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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 208 | 现货 | |
5 mg | ¥ 478 | 现货 | |
10 mg | ¥ 697 | 现货 | |
25 mg | ¥ 1,160 | 现货 | |
50 mg | ¥ 1,480 | 现货 | |
100 mg | ¥ 2,320 | 现货 | |
500 mg | ¥ 5,520 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 615 | 现货 |
产品描述 | DOTA-NHS-ester is a linker of affibody molecules for small animal PET, SPECT and CT. DOTA-NHS-ester can be used to label radiotherapeutic agents or imaging probes for tumor detection. |
体外活性 | DOTA-NHS-酯可用于修饰人血清白蛋白(HSA),生成DOTA-HSA。DOTA-HSA进一步通过Sulfo-SMCC修饰,获得DOTA-HSA-SMCC。DOTA-HSA-SMCC与ZHER2:342偶联,最终产物为DOTA-HSA-ZHER2:342[1]。在细胞摄取实验中,标记了64Cu的DOTA-HSA-ZHER2:342(0.5-2小时)在SKOV3细胞中缓慢累积,0.5小时时达到施加活性的0.71%,2小时时摄取量增加至1.58%[1]。 |
分子量 | 501.49 |
分子式 | C20H31N5O10 |
CAS No. | 170908-81-3 |
存储 | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 50 mg/mL (99.70 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||
DMSO
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