoptosis; Antioxidant Apoptosis; oxidation-reduction
D609 (Tricyclodecan-9-yl-Xanthogenate) 具有广泛的生物活性,包括抗氧化、抗凋亡、抗胆碱能、抗肿瘤、抗炎、抗病毒、抗增殖和神经保护活性。D609 通过引起磷脂酰胆碱 (PC) 特异性磷脂酶 C (PC-PLC) 和鞘磷脂合酶 (SMS) 的竞争性抑制来发挥作用。
T65167 EDTA copper(II) disodium salt

Antibiotic Microbiology/Virology
EDTA copper(II) disodium salt 是一种金属螯合剂,具有抗菌、抗炎、抗氧化活性,可减缓金属离子造成的损伤,可维持蛋白纯化过程中的渗透压,可用于研究神经系统疾病。
T50003 Debrisoquin hydriodide

1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide

Others Others
Debrisoquin hydriodide (1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide) 具有抗氧化、抗炎和神经保护特性,也被发现可以调节某些神经递质的活性,包括多巴胺和血清素,使其成为治疗帕金森病和抑郁症等神经疾病的有前途的候选药物。
T4632 NSC 6038

4-chloro-N,N-dipropylbenzamide,4-Chloro-N,N-di-n-propylbenzaMide,4-氯-N,N-二-N-丙基苯甲酰胺

Others Others
NSC-6038 (4-chloro-N,N-dipropylbenzamide) 是一种苯甲酰胺类生物活性化合物,具有广泛的生物活性,已被证明具有抗炎、抗氧化和抗血管生成的活性,也被证明能有效治疗多种疾病,如癌症、糖尿病和心血管疾病。
T7911 Arbidol

Umifenovir

Antiviral; SARS-CoV Immunology/Inflammation; Microbiology/Virology
Arbidol (Umifenovir) 是一种具有口服活性广谱抗病毒化合物,属于融合抑制剂,可与 SARS-CoV-2 刺突蛋白相互作用。Arbidol 对多种冠状病毒显示出抑制活性。Arbidol 具有抗炎抗氧化活性,可用于研究浓度感染。
T5509 FPTQ

GluR Neuroscience
FPTQ,一种mGluR 1的高效拮抗剂,在人类和小鼠mGluR1上展示出6 nM和1.4 nM的IC50值[1]。除了其强大的抑制特性外,FPTQ在体外和体内实验中均表现出显著的抗氧化和抗炎效应[2]。
T50071 Xanthine dehydrogenase Inhibitor 1

Others Others
5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile 是一种用作分子结构单元的化合物,被认为是 COX-2、5-LOX 等酶的抑制剂,具有多种生化和生理作用,包括抗肿瘤活性、抗炎作用和抗氧化活性。
T50069 1-pentyl-1H-indole-3-carboxylic acid

Others Others
1-pentyl-1H-indole-3-carboxylic acid 是一种天然存在的吲哚生物碱类化合物,具有多种生物活性,包括抗炎、镇痛、抗氧化和抗真菌、抗肿瘤活性等;它通过结合体内的各种受体和酶发挥作用,包括血清素受体、大麻素受体、PPARγ受体和PDE4酶。
T32535 Ladostigil

TV-3326,Ladostigil,TV 3326,TV3326,Ladostigil free base

Antioxidant; MAO; AChE Metabolism; Neuroscience; oxidation-reduction
Ladostigil (Ladostigil free base) 是一种具有口服活性的胆碱酯酶和脑选择性单胺氧化酶(MAO)双重抑制剂,对 MAO-B 和 AChE 具有抑制作用,IC50值分别为37.1和31.8μM。Ladostigil 具有抗炎、抗氧化和神经保护活性,可用于研究抑郁症和阿尔茨海默病。
T38164 MnTBAP chloride

Mn(III)TBAP

Others Others
MnTBAP chloride (Mn(III)TBAP) 是一种具有细胞渗透性的超氧化物歧化酶 (SOD) 模拟物和过氧亚硝酸盐清除剂,能使SOD-大肠杆菌的加倍时间减少了2倍。 MnTBAP chloride 通过上调 BMPR-II 和抑制 NFκB 信号传导展现抗炎作用。MnTBAP chloride 是一种锰卟啉配合物,具有抗氧化性能,具有用于研究慢性肾脏疾病 (CKDs) 纤维化反应的潜力。
T28222 5-Hydroxy-1-methylhydantoin

HD-003,HD003,5-羟基-1-甲基咪唑啉-2,4-二酮,NZ419,NZ-419,HD 003,NZ 419

Bradykinin Receptor GPCR/G Protein
5-Hydroxy-1-methylhydantoin (HD-003) 是一种可能用于治疗肾衰竭的抗氧化剂。它是肌酐代谢物,是一种羟基自由基清除剂,此前已显示通过抑制大鼠慢性肾病的进展来提供肾脏保护。 它是一种新型抗氧化药物,可完全抑制 B2-激肽受体(B2KR) 对 VSMC 中高葡萄糖 (25 mM) 刺激的反应,并且还显示可减弱 BK 对 VSMC 重塑的影响。它抑制 BK 诱导的 MAPK 磷酸化增加并减弱 VSMC 中结缔组织生长因子 (CTGF) 蛋白水平的增加。这些研究结果表明,它可能通过其抗氧化特性赋予血管保护免受高葡萄糖浓度和 BK 刺激以改善血管损伤和重塑。
T36674 DMU-212

Apoptosis; ERK Apoptosis; MAPK
DMU-212 是具有口服活性的白藜芦醇的甲基化衍生物,表现出抗分裂、抗增殖、抗氧化和促进细胞凋亡的活性。它通过诱导凋亡和激活ERK1/2蛋白阻止有丝分裂。
T27901 LY 221068

LY221068,LY-221068

Others Others
LY 221068 is a potent antioxidant with anti-inflammatory activity.
T25735 Linearol

Others Others
Linearol is a diterpene found in Sideritis L. spp. (Lamiaceae) with a broad range of demonstrated properties including antioxidant, anti-inflammatory, and anti-apoptotic activities.
T83030 Antioxidant agent-11

Others Others
Antioxidant agent-11 (compound 3d) 是具备抗氧化以及轻度抗癌活性的化学化合物。
T24261 KHG26693

KHG-26693,KHG 26693

Others Others
KHG26693 is an anti-inflammatory and antioxidant agent that acts by significantly decreasing blood glucose, triglycerides, cholesterol and increased insulin.
T14861 Camobucol

AGIX 4207

Others Others
Camobucol is an orally active, anti-inflammatory compound. It also is a phenolic antioxidant with antirheumatic properties.
T27908 LY 269415

LY269415,LY-269415

Others Others
LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis.
T17112 Todralazine

Ecarazine

Others Others
Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.
T23697 AL-8417

J1.090.276B,AL8417,(2R)-AL-5898

Others Others
AL-8417 is an enzyme inhibitor. It acting as an antioxidant, anti-inflammatory, and cytostatic agent. It also has the ability to suppress vitrectomy-induced posterior lens fiber changes.
T37252 Chitoheptaose heptahydrochloride

Others Others
Chitoheptaose heptahydrochloride is a chitosan oligosaccharide with antioxidant, anti-inflammatory, antiapoptotic, and cardioprotective properties. It effectively promotes the growth and photosynthesis parameters of wheat seedlings[1][2].
T13773 Mito-apocynin (C11)

Others Others
Mito-apocynin (C11)是一种线粒体靶向抗氧化剂,通过靶向和中和细胞呼吸过程中产生的活性氧(ROS)发挥作用。三苯基溴化鏻已被发现能有效预防线粒体功能障碍,线粒体功能障碍是衰老过程和各种疾病的主要原因。它具有抗炎、抗凋亡和抗氧化活性。
T36178 Aspalatone

Others Others
Aspalatone is an anti-platelet aggregator (IC50 = 180 μM, in vitro) that prolongs bleeding time significantly in a rodent model of thromboembolism. Additionally at a minimal effective dose of 24 mg/kg, aspalatone generates antioxidant and neuroprotective effects against kainic acid-induced epilepsy in rat hippocampus.
T67870 DKI5

(E)-N'-benzylidenehydrazinecarbothiohydrazide

Lipoxygenase Metabolism
DKI5 ((E)-N'-benzylidenehydrazinecarbothiohydrazide) 是一种 LOX-1 抑制剂,IC50 值为 22.5 μM。DKI5 可能具有抗炎和抗氧化活性,在体外生物测定中显示出抗脂质过氧化活性。
T83048 Anti-inflammatory agent 64

ROS Kinase Tyrosine Kinase/Adaptors
Anti-inflammatory agent 64(compound 4b)能抑制IL-6和TNF-α的分泌,具备抗氧化及抗炎活性,无论在体内外均有效,能显著减轻足跖水肿。
T79538 PDE4-IN-13

Others Others
PDE4-IN-13 is a phosphodiesterase 4 inhibitor with an IC50 value of 1.56 μM, exhibiting anti-inflammatory and antioxidative properties. It is utilized in the study of chronic obstructive pulmonary disease (COPD).

化合物

cyclo(L-Pro-L-Tyr)
Cat.No: TP2333
Synonym:
Target: Others
DPN
Cat.No: T7644
Synonym: Diarylpropionitrile,2,3-双(4-羟苯基)丙腈
Target: Apoptosis, Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
Dihydrolipoic acid
Cat.No: T21233
Synonym: Reduced thioctic acid,Reduced lipoic acid,DHLA,USAF XR-12,6,8-Dihydrothioctic acid,二氢硫辛酸
Target: Antioxidant
Prifelone
Cat.No: T25985
Synonym: R-830,R830,S-16820,S 16820,R 830
Target: Others
GLP-1(28-36)amide acetate
Cat.No: T37890L
Synonym: GLP-1(28-36)amide acetate(1225021-13-5 Free base)
Target: Antioxidant, Glucagon Receptor
LDL-IN-3
Cat.No: T10063
Synonym:
Target: Antioxidant
Todralazine hydrochloride
Cat.No: T17111
Synonym: Ecarazine hydrochloride,盐酸托屈嗪
Target: Adrenergic Receptor
Se-DMC
Cat.No: T39527
Synonym:
Target: Antioxidant
N-Arachidonylglycine
Cat.No: T23040
Synonym: NA-Gly,N-Arachidonyl Glycine
Target: Antioxidant
Succinobucol
Cat.No: T4287
Synonym: Probucol monosuccinate,AGI-1067
Target: Antioxidant, Reactive Oxygen Species
Polaprezinc
Cat.No: T4510
Synonym: Zinc L-carnosine,聚普瑞锌,L-肌肽锌
Target: Others
Nrf2 activator-3
Cat.No: T78650
Synonym:
Target: Antioxidant, Nrf2
(R)-3-hydroxy Myristic Acid
Cat.No: T38041
Synonym:
Target: Antioxidant, Serine Protease, Antifungal
Geranylacetone(Z/E)
Cat.No: T8368
Synonym: 6,10-二甲基-5,9-十一双烯-2-酮,Dihydropseudoionone
Target: Others
Quercetin pentaacetate
Cat.No: T38343
Synonym: Pentaacetylquercetin
Target: RSV
AFMK
Cat.No: T41345
Synonym: Formyl-N-acetyl-5-methoxykynurenamine,Acetyl-N-formyl-5-methoxykynurenamine
Target: Apoptosis, Free radical scavengers, Antioxidant, Endogenous Metabolite
Riparin III
Cat.No: T26091
Synonym: Riparin
Target: Antioxidant, Calcium Channel
beta-Glucogallin
Cat.No: T126022
Synonym: 1-O-Galloyl-β-D-glucose,β-Glucogallin
Target: Reductase
Obestatin (rat) acetate
Cat.No: TP2279L
Synonym:
Target: GHSR
TNF/IFNγ-IN-1
Cat.No: T83628
Synonym:
Target: Antioxidant, TNF, COX
Elsibucol
Cat.No: T31615
Synonym: AGI-1096,UNII-O7T92N1Y8T,AGI 1096
Target: Antioxidant
NSC 409012
Cat.No: T4184
Synonym: 5-(4-iodobenzylidene)rhodanine,5-(4-碘苯亚甲基)罗丹宁
Target: Others
Homocarnosine acetate
Cat.No: T32098L
Synonym:
Target: GABA Receptor, Endogenous Metabolite
Isourolithin A
Cat.No: T125575
Synonym:
Target: Others
D609
Cat.No: T15044
Synonym:
Target: Apoptosis, Antioxidant
EDTA copper(II) disodium salt
Cat.No: T65167
Synonym:
Target: Antibiotic
Debrisoquin hydriodide
Cat.No: T50003
Synonym: 1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide
Target: Others
NSC 6038
Cat.No: T4632
Synonym: 4-chloro-N,N-dipropylbenzamide,4-Chloro-N,N-di-n-propylbenzaMide,4-氯-N,N-二-N-丙基苯甲酰胺
Target: Others
Arbidol
Cat.No: T7911
Synonym: Umifenovir
Target: Antiviral, SARS-CoV
FPTQ
Cat.No: T5509
Synonym:
Target: GluR
Xanthine dehydrogenase Inhibitor 1
Cat.No: T50071
Synonym:
Target: Others
1-pentyl-1H-indole-3-carboxylic acid
Cat.No: T50069
Synonym:
Target: Others
Ladostigil
Cat.No: T32535
Synonym: TV-3326,Ladostigil,TV 3326,TV3326,Ladostigil free base
Target: Antioxidant, MAO, AChE
MnTBAP chloride
Cat.No: T38164
Synonym: Mn(III)TBAP
Target: Others
5-Hydroxy-1-methylhydantoin
Cat.No: T28222
Synonym: HD-003,HD003,5-羟基-1-甲基咪唑啉-2,4-二酮,NZ419,NZ-419,HD 003,NZ 419
Target: Bradykinin Receptor
DMU-212
Cat.No: T36674
Synonym:
Target: Apoptosis, ERK
LY 221068
Cat.No: T27901
Synonym: LY221068,LY-221068
Target: Others
Linearol
Cat.No: T25735
Synonym:
Target: Others
Antioxidant agent-11
Cat.No: T83030
Synonym:
Target: Others
KHG26693
Cat.No: T24261
Synonym: KHG-26693,KHG 26693
Target: Others
Camobucol
Cat.No: T14861
Synonym: AGIX 4207
Target: Others
LY 269415
Cat.No: T27908
Synonym: LY269415,LY-269415
Target: Others
Todralazine
Cat.No: T17112
Synonym: Ecarazine
Target: Others
AL-8417
Cat.No: T23697
Synonym: J1.090.276B,AL8417,(2R)-AL-5898
Target: Others
Chitoheptaose heptahydrochloride
Cat.No: T37252
Synonym:
Target: Others
Mito-apocynin (C11)
Cat.No: T13773
Synonym:
Target: Others
Aspalatone
Cat.No: T36178
Synonym:
Target: Others
DKI5
Cat.No: T67870
Synonym: (E)-N'-benzylidenehydrazinecarbothiohydrazide
Target: Lipoxygenase
Anti-inflammatory agent 64
Cat.No: T83048
Synonym:
Target: ROS Kinase
PDE4-IN-13
Cat.No: T79538
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5660 Menthone

IL Receptor; TNF; NF-κB; Parasite Apoptosis; Immunology/Inflammation; Microbiology/Virology; NF-κB
Menthone 是一种从植物和薄荷油中提取的单萜,是精油的主要挥发性成分,具有抗炎和抗氧化特性。
T5712 zerumbone

花薑酮,球姜酮

Antioxidant; HSV Microbiology/Virology; oxidation-reduction
Zerumbone 是从Zingiber zerumbetSmith 的根茎中分离的一种单环倍半萜烯,可有效抑制Epstein-Barr 病毒的激活,IC50为 0.14 mM,具有抗癌、抗炎、抗氧化和抗增殖的作用。
TN1990 Norathyriol

芒果苷元

Akt; DNA/RNA Synthesis; AMPK; PPAR Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Norathyriol 是来自芒果的芒果苷代谢物,具有抗氧化、抗癌、抗菌和抗炎活性。它以非竞争性方式抑制 α-葡萄糖苷酶,IC50为 3.12 μM。它还抑制PPARα、PPARβ和PPARγ,IC50分别为 92.8、102.4 和 153.5 µM。
TN1686 Ginsenoside Rg4

人参皂苷 RG4

Antibacterial Microbiology/Virology
Ginsenoside Rg4 是分离自Panax ginsengC. A. Meyer 叶子中的一种人参三醇型人参皂苷。人参三醇型人参皂苷具有多种生物活性,包括防腐,抗糖尿病,伤口愈合,免疫刺激和抗氧化活性等。
T4518 Licochalcone D

ERK; NF-κB MAPK; NF-κB
Licochalcone D 是一种 NF-κB p65的有效抑制剂,是一种存在于 Glycyrrhiza inflate 中的黄酮类化合物,具有抗氧化、抗炎、抗癌等作用。
T9135 Epirosmanol

Others Others
Epirosmanol 是含有内酯部分的二萜类化合物。 Epirosmanol 是一种极弱碱性(基本中性)的化合物(基于其 pKa)。
T5814 Aurantiamide

TMC-58B,橙黄胡椒酰胺

p38 MAPK; NF-κB MAPK; NF-κB
Aurantiamide 是马齿苋的活性成分,具有多种生物活性(如抗氧化、抗血小板、抗炎、抗肿瘤活性等),具有口服活性。
T6917 Oleuropein

洋橄榄苦甙,橄榄苦苷

Apoptosis; Aromatase; ROS; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。
TN5634 Aureusidin

Auresudidin,金鱼草素,Auresidin

Antioxidant; Reactive Oxygen Species; Lipoxygenase Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。
T6S1572 Sauchinone

ERK; p38 MAPK; NF-κB MAPK; NF-κB
Sauchinone 是一种从Saururus chinensis 中获得的非对映异构的木脂素。它通过抑制I-κBα磷酸化和p65核易位来抑制 LPS 诱导的 iNOS,TNF-α 和 COX-2 表达。它具有抗炎和抗氧化活性。
T11685 Isolongifolene

异长叶烯,(-)-Isolongifolene

Apoptosis; Others Apoptosis; Others
Isolongifolene ((-)-Isolongifolene) 是一种从调料九里香中分离的三环倍半萜烯,具有抗氧化,抗炎,抗癌和神经保护的特性。它通过调节 PI3K/AKT/GSK-3β 信号通路来减轻鱼藤酮诱导的氧化应激,线粒体功能障碍和细胞凋亡。
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
T2899 Liquiritin

Liquiritigenin-4'-O-glucoside,Liquiritoside,甘草苷

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Liquiritin (Liquiritigenin-4'-O-glucoside) 是一种从甘草中分离出的类黄酮,是一种竞争性的 AKR1C1 抑制剂,对 AKR1C1,AKR1C2 和 AKR1C3 的 IC50分别为 0.62 μM,0.61 μM 和 3.72 μM,在体内有效抑制 AKR1C1 介导的孕酮代谢。它是一种抗氧化剂,具有神经保护、抗癌、抗炎的活性。
T3921 Punicalagin

安石榴甙,安石榴苷

SARS-CoV; HBV Microbiology/Virology
Punicalagin 是一种在石榴中发现的主要鞣花单宁,是可逆且非竞争性的 3CLpro 抑制剂。Punicalagin 具有抗氧化、抗炎和抗肿瘤活性。
T6569 Mimosine

Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine

Others Others
Mimosine (Leucenol) 是一种酪氨酸类似物,具有抗癌和抗炎等活性。它可通过其强大的铁结合活性作为抗氧化剂,是一种 Fe(III) 螯合剂。它作用于人类白血病细胞,通过金属离子螯合、线粒体激活和诱导活性氧产生来诱导细胞凋亡。
T6S1653 Albiflorin

Alibiflorin,芍药内酯苷

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分,是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。
T8733 Antrodin A

(2-氯苯基)二苯基甲醇,camphorataanhydride A

Others Others
Antrodin A (camphorataanhydride A) 是固体发酵樟脑菌菌丝体的一种主要活性成分。它能够增强肝脏的抗炎及抗氧化能力,维持肠道菌群的稳定,避免酒精对肝脏的损伤。
T2957 Arctigenin

牛蒡苷元,牛蒡子苷元,(-)-Arctigenin

Apoptosis; MMP; Influenza Virus; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。
TN1237 3-O-Methylgallic acid

3,4-Dihydroxy-5-methoxybenzoic acid,3-O-甲基没食子酸

Apoptosis; NF-κB; OCT; DNA/RNA Synthesis; STAT Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; JAK/STAT signaling; Membrane transporter/Ion channel; NF-κB; Stem Cells
3-O-Methylgallic acid (3,4-Dihydroxy-5-methoxybenzoic acid) 是一种花青素代谢产物,具有强大的抗氧化能力。它还诱导细胞凋亡并具有抗癌作用,可抑制 Caco-2 细胞增殖,IC50值为 24.1 μM。
T3416 Aucubin

Aucuboside,桃叶珊瑚苷,Rhinanthin

IL Receptor; NF-κB; Antibacterial Immunology/Inflammation; Microbiology/Virology; NF-κB
Aucubin (Rhinanthin) 是一种可从许多传统的草药中提取的环烯醚萜苷,有许多生物学活性。
T8516 Levomenol

没药醇,(-)-α-BISABOLOL,(-)-α-红没药醇

Others Others
Levomenol ((-)-α-BISABOLOL) 是一种单环倍半萜醇,具有有神经保护、抗氧化、抗炎和抗凋亡的作用。它可减轻三叉神经性疼痛啮齿动物模型的伤害性行为和中枢敏感性。它通过减少小鼠永久性局灶性脑缺血诱导的促炎标志物,防止神经元损伤和记忆缺陷。
T2950 Schisandrin

Wuweizi alcohol-A,Wuweizichun-A,Schizandrol-A,Schizandrol,五味子醇甲

Autophagy Autophagy
Schisandrin (Wuweizi alcohol-A) 是一种从五味子中分离出来的联苯环辛烯类木脂素,可逆转大鼠的记忆障碍,具有保肝、抗氧化、抗哮喘、抗癌和抗炎作用。
T0795 Rutin

Quercetin 3-O-rutinoside,芦丁,Rutoside

Beta Amyloid; Prostaglandin Receptor; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rutin (Quercetin 3-O-rutinoside) 属于黄酮类天然产物,具有血脑屏障渗透性。Rutin 具有广泛的生物活性,包括抗氧化、抗炎、抗肿瘤、降血糖、神经保护、抗菌、抗衰老等等。
T3363 Jervine

蒜黎芦碱,Iervin,11-Ketocyclopamine,Jerwiny

Hedgehog/Smoothened; Smo GPCR/G Protein; Stem Cells
Jervine (Jerwiny) 是一种有效的刺猬 (Hh) 抑制剂(IC50:500-700 nM)。它是一种天然致畸性甾体生物碱,来自于 Veratrumalbum 的根茎,具有抗炎和抗氧化作用。
T5S1923 Schisandrin C

五味子丙素,Schizandrin-C,Wuweizisu-C

Apoptosis; Others; Virus Protease Apoptosis; Microbiology/Virology; Others
Schisandrin C (Wuweizisu-C) 是从五味子中分离得到的一种植物化学木脂素。它具有抗癌、抗炎和抗氧化等多种生物活性,可研究癌症、阿尔茨海默病、肝病。
T0492 Dimethyl fumarate

富马酸二甲酯,DMF

Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂,可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物,可作抗炎和免疫调节剂,可研究多发性硬化症。
T26288 Clovamide

trans-Clovamide,N-trans-Caffeoy-L-dopa

Apoptosis; Influenza Virus; ROS; Antibacterial Apoptosis; Immunology/Inflammation; Microbiology/Virology
Clovamide (trans-Clovamide) 是一种天然存在的咖啡酰结合物,具有抗菌、抗炎、抗氧化和神经保护作用。它是一种极好的活性氧和氧自由基清除剂。
T5728 OsMundacetone

4-(3,4-Dihydroxyphenyl)-3-buten-2-one

Apoptosis; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB
OsMundacetone (4-(3,4-Dihydroxyphenyl)-3-buten-2-one) 是从白桦茸中分离出的一种天然产物,具有抗凋亡作用。它具有DPPH 清除活性,保护神经细胞免受氧化应激,可研究神经退行性疾病。
TN4893 Rapanone

拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌

Apoptosis; Phospholipase; Antibacterial; Parasite Apoptosis; Metabolism; Microbiology/Virology
Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) 是一种具有广泛生物活性的天然苯醌,如抗肿瘤、抗氧化、抗炎、抗菌和抗寄生虫活性。它还是选择性人滑膜 PLA2抑制剂,IC50值为 2.6 μM。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
T22417 Rutin hydrate

芦丁,Rutoside,Sophorin,Quercetin-3-O-rutinoside

Beta Amyloid; Others; Autophagy Autophagy; Neuroscience; Others
Rutin hydrate (Sophorin) 是一种广泛存在于多种植物中的黄酮类天然产物,具有降糖、抗炎、抗氧化、神经保护、肾脏保护、肝脏保护和降低 Aβ 低聚物活性等多种生物活性。它能穿过血脑屏障,通过抑制细胞凋亡、线粒体功能紊乱和氧化应激抑制万古霉素诱导的肾小管细胞凋亡。
TN1238 3,4-O-Isopropylidene-shikimic acid

3,4-O-异亚丙基莽草酸,3,4-O-Isopropylidene shikimic acid

NOS; NO Synthase Immunology/Inflammation
3,4-O-Isopropylidene-shikimic acid (3,4-O-Isopropylidene shikimic acid) 是一种从Hypericum wightianum 中提取得到的天然产物。它具有抗炎症和抗氧化作用。
T2S1158 4,5-Dicaffeoylquinic acid

3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C

Others; HBV; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。
TN1353 N-Benzyllinoleamide

(9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺

Others Others
N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) 是一种分离自 Lepidium meyeniiWalp,能够抗运动性疲劳的药物。
T4S1659 Xanthotoxol

8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene

Reactive Oxygen Species; 5-HT Receptor; Endogenous Metabolite GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Xanthotoxol (Psoralen) 是一种具有生物活性的线性呋喃香豆素,具有很强的抗炎、抗氧化、5-HT 拮抗和神经保护作用等药理活性。
T6S1917 Schisandrol B

Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B

P450; Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Schisandrol B (Besigomsin) 是华中五味子的主要活性成分,具有保肝、抗炎、抗糖尿病和抗氧化的作用。它抑制活性氧的产生,也抑制 P-糖蛋白和CYP3A 的活性。
TN6732 Oenothein B

Apoptosis; HCV Protease; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Proteases/Proteasome
Oenothein B 是一种聚(ADP-核糖)糖水解酶的特异性抑制剂。 Oenothein B 具有抗氧化、抗炎、抗真菌、抗 HCV 和抗肿瘤特性。
T5145 Oxytocin acetate

Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。
T6S1101 Astragalin

Kaempferol 3-D-glucoside,Kaempferol 3-O-glucoside,kaempferol-3-glucoside,3-Glucosylkaempferol,Astragaline,紫云英苷,Kaempferol 3-β-D-glucopyranoside

Apoptosis; NF-κB Apoptosis; NF-κB
Astragalin (Kaempferol 3-O-glucoside) 是一种具有生物活性的天然黄酮类化合物。 它具有多种药理特性,包括抗氧化、抗炎、抗癌、神经保护和心脏保护特性。
T2S2104 Sinigrin hydrate

黑芥子苷,Sinigrin monohydrate,芥子甙单水合物,Allylglucosinolate monohydrate

Antibacterial Microbiology/Virology
Sinigrin hydrate (Allylglucosinolate monohydrate) 是一种天然脂肪族芥子油苷,存在于十字花科植物中。它具有消炎、抗癌、抗真菌、抗菌、抗氧化作用。
T3376 Cynaroside

朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside

Others; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。
TQ0188 Miquelianin

槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide

stilbene oxidase; Endogenous Metabolite Metabolism
Miquelianin (Quercetin 3-glucuronide) 是槲皮素的代谢产物,属于类黄酮化合物。
TN2233 Spathulenol

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Spathulenol 是一种来自 Aristolochia yunnanensis 的天然成分,具有抗炎、抗氧化、抗增殖、抗溃疡和抗分枝杆菌活性。 Spathulenol 在 DPPH 系统中显示出显著的抗氧化活性,IC50 为 85.60 μg/mL。
TN1599 Eburicoic acid

Eburicoicacid,MFCD00238594,ZINC4655149,齿孔菌酸

Antioxidant; TNF; NOS; NO Synthase; CCR; Immunology/Inflammation related Apoptosis; Immunology/Inflammation; Microbiology/Virology; oxidation-reduction
Eburicoic acid (ZINC4655149) 具有抗炎和抗氧化活性,从而保护肝脏免受 CCl4 引起的肝损伤,可用于抗肝癌研究。
TN1438 beta-Amyrin acetate

beta-香树脂醇乙酸酯

Antioxidant; HMG-CoA Reductase; Epoxide Hydrolase; Antifungal Metabolism; Microbiology/Virology; oxidation-reduction
beta-Amyrin acetate 抑制 HMG-CoA 还原酶 (HMGCR) 和 sEH 活性,IC50 为 3.4 μM。 beta-Amyrin acetate 具有抗炎、抗真菌、抗氧化和抗高血脂活性。
T2837 Chrysin

5, 7-Dihydroxyflavone,NSC 407436,白杨素,5,7-Dihydroxyflavone

Estrogen Receptor/ERR; Antioxidant Endocrinology/Hormones; oxidation-reduction
Chrysin (5,7-Dihydroxyflavone) 是一种雌激素阻断剂。
T5098 Isochlorogenic acid A

3,5-CQA,异绿原酸 A,3,5-Dicaffeoylquinic acid,金银花

Reactive Oxygen Species; HBV; Endogenous Metabolite Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Isochlorogenic acid A (3,5-Dicaffeoylquinic acid) 是一种天然酚酸,具有抗氧化和抗炎活性。
TN1432 Bacopasaponin C

(-)-假马齿苋皂苷 C,假马齿苋皂苷C

Anti-infection; GABA Receptor; NMDAR Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷,具有抗肿瘤和抗利什曼原虫作用。
T2912 Ergosterol

麦角固醇,Provitamin D,Ergosterin,Provitamin D2

Others; Antioxidant; Endogenous Metabolite Metabolism; Others; oxidation-reduction
Ergosterol 是真菌中的主要固醇类,具有抗炎,抗氧化和抗增殖的作用。
T1368 Methyl 3,4-dihydroxybenzoate

3,4-Dihydroxybenzoic acid methyl ester,Methyl protocatechuate,原儿茶酸甲酯,3,4-二羟基苯甲酸甲酯,Protocatechuic acid methyl ester

Apoptosis; Antioxidant; Nrf2 Apoptosis; Immunology/Inflammation; oxidation-reduction
Methyl 3,4-dihydroxybenzoate (Protocatechuic acid methyl ester) 是绿茶中发现的主要代谢产物,是一种多酚,有抗氧化和抗炎作用。
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天然产物

Menthone
Cat.No: T5660
Synonym:
Target: IL Receptor, TNF, NF-κB, Parasite
zerumbone
Cat.No: T5712
Synonym: 花薑酮,球姜酮
Target: Antioxidant, HSV
Norathyriol
Cat.No: TN1990
Synonym: 芒果苷元
Target: Akt, DNA/RNA Synthesis, AMPK, PPAR
Ginsenoside Rg4
Cat.No: TN1686
Synonym: 人参皂苷 RG4
Target: Antibacterial
Licochalcone D
Cat.No: T4518
Synonym:
Target: ERK, NF-κB
Epirosmanol
Cat.No: T9135
Synonym:
Target: Others
Aurantiamide
Cat.No: T5814
Synonym: TMC-58B,橙黄胡椒酰胺
Target: p38 MAPK, NF-κB
Oleuropein
Cat.No: T6917
Synonym: 洋橄榄苦甙,橄榄苦苷
Target: Apoptosis, Aromatase, ROS, PPAR
Aureusidin
Cat.No: TN5634
Synonym: Auresudidin,金鱼草素,Auresidin
Target: Antioxidant, Reactive Oxygen Species, Lipoxygenase
Sauchinone
Cat.No: T6S1572
Synonym:
Target: ERK, p38 MAPK, NF-κB
Isolongifolene
Cat.No: T11685
Synonym: 异长叶烯,(-)-Isolongifolene
Target: Apoptosis, Others
3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
Liquiritin
Cat.No: T2899
Synonym: Liquiritigenin-4'-O-glucoside,Liquiritoside,甘草苷
Target: Reactive Oxygen Species
Punicalagin
Cat.No: T3921
Synonym: 安石榴甙,安石榴苷
Target: SARS-CoV, HBV
Mimosine
Cat.No: T6569
Synonym: Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine
Target: Others
Albiflorin
Cat.No: T6S1653
Synonym: Alibiflorin,芍药内酯苷
Target: Reactive Oxygen Species
Antrodin A
Cat.No: T8733
Synonym: (2-氯苯基)二苯基甲醇,camphorataanhydride A
Target: Others
Arctigenin
Cat.No: T2957
Synonym: 牛蒡苷元,牛蒡子苷元,(-)-Arctigenin
Target: Apoptosis, MMP, Influenza Virus, Autophagy
3-O-Methylgallic acid
Cat.No: TN1237
Synonym: 3,4-Dihydroxy-5-methoxybenzoic acid,3-O-甲基没食子酸
Target: Apoptosis, NF-κB, OCT, DNA/RNA Synthesis, STAT
Aucubin
Cat.No: T3416
Synonym: Aucuboside,桃叶珊瑚苷,Rhinanthin
Target: IL Receptor, NF-κB, Antibacterial
Levomenol
Cat.No: T8516
Synonym: 没药醇,(-)-α-BISABOLOL,(-)-α-红没药醇
Target: Others
Schisandrin
Cat.No: T2950
Synonym: Wuweizi alcohol-A,Wuweizichun-A,Schizandrol-A,Schizandrol,五味子醇甲
Target: Autophagy
Rutin
Cat.No: T0795
Synonym: Quercetin 3-O-rutinoside,芦丁,Rutoside
Target: Beta Amyloid, Prostaglandin Receptor, Autophagy
Jervine
Cat.No: T3363
Synonym: 蒜黎芦碱,Iervin,11-Ketocyclopamine,Jerwiny
Target: Hedgehog/Smoothened, Smo
Schisandrin C
Cat.No: T5S1923
Synonym: 五味子丙素,Schizandrin-C,Wuweizisu-C
Target: Apoptosis, Others, Virus Protease
Dimethyl fumarate
Cat.No: T0492
Synonym: 富马酸二甲酯,DMF
Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy
Clovamide
Cat.No: T26288
Synonym: trans-Clovamide,N-trans-Caffeoy-L-dopa
Target: Apoptosis, Influenza Virus, ROS, Antibacterial
OsMundacetone
Cat.No: T5728
Synonym: 4-(3,4-Dihydroxyphenyl)-3-buten-2-one
Target: Apoptosis, Reactive Oxygen Species
Rapanone
Cat.No: TN4893
Synonym: 拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌
Target: Apoptosis, Phospholipase, Antibacterial, Parasite
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
Rutin hydrate
Cat.No: T22417
Synonym: 芦丁,Rutoside,Sophorin,Quercetin-3-O-rutinoside
Target: Beta Amyloid, Others, Autophagy
3,4-O-Isopropylidene-shikimic acid
Cat.No: TN1238
Synonym: 3,4-O-异亚丙基莽草酸,3,4-O-Isopropylidene shikimic acid
Target: NOS, NO Synthase
4,5-Dicaffeoylquinic acid
Cat.No: T2S1158
Synonym: 3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C
Target: Others, HBV, Endogenous Metabolite
N-Benzyllinoleamide
Cat.No: TN1353
Synonym: (9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺
Target: Others
Xanthotoxol
Cat.No: T4S1659
Synonym: 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene
Target: Reactive Oxygen Species, 5-HT Receptor, Endogenous Metabolite
Schisandrol B
Cat.No: T6S1917
Synonym: Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B
Target: P450, Reactive Oxygen Species, Autophagy
Oenothein B
Cat.No: TN6732
Synonym:
Target: Apoptosis, HCV Protease, Antibacterial, Antifungal
Oxytocin acetate
Cat.No: T5145
Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素
Target: Oxytocin Receptor
Astragalin
Cat.No: T6S1101
Synonym: Kaempferol 3-D-glucoside,Kaempferol 3-O-glucoside,kaempferol-3-glucoside,3-Glucosylkaempferol,Astragaline,紫云英苷,Kaempferol 3-β-D-glucopyranoside
Target: Apoptosis, NF-κB
Sinigrin hydrate
Cat.No: T2S2104
Synonym: 黑芥子苷,Sinigrin monohydrate,芥子甙单水合物,Allylglucosinolate monohydrate
Target: Antibacterial
Cynaroside
Cat.No: T3376
Synonym: 朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside
Target: Others, Influenza Virus, DNA/RNA Synthesis
Miquelianin
Cat.No: TQ0188
Synonym: 槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide
Target: stilbene oxidase, Endogenous Metabolite
Spathulenol
Cat.No: TN2233
Synonym:
Target: Antioxidant, Antifungal
Eburicoic acid
Cat.No: TN1599
Synonym: Eburicoicacid,MFCD00238594,ZINC4655149,齿孔菌酸
Target: Antioxidant, TNF, NOS, NO Synthase, CCR, Immunology/Inflammation related
beta-Amyrin acetate
Cat.No: TN1438
Synonym: beta-香树脂醇乙酸酯
Target: Antioxidant, HMG-CoA Reductase, Epoxide Hydrolase, Antifungal
Chrysin
Cat.No: T2837
Synonym: 5, 7-Dihydroxyflavone,NSC 407436,白杨素,5,7-Dihydroxyflavone
Target: Estrogen Receptor/ERR, Antioxidant
Isochlorogenic acid A
Cat.No: T5098
Synonym: 3,5-CQA,异绿原酸 A,3,5-Dicaffeoylquinic acid,金银花
Target: Reactive Oxygen Species, HBV, Endogenous Metabolite
Bacopasaponin C
Cat.No: TN1432
Synonym: (-)-假马齿苋皂苷 C,假马齿苋皂苷C
Target: Anti-infection, GABA Receptor, NMDAR
Ergosterol
Cat.No: T2912
Synonym: 麦角固醇,Provitamin D,Ergosterin,Provitamin D2
Target: Others, Antioxidant, Endogenous Metabolite
Methyl 3,4-dihydroxybenzoate
Cat.No: T1368
Synonym: 3,4-Dihydroxybenzoic acid methyl ester,Methyl protocatechuate,原儿茶酸甲酯,3,4-二羟基苯甲酸甲酯,Protocatechuic acid methyl ester
Target: Apoptosis, Antioxidant, Nrf2
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Cat. No. Product Name Species Expression System
TMPY-02084 Thioredoxin 2/TRX2 Protein, Human, Recombinant (His)

MT-TRX,RP5-1119A7. 13-005,TRX2,MTRX,thioredoxin 2

Human E. coli
Thioredoxin-2, also known as TXN2, MTRX and TRX2, is a member of the thioredoxin family. Tryparedoxins (TXN) are thioredoxin-related proteins which, as trypanothione:peroxiredoxin oxidoreductases, constitute the trypanothione-dependent antioxidant defense and may also serve as substrates for ribonucleotide reductase in trypanosomatids. Thioredoxin-2 / TXN2 contains one thioredoxin domain. It is widely expressed in adult (at protein level) and fetal tissues. Human Thioredoxin-2 / TXN2 is a small ...
TMPY-04122 ATOX1 Protein, Human, Recombinant (His)

HAH1,ATX1,antioxidant 1 copper chaperone

Human E. coli
ATOX1 is a cytoplasmic copper chaperone that interacts with the copper-binding domain of the membrane copper transporters ATP7A and ATP7B. ATOX1 has also been suggested to have a potential anti-oxidant activity. As the trace element copper is essential, but extremely toxic in high concentrations, intracellular copper concentrations are tightly controlled. Once in the cell, copper is distributed by metallochaperones, including the small cytoplasmic protein ATOX1. ATOX1 plays an important role in ...
TMPJ-01106 NAD(P) transhydrogenase/NNT Protein, Human, Recombinant (His)

NAD(P) transhydrogenase,NNT

Human E. coli
NAD(P)+transhydrogenase (NNT) is located in the inner mitochondrial membrane and catalyzes a reversible hydride transfer between NAD(H) and NADP(H) that is coupled to proton translocation between the intermembrane space and mitochondrial matrix. NNT activity has an essential role in maintaining the NADPH supply for antioxidant defense and biosynthetic pathways. Structurally, NNT is composed of three domains; domains I and III are hydrophilic and have binding sites for NAD and NADP, respectively,...
TMPY-00186 GHRH Protein, Human, Recombinant (hFc)

GRF,INN,growth hormone releasing hormone,GHRF

Human HEK293 Cells
The role of hypothalamic growth hormone-releasing hormone (GHRH) in the release of growth hormone (GH) from the pituitary is well established. Extra-hypothalamic growth hormone-releasing hormone (GHRH) plays an important role in infertility. Growth hormone releasing hormone (GHRH) has recently been shown to increase the level of gamma-aminobutyric acid (GABA) and activate GABA receptors (GABARs) in the cerebral cortex. GABA is an inhibitory neurotransmitter that can inhibit seizures. GHRH may pl...

重组蛋白

Thioredoxin 2/TRX2 Protein, Human, Recombinant (His)
Cat.No: TMPY-02084
Species: Human
Expression System: E. coli
ATOX1 Protein, Human, Recombinant (His)
Cat.No: TMPY-04122
Species: Human
Expression System: E. coli
NAD(P) transhydrogenase/NNT Protein, Human, Recombinant (His)
Cat.No: TMPJ-01106
Species: Human
Expression System: E. coli
GHRH Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00186
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
T10901 Curcumin-d6

Turmeric yellow D6,Natural Yellow 3 D6,Curcumin D6,Diferuloylmethane D6

Others Others
Curcumin D6 (difluoroformylmethane D6) is deuterium-labeled curcumin (Turmeric yellow). Curcumin (Turmeric yellow) is a natural phenolic compound with various pharmacological effects, including anti-inflammatory, antioxidant, anti-proliferative and anti-a
TMIH-0181 Demethoxy Curcumin-d4

Demethoxy Curcumin-d4 是 Demethoxy Curcumin 的氘代化合物。Demethoxy Curcumin 的 CAS 号为 22608-11-3。Demethoxycurcumin是姜黄素的主要活性成分,有抗炎和抗癌作用。
TMIJ-0194 Tetramethylpyrazine-d12

Tetramethylpyrazine-d12 是 Tetramethylpyrazine 的氘代化合物。Tetramethylpyrazine 的 CAS 号为 1124-11-4。Tetramethylpyrazine 是从Ligusticum wallichii中提取的一种烷基吡嗪,常在薯条、面包、茶、乳制品、豆制品等食物中作为香精。它对大鼠具有潜在的抗神经和抗炎活性。
TMID-0254 Linalool-d3

Linalool-d3 是 Linalool 的氘代化合物。Linalool 的 CAS 号为 78-70-6。Linalool 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。

同位素标记化合物

Curcumin-d6
Cat.No: T10901
Synonym: Turmeric yellow D6,Natural Yellow 3 D6,Curcumin D6,Diferuloylmethane D6
Target: Others
Demethoxy Curcumin-d4
Cat.No: TMIH-0181
Synonym:
Target:
Tetramethylpyrazine-d12
Cat.No: TMIJ-0194
Synonym:
Target:
Linalool-d3
Cat.No: TMID-0254
Synonym:
Target:
TargetMol Loading
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