VU6010572

Name: VU6010572
Brand: TargetMol
SKU: T61070
Price: 122 USD
Availability: InStock
Rating: 4.5 (1 reviews)

还可以

产品编号 T61070Cas号 2126784-39-0

VU6010572 is a highly potent and selective negative allosteric modulator of mGlu3, exhibiting an IC50 of 245 nM. Additionally, VU6010572 displays high central nervous system penetrance [1] [2].

VU6010572

还可以

产品编号 T61070Cas号 2126784-39-0

VU6010572 is a highly potent and selective negative allosteric modulator of mGlu3, exhibiting an IC50 of 245 nM. Additionally, VU6010572 displays high central nervous system penetrance [1] [2].

规格	价格	库存
25 mg	¥ 14,900	6-8周
50 mg	¥ 19,420	6-8周
100 mg	¥ 24,625	6-8周

大包装 & 定制

加入购物车

实验操作小课堂

联系我们获取更多批次信息

资源下载

产品操作手册

TargetMol 的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。

产品介绍

生物活性

产品描述	VU6010572 is a highly potent and selective negative allosteric modulator of mGlu3, exhibiting an IC50 of 245 nM. Additionally, VU6010572 displays high central nervous system penetrance [1] [2].
体内活性	VU6010572 (3 mg/kg; i.p.) shows robust efficacy [1]. VU6010572 (3 mg/kg; i.p.; 45 minutes) produces lasting anxiolytic-like behavioral effects [2]. Animal Model: CD-1 mice [1] Dosage: 3 mg/kg Administration: I.p. Result: Showed robust efficacy. Animal Model: Rats [2] Dosage: 3 mg/kg Administration: I.p.; 45 minutes Result: Produced lasting anxiolytic-like behavioral effects.