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Search Results for " antibacterial activity "
Targets Recommended: MMP Antibacterial Antibiotic

283

抑制剂 & 化合物

175

天然产物

7

化合物库

1

TargetMol 试剂盒

20

重组蛋白

5

同位素标记化合物

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Cat. No. Product Name
L4520 抗菌活性库

904 compounds
904 种具有抗菌活性的化合物,是抗菌药物研发的有力工具;
L9300 大环化合物库

210 compounds
210 种活性已知的大环化合物,用于高通量、高内涵筛选;
L4400 抗生素库

692 compounds
692 个具有抗菌活性化合物的独特集合,是医药研究的优良工具库和药物筛选的有效载体;
L6110 生物碱类天然产物库

500 compounds
500 种生物碱类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L6120 黄酮类天然产物库

514 compounds
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L9240 农药化合物库

270 compounds
270种农药相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L6610 抗感染天然产物库

1060 compounds
1060 个抗感染相关的天然产物集合,是药物开发、药理研究的有效工具;

化合物库

抗菌活性库
Cat.No: L4520
Compounds: 904
大环化合物库
Cat.No: L9300
Compounds: 210
抗生素库
Cat.No: L4400
Compounds: 692
生物碱类天然产物库
Cat.No: L6110
Compounds: 500
黄酮类天然产物库
Cat.No: L6120
Compounds: 514
农药化合物库
Cat.No: L9240
Compounds: 270
抗感染天然产物库
Cat.No: L6610
Compounds: 1060
Cat. No. Product Name Form Specificity Of Inhibition
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
Cat. No. Product Name Target Signaling Pathways
T1140 Doxycycline hydrochloride

Doxylin,盐酸多西环素,Vibramycin,Hyclate

MMP; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hydrochloride (Hyclate) 是一种四环素抗生素,是口服有效的广谱金属蛋白酶抑制剂,具有抗菌活性。
T22330 Fenamic acid

N-苯基邻氨基苯甲酸,2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid

Chloride channel Membrane transporter/Ion channel
Fenamic acid (N-Phenylanthranilic acid) 是氯通道阻滞剂。
T1616 Cefotiam hydrochloride

盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor

Antibacterial; Antibiotic Microbiology/Virology
Cefotiam hydrochloride (SCE-963 hydrochloride) 是一种肠外头孢菌素类广谱抗生素,对革兰氏阳性菌和革兰氏阴性菌有活性。
T20766 Sulfisoxazole acetyl

Gantrisin,Acetylsulfisoxazole,Gantrisin Pediatric,Lipo Gantrisin,乙酰磺胺异噁唑

Antibacterial Microbiology/Virology
Sulfisoxazole acetyl (Gantrisin) 是 Sulfisoxazole 的一种衍生物,是口服有效的二氢蝶酸合酶抑制剂。Sulfisoxazole acetyl 显示出抗菌作用。
T10214 A7132

Antibacterial Microbiology/Virology
A7132是一种抗菌剂,具有广泛而有效的抗菌活性。
T9612 Antibacterial agent 27 

Anti-infection Microbiology/Virology
Antibacterial agent 27 是抗菌化合物,显示出有效的抗念珠菌活性。
T6411 Biapenem

CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Antibacterial; Antibiotic Microbiology/Virology
Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T9990 c-Met-IN-15

Antibacterial Microbiology/Virology
c-Met-IN-15 具有抗菌活性。
T7432 2'-​Hydroxy-​2-​methoxychalcone

2'-Hydroxy-2-methoxychalcone,2'-羟基-2-甲氧基查尔酮

Others; Antibacterial Microbiology/Virology; Others
2'-​Hydroxy-​2-​methoxychalcone 是一个合成的查尔酮,具有抗菌活性。
T60000 STING (WT/R232) activity regulator 126

STING Immunology/Inflammation
STING (WT/R232) activity regulator 126 是一种具有抗菌和抗病毒作用的 STING 调节剂。
T60073 Antimycobacterial agent-4

4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide

Antibacterial Microbiology/Virology
Antimycobacterial agent-4 (4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide) 对结核分枝杆菌具有抗菌活性。
T60093 CHEMBL1380345

N,N'-(Ethane-1,2-diyl)bis(3-methylbenzenesulfonamide)

Antibacterial Microbiology/Virology
CHEMBL1380345 对金黄色葡萄球菌、蜡状芽孢杆菌和大肠杆菌具有抗菌活性,pMIC 值分别为 3.64、3.56 和 3.70。
T8365 Methenamine Hippurate

Antibacterial Microbiology/Virology
Methenamine hippurate 是一种口服活性尿液广谱抗菌剂。它对大多数常见的尿路病原体有效。
T4270 Cefquinome sulfate

硫酸头孢喹肟,硫酸头孢喹诺

Antibacterial; Antibiotic Microbiology/Virology
Cefquinome sulfate 是一种半合成的头孢烯广谱抗生素,具有抗菌活性。
T11227L1 Eravacycline HCl

Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl

Antibiotic Microbiology/Virology
Eravacycline HCl (TP-434 HCl) 是一种具有广谱抗菌活性的强效抗生素。
T11933 MAC13772

Others Others
MAC13772 是一种 BioA 酶的有效抑制剂,IC50 为 250 nM,从而抑制生物素的生物合成。 MAC13772 具有抗菌活性。
T8323 LolCDE-IN-1

Antibacterial Microbiology/Virology
LolCDE-IN-1 是一种有抗菌活性的LolCDE 复合物抑制。
T33470 Monoctanoin

辛酸2,3-二羟基酯,Glyceryl 1-caprylate,Moctanin

Antibacterial Microbiology/Virology
Monoctanoin (Glyceryl 1-caprylate) 对金黄色葡萄球菌和大肠杆菌具有抗菌活性。
T72310 Antibacterial agent 132

Antifungal Microbiology/Virology
Antibacterial agent 132 对 C. parapsilosis (ATCC 22019) 和 C. krusei (ATCC 6258) 实验中显示出抗菌作用,MIC90 值分别为 <0.06 μg/mL 和 62.50 μg/mL。Antibacterial agent 132 对芳香化酶 (aromatase enzyme)具有抑制作用,IC50 为 0.047μM。
T7669 RPW-24

Antibacterial Microbiology/Virology
RPW-24 刺激线虫的宿主免疫反应,保护秀丽隐杆线虫免受细菌感染。它具有抗菌活性。
T72047 Antibacterial agent 125

Antibacterial Microbiology/Virology
Antibacterial agent 125 是一种抗菌剂。Antibacterial agent 125 对临床相关的革兰氏阳性病原体具有有效的抗菌活性,MIC50值范围为 0.25 - 8 μM。Antibacterial agent 125 可用于抗菌药物耐药性研究。
T17254 Amifloxacin

Win49375,氨氟沙星

Antibacterial Microbiology/Virology
Amifloxacin (Win49375) 是有效的喹诺酮类抗菌剂。
T80665 Leu-Val

L-leucyl-L-valine

Parasite; Antifungal Microbiology/Virology
Leu-Val (L-leucyl-L-valine) 是一种新型有效的二肽,具有抗菌和抗疟活性。
T40473L rCRAMP (rat) acetate

rCRAMP (rat) acetate (376364-38-4 Free base)

Antibacterial Microbiology/Virology
rCRAMP (rat) acetate 是一种与cathelin 相关的抗菌肽,在大鼠脑肽/蛋白质提取物中表现出抗菌活性。
T8390 Cefazolin

头孢唑林,头孢唑啉

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin 是一种头孢类抗生素, 用于多种细菌感染的研究。
T1444 Lomefloxacin

洛美沙星,SC47111A

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T77716 Wnt pathway inhibitor 4

Antibacterial Microbiology/Virology
Wnt pathway inhibitor 4 是一种小分子抗菌剂,具有抗菌和抗癌细胞增殖活性。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T12470 Picloxydine

Antibacterial Microbiology/Virology
Picloxydine 是一种杂环双胍,有抗细菌和牙菌斑活性。
T0396 Pipemidic acid

吡哌酸,Acido pipemidico

Antibacterial; Antibiotic Microbiology/Virology
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。
T0751 Furazolidone

呋喃唑酮,Furoxone

Apoptosis; MAO; Antibacterial; Antibiotic Apoptosis; Metabolism; Microbiology/Virology; Neuroscience
Furazolidone (Furoxone) 是一种具有抗菌和抗原虫活性的硝基呋喃衍生物,抑制AML1-ETO 转化细胞,IC50为12.7 μM。
T77619 WAY-322243

CDK Cell Cycle/Checkpoint
WAY-322243 具有抗菌抗炎活性,对 CLK-1 有抑制作用,可用于研究阿尔茨海默症。
T5024 Cefotiam Hexetil Hydrochloride

盐酸头孢替安酯,头孢替安海替酯盐酸盐

Antibacterial; Antibiotic Microbiology/Virology
Cefotiam hexetil hydrochloride 是一种可口服头孢菌素,是抗生素 cefotiam 的前药,但无抗菌作用。
T12096L Morinidazole

Antibacterial Microbiology/Virology
Morinidazole 具有抗菌活性,可用于厌氧菌引起的阑尾炎、盆腔炎等细菌感染研究。
T0495 Aminothiazole

2-Aminothiazole,2-氨基噻唑,2-Thiazolylamine,氨噻唑

Virus Protease; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Aminothiazole (2-Aminothiazole) 是一种甲状腺抑制剂,具有抗菌活性。它是一种典型的杂环胺,是合成多种生物活性分子的前体,包括染料,抗生素,硫磺药物,杀真菌剂和化学反应促进剂。
T15237 Eperezolid

PNU-100592

Antibacterial; Antibiotic Microbiology/Virology
Eperezolid (PNU-100592) 是一种在体外表现出良好抑制活性的恶唑烷酮类抗生素。
T4405 Ceftibuten dihydrate

头孢布烯二水合物,Sch-39720 dihydrate

Antibacterial; Antibiotic Microbiology/Virology
Ceftibuten dihydrate (Sch-39720 dihydrate) 是一种具有口服活性的头孢菌素,在体外对多种革兰氏阴性和某些革兰氏阳性病原体有抗菌活性。
T67978 Cefuzonam

Antibiotic Microbiology/Virology
Cefuzonam 是一种新型头孢菌素,具有抗炎抗菌活性,可用于研究呼吸道感染、扁桃体炎和肝胆感染。
T35346 Tiamulin fumarate

Thiamutilin fumarate

Antibacterial Microbiology/Virology
Tiamulin fumarate (Thiamutilin fumarate)是一种半合成的二萜类抗生素,具有抗菌活性,抑制蛋白质合成,可用于研究气囊炎。
T6268 Ceftiofur hydrochloride

头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur hydrochloride (U-67279A) 是头孢噻呋的盐酸盐形式,是一种β-内酰胺酶稳定的半合成广谱头孢菌素,具有抗菌活性。
T26748 BB-78485

BB78485,BB 78485

Others Others
BB-78485 是一种有效的 LpxC 金属酶小分子抑制剂,具有抗菌作用。 BB-78485 对 LpxC 的 IC50 值为 160 nM。 BB-78485 可用于研究革兰氏阴性菌感染。
T7897 PK150

Others; Antibacterial Microbiology/Virology; Others
PK150 是一种 Sorafenib 类似物,具有抗菌活性。它抑制甲氧西林敏感金黄色葡萄球菌,耐甲氧西林金黄色葡萄球菌,万古霉素中介金黄色葡萄球菌的 MIC 分别为 0.3,0.3-1,0.3 µM。
TN6672 Cyclo(L-Phe-L-Pro)

Free radical scavengers; COX; Antibacterial; Antifungal Immunology/Inflammation; Microbiology/Virology; Neuroscience; oxidation-reduction
Cyclo(L-Phe-L-Pro) 具有广谱抗菌和抗真菌活性。 Cyclo(L-Phe-L-Pro) 对耐甲氧西林金黄色葡萄球菌和棉子肠球菌具有活性。
T50016 2-amino-4-methyl-1,3-thiazole-5-carbohydrazide

Others Others
2-amino-4-methyl-1,3-thiazole-5-carbohydrazide (AMTCH)具有抗肿瘤活性,通过诱导细胞凋亡或细胞程序性死亡抑制癌细胞的生长,也具有抗细菌和真菌活性。
T64396 Antiviral agent 38

Antiviral Immunology/Inflammation
Antiviral agent 38具有抗菌和抗病毒活性,可用来研究乙肝病毒。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T67717L Questiomycin A derivatives 18 TFA

Others Others
Questiomycin A derivatives 18 TFA 是一种Questiomycin A 衍生物,Questiomycin A 具有抗菌和抗癌活性 ,对细胞保护性 ER 伴侣蛋白 GRP78 的表达具有抑制作用。
T3279 Silver sulfadiazine

Silvadene,磺胺嘧啶银,Dermazin,Flamazine

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Silver sulfadiazine (Dermazin) 是一种磺胺类抗生素,具有抗菌和抗真菌活性。它的通磺胺部分(SD-SDZ) 对细菌生长有双重抑制作用,可阻止细菌叶酸吸收以及 DNA 合成。它释放的银结合并破坏 DNA 结构,阻止细菌 DNA 复制。
T0750 Sulfisoxazole

NU-445,磺胺二甲异唑,Sulfafurazole,磺胺异恶唑

Endothelin Receptor; Antibacterial; Antibiotic; Autophagy Autophagy; GPCR/G Protein; Microbiology/Virology
Sulfisoxazole (Sulfafurazole) 是一种内皮素受体拮抗剂,是磺胺类抗生素。它靶向内皮素受体 A,抑制乳腺癌外显子释放。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。

化合物

Doxycycline hydrochloride
Cat.No: T1140
Synonym: Doxylin,盐酸多西环素,Vibramycin,Hyclate
Target: MMP, Antibacterial, Antibiotic
Fenamic acid
Cat.No: T22330
Synonym: N-苯基邻氨基苯甲酸,2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid
Target: Chloride channel
Cefotiam hydrochloride
Cat.No: T1616
Synonym: 盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor
Target: Antibacterial, Antibiotic
Sulfisoxazole acetyl
Cat.No: T20766
Synonym: Gantrisin,Acetylsulfisoxazole,Gantrisin Pediatric,Lipo Gantrisin,乙酰磺胺异噁唑
Target: Antibacterial
A7132
Cat.No: T10214
Synonym:
Target: Antibacterial
Antibacterial agent 27 
Cat.No: T9612
Synonym:
Target: Anti-infection
Biapenem
Cat.No: T6411
Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627
Target: Antibacterial, Antibiotic
c-Met-IN-15
Cat.No: T9990
Synonym:
Target: Antibacterial
2'-​Hydroxy-​2-​methoxychalcone
Cat.No: T7432
Synonym: 2'-Hydroxy-2-methoxychalcone,2'-羟基-2-甲氧基查尔酮
Target: Others, Antibacterial
STING (WT/R232) activity regulator 126
Cat.No: T60000
Synonym:
Target: STING
Antimycobacterial agent-4
Cat.No: T60073
Synonym: 4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide
Target: Antibacterial
CHEMBL1380345
Cat.No: T60093
Synonym: N,N'-(Ethane-1,2-diyl)bis(3-methylbenzenesulfonamide)
Target: Antibacterial
Methenamine Hippurate
Cat.No: T8365
Synonym:
Target: Antibacterial
Cefquinome sulfate
Cat.No: T4270
Synonym: 硫酸头孢喹肟,硫酸头孢喹诺
Target: Antibacterial, Antibiotic
Eravacycline HCl
Cat.No: T11227L1
Synonym: Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl
Target: Antibiotic
MAC13772
Cat.No: T11933
Synonym:
Target: Others
LolCDE-IN-1
Cat.No: T8323
Synonym:
Target: Antibacterial
Monoctanoin
Cat.No: T33470
Synonym: 辛酸2,3-二羟基酯,Glyceryl 1-caprylate,Moctanin
Target: Antibacterial
Antibacterial agent 132
Cat.No: T72310
Synonym:
Target: Antifungal
RPW-24
Cat.No: T7669
Synonym:
Target: Antibacterial
Antibacterial agent 125
Cat.No: T72047
Synonym:
Target: Antibacterial
Amifloxacin
Cat.No: T17254
Synonym: Win49375,氨氟沙星
Target: Antibacterial
Leu-Val
Cat.No: T80665
Synonym: L-leucyl-L-valine
Target: Parasite, Antifungal
rCRAMP (rat) acetate
Cat.No: T40473L
Synonym: rCRAMP (rat) acetate (376364-38-4 Free base)
Target: Antibacterial
Cefazolin
Cat.No: T8390
Synonym: 头孢唑林,头孢唑啉
Target: Others, Antibacterial, Antibiotic
Lomefloxacin
Cat.No: T1444
Synonym: 洛美沙星,SC47111A
Target: Topoisomerase, Antibacterial, Antibiotic
Wnt pathway inhibitor 4
Cat.No: T77716
Synonym:
Target: Antibacterial
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Picloxydine
Cat.No: T12470
Synonym:
Target: Antibacterial
Pipemidic acid
Cat.No: T0396
Synonym: 吡哌酸,Acido pipemidico
Target: Antibacterial, Antibiotic
Furazolidone
Cat.No: T0751
Synonym: 呋喃唑酮,Furoxone
Target: Apoptosis, MAO, Antibacterial, Antibiotic
WAY-322243
Cat.No: T77619
Synonym:
Target: CDK
Cefotiam Hexetil Hydrochloride
Cat.No: T5024
Synonym: 盐酸头孢替安酯,头孢替安海替酯盐酸盐
Target: Antibacterial, Antibiotic
Morinidazole
Cat.No: T12096L
Synonym:
Target: Antibacterial
Aminothiazole
Cat.No: T0495
Synonym: 2-Aminothiazole,2-氨基噻唑,2-Thiazolylamine,氨噻唑
Target: Virus Protease, Antibacterial, Antibiotic, Antifungal
Eperezolid
Cat.No: T15237
Synonym: PNU-100592
Target: Antibacterial, Antibiotic
Ceftibuten dihydrate
Cat.No: T4405
Synonym: 头孢布烯二水合物,Sch-39720 dihydrate
Target: Antibacterial, Antibiotic
Cefuzonam
Cat.No: T67978
Synonym:
Target: Antibiotic
Tiamulin fumarate
Cat.No: T35346
Synonym: Thiamutilin fumarate
Target: Antibacterial
Ceftiofur hydrochloride
Cat.No: T6268
Synonym: 头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
BB-78485
Cat.No: T26748
Synonym: BB78485,BB 78485
Target: Others
PK150
Cat.No: T7897
Synonym:
Target: Others, Antibacterial
Cyclo(L-Phe-L-Pro)
Cat.No: TN6672
Synonym:
Target: Free radical scavengers, COX, Antibacterial, Antifungal
2-amino-4-methyl-1,3-thiazole-5-carbohydrazide
Cat.No: T50016
Synonym:
Target: Others
Antiviral agent 38
Cat.No: T64396
Synonym:
Target: Antiviral
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Questiomycin A derivatives 18 TFA
Cat.No: T67717L
Synonym:
Target: Others
Silver sulfadiazine
Cat.No: T3279
Synonym: Silvadene,磺胺嘧啶银,Dermazin,Flamazine
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Sulfisoxazole
Cat.No: T0750
Synonym: NU-445,磺胺二甲异唑,Sulfafurazole,磺胺异恶唑
Target: Endothelin Receptor, Antibacterial, Antibiotic, Autophagy
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
T3947 Nonanoic acid

pelargonic acid,Nonoic acid,壬酸

Others; Antibacterial Microbiology/Virology; Others
Nonanoic acid (Nonoic acid) 是一种天然存在的具有九个碳原子的饱和脂肪酸。它减少细菌易位,增强抗菌活性,并增加猪 β-防御素 1 (pBD-1) 和 pBD-2 的分泌。
T1687 Doxycycline

Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素

MMP; ribosome; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
T6702 Terbinafine

Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine (TDT 067) 是念珠菌属的角鲨烯环氧化酶有效的非竞争性抑制剂,Ki 值为 30 nM。它具有抗真菌感染活性。
T1411 Terbinafine hydrochloride

KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。
T20345 Benzoylacetone

AI3 10572,苯甲酰丙酮,AI3-10572,AI310572

Antibacterial Microbiology/Virology
Benzoylacetone (AI3 10572) 具有抗菌活性。
TN6780 Carvacrol methyl ether

Methyl carvacrol,Methyl carvacryl ether

Antibacterial Microbiology/Virology
Carvacrol methyl ether 来源于植物挥发油,具有抗菌活性。
T20550 Thiobarbituric acid

NSC4733,NSC 4733,4,6-二羟基-2-巯基嘧啶,NSC-4733

Antibacterial Microbiology/Virology
Thiobarbituric acid (NSC-4733) 具有抗菌活性。
T5757 Loganetin

Antibacterial Microbiology/Virology
Loganetin 是无毒的天然产物,来源于Cornus officinalis Sieb. et Zucc.,可用于耐多药革兰氏阴性菌感染的研究。
T5S1959 (-)-Asarinin

Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin

Antibacterial Microbiology/Virology
(-)-Asarinin (Eleutheroside B4) 是一种主要从 Zanthoxylum armatum 根部提取到的木脂素。
TN1469 Cassiaside B

Others; Antibacterial Microbiology/Virology; Others
Cassiaside B 是一种具有强效抗菌活性的天然产物。
T37886 1-Heptadecanol

Antibacterial Microbiology/Virology
1-Heptadecanol 是分离自Solena amplexicaulis 的长链伯醇,显示出抗菌活性。
T9112 (-)-Perillaldehyde

AhR; ROS; Nrf2 Immunology/Inflammation; Metabolism
L-Perillaldehyde 是紫苏草精油的主要成分,吸入后经由嗅觉神经功能表现出抗抑郁功能。
TN1041 Quercimeritrin

槲皮素-7-O-葡萄糖苷,槲皮素-7-0-葡萄苷,Quercetin-7-O-beta-D-glucopyranoside

Anti-infection; COX; NO Synthase Immunology/Inflammation; Microbiology/Virology; Neuroscience
Quercimeritrin (Quercetin-7-O-beta-D-glucopyranoside) 是分离自齿状苦艾叶中,具淀粉酶作用。
T3S0970 Thermopsine

Thermospine,黄华碱

Antibacterial Microbiology/Virology
Thermopsine (Thermospine) 是从槐豆亚种的果实,豆荚和茎皮中分离出来的一种喹诺酮类生物碱,具有抗菌活性。
T5982 3-Methoxybenzoic acid

m-Methoxybenzoic acid,NSC 9264,3-甲氧基苯甲酸,NSC 27014,3-Anisic acid

Endogenous Metabolite Metabolism
3-Methoxybenzoic acid (NSC 27014) 能够用于合成3-甲氧基苯甲醚(III) 和钆 (III) 。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T4S0578 Guaijaverin

番石榴苷,Guajaverin,Quercetin-3-Arabinoside

Others; Antioxidant; Antibacterial Microbiology/Virology; Others; oxidation-reduction
Guaijaverin (Quercetin-3-Arabinoside) 是一种尿素酶抑制剂,IC50值为 120 μM,有抗氧化和抗变形链球菌作用。
T8258 Chloramphenicol succinate sodium

Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。
TN5173 Trichorabdal A

Antifection Microbiology/Virology
Trichorabdal A 是一种二萜化合物,分离自 Rabdosia trichocarpa,抗肿瘤作用强大。
TN4375 Kamebanin

Antifection Microbiology/Virology
Kamebanin 是一种天然二萜类化合物,具有抗菌活性。它对 HeLa 和 HL-60 细胞显示出有效的细胞毒活性。
TN7051 2,4-Dihydroxybenzaldehyde

2,4-二羟基苯甲醛,4-Formylresorcinol,beta-Resorcylaldehyde,4-Hydroxysalicylaldehyde

Endogenous Metabolite Metabolism
2,4-Dihydroxybenzaldehyde (4-Formylresorcinol) 是内源性代谢产物的一种。
T3629 Gamithromycin

ML-1709460,加米霉素

Antibacterial; Antibiotic Microbiology/Virology
Gamithromycin (ML-1709460) 是一种可抑制 MmmSC 菌株 B237 和 Tan8 生长的大环内酯类抗菌剂,MIC 值分别为 0.00012 和 0.00006 μg/mL。
T6S2024 Harpagide

Antibacterial; Parasite Microbiology/Virology
Harpagide 是从Scrophularia cryptophila 中分离出来的一种鸢尾糖苷,具有抗炎和抗寄生虫活性,对T.b. rhodesiense 具有体外锥虫杀虫活性,IC50为 21 μg/mL,它对L. donovani 的IC50值为 2.0 μg/mL。
T8247 (+)-Aromadendrene

Anti-infection Microbiology/Virology
(+)-Aromadendrene 是一种天然产物,对革兰氏阳性菌和革兰氏阴性菌具有显着的抗菌活性。
TMO2685 10-Hydroxydecanoic Acid

NSC 15139,10-羟基癸烯酸,10-羟基癸酸

Antibacterial Microbiology/Virology
10-Hydroxydecanoic Acid (NSC 15139) 是一种存在于蜂王浆中的 10-hydroxy-trans-2-decenoic acid 的饱和脂肪酸,具有抗炎活性。
T8335 Lycobetaine acetate

氧化石蒜碱乙酸盐,Oxylycorine

Others Others
Lycobetaine acetate (Oxylycorine) 是一种潜在的抗罗克福提青霉和黑曲霉的生物杀菌剂。
TN1530 Cowaxanthone B

β-倒捻子素类似物2号

Antioxidant; Parasite Microbiology/Virology; oxidation-reduction
Cowaxanthone B 是从小叶藤黄果实中分离出的新的四氧氧杂蒽酮。Cowaxanthone B 具有潜在的抗菌活性。
T8261 Ceftazidime Pentahydrate

头孢他啶五水合物,头孢他啶

Antibacterial; Antibiotic Microbiology/Virology
Ceftazidime pentahydrate 是一种β-内酰胺类抗菌剂,对革兰氏阳性和革兰氏阴性需氧细菌有广谱活性,可静脉内或肌肉给药。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。
T5707 3-O-Methylgalangin

3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚

Antibacterial Microbiology/Virology
3-O-Methylgalangin (GALANGIN-3-METHYLETHER) 是一种来源于高良姜根茎的天然黄酮,具有抗菌活性,抑制胰腺脂肪酶。
T8185 (+)-Viroallosecurinine

别一叶萩碱,Viroallosecurinine

Antibacterial Microbiology/Virology
(+)-Viroallosecurinine (Viroallosecurinine) 是一种具有抗菌活性的天然生物碱,抑制Ps. Aeruginosa 和Staph. aureus,MIC 为 0.48 μg/mL。
T8066 Sulbenicillin disodium

磺苄西林钠,Sulbenicillin Sodium

Antibacterial; Antibiotic Microbiology/Virology
Sulbenicillin disodium (Sulbenicillin Sodium) 是 Sulbenicillin 的二钠盐。Sulbenicillin 是一种青霉素抗生素,对Pseudomonas aeruginosa 的许多粘液型和非粘液型菌株具有抗菌活性。
TN1008 Psoralenoside

CaMK; Calcium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T3S1534 Secoxyloganin

断氧化马钱苷,幼枝含断氧化马钱子甙,金银花

Anti-infection Microbiology/Virology
Secoxyloganin 是从Lonicera japonicaThunb 提取得到,能够抑制血流量减少,具有抗过敏活性。
TN1209 2-Hydroxy-1-methoxyanthraquinone

Alizarin 1-methyl ether

Antibacterial Microbiology/Virology
2-Hydroxy-1-methoxyanthraquinone (Alizarin 1-methyl ether) 是一种从 Morinda lucida Benth. (Rubiaceae) 中分离得到具有抗菌活性的天然产物。
TN1466 Canthin-6-one

NSC 103003

Antifungal Microbiology/Virology
Canthin-6-one(NSC 103003) 是一种从 Allium neapolitanum 分离出来的生物碱,具有抗菌活性,对结核分枝杆菌具有抑制作用。
TN1492 Chrysophanein

Chrysophanol 1-O-glucoside

Antioxidant; Antiviral; Antibacterial Immunology/Inflammation; Microbiology/Virology; oxidation-reduction
Chrysophanein (Chrysophanol 1-O-glucoside) 是来自芦荟 (Aloe hijazensis) 叶和根的羟醌化合物,具有抗菌、抗真菌和抗氧化活性,MIC 值为8-256 μg/mL。Chrysophanein 可用于研究真菌感染。
T1465 Mupirocin

Pseudomonic acid,莫匹罗星,BRL-4910A

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Mupirocin (BRL-4910A) 是从Pseudomonas fluorescens 中分离得到的一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起抗菌作用。
T5S2245 Alisol C 23-acetate

泽泻醇 C-23-醋酸酯,Alisol C monoacetate

Others Others
Alisol C 23-acetate (Alisol C monoacetate) 是一种提取自东方泽泻中的天然产物,可以显著减少迟发型超敏反应。
T6389 Anacardic Acid

漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid

Others; Epigenetic Reader Domain; Histone Acetyltransferase; Antibacterial Chromatin/Epigenetic; Microbiology/Virology; Others
Anacardic Acid (6-pentadecylsalicylic Acid) 是从腰果壳中提取液中分离到的酸类物质,是一种组蛋白乙酰转移酶抑制剂,对 p300 和 PCAF 的 IC50值分别为 ∼8.5 μM 和 ∼5 μM。
T5781 taraxasteryl acetate

蒲公英甾醇醋酸酯,醋酸蒲公英酯

Antibacterial Microbiology/Virology
Taraxasteryl acetate 是分离自矢状疟原虫中,具有广谱的抗炎活性。它能够改善右旋糖酐、酵母聚糖及花生四烯酸诱导的大鼠后爪水肿。它可用于研究局部炎症。
T13305 Viridicatol

Anti-infection; Antifungal Microbiology/Virology
Viridicatol 是从夹竹桃的内生真菌青霉菌属的发酵中分离出的一种喹诺酮类生物碱,对金黄色葡萄球菌有抗菌活性,MIC 值为 15.6 μg/mL。
T4S1616 Sanggenon D

Sanggenone D

GABA Receptor; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Sanggenon D (Sanggenone D) 是来自桑白皮的小分子化合物,是GABA(A)受体调节剂,具有抗氧化抗菌活性,抑制乳腺癌细胞增殖,通过调节脂肪酸生物合成系统来抑制金黄色葡萄球菌的生长。
T10164 5,6-Dihydroxyindole

Dopamine lutine

Endogenous Metabolite Metabolism
5,6-Dihydroxyindole (Dopamine lutine) 是黑色素的前体,显示出广谱的抗菌,抗真菌,抗病毒,抗寄生虫活性。5,6-Dihydroxyindole 也显示出细胞毒性作用。
T67867 Mycaminosyltylonolide

Antibacterial Microbiology/Virology
Mycaminosyltylonolide 是一种大环内酯类抗生素,它是 tyololide 在位置5上具有β - d -mycaminosyl 残基。Mycaminosyltylonolide 是一种有效的抗生素,具有抗菌活性和抑制荧光素酶的合成。
T4S1452 Artemisic acid

(+)-Artemisinic Acid,青蒿酸,Artemisinic acid

Antibacterial Microbiology/Virology
Artemisic acid ((+)-Artemisinic Acid) 是黄花蒿中分离得到的一种倍半萜,具有多种药理活性,如抗疟、抗菌和抗肿瘤活性,以及解热、化感和抗脂肪生成作用。
TN1905 Magnolioside

七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷

Antifection Microbiology/Virology
Magnolioside 是分离自Angelica gigas Nakai(Umbelliferae) 中,对谷氨酸诱导的毒性有显著的神经保护作用。 它显示出对金黄色葡萄球菌 CIP 53.154 的中等抗菌活性。它具有抗疟原虫活性,对氯喹敏感的恶性疟原虫菌株具有强烈的生长抑制作用。
T3733 (E)-Methyl 4-coumarate

Methyl trans-p-Coumarat,OMpCA,反式对羟基肉桂酸,Methyl 4-hydroxycinnamate

Apoptosis; Others; Antibacterial Apoptosis; Microbiology/Virology; Others
Methyl (E)-4-hydroxycinnamatee在几种植物中发现,如洋葱或海巴戟叶中。它与 Carnosic Acid 联用可诱导细胞凋亡,杀死急性髓性白血病细胞。它具有抗氧化和抗菌活性。
T5070 LC3-mHTT-IN-AN2

5,7-二羟基-4-苯基香豆素,5,7-Dihydroxy-4-phenylcoumarin

Antibacterial; Autophagy; ATTECs Autophagy; Microbiology/Virology; PROTAC
LC3-mHTT-IN-AN2 (5,7-Dihydroxy-4-phenylcoumarin) 是一种 mHTT-LC3 接头化合物,可与突变亨廷顿蛋白(mHTT) 和 LC3B 相互作用。 它将 mHTT 靶向自噬体以等位基因选择性方式降低培养的亨廷顿病小鼠神经元中的 mHTT 水平。它存在于西番莲植物中,具有抗菌活性。
TN3972 Epimedokoreanin B

Apoptosis; Others; Antibacterial Apoptosis; Microbiology/Virology; Others
Epimedokoreanin B (EKB) 是一种从韩国淫羊藿中分离出的异戊烯化类黄酮,在人非小细胞肺癌(NSCLC)A549和NCI-H292细胞中展现出抗癌活性。Epimedokoreanin B 还具有抗炎和抗菌活性,可有清除 DPPH 自由基的活性,能以剂量依赖的方式抑制 MCF-7 和 HepG2 的增殖。Epimedokoreanin B 能显著抑制 N (δ) -(羧甲基)赖氨酸(CML)和 N (Ï) -(羧甲基)精氨酸(CMA)的形成,可通过抑制高级糖化终产物(AGEs)预防糖尿病的临床并发症。
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天然产物

Nonanoic acid
Cat.No: T3947
Synonym: pelargonic acid,Nonoic acid,壬酸
Target: Others, Antibacterial
Doxycycline
Cat.No: T1687
Synonym: Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Terbinafine
Cat.No: T6702
Synonym: Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067
Target: Antibacterial, Antibiotic, Antifungal
Terbinafine hydrochloride
Cat.No: T1411
Synonym: KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride
Target: Antibacterial, Antibiotic, Antifungal
Benzoylacetone
Cat.No: T20345
Synonym: AI3 10572,苯甲酰丙酮,AI3-10572,AI310572
Target: Antibacterial
Carvacrol methyl ether
Cat.No: TN6780
Synonym: Methyl carvacrol,Methyl carvacryl ether
Target: Antibacterial
Thiobarbituric acid
Cat.No: T20550
Synonym: NSC4733,NSC 4733,4,6-二羟基-2-巯基嘧啶,NSC-4733
Target: Antibacterial
Loganetin
Cat.No: T5757
Synonym:
Target: Antibacterial
(-)-Asarinin
Cat.No: T5S1959
Synonym: Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin
Target: Antibacterial
Cassiaside B
Cat.No: TN1469
Synonym:
Target: Others, Antibacterial
1-Heptadecanol
Cat.No: T37886
Synonym:
Target: Antibacterial
(-)-Perillaldehyde
Cat.No: T9112
Synonym:
Target: AhR, ROS, Nrf2
Quercimeritrin
Cat.No: TN1041
Synonym: 槲皮素-7-O-葡萄糖苷,槲皮素-7-0-葡萄苷,Quercetin-7-O-beta-D-glucopyranoside
Target: Anti-infection, COX, NO Synthase
Thermopsine
Cat.No: T3S0970
Synonym: Thermospine,黄华碱
Target: Antibacterial
3-Methoxybenzoic acid
Cat.No: T5982
Synonym: m-Methoxybenzoic acid,NSC 9264,3-甲氧基苯甲酸,NSC 27014,3-Anisic acid
Target: Endogenous Metabolite
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
Guaijaverin
Cat.No: T4S0578
Synonym: 番石榴苷,Guajaverin,Quercetin-3-Arabinoside
Target: Others, Antioxidant, Antibacterial
Chloramphenicol succinate sodium
Cat.No: T8258
Synonym: Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠
Target: Others, Antibacterial, Antibiotic
Trichorabdal A
Cat.No: TN5173
Synonym:
Target: Antifection
Kamebanin
Cat.No: TN4375
Synonym:
Target: Antifection
2,4-Dihydroxybenzaldehyde
Cat.No: TN7051
Synonym: 2,4-二羟基苯甲醛,4-Formylresorcinol,beta-Resorcylaldehyde,4-Hydroxysalicylaldehyde
Target: Endogenous Metabolite
Gamithromycin
Cat.No: T3629
Synonym: ML-1709460,加米霉素
Target: Antibacterial, Antibiotic
Harpagide
Cat.No: T6S2024
Synonym:
Target: Antibacterial, Parasite
(+)-Aromadendrene
Cat.No: T8247
Synonym:
Target: Anti-infection
10-Hydroxydecanoic Acid
Cat.No: TMO2685
Synonym: NSC 15139,10-羟基癸烯酸,10-羟基癸酸
Target: Antibacterial
Lycobetaine acetate
Cat.No: T8335
Synonym: 氧化石蒜碱乙酸盐,Oxylycorine
Target: Others
Cowaxanthone B
Cat.No: TN1530
Synonym: β-倒捻子素类似物2号
Target: Antioxidant, Parasite
Ceftazidime Pentahydrate
Cat.No: T8261
Synonym: 头孢他啶五水合物,头孢他啶
Target: Antibacterial, Antibiotic
3-O-Methylgalangin
Cat.No: T5707
Synonym: 3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚
Target: Antibacterial
(+)-Viroallosecurinine
Cat.No: T8185
Synonym: 别一叶萩碱,Viroallosecurinine
Target: Antibacterial
Sulbenicillin disodium
Cat.No: T8066
Synonym: 磺苄西林钠,Sulbenicillin Sodium
Target: Antibacterial, Antibiotic
Psoralenoside
Cat.No: TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Secoxyloganin
Cat.No: T3S1534
Synonym: 断氧化马钱苷,幼枝含断氧化马钱子甙,金银花
Target: Anti-infection
2-Hydroxy-1-methoxyanthraquinone
Cat.No: TN1209
Synonym: Alizarin 1-methyl ether
Target: Antibacterial
Canthin-6-one
Cat.No: TN1466
Synonym: NSC 103003
Target: Antifungal
Chrysophanein
Cat.No: TN1492
Synonym: Chrysophanol 1-O-glucoside
Target: Antioxidant, Antiviral, Antibacterial
Mupirocin
Cat.No: T1465
Synonym: Pseudomonic acid,莫匹罗星,BRL-4910A
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Alisol C 23-acetate
Cat.No: T5S2245
Synonym: 泽泻醇 C-23-醋酸酯,Alisol C monoacetate
Target: Others
Anacardic Acid
Cat.No: T6389
Synonym: 漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid
Target: Others, Epigenetic Reader Domain, Histone Acetyltransferase, Antibacterial
taraxasteryl acetate
Cat.No: T5781
Synonym: 蒲公英甾醇醋酸酯,醋酸蒲公英酯
Target: Antibacterial
Viridicatol
Cat.No: T13305
Synonym:
Target: Anti-infection, Antifungal
Sanggenon D
Cat.No: T4S1616
Synonym: Sanggenone D
Target: GABA Receptor, Antibiotic
5,6-Dihydroxyindole
Cat.No: T10164
Synonym: Dopamine lutine
Target: Endogenous Metabolite
Mycaminosyltylonolide
Cat.No: T67867
Synonym:
Target: Antibacterial
Artemisic acid
Cat.No: T4S1452
Synonym: (+)-Artemisinic Acid,青蒿酸,Artemisinic acid
Target: Antibacterial
Magnolioside
Cat.No: TN1905
Synonym: 七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷
Target: Antifection
(E)-Methyl 4-coumarate
Cat.No: T3733
Synonym: Methyl trans-p-Coumarat,OMpCA,反式对羟基肉桂酸,Methyl 4-hydroxycinnamate
Target: Apoptosis, Others, Antibacterial
LC3-mHTT-IN-AN2
Cat.No: T5070
Synonym: 5,7-二羟基-4-苯基香豆素,5,7-Dihydroxy-4-phenylcoumarin
Target: Antibacterial, Autophagy, ATTECs
Epimedokoreanin B
Cat.No: TN3972
Synonym:
Target: Apoptosis, Others, Antibacterial
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Cat. No. Product Name Species Expression System
TMPY-00672 Azurocidin/CAP37 Protein, Human, Recombinant (His)

AZU,NAZC,azurocidin 1,hHBP,AZAMP,HUMAZUR,CAP37,HBP,AZU1

Human HEK293 Cells
Azurocidin (AZU1), also known as heparin-binding protein (HBP) or cationic antimicrobial protein 37 (CAP37), is an azurophil granule antibiotic protein, with monocyte chemotactic and antibacterial activity. The Azurophil granules, specialized lysosomes of the neutrophil, contain at least 10 proteins implicated in the killing of microorganisms. Azurocidin is a member of the serine protease family that includes Cathepsin G, neutrophil elastase (NE), and proteinase 3 (PR3), however, Azurocidin is n...
TMPH-02543 DEFB33 Protein, Mouse, Recombinant (His & Myc & SUMO)

BD-33,Defb33,mBD-33,Defensin, beta 33,Beta-defensin 33

Mouse E. coli
Has antibacterial activity.
TMPH-02542 DEFB19 Protein, Mouse, Recombinant (His & Myc)

Defensin, beta 19,Tdl,Testis-specific beta-defensin-like pro...

Mouse E. coli
Has antibacterial activity.
TMPH-01006 DEFB129 Protein, Human, Recombinant (His & Myc)

DEFB129,C20orf87,Beta-defensin 129,DEFB29,DEFB-29,Beta-defen...

Human P. pastoris (Yeast)
Has antibacterial activity. DEFB129 Protein, Human, Recombinant (His & Myc) is expressed in yeast with C-6xHis-Myc tag. The predicted molecular weight is 21.8 kDa and the accession number is Q9H1M3.
TMPH-00512 Lysenin-related protein 2 Protein, Eisenia foetida, Recombinant (His & Myc)

Hemolysin,Lysenin-related protein 2,Fetidin,Lysenin-3,efL3

Eisenia fetida E. coli
Pore-forming toxin that specifically binds sphingomyelin in the plasma membrane of various cells. Has hemolytic activity. It also has antibacterial activities against B.megaterium.
TMPH-01005 DEFB128 Protein, Human, Recombinant (His & Myc)

DEFB-28,Beta-defensin 128,DEFB28,Beta-defensin 28,Defensin, ...

Human E. coli
Has antibacterial activity. DEFB128 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 16.0 kDa and the accession number is Q7Z7B8.
TMPH-02545 DEFB6 Protein, Mouse, Recombinant (His & KSI)

Defb6,Beta-defensin 6,Defensin, beta 6,mBD-6,BD-6

Mouse E. coli
Has potent antibacterial activity against E.coli (ATCC 25922). DEFB6 Protein, Mouse, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 19.8 kDa and the accession number is Q91VD6.
TMPH-03082 DEFB106A Protein, Pan troglodytes, Recombinant (His & KSI)

BD-6,cBD-6,DEFB6,DEFB106,DEFB106A,Defensin, beta 106,Beta-de...

Chimpanzee E. coli
Has antibacterial activity. Acts as a ligand for C-C chemokine receptor CCR2. DEFB106A Protein, Pan troglodytes, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 20.4 kDa and the accession number is Q5IAB3.
TMPH-01058 Cathelicidin antimicrobial peptide Protein, Human, Recombinant (His & Myc & SUMO)

CAP18,Cathelicidin antimicrobial peptide,CAMP,FALL39,CAP-18,...

Human E. coli
Binds to bacterial lipopolysaccharides (LPS), has antibacterial activity. Cathelicidin antimicrobial peptide Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 24.7 kDa and the accession number is P49913.
TMPH-00064 MRJP1 Protein, Apis mellifera, Recombinant (His)

Royalactin,Major royal jelly protein 1,Apalbumin 1,MRJP1,56-...

Apis mellifera P. pastoris (Yeast)
Induces the differentiation of honeybee larvae into queens through an Egfr-mediated signaling pathway. Promotes body size increase by activating p70 S6 kinase, stimulates ovary development by augmenting the titer of vitellogenin (Vg) and juvenile hormone, and reduces developmental time by increasing the activity of mitogen-activated protein kinase and inducing the 20-hydroxyecdysone protein (20E). Most abundant protein found in the royal jelly which is the food of the queen honey bee larva. The ...
TMPH-02503 DEFA1 Protein, Mouse, Recombinant (GST & His)

HP-1,HNP-1,Defensin, alpha 1,DEFA1,DEFA2,MRS,Neutrophil defe...

Mouse E. coli
Probably contributes to the antimicrobial barrier function of the small bowel mucosa. Has antibacterial activity against attenuated mutants of S.typhimurium. DEFA1 Protein, Mouse, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predicted molecular weight is 34.1 kDa and the accession number is P11477.
TMPH-01772 DEFA1 Protein, Human, Recombinant (GST)

MRS,HP1,HP-1,DEFA1,DEF1,Defensin, alpha 1,Neutrophil defensi...

Human E. coli
Defensin 1 and defensin 2 have antibacterial, fungicide and antiviral activities. Has antimicrobial activity against Gram-negative and Gram-positive bacteria. Defensins are thought to kill microbes by permeabilizing their plasma membrane. DEFA1 Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 37.2 kDa and the accession number is P59665.
TMPH-02875 ROMO1 Protein, Mouse, Recombinant (His)

Protein MGR2 homolog,Romo1,Reactive oxygen species modulator...

Mouse E. coli
Has antibacterial activity against a variety of bacteria including S.aureus, P.aeruginosa and M.tuberculosis. Acts by inducing bacterial membrane breakage.; Induces production of reactive oxygen species (ROS) which are necessary for cell proliferation. May play a role in inducing oxidative DNA damage and replicative senescence. May play a role in the coordination of mitochondrial morphology and cell proliferation.
TMPJ-00574 RNASE3 Protein, Human, Recombinant (His)

RNase 3,RNS3,ECP,Eosinophil Cationic Protein,RNASE3,Ribonucl...

Human HEK293 Cells
Ribonuclease 3 (RNASE3) is a basic protein that is localized to the eosinophil primary matrix and belongs to the pancreatic ribonuclease family. RNASE3 is released during degranulation of eosinophils. RNASE3 possesses a wide variety of biological activities. RNASE3 interacts with bacterial lipopolysaccharide (LPS) and lipoteichoic acid (LTA). RNASE3 exhibits antibacterial activity, including cytoplasmic membrane depolarization of preferentially Gram-negative, but also Gram-positive strains. It p...
TMPY-02163 PGLYRP1 Protein, Mouse, Recombinant (His)

Tnfsf3l,peptidoglycan recognition protein 1,PGRP,Tasg7,Tag7,...

Mouse HEK293 Cells
Peptidoglycan recognition protein 1, also known as Peptidoglycan recognition protein short, PGRP-S, PGLYRP1, PGLYRP, PGRP and TNFSF3L, is a secreted protein that belongs to the N-acetylmuramoyl-L-alanine amidase 2 family. PGLYRP1 / PGLYRP is highly expressed in bone marrow. It is weakly expressed in kidney, liver, small intestine, spleen, thymus, peripheral leukocyte, lung, fetal spleen and neutrophils. PGLYRP1 / PGLYRP is a pattern receptor that binds to murein peptidoglycans (PGN) of Gram-posi...
TMPH-03266 CHI3L1 Protein, Rat, Recombinant (His)

Chi3l1,Cartilage glycoprotein 39,CGP-39,GP-39,Chitinase-3-li...

Rat E. coli
Carbohydrate-binding lectin with a preference for chitin. Has no chitinase activity. May play a role in tissue remodeling and in the capacity of cells to respond to and cope with changes in their environment. Plays a role in T-helper cell type 2 (Th2) inflammatory response and IL-13-induced inflammation, regulating allergen sensitization, inflammatory cell apoptosis, dendritic cell accumulation and M2 macrophage differentiation. Facilitates invasion of pathogenic enteric bacteria into colonic mu...
TMPY-01812 Enoyl-ACP Reductase Protein, E. coli, Recombinant (His)

b1288,JW1281,gts,ECK1283,qmeA,envM

E. coli E. coli
Enoyl-ACP reductase, also known as NADH-dependent enoyl-ACP reductase and FABI, is a cell inner membrane and peripheral membrane protein which belongs to theshort-chain dehydrogenases/reductases (SDR) family and FabI subfamily. Microorganisms produce many kinds of antibiotics which function in an antagonistic capacity in nature where they have much competition. Bacterial FAS provides essential fatty acids for use in the assembly of key cellular components. Among them, FABI is an enoyl-ACP...
TMPY-01644 Cystatin S Protein, Human, Recombinant (His)

MGC71923,cystatin S,CST4

Human HEK293 Cells
Cystatin-S, also known as Cystatin-4, Salivary acidic protein 1, Cystatin-SA-III and CST4, is a secreted protein which belongs to thecystatin family. Cystatin-4 / CST4 is expressed in submandibular and sublingual saliva but not in parotid saliva (at protein level). It is also expressed in saliva, tears, urine and seminal fluid. The cystatin superfamily encompasses proteins that contain multiple cystatin-like sequences. Some of the members are active cysteine protease inhibitors, while oth...
TMPY-05252 Myeloperoxidase/MPO Protein, Human, Recombinant (His)

myeloperoxidase

Human HEK293 Cells
MPO (myeloperoxidase) is a peroxidase enzyme secreted by activated leukocytes that plays a pathogenic role in cardiovascular disease, mainly by initiating endothelial dysfunction. Myeloperoxidase (MPO) is an important enzyme, which is one of the components of the antibacterial system in neutrophils and monocytes. MPO participates in the inflammatory response in multiple locations in the body, including the mammary glands. Myeloperoxidase (MPO), a specific polymorphonuclear leukocyte enzyme, has ...
TMPH-01552 IRF1 Protein, Human, Recombinant (GST & His)

IRF1,Interferon regulatory factor 1

Human Baculovirus Insect Cells
Transcriptional regulator which displays a remarkable functional diversity in the regulation of cellular responses. Regulates transcription of IFN and IFN-inducible genes, host response to viral and bacterial infections, regulation of many genes expressed during hematopoiesis, inflammation, immune responses and cell proliferation and differentiation, regulation of the cell cycle and induction of growth arrest and programmed cell death following DNA damage. Stimulates both innate and acquired imm...

重组蛋白

Azurocidin/CAP37 Protein, Human, Recombinant (His)
Cat.No: TMPY-00672
Species: Human
Expression System: HEK293 Cells
DEFB33 Protein, Mouse, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-02543
Species: Mouse
Expression System: E. coli
DEFB19 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02542
Species: Mouse
Expression System: E. coli
DEFB129 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01006
Species: Human
Expression System: P. pastoris (Yeast)
Lysenin-related protein 2 Protein, Eisenia foetida, Recombinant (His & Myc)
Cat.No: TMPH-00512
Species: Eisenia fetida
Expression System: E. coli
DEFB128 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01005
Species: Human
Expression System: E. coli
DEFB6 Protein, Mouse, Recombinant (His & KSI)
Cat.No: TMPH-02545
Species: Mouse
Expression System: E. coli
DEFB106A Protein, Pan troglodytes, Recombinant (His & KSI)
Cat.No: TMPH-03082
Species: Chimpanzee
Expression System: E. coli
Cathelicidin antimicrobial peptide Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-01058
Species: Human
Expression System: E. coli
MRJP1 Protein, Apis mellifera, Recombinant (His)
Cat.No: TMPH-00064
Species: Apis mellifera
Expression System: P. pastoris (Yeast)
DEFA1 Protein, Mouse, Recombinant (GST & His)
Cat.No: TMPH-02503
Species: Mouse
Expression System: E. coli
DEFA1 Protein, Human, Recombinant (GST)
Cat.No: TMPH-01772
Species: Human
Expression System: E. coli
ROMO1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02875
Species: Mouse
Expression System: E. coli
RNASE3 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00574
Species: Human
Expression System: HEK293 Cells
PGLYRP1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02163
Species: Mouse
Expression System: HEK293 Cells
CHI3L1 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03266
Species: Rat
Expression System: E. coli
Enoyl-ACP Reductase Protein, E. coli, Recombinant (His)
Cat.No: TMPY-01812
Species: E. coli
Expression System: E. coli
Cystatin S Protein, Human, Recombinant (His)
Cat.No: TMPY-01644
Species: Human
Expression System: HEK293 Cells
Myeloperoxidase/MPO Protein, Human, Recombinant (His)
Cat.No: TMPY-05252
Species: Human
Expression System: HEK293 Cells
IRF1 Protein, Human, Recombinant (GST & His)
Cat.No: TMPH-01552
Species: Human
Expression System: Baculovirus Insect Cells
Cat. No. Product Name Target Signaling Pathways
TMIH-0305 Lomefloxacin-d5 hydrochloride

Lomefloxacin-d5 hydrochloride 是 Lomefloxacin hydrochloride 的氘代化合物。Lomefloxacin hydrochloride 的 CAS 号为 98079-51-7。Lomefloxacin是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
TMID-0286 Rifaximin-d6

Rifaximin-d6 是 Rifaximin 的氘代化合物。Rifaximin 的 CAS 号为 80621-81-4。Rifaximin是一种胃肠道选择性抗生素,与细菌 DNA 依赖性 RNA 聚合酶的 β 亚基结合,抑制细菌 RNA 合成。与革兰氏阴性菌(MIC:8-50 毫克/毫升)相比,它对革兰氏阳性菌株(MIC:0.03-5 毫克/毫升)的敏感性更高。
TMID-0072 Imipenem-d4

Imipenem-d4 是 Imipenem 的氘代化合物。Imipenem 的 CAS 号为 64221-86-9。Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。
TMIH-0530 Sulbactam-d2

Sulbactam-d2 是 Sulbactam 的氘代化合物。Sulbactam 的 CAS 号为 68373-14-8。Sulbactam是一种竞争性、不可逆的 β-内酰胺酶抑制剂,抑制耐多药不动杆菌-鲍曼不动杆菌复合物。它具有抗菌活性。
T36021 Flumequine-13C3

Flumequine-13C3

Flumequine-13C3is intended for use as an internal standard for the quantification of flumequine by GC- or LC-MS. Flumequine is a fluoroquinolone antibiotic.1It is active againstS. aureus, S. pyogenes, B. subtilis, E. coli, P. aeruginosa, S. faecalis, andK. pneumoniae(MICs = 1-100 μg/ml). Flumequine is also active against field isolates of B. hyodysenteriae (MICs = 6.25-200 μg/ml).2It inhibits DNA gyrase, disrupting supercoiling of bacterial DNA to block transcription and replication.3In vivo, fl...

同位素标记化合物

Lomefloxacin-d5 hydrochloride
Cat.No: TMIH-0305
Synonym:
Target:
Rifaximin-d6
Cat.No: TMID-0286
Synonym:
Target:
Imipenem-d4
Cat.No: TMID-0072
Synonym:
Target:
Sulbactam-d2
Cat.No: TMIH-0530
Synonym:
Target:
Flumequine-13C3
Cat.No: T36021
Synonym: Flumequine-13C3
Target:
TargetMol Loading
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