24
194
2
2
1
Cat. No. | Product Name | ||
---|---|---|---|
L6120 | 黄酮类天然产物库 | 514 compounds | |
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L6140 | 糖类及苷类化合物库 | 595 compounds | |
595 种糖类或苷类的化合物,可用于高通量筛选和高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0723 |
Cloperastine hydrochloride
HT-11 hydrochloride,盐酸氯哌斯丁 |
Potassium Channel; 5-HT Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Cloperastine hydrochloride (HT-11 hydrochloride) 是 hERG K+电流的抑制剂,IC50为 27 nM,具有浓度依赖性。 | |||
T84296 |
4'-Hydroxyflavone
|
||
4'-Hydroxyflavone 是一种从黄芩根部分离得到的黄酮化合物,具有抗炎活性。 | |||
T125076 |
Hispidulin 7-glucuronide
|
IL Receptor | Immunology/Inflammation |
Hispidulin 7-glucuronide是一种可从槲皮的叶中提取到的黄酮类化合物,具有潜在的抗炎活性,可抑制IL-6的释放。 | |||
T5941 |
Anthraflavic acid
2,6-二羟基蒽醌,2,6-Dihydroxyanthraquinone |
Others | Others |
Anthraflavic acid (2,6-Dihydroxyanthraquinone) 是一种特异性细胞色素 P-448抑制剂,细胞色素 P-448 是与许多化学致癌物质的激活密切相关的酶系统。它是一种类黄酮,有效的IQ 诱变性抑制剂,能够抑制微粒体和胞质激活途径。 | |||
T36488 |
LYG-202
LYG202,LYG 202 |
Apoptosis; ROS | Apoptosis; Immunology/Inflammation |
LYG-202是一种具有哌嗪替代的新型类黄酮,在体内和体外都具有抗肿瘤作用。LYG-202 诱导 MCF-7、MDA-MB-231 和 MDA-MB-435 细胞凋亡, 增加了细胞内 ROS 的产生。 | |||
T125575 |
Isourolithin A
|
Others | Others |
Isourolithin A 是一种天然存在的化合物,存在于各种植物中,包括欧芹、芹菜和洋甘菊。Isourolithin A 是类黄酮家族的一员,以其抗氧化和抗炎特性而闻名。 | |||
T32721 |
Lew 10
Lew-10,Lew10 |
Others | Others |
Lew 10 is a flavonoid and derivative of diosmin. | |||
T10496 |
Bencianol
ZY15051,苯西阿诺 |
Others | Others |
Bencianol is a semisynthetic flavonoid with anti-spasmogenic activities. | |||
T32761 |
Linariifolioside
|
Others | Others |
Linariifolioside is a flavonoid glycoside extracted from Veronica linariifolia. | |||
T84867 |
5-Demethoxynobiletin
2-(3,4-dimethoxyphenyl)-6,7,8-trimethoxychromen-4-one |
Others | Others |
5-Demethylnobiletin (2-(3,4-dimethoxyphenyl)-6,7,8-trimethoxychromen-4-one), a distinctive flavonoid present in citrus fruits, shows potential as a chemopreventive agent against human cancers. | |||
T24749 |
S 5682
Capiven,S-5682,Detralex,Arvenum 500,S5682 |
Others | Others |
S 5682 is a purified flavonoid fraction composed. S 5682 has anti-oedematous effect anti-inflammatory properties. | |||
T24177 |
Isariin C
|
Others | Others |
Isariin C is a flavonoid glucoside derived from the Epimedium plant genus. It stimulates angiogenesis and exhibits antioxidant activity. | |||
T32876 |
Loquatoside
|
Others | Others |
Loquatoside belongs to the class of organic compounds known as flavonoid-3-o-glycosides. These are phenolic compounds containing a flavonoid moiety which is O-glycosidically linked to carbohydrate moiety at the C3-position. Loquatoside exists as a solid, | |||
T11268 |
FD 12-9
Ac12Az9 |
Others | Others |
FD 12-9, Anti-glioblastoma activity. is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. | |||
T79005 |
6-Hydroxyluteolin
|
Others | Others |
6-Hydroxyluteolin (Compound 17),一种类黄酮化合物,对醛糖还原酶 (AR) 表现出抑制活性。 | |||
T1729 |
3',4',5',5,7-Pentamethoxyflavanone
|
Others | Others |
3',4',5',5,7-Pentamethoxyflavanone 是一种天然黄酮化合物,在 Neoraptua magnifica var. magnifica 中发现。 | |||
T83007 |
Antitumor agent-120
|
Others | Others |
Antitumor agent-120 (compound 1) 为一类黄酮化合物,来源于葛根提取。本化合物对LNCaP和PC3癌细胞的抑制作用不明显,表现出IC50s均大于50 μM。 | |||
T81970 |
Kuwanon T
|
Others | Others |
Kuwanon T为一种源自桑树根皮的异戊二烯黄酮类化合物,能抵御t-BHP诱导的氧化应激,其EC50值为30.32 μM。 | |||
T37809 |
Alphitonin
|
Others | Others |
Alphitonin is a flavonoid that has been found in L. leptolepis wood.1 It is also a metabolic intermediate that is formed during the catabolism of quercetin by the human gut bacteria E. ramulus.2,3 |1. Chen, K., Ohmura, W., Doi, S., et al. Termite feeding deterrent from Japanese larch wood. Bioresour. Technol. 95(2), 129-134 (2004).|2. Braune, A., Gütschow, M., Engst, W., et al. Degradation of quercetin and luteolin by Eubacterium ramulus. Appl. Environ. Microbiol. 67(12), 5558-55567 (2001).|3. J... | |||
T73228 |
Artonin E
5'-Hydroxymorusin |
Others | Others |
Artonin E (5'-Hydroxymorusin) 是一种已知的异戊二烯化类黄酮,可以诱导细胞凋亡 (apoptosis),使细胞周期停滞在S 期。Artonin E 可以通过线粒体通路失调诱导抗增殖作用,可以用于癌症研究。 | |||
T75501 |
Morin 3-O-β-D-glucopyranoside
|
Others | Others |
Morin 3-O-β-D-glucopyranoside 是一种天然类黄酮,具有抗真菌、抗癌和抗氧化活性。Morin 3-O-β-D-glucopyranoside 抑制逆转录酶、蛋白酪氨酸激酶和黄嘌呤氧化酶,还具有抗 HIV、抗动脉硬化和超氧化物清除活性。 | |||
T73885 |
Methyl gerfelin
|
Others | Others |
Methyl gerfelin通过与三种关键细胞蛋白乙二醛酶 1 (GLO1)、固醇结合蛋白 2 (SCP2) 和富含谷氨酰胺的四肽重复蛋白 A (SGTA) 结合,抑制破骨细胞的分化。研究表明,Methyl gerfelin是一种与类黄酮相关的强效GLO1抑制剂。 | |||
T36471 |
Ternatin
|
Others | Others |
Ternatin is a cyclic heptapeptide first isolated from the mushroom C. versicolor that has been shown to have cytotoxic and anti-adipogenic effects in vitro. It inhibits adipogenesis with an IC50 value of 27 nM and becomes cytotoxic to 3T3-L1 mouse adipocytes at 10-fold higher concentrations. Ternatin is reported to inhibit HCT116 cell proliferation with an IC50 value of 71 nM. Note that this metabolite should not be confused with the plant flavonoid of the same name. | |||
T78858 |
cGAS-IN-1
|
Others | Others |
cGAS-IN-1(化合物C20)是一种黄酮类化合物,作为Cyclic GMP-AMP Synthase(cGAS)的抑制剂,其IC50分别为2.28 μM(针对人类cGAS)和1.44 μM(针对小鼠cGAS)。由于cGAS异常激活与众多免疫介导的炎症性疾病相关,cGAS-IN-1显示出了其抗炎潜力。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1040 |
Skullcapflavone II
|
COX; Antibacterial; TGF-beta/Smad | Immunology/Inflammation; Microbiology/Virology; Neuroscience; Stem Cells |
Skullcapflavone II 是从黄芩中提取的黄酮,具有抗炎作用。它对 M. aurum 和 M. bovisBCG 具有较强的抗菌活性。它还调节破骨细胞的分化、存活和功能。 | |||
TN1740 |
Homoeriodictyol
高胜草酚,高圣草酚 |
5-HT Receptor; transporter; Sodium Channel; Drug Metabolite | GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Homoeriodictyol 是 Eriocitrin 的代谢物,属于黄酮类。Eriocitrin 是强效抗氧化剂。 | |||
T7994 |
3-Methoxyflavone
|
Antiviral | Immunology/Inflammation |
3-Methoxyflavone 是一种黄酮类化合物,分离自 Artemisia incanescens,具有抗病毒作用。 | |||
TN2151 |
Rhamnocitrin
|
Others | Others |
Rhamnocitrin 是一种分离自黄芪(沙源子)中的类黄酮,具有抗氧化,抗炎和抗动脉粥样硬化活性。它是 DPPH 的清除剂(IC50:28.38 mM)。 | |||
TN3209 |
3′,4′,7-Trihydroxyflavone
|
ATPase; Others; p38 MAPK; NF-κB | MAPK; Membrane transporter/Ion channel; NF-κB; Others |
3',4',7-Trihydroxyflavone 是分离自蚕豆荚的黄酮苷元化合物。 | |||
T6S0139 |
Neobavaisoflavone
|
Apoptosis; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Neobavaisoflavone 是一种从Psoralea corylifolia 的种子中分离出来的类黄酮。它具有抗炎,抗癌和抗氧化的作用。它在中至高浓度下可抑制 DNA 聚合酶,也可抑制血小板聚集。 | |||
T3882 |
4”-O-Glucosylvitexin
glucosylvitexin,牡荆素葡萄糖苷 |
Thrombopoietin Receptor | Immunology/Inflammation |
4”-O-Glucosylvitexin (glucosylvitexin) 是一种黄酮类化合物,提取自山楂叶中,具有生物活性。 | |||
TN1621 |
Eriodictyol-7-O-glucoside
|
Nrf2 | Immunology/Inflammation |
Eriodictyol-7-O-glucoside 是一种 Nrf2 激活剂,可防止顺铂诱导的毒性。 Eriodictyol-7-O-glucoside 是一种类黄酮和自由基清除剂,在开心果皮中具有抗氧化活性。 | |||
T5722 |
Nevadensin
Pedunculin,石吊兰素,5,7-二羟基-6,8,4'-三甲氧基黄酮 |
Anti-infection; Antibacterial | Microbiology/Virology |
Nevadensin 是一种重要的草本成分,可抑制雌二醇的生物活化。 它具有抗结核分枝杆菌、镇咳、抗炎、抗高血压等多种药理作用。 | |||
T5773 |
Moslosooflavone
5-羟基-7,8-二甲氧基黄酮,5-hydroxy-7,8-dimethoxyflavone |
NF-κB; Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Moslosooflavone (5-hydroxy-7,8-dimethoxyflavone) 是一种从雪莲中分离出来的类黄酮,具有抗缺氧和抗炎作用。 | |||
T0795 |
Rutin
Quercetin 3-O-rutinoside,芦丁,Rutoside |
Beta Amyloid; Prostaglandin Receptor; Autophagy | Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Rutin (Quercetin 3-O-rutinoside) 属于黄酮类天然产物,具有血脑屏障渗透性。Rutin 具有广泛的生物活性,包括抗氧化、抗炎、抗肿瘤、降血糖、神经保护、抗菌、抗衰老等等。 | |||
TN2158 |
Robinetin
3,3',4',5',7-Pentahydroxyflavone,洋槐黄素 |
Anti-infection; HIV Protease; Antibacterial | Microbiology/Virology; Proteases/Proteasome |
Robinetin (3,3',4',5',7-Pentahydroxyflavone) 是一种天然黄酮,具有显著的“两种颜色”固有荧光特性。它具有抗真菌、抗病毒、抗菌、抗突变、抗氧化和抗自由基活性,高效抑制 EYPC 膜脂质过氧化和 HbA 糖基化。 | |||
T22417 |
Rutin hydrate
芦丁,Rutoside,Sophorin,Quercetin-3-O-rutinoside |
Beta Amyloid; Others; Autophagy | Autophagy; Neuroscience; Others |
Rutin hydrate (Sophorin) 是一种广泛存在于多种植物中的黄酮类天然产物,具有降糖、抗炎、抗氧化、神经保护、肾脏保护、肝脏保护和降低 Aβ 低聚物活性等多种生物活性。它能穿过血脑屏障,通过抑制细胞凋亡、线粒体功能紊乱和氧化应激抑制万古霉素诱导的肾小管细胞凋亡。 | |||
T4S0094 |
Hydroxygenkwanin
羟基芫花素,Luteolin 7-methylether,7-O-Methylluteolin |
Antioxidant | oxidation-reduction |
Hydroxygenkwanin (Luteolin 7-methylether) 是一种丁香达芙妮的主要成分,是一种天然的类黄酮化合物。它具有抗氧化,抗神经胶质瘤能力和抗癌作用。 | |||
T1686 |
Hematoxylin
苏木精,Hydroxybrazilin,Natural Black 1,Haematoxylin |
Beta Amyloid; Others | Neuroscience; Others |
Hematoxylin (Natural Black 1) 是一种天然存在的类黄酮化合物,衍生自木柴树Haematoxylon campechianum。它是一种组织学上的核染色剂,也是一种有效的Aβ42原纤维形成的抑制剂,IC50=1.6 µM。 | |||
TN1259 |
Complanatoside B
3-O-Β-D-芹糖(1-2)-Β-D-葡萄糖-鼠李柠檬素4'-O-Β-D-葡萄糖苷,沙苑子苷B |
Others | Others |
Complanatoside B 是一种黄酮类化合物,具有抗炎作用。 | |||
T7437 |
3-(3-Hydroxyphenyl)propionic Acid
m-Hydroxyphenylpropionic acid,3-Hydroxyhydrocinnamic acid,3-(3-羟基苯基)丙酸 |
Others; Endogenous Metabolite | Metabolism; Others |
3-(3-Hydroxyphenyl)propionic Acid (m-Hydroxyphenylpropionic acid) 是一种黄酮类代谢产物,由人体微生物区系形成,具有舒张血管的特性。 | |||
TN2130 |
Manghaslin
槲皮素-3-O-芸香糖-(1→2)-O-鼠李糖苷,Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside |
AChE; Glucosidase | Metabolism; Neuroscience |
Manghaslin (Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside) 是具有抗炎活性的黄酮苷,对 AChE 具有抑制活性,IC50=94.92 µM。 | |||
TN5028 |
Sinensin
ZINC38908691 |
Others | Others |
Sinensin 是一种来自 Cudrania cochinchinensis 的草本植物中的类黄酮。 | |||
TN1808 |
Isovitexin 2''-O-arabinoside
|
Others | Others |
Isovitexin 2''-O-arabinoside 是一种在紫花苜蓿植物中发现黄酮类化合物。 | |||
TN1489 |
3'-Methoxyapiin
Graveobioside B,3'-Methoxy apiin,Chrysoeriol 7-apiosylglucoside,3'-甲氧基芹菜苷 |
Others | Others |
3'-Methoxyapiin (Graveobioside B) 是一种来自 Eminium spiculatum 植物的类黄酮。 | |||
TN7128 |
4,6,3',4'-Tetrahydroxyaurone
aureusidin |
Others | Others |
4,6,3',4'-Tetrahydroxyaurone 是一种来自 Heleocharis dulcis 草本的类黄酮。 | |||
TN2883 |
3',4'-Dimethoxyflavone
|
Others; PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair; Others |
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。 | |||
T2O2770 |
Agarotetrol
|
Others | Others |
Agarotetrol 是一种色酮衍生物,从沉香中分离得到。 | |||
T3242 |
Breviscapin
Scutellarin,红盏花素,Scutellarin B |
Others | Others |
Breviscapin (Scutellarin) 是从Erigeron breviscapus 全草中提取的总黄酮成分(含量≥85%)。 | |||
T13761 |
Luteolin 7-diglucuronide
|
Others | Others |
Luteolin 7-diglucuronide 是一种从马鞭草 Verbena officinalis 和三叶草 Aloysia triphylla 中提取的类黄酮。 | |||
TN3689 |
Comanthoside A
Comanthosid A |
Others | Others |
Comanthoside A (Comanthosid A) 是一种可从 Comanthosphace japonica 中分离的天然黄酮苷。Comanthoside A 也 是合成 Linaroside和 Comanthoside B 的关键中间体。 | |||
TN3120 |
5-Hydroxy-7-acetoxy-8-methoxyflavone
|
Histone Demethylase; Antiviral | Chromatin/Epigenetic; Immunology/Inflammation |
5-Hydroxy-7-acetoxy-8-methoxyflavone 是一种类黄酮化合物,可以抑制脂质过氧化,可能具有抗流感病毒活性。 | |||
T8263 |
3,4'-Dihydroxyflavone
|
Influenza Virus | Microbiology/Virology |
3,4'-Dihydroxyflavone 是一种口服活性黄酮类化合物,具有抗甲型流感病毒的抗病毒活性。 | |||
T13514 |
5-MethoxyPinocembroside
|
Others | Others |
5-MethoxyPinocembroside 是一种黄酮类天然产物,存在于辣木 Moringa oleifera 的叶子中。 | |||
T0228 |
Methyl-Hesperidin
甲基橙皮甙 |
Akt; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Methyl hesperidin 是一种血管扩张剂。 | |||
T5S1526 |
Apigenin-7-O-(2G-rhamnosyl)gentiobioside
Apigenin 7-O-(2G-rhamnosyl)gentiobioside,芹菜素-7-0-(2G-鼠李糖)龙胆糖苷,Apigenin 7-(2-Rhamnosylgentiobioside),金银花 |
Others | Others |
Apigenin-7-O-(2G-rhamnosyl)gentiobioside 是一种黄酮类苷化合物,从Lonicera gracilipes var. glandulosa 中提取得到。 | |||
TN1039 |
Tamarixetin
柽柳黄素,4'-O-Methyl Quercetin |
Endogenous Metabolite; Immunology/Inflammation related | Immunology/Inflammation; Metabolism |
Tamarixetin (4'-O-Methyl Quercetin) 是一种槲皮素的天然类黄酮衍生物,具有抗氧化、抗炎作用,能够防止心肌肥厚。 | |||
T2987 |
(-)-Epigallocatechin
表没食子儿茶素,(-)-表没食子儿茶素,l-Epigallocatechin,Epigallocatechin,EGC |
MMP; Autophagy | Autophagy; Proteases/Proteasome |
(-)-Epigallocatechin (Epigallocatechin) 是绿茶中含量最丰富的黄酮类天然产物,可与未折叠的天然多肽结合,阻止转化为淀粉样蛋白原纤维。 | |||
T4130 |
Complanatuside
沙苑子苷,Complanatoside |
Others | Others |
Complanatuside (Complanatoside) 是一种黄酮类化合物,存在于中药沙苑子中。 | |||
T10822 |
Cirsimarin
Cirsitakaoside |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Cirsimarin (Cirsitakaoside) 是一种从 Microtea debilis 中分离出来的黄酮类化合物。它具有很强的抗脂肪生成作用,能减少小鼠脂肪组织的沉积。Cirsimarin 对腺苷 A1 受体有拮抗作用,对磷酸二酯酶有抑制作用 | |||
T5S2139 |
Epimedin A1
朝藿定A1,Hexandraside F |
Others | Others |
Epimedin A1 (Hexandraside F) 是一种黄酮类化合物,从常用中药淫羊藿中提取得到。 | |||
T2933 |
Wogonin
Vogonin,汉黄芩素 |
Apoptosis; Wnt/beta-catenin; CDK; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells |
Wogonin (Vogonin) 是一种具有细胞渗透性的口服类黄酮,具有抗炎和抗癌特性,能够抑制 CDK8和 Wnt 的活性。 | |||
T3881 |
Vaccarin
|
Integrin; Akt; PERK; AMPK | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Vaccarin 是从王不留行中提取的一种黄酮糖苷,可显著促进伤口愈合以及伤口部位的内皮和成纤维细胞增殖。它通过激活 AMPK 信号通路改善胰岛素抵抗和脂肪变性。 | |||
T2778 |
(+)-Catechin Hydrate
一水合儿茶素,(+)-水合儿茶素 |
Antioxidant; COX | Immunology/Inflammation; Neuroscience; oxidation-reduction |
(+)-Catechin hydrate 是来自茶树的抗氧化类黄酮,可抑制环加氧酶-1,IC50为 1.4 μM。它是一种自由基清除剂,可防止多种生物系统中自由基介导的损害。 | |||
T0579 |
Myricetin
Cannabiscetin,杨梅素 |
Apoptosis; PI3K; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Metabolism; PI3K/Akt/mTOR signaling |
Myricetin (Cannabiscetin) 是一种存在于常见植物中的类黄酮,具有强抗氧化,抗糖尿病,抗癌和抗炎活性。 | |||
TN1082 |
Apigenin 7-O-malonylglucoside
Apigenin 7-O-(6''-O-malonylglucoside) |
||
Apigenin 7-O-malonylglucoside (Apigenin 7-O-(6''-O-malonylglucoside)) 存在于菊花中,是一种黄酮,也是一种糖苷。 | |||
TN1819 |
Kaempferol 3-neohesperidoside
Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷 |
GSK-3; MEK; PI3K | MAPK; PI3K/Akt/mTOR signaling; Stem Cells |
Kaempferol 3-neohesperidoside (Kaempferol 3-O-neohesperidoside) 是一种类黄酮,对大鼠比目鱼肌具有拟胰岛素作用。 | |||
T2757 |
Myricitrin
杨梅苷,Myricetrin,Myricitrine |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Myricitrin (Myricitrine) 是从杨梅根皮中分离出来的类黄酮化合物,具有镇痛作用。它是主要的抗氧化剂。 | |||
T2O2744 |
alpha-Naphthoflavone
苯并黄素;α-萘黄酮;7,8-苯并黄酮,7,8-benzoflavone,α-萘黄酮 |
Aromatase | Endocrinology/Hormones |
alpha-Naphthoflavone (7,8-benzoflavone) 是合成的黄酮类化合物,是一种竞争性芳香酶抑制剂,其IC50=0.5 μM,Ki=0.2 μM。 | |||
T2S2150 |
Noricaritin
诺里卡汀,去甲淫羊藿黄素 |
Others | Others |
Noricaritin 是一种来源于淫羊藿根的黄酮类化合物,可诱导肺组织细胞增殖,抑制人肺上皮细胞中促炎细胞因子和趋化因子的产生。 | |||
T3325 |
Liquiritigenin
4',7-Dihydroxyflavanone,甘草素 |
Estrogen Receptor/ERR; Estrogen/progestogen Receptor | Endocrinology/Hormones |
Liquiritigenin (4',7-Dihydroxyflavanone) 是一种黄烷酮,从甘草中分离得到,是高度选择性的雌激素受体β 激动剂,用于活化 ERE tk-Luc 的 EC50值为36.5 nM。 | |||
T4S0217 |
HOMOPLANTAGININ
|
TNF; NF-κB | Apoptosis; NF-κB |
Homoplantaginin 是来自中药荔枝草的一种类黄酮,具有抗炎和抗氧化活性。 | |||
TN7233 |
Pseudobaptigenin
Psi-baptigenin |
Others | Others |
Pseudobaptigenin (Psi-baptigenin) 是一种异黄酮,是一种黄酮类脂质分子,是在Pterocarpus marsupium、Dalbergia spruceana 中发现的一种天然产品。 | |||
T10183 |
6-Methoxytricin
|
Reductase | Endocrinology/Hormones; Metabolism |
6-Methoxytricin 是从积雪草中分离的黄酮类化合物,是醛糖还原酶 (AR) 和晚期糖基化终产物 (AGE) 的抑制剂,抑制生物细胞中的T细胞增殖和活化。 | |||
------------------------ 更多 ------------------------ |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-03512 |
GT Protein, Solanum melongena, Recombinant (His & Myc)
GT,UDP-glucose flavonoid 3-O-glucosyltransferase,An... |
Solanum melongena | Baculovirus Insect Cells |
In the presence of other necessary color factors, this glycosylation reaction allows the accumulation of anthocyanin pigments. GT Protein, Solanum melongena, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 52.2 kDa and the accession number is Q43641. | |||
TMPY-01579 |
GBA3 Protein, Human, Recombinant (His)
glucosidase, beta, acid 3 (gene/pseudogene),GBA3,MGC126878,K... |
Human | Baculovirus Insect Cells |
Cytosolic beta-glucosidase, also known as Cytosolic beta-glucosidase-like protein 1, GBA3, CBG and CBGL1 is a cytoplasm protein which belongs to theglycosyl hydrolase 1 family and Klotho subfamily. GBA3 / CBGL1 is a glycosidase probably involved in the intestinal absorption and metabolism of dietary flavonoid glycosides. GBA3 / CBGL1 is present in small intestine (at protein level). GBA3 / CBGL1 is expressed in liver, small intestine, colon, spleen and kidney. GBA3 / CBGL1 is down-regulated in r... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0618 |
Quercetin-d5
|
||
Quercetin-d5 是 Quercetin 的氘代化合物。Quercetin 的 CAS 号为 117-39-5。Quercetin 是一种存在于蔬菜、水果和葡萄酒中的天然黄酮,可激活或抑制许多蛋白质的活性。它是重组 SIRT1 的刺激剂,也是 PI3K 抑制剂,抑制 PI3Kγ,PI3Kδ,PI3Kβ 的IC50分别为 2.4 μM, 3.0 μM, 5.4 μM。 |