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Search Results for " wide spectrum "

Targets Recommended: Antibacterial Antibiotic

25

抑制剂 & 化合物

5

天然产物

2

化合物库

8

重组蛋白

2

同位素标记化合物

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Cat. No.	Product Name
L9500	表型筛选靶点鉴定库		1796 compounds
	1796 种靶点明确的已知活性化合物，适合表型筛选；
L2170	肿瘤免疫治疗小分子化合物库		449 compounds
	449 种靶向肿瘤免疫治疗靶点的小分子，可用于高通量和高内涵筛选，是研究肿瘤免疫治疗的有力工具；

化合物库

表型筛选靶点鉴定库

Cat.No: L9500

Compounds: 1796

肿瘤免疫治疗小分子化合物库

Cat.No: L2170

Compounds: 449

Cat. No.	Product Name	Target	Signaling Pathways
T8134	Cefathiamidine	Antibacterial; Antibiotic	Microbiology/Virology
	Cefathiamidine 是一种头孢菌素抗菌剂，可研究由易感细菌引起的感染，还可用于呼吸道、肝脏、五官感觉、尿路感染以及心内膜炎和败血症的研究。
T21995	XAP044	GluR	Neuroscience
	XAP044 是高效的选择性mGlu7拮抗剂。代谢型谷氨酸受体亚型 7 是哺乳动物 CNS 中神经传递的重要突触前调节剂。它在啮齿动物行为测试中表现出较好的大脑暴露、广谱抗应激、抗抑郁以及抗焦虑作用。
T4017	Relebactam 瑞来巴坦,MK-7655	Antibacterial	Microbiology/Virology
	Relebactam (MK-7655) 是一种有广谱抗β内酰胺酶活性的二氮杂双环辛烷抑制剂。
T8620	piperacillin Pipril,Pipracil,哌拉西林,Pipercillin	Antibacterial	Microbiology/Virology
	Piperacillin (Pipercillin) 是半合成青霉素，可以作用于革兰氏阳性和革兰氏阴性需氧和厌氧菌。与其他青霉素相比，它对产生 β-内酰胺酶的菌类表现出更强的活性。
T9449	Nitrofural [(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺	Antibacterial	Microbiology/Virology
	Nitrofural 是 20 世纪已在临床应用中确立的硝基呋喃。 Nitrofural 在临床上对广泛的革兰氏阳性和革兰氏阴性细菌（包括许多常见的泌尿道病原体菌株）仍然有效。
T37071	Pyrimethanil	Antifungal	Microbiology/Virology
	Pyrimethanil 是苯胺嘧啶类广谱接触杀菌剂，用于控制多种作物上的Botrytis spp.。它抑制灰霉病菌中氨基酸的生物合成，可用于霉菌感染的水果、蔬菜和观赏植物真菌病害防治的相关研究。
T10491	Galidesivir BCX4430,Immucillin-A	Others	Others
	Galidesivir (BCX4430) 是一种广谱抗病毒化合物，是一种腺苷类似物，能抑制病毒 RNA 依赖的 RNA 聚合酶 (RdRp) 活性。Galidesivir 在体外对多种 RNA 病毒病原体有抑制作用，可减少受感染动物的肺部感染。
T19860	Clavulanic Acid BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151	Antibacterial; Antifungal	Microbiology/Virology
	Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素，是一种强效的细菌 β-内酰胺酶抑制剂，用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性，对多种革兰氏阳性和革兰氏阴性细菌均有活性。
T4501	Ceftizoxime 头孢唑肟,Epocelin	Antibacterial; Antibiotic	Microbiology/Virology
	Ceftizoxime (Epocelin) 是一种强效抗菌剂，它通过干扰细菌细胞壁合成和抑制肽聚糖的交联起作用。它对广谱的 β-内酰胺酶具有高度抗性，并且对多种需氧和厌氧的革兰氏阳性和革兰氏阴性微生物均有效。
T27794	λ-Cyhalothrin lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon	Sodium Channel; Parasite	Membrane transporter/Ion channel; Microbiology/Virology
	λ-Cyhalothrin (Icon) 是广谱的 II 型合成除虫菊酯杀虫剂，含有 α-氰基，用于防治多种害虫。它是一种钠通道神经毒素，靶向中枢神经系统中神经元膜。
T20196	Cefamandole 头孢孟多,Compound 83405,L-Cefamandole,Mancef,Mandol	Others	Others
	Cefamandole is a semisynthetic wide-spectrum cephalosporin with prolonged action. It is used also as the nafate.
T1101	Minocycline hydrochloride Minocycline HCl,盐酸米诺环素,美满霉素	HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic	Chromatin/Epigenetic; Metabolism; Microbiology/Virology
	Minocycline hydrochloride (Minocycline HCl) 属于四环素类抗生素，具有出色的吸收和组织渗透性。Minocycline hydrochloride 是一种广谱的抗菌剂，可用于多种细菌感染以及痤疮的治疗。
T28576	Ro 24-6392 Ro 246392,Ro-24-6392	Others	Others
	Ro 24-6392 is an ester-linked co-drug combining ciprofloxacin and desacetylcefotaxime. Ro 24-6392 demonstrats activity against a wide spectrum of aerobic bacteria.
T20107	Ertapenem Invanz,MK0826,MK-0826,MK 0826	Others	Others
	Ertapenem is a parenteral carbapenem. It has a broad spectrum of antimicrobial activity. It is highly resistant to inactivation by a wide variety of beta-lactamases.
TP2064	ω-Conotoxin MVIIC
	Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.
T17106	TMC310911	Others	Others
	TMC310911 is an effective and orally active HIV type-1 protease inhibitor (EC50: ranged from 2.2 nM to 14.2 nM for wild-type HIV-1). TMC310911 has effective activity against a wide spectrum of recombinant HIV-1 isolates.
T69388	PD 0305970	Others	Others
	PD 0305970 is new bacterial gyrase and topoisomerase inhibitor that possess outstanding in vitro and in vivo activities against a wide spectrum of bacterial species including quinolone- and multidrug-resistant gram-positive and fastidious organism groups.
T24690	Pyrromecaine HCl Bumecaine hydrochloride,Pyrromecaine	Others	Others
	Pyrromecaine is a local anesthetic used for surface anesthesia. Pyromecaine has a wide spectrum of antiarrhythmic action, exerts a favorable effect on the contractility of the left ventricle, and on the myocardial blood flow following the ligation of the
T39206	HKSOX-1m (5/6-mixture)
	HKSOX-1m (5/6-mixture) serves as a mitochondria-targeting O2 fluorescent probe with an excitation/emission wavelength of 509/534nm (green), showcasing exceptional selectivity and sensitivity for O2 across a wide pH spectrum and in the presence of strong oxidants and prevalent reductants within cells.
T75345	HKSOX-1m (5/6-mixture) (hydrobromide)
	HKSOX-1m (5/6-mixture) hydrobromide 是靶向线粒体的 O2•−荧光探针(Ex/Em=509/534 nm; 绿色)，具有极好的选择性，且在较大范围的 pH 值区间，细胞中即使有大量强氧化剂和还原剂的时候依然有效。
T82410	Fenquinotrione	Others	Others
	Fenquinotrione为4-羟基苯丙酮酸双加氧酶(HPPD)抑制剂，水稻HPPD (OsHPPD) 及拟南芥HPPD (AtHPPD) 的IC50分别达27.2及44.7nM。此化合物作为除草剂，对多种阔叶及芦苇杂草具有广泛防治效果，并展现出对水稻的高选择性。
T81011	Tetanus Toxin (830–844)
	Tetanus Toxin (830–844) 是具有生物活性的肽类化合物。它是破伤风毒素衍生的 TT830–844 CD4+ T 细胞表位，能与多种 HLA-DRB 分子结合。该 CD4+ T 细胞表位由于与广泛的 HLA-DRB 分子具有亲和力，有潜力在大范围人群中诱发 CD4+ T 细胞应答。
T75281	Cephalexin hydrochloride monohydrate	Others	Others
	Cephalexin (Cefalexin) hydrochloride monohydrate 是一种口服有效的半合成头孢菌素类抗生素（antibiotic），对广泛的革兰氏阳性及革兰氏阴性细菌展现出抗菌活性。该化合物通过靶向青霉素结合蛋白（PBPs）抑制细菌细胞壁的组装，应用于包括肺炎、链球菌性咽喉炎、细菌性心内膜炎在内的疾病研究。
T23451	Tedizolid HCl (856866-72-3 free base) Tedizolid HCl	Others	Others
	Tedizolid HCl is a reversible, novel oxazolidinone antibiotic (IC50: for MAO-A (monoamine oxidase-A), 8.7 uM; for MAO-B, 5.7 uM). It is the first oxazolidinone to be approved since linezolid in 2000. Tedizolid phosphate is the second commercially availabl
T38174	Mpro inhibitor N3 hemihydrate	Others	Others
	Mpro inhibitor N3 hemihydrate is a potent inhibitor of SARS-CoV-2 Mpro with an EC50 of 16.77 μM for SARS-CoV-2. Mpro inhibitor N3 hemihydrate specifically inhibits Mpro from multiple coronaviruses, including SARS-CoV and MERS-CoV. Mpro inhibitor N3 hemihydrate displays inhibition against HCoV-229E, FIPV, and MHV-A59 with individual IC50 of 4.0 μM, 8.8 μM, and 2.7 μM, respectively[1][2]. Mpro inhibitor N3 hemihydrate (0-0.64 μM) is able to penetrate cells to inhibit the replication of IBV viruses...

化合物

Cat.No: T8134

Target: Antibacterial, Antibiotic

Cat.No: T21995

Target: GluR

Cat.No: T4017

Synonym: 瑞来巴坦,MK-7655

Target: Antibacterial

Cat.No: T8620

Synonym: Pipril,Pipracil,哌拉西林,Pipercillin

Target: Antibacterial

Cat.No: T9449

Synonym: [(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺

Target: Antibacterial

Cat.No: T37071

Target: Antifungal

Cat.No: T10491

Synonym: BCX4430,Immucillin-A

Target: Others

Clavulanic Acid

Cat.No: T19860

Synonym: BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151

Target: Antibacterial, Antifungal

Cat.No: T4501

Synonym: 头孢唑肟,Epocelin

Target: Antibacterial, Antibiotic

Cat.No: T27794

Synonym: lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon

Target: Sodium Channel, Parasite

Cat.No: T20196

Synonym: 头孢孟多,Compound 83405,L-Cefamandole,Mancef,Mandol

Target: Others

Minocycline hydrochloride

Cat.No: T1101

Synonym: Minocycline HCl,盐酸米诺环素,美满霉素

Target: HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic

Cat.No: T28576

Synonym: Ro 246392,Ro-24-6392

Target: Others

Cat.No: T20107

Synonym: Invanz,MK0826,MK-0826,MK 0826

Target: Others

ω-Conotoxin MVIIC

Cat.No: TP2064

Cat.No: T17106

Target: Others

Cat.No: T69388

Target: Others

Pyrromecaine HCl

Cat.No: T24690

Synonym: Bumecaine hydrochloride,Pyrromecaine

Target: Others

HKSOX-1m (5/6-mixture)

Cat.No: T39206

HKSOX-1m (5/6-mixture) (hydrobromide)

Cat.No: T75345

Cat.No: T82410

Target: Others

Tetanus Toxin (830–844)

Cat.No: T81011

Cephalexin hydrochloride monohydrate

Cat.No: T75281

Target: Others

Tedizolid HCl (856866-72-3 free base)

Cat.No: T23451

Synonym: Tedizolid HCl

Target: Others

Mpro inhibitor N3 hemihydrate

Cat.No: T38174

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T1326	Gentamicin sulfate SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素	ribosome; DHFR; Antibacterial; Antibiotic	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
	Gentamicin sulfate (SCH9724) 是一种广谱的氨基糖苷类抗生素，具有口服活性。Gentamicin sulfate 可以用于抑制敏感生物体中的蛋白质合成。
TN6718	Dehydrocostuslactone	Others	Others
	Dehydrocostuslactone 是一种从奥克兰提取的天然产物。它具有广泛的生物作用，包括抗炎、抗癌、抗病毒、抗菌、抗真菌、抗氧化、抗糖尿病、抗溃疡和驱虫活性。
T1304	Chlortetracycline hydrochloride Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素	ribosome; Antibacterial; Antibiotic	Microbiology/Virology
	Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T3893	Forsythoside B 连翘酯苷 B,连翘脂苷B	TNF; NF-κB	Apoptosis; NF-κB
	Forsythoside B 是传统中药植物独一味叶子中分离的一种苯乙醇苷。它可抑制 TNF-alpha，IL-6，IκB，调节 NF-κB。它抑制炎症反应，具有抗氧化和神经保护作用。
T20779	Kitasamycin tartrate Leucomycin tartrate	Others	Others
	Kitasamycin tartrate, a macrolide antibiotic produced by Streptomyces kitasatoensis, has a wide spectrum of antimicrobial activity.

天然产物

Gentamicin sulfate

Cat.No: T1326

Synonym: SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素

Target: ribosome, DHFR, Antibacterial, Antibiotic

Dehydrocostuslactone

Cat.No: TN6718

Target: Others

Chlortetracycline hydrochloride

Cat.No: T1304

Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

Target: ribosome, Antibacterial, Antibiotic

Cat.No: T3893

Synonym: 连翘酯苷 B,连翘脂苷B

Target: TNF, NF-κB

Kitasamycin tartrate

Cat.No: T20779

Synonym: Leucomycin tartrate

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-02030	CD82 Protein, Human, Recombinant (His) CD82 molecule,SAR2,R2,KAI-1,4F9,KAI1,C33,TSPAN27,ST6,IA4,GR1...	Human	HEK293 Cells
	CD82, also known as KAI-1, structurally belongs to tetraspanin family while categorised as metastasis suppressor gene on functional grounds. KAI1/CD82 is localized on cell membrane and form interactions with other tetraspanins, integrins and chemokines which are respectively responsible for cell migration, adhesion and signalling. Downregulation of CD82 expression is associated with the advanced stages of many human cancers and correlates with the acquisition of metastatic potential. Recent stud...
TMPY-00828	Iduronate 2 sulfatase/IDS Protein, Human, Recombinant (His) MPS2,IDS,SIDS,iduronate 2-sulfatase	Human	HEK293 Cells
	Iduronate 2-Sulfatase, also known as IDS, is a member of the highly conserved sulfatase family of enzymes that catalyze the hydrolysis of O- and N-sulfate esters from a variety of substrates. The human Iduronate 2-Sulfatase/IDS consists of a signal peptide, a propeptide, and a mature chain that may be further processed into two chains. Among the identified 18 human sulfatases, Iduronate 2-Sulfatase/IDS is required for the lysosomal degradation of the glycosaminoglycans (GAG), heparan sulfate, an...
TMPY-03296	SHP-1 Protein, Mouse, Recombinant (aa 207-597, His & GST) SH-PTP1,Hcph,70Z-SHP,Ptp1C,protein tyrosine phosphatase, non...	Mouse	Baculovirus Insect Cells
	PTPN6 is an enzyme that belongs to the protein tyrosine phosphatase (PTP) family. PTPs are signaling molecules that regulate a variety of cellular processes including cell growth, differentiation, mitotic cycle, and oncogenic transformation. N-terminal part of PTPN6 contains two tandem Src homolog (SH2) domains, which act as protein phospho-tyrosine binding domains, and mediate the interaction of PTPN6 with its substrates. PTPN6 is expressed primarily in hematopoietic cells, and functions as an ...
TMPY-02511	PTP alpha/PTPRA Protein, Human, Recombinant (aa 174-793, His & GST) LRP,PTP α/PTPRA Protein, Human, Recombinant (aa 174-793, His...	Human	Baculovirus Insect Cells
	PTPRA is reported to be involved in cancer development and progression through activating the Src family kinase (SFK) signaling pathways. The higher PTPRA level was associated with worse prognosis of SCC patients and PTPRA could promote the cell cycle progression through stimulating the c-Src signaling pathways. The PTPRA gene, which encodes the protein RPTP-alpha, is critical to neurodevelopment. Previous linkage studies, genome-wide association studies, controlled expression analyses and anima...
TMPJ-00931	Serpin A4 Protein, Human, Recombinant (His) Kallistatin,Peptidase Inhibitor 4,KST,Kallikrein Inhibitor,S...	Human	HEK293 Cells
	Serpin Peptidase Inhibitor, Clade A (α-1 Antiproteinase, Antitrypsin), Member 4 (Serpin A4) is a member of the Serpin family. Serpin A4 exists as a monomer and some homodimers. Serpin A4 is expressed by the liver and secreted in plasma. Serpin A4 is a regulator of vascular homeostasis capable of controlling a wide spectrum of biological actions in the cardiovascular and renal systems. It can inhibit intracellular reactive oxygen species formation in cultured cardiac and renal cells. In addition,...
TMPY-05088	CNTN6 Protein, Human, Recombinant (hFc) NB3,contactin 6	Human	HEK293 Cells
	Copy number variations (CNVs) of the human CNTN6 gene caused by megabase-scale microdeletions or microduplications in the 3p26.3 region are often the cause of neurodevelopmental disorders, including intellectual disability and developmental delay. Contactin genes CNTN5 and CNTN6 code for neuronal cell adhesion molecules that promote neurite outgrowth in sensory-motor neuronal pathways. The deletion or duplication of the CNTN6 gene is associated with a wide spectrum of neurodevelopmental behavior...
TMPY-00344	ARL6IP6 Protein, Human, Recombinant (mFc) PFAAP1,AIP-6,ADP-ribosylation factor-like 6 interacting prot...	Human	HEK293 Cells
	It had been found that a homozygous truncating mutation in ARL6IP6 as the likely cause of a syndromic form of CMTC associated with major dysmorphism, developmental delay, transient ischemic attacks and cerebral vascular malformations. This gene was previously implicated by genome wide association study (GWAS) as a susceptibility locus to ischemic stroke in young adults. We identify ARL6IP6 as a novel candidate gene for a syndromic form of CMTC. This suggests that ischemic stroke or transient isc...
TMPH-01239	XPC Protein, Human, Recombinant (His) Xeroderma pigmentosum group C-complementing protein,p125,XPC...	Human	E. coli
	Involved in global genome nucleotide excision repair (GG-NER) by acting as damage sensing and DNA-binding factor component of the XPC complex. Has only a low DNA repair activity by itself which is stimulated by RAD23B and RAD23A. Has a preference to bind DNA containing a short single-stranded segment but not to damaged oligonucleotides. This feature is proposed to be related to a dynamic sensor XPC can rapidly screen duplex DNA for non-hydrogen-bonded bases by forming a transient nucleoprotein i...

重组蛋白

CD82 Protein, Human, Recombinant (His)

Cat.No: TMPY-02030

Species: Human

Expression System: HEK293 Cells

Iduronate 2 sulfatase/IDS Protein, Human, Recombinant (His)

Cat.No: TMPY-00828

Species: Human

Expression System: HEK293 Cells

SHP-1 Protein, Mouse, Recombinant (aa 207-597, His & GST)

Cat.No: TMPY-03296

Species: Mouse

Expression System: Baculovirus Insect Cells

PTP alpha/PTPRA Protein, Human, Recombinant (aa 174-793, His & GST)

Cat.No: TMPY-02511

Species: Human

Expression System: Baculovirus Insect Cells

Serpin A4 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00931

Species: Human

Expression System: HEK293 Cells

CNTN6 Protein, Human, Recombinant (hFc)

Cat.No: TMPY-05088

Species: Human

Expression System: HEK293 Cells

ARL6IP6 Protein, Human, Recombinant (mFc)

Cat.No: TMPY-00344

Species: Human

Expression System: HEK293 Cells

XPC Protein, Human, Recombinant (His)

Cat.No: TMPH-01239

Species: Human

Expression System: E. coli

Cat. No.	Product Name	Target	Signaling Pathways
TMIH-0438	Piperacillin-d5
	Piperacillin-d5 是 Piperacillin 的氘代化合物。Piperacillin 的 CAS 号为 61477-96-1。Piperacillin 是半合成青霉素，可以作用于革兰氏阳性和革兰氏阴性需氧和厌氧菌。与其他青霉素相比，它对产生 β-内酰胺酶的菌类表现出更强的活性。
TMIJ-0232	Piperacillin-d5 (N-ethyl-d5)
	Piperacillin-d5 (N-ethyl-d5) 是 Piperacillin 的氘代化合物。Piperacillin 的 CAS 号为 61477-96-1。Piperacillin 是半合成青霉素，可以作用于革兰氏阳性和革兰氏阴性需氧和厌氧菌。与其他青霉素相比，它对产生 β-内酰胺酶的菌类表现出更强的活性。

同位素标记化合物

Piperacillin-d5

Cat.No: TMIH-0438

Piperacillin-d5 (N-ethyl-d5)

Cat.No: TMIJ-0232

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