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Targets Recommended: Cysteine Protease Parasite

81

抑制剂 & 化合物

7

天然产物

3

化合物库

13

重组蛋白

3

同位素标记化合物

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Cat. No.	Product Name
L9860	抗抑郁症化合物库		1163 compounds
	1163 种与抑郁症相关的化合物，可以用于高通量和高内涵筛选
L9830	抗帕金森病化合物库		857 compounds
	857 种帕金森病相关的化合物集合，可用于高通量和高内涵筛选；
L7110	抗高血压化合物库		678 compounds
	678 种高血压相关的小分子，用于高通量和高内涵筛选；

化合物库

抗抑郁症化合物库

Cat.No: L9860

Compounds: 1163

抗帕金森病化合物库

Cat.No: L9830

Compounds: 857

抗高血压化合物库

Cat.No: L7110

Compounds: 678

Cat. No.	Product Name	Target	Signaling Pathways
T12909	SID 26681509	Cysteine Protease; Parasite	Microbiology/Virology; Proteases/Proteasome
	SID 26681509 是可逆的，竞争性的人组织蛋白酶 L 选择性抑制剂，IC50为 56 nM。它抑制Plasmodium falciparum 的体外繁殖，IC50为15.4 μM，抑制Leishmania major，IC5012.5 μM。
T11831	LDN-27219	Others	Others
	LDN-27219 是一种人组织型转谷氨酰胺酶抑制剂(IC50:600 nM)。
T24421	LY-2624803 DB-7,LY2624803,HY-10275,LY 2624803	5-HT Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	LY-2624803 是一种 5-HT2A 受体拮抗剂和组胺受体反向激动剂，可用于改善慢波睡眠。
T24932	Vatanidipine AE-0047,AE 0047,AE0047	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Vatanidipine (AE0047) 是一种新型的双氢吡啶(DHP)型钙通道阻滞剂，具有缓慢起效的药理作用。在各种实验性高血压模型中观察到缓慢起效和持久的降压作用。
T9597	H2S Donor 5a N-(苯甲酰基硫基)苯甲酰胺	Endogenous Metabolite	Metabolism
	H2S Donor 5a 是一种稳定的、半胱氨酸活化的的 H2S 供体。它是研究 H2S 的有用工具。
T20206	Oxymethurea CSI Paste,1'3-双羟甲基脲,Carbamol,Caurite,Dimethylolurea	Others	Others
	Oxymethurea (CSI Paste) 是一种改性尿素，可在农田中用作缓释肥料。
T70470L	isomer-CM 352 isomer-1542205-83-3	MMP	Proteases/Proteasome
	isomer-CM 352 是一种金属酶抑制剂，可用于减缓脑损伤。
T28748	Selodenoson RG14202,DTI0009,DTI-0009,RG-14202,DT-009,DT009	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Selodenoson (RG-14202) 是一种选择性腺苷 A1 受体激动剂，可用于减慢心房颤动患者的心率，治疗心律失常。
T25372	EMD57033 EMD-57033,(+)-EMD 57033,EMD 57033	Calcium Channel; Carbonic Anhydrase	Membrane transporter/Ion channel; Metabolism
	EMD57033是一种心脏肌钙蛋白C（cTnC）激活剂，是一种显性的Ca2+增敏剂。EMD57033通过与心脏/慢速骨骼肌钙蛋白C 异构体结合从而发挥促进心脏收缩的功能。
TP1545L1	FFAGLDD amine salt	Others	Others
	FFAGLDD amine salt 是MMP9选择性裂解肽，用于多柔比星（DOX）的胞浆递送，实现时间和空间可控的缓慢药物递送和释放。
T11805	L-NIL	NOS	Immunology/Inflammation
	L-NIL 是选择性一氧化氮合成酶 (iNOS) 抑制剂，可逆转大鼠骨骼肌中烧伤诱导的糖原合酶激酶-3β激活，可延缓鳞状细胞癌肺的进程。
T21769L	β-Pompilidotoxin Acetate β-Pompilidotoxin Acetate(216064-36-7 Free base)	Sodium Channel	Membrane transporter/Ion channel
	β-Pompilidotoxin Acetate 是一种黄蜂毒肽。它可以减缓钠通道的失活并增加细胞中的稳态钠电流。
T26822	Bisaramil hydrochloride RGH-2957,NK 1556,NK1556,Bisaramil,NK-1556,RGH 2957	Potassium Channel; Adrenergic Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Bisaramil hydrochloride (Bisaramil) 是一种新型二氮双环壬烷抗心律失常化合物，抑制自由基生成。Bisaramil hydrochloride 可阻断钠电流，抑制异丙肾上腺素在 K（+）去极化肌上诱导的缓慢 Ca（2+）动作电位。
T30188L	Atagabalin HCl PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base）	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Atagabalin HCl 是一种新型电压依赖性钙通道（VDCC）α2δ亚基（1 和 2）配体，会影响慢波睡眠,可用于治疗失眠。
T22830	GYY4137 GYY 4137 morpholine salt	Others	Others
	GYY4137 (GYY 4137 morpholine salt) 是一种缓释H2S 供体，具有抗炎和抗癌作用，也具有血管扩张和抗高血压活性。
T0377	Clofazimine NSC-141046,氯法齐明,氯苯吩嗪	DNA; Antibacterial; Antibiotic	DNA Damage/DNA Repair; Microbiology/Virology
	Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料，与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。
T7502L	PF 05089771 PF-05089771,PF05089771	Sodium Channel	Membrane transporter/Ion channel
	PF 05089771是具有口服有效的、选择性的 Nav1.7丙烯酰胺抑制剂。PF-05089771在疼痛和糖尿病神经性疾病的研究中具有价值。
T3193	Pimelic diphenylamide 106 Histone Deacetylase Inhibitor VII,TC-H 106,RGFA-8	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Pimelic diphenylamide 106 (RGFA-8) 是一种缓慢和紧密结合的I 类HDAC 抑制剂，对HDAC1、 2和3的IC50值分别150、760和370 nM。
T15673	KU 59403 KU-59403,KU59403	ATM/ATR	DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
	KU 59403 是一种具有选择性和高效性的 ATM 抑制剂，具有抗肿瘤和抗癌活性，抑制 ATM、DNA-PK 和 PI3K，常与PARP或ATR抑制剂的联合治疗来延缓癌症的进程。
T0029	Procaine Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因	Histone Demethylase; DNA/RNA Synthesis; Sodium Channel	Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Membrane transporter/Ion channel
	Procaine (Vitamin H3) 是DNA 脱甲基剂，是一种酯类局部麻醉剂。它起效缓慢，作用持续时间短，主要用于浸润麻醉、周围神经阻滞和脊髓阻滞。
T1439	Lacidipine SN-305,拉西地平,GX-1048,GR-43659X	Apoptosis; Calcium Channel; Reactive Oxygen Species	Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
	Lacidipine (SN-305) 是一种L 型钙离子通道阻断剂。
T40870	Leukotriene E4 LTE4	Endogenous Metabolite	Metabolism
	Leukotriene E4 (LTE4)（LTE4）通过二肽酶对LTD4 上的作用生成，是过敏性休克慢反应物质（SRS-A）的成分之一。LTE4 存在于血浆和尿液中，可用于检测哮喘。
T5117	Hexaflumuron	Others	Others
	Hexazinone 是一种三嗪家族的非选择性除草剂。它能够同光系统 II 电子传递链的 D-1 醌蛋白结合，抑制光合作用的发生。
T61111	UCB-5307	TNF	Apoptosis
	UCB-5307 是一种小分子化合物，可在体外抑制 TNFR1 信号转导和下游功能。人 TNFα 的 KD 为 9 nM。 TNF 直接通过缓慢的结合动力学结合，KD = 6 nM。 UCB-5307 可以通过预制的 hTNF/hTNFR1 复合物。
T24415	Lotrifen Privaprol,L-12717,DL 717-IT,L 12717,L12717,Canocenta	Others	Others
	Lotrifen (Privaprol) 是一种非激素抗生育药物，Lotrifen 引起妊娠停止和复旧。在胚泡着床后，它直接作用于受精卵，受精卵经历一个缓慢而逐渐的退化过程，并以受精卵的再吸收或排出而结束。
T4440	Saclofen	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Saclofen 是竞争性GABAB 受体拮抗剂(IC50:7.8 μM)。它可研究 GABAB 受体调节大脑中缓慢抑制性突触后电位的功能。
T6541	Ibutilide Fumarate Corvert Fumarate,U70226E,富马酸伊布利特	Calcium Channel; Sodium Channel	Membrane transporter/Ion channel; Metabolism
	Ibutilide Fumarate (U70226E) 是一种 III 类抗心律失常药物，可作用于急性心梗阻塞。
T12425	PF-06424439 methanesulfonate	Acyltransferase; Transferase	Metabolism
	PF-06424439 methanesulfonate 是一种口服有效咪唑并吡啶二酰基甘油酰基转移酶 2 (DGAT2)选择性抑制剂，IC50是14 nM。PF-06424439 methanesulfonate 具有缓慢可逆，时间依赖性的特点，其相对于酰基-CoA 底物以非竞争性模式抑制 DGAT2。
T17197	UCL 2077	Others	Others
	UCL 2077 是癫痫相关 KCNQ 通道的亚型选择性阻滞剂，也是一种选择性慢后超极化通道阻滞剂，在培养的海马神经元中 IC50 为 500 nM，对 Ca2+ 通道、动作电位、输入电阻的影响小，以及超极化后的介质。
T15257	Etripamil MSP-2017,(-)-MSP-2017	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Etripamil (MSP-2017) 是一种短效L 型钙通道拮抗剂，可用于治疗阵发性室上性心动过速的研究。它通过抑制房室结细胞中钙慢通道的钙离子流入，显示房室结传导并延长房室结不应期
T13387L	Zatebradine hydrochloride UL-FS-49CL,UL-FS-49	Others; HCN Channel	Membrane transporter/Ion channel; Others
	Zatebradine hydrochloride (UL-FS-49CL) 是一种高效的、有效的HCN Channel 抑制剂( IC50 ：1.96 µM)。 HCN Channel 是一种有效的超极化激活环核苷酸门控通道。 Zatebradine hydrochloride 阻止通过人类 HCN1，HCN2，HCN3 和 HCN4 通道的缓慢内向电流，其 IC50 值分别为 1.83 µM，2.21 µM，1.90 µM 和 1.88 µM。
T1641	Strontium ranelate Distrontium renelate,S12911,雷尼酸锶	Calcium Channel; CaSR	GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
	Strontium ranelate (S12911) 是抗骨质疏松的药物，能够抑制骨吸收，促进骨形成，进而促使正骨平衡。它还能够激活非骨骼细胞中的钙敏感受体 (CaSR)，进而促进肌醇 1，4，5-三磷酸的生成及丝裂原活化的蛋白激酶信号转导。
T0866	Propafenone Rythmol,普罗帕酮,Propafenonum	Potassium Channel; MRP; Sodium Channel	Immunology/Inflammation; Membrane transporter/Ion channel
	Propafenone (Propafenonum) 是钠通道阻滞剂，它对 β 受体具有高亲和力 (IC50=32 nM)。它能够阻断瞬时外向钾电流 (Ito) (IC50: 4.9 nM) 和持续延迟整流器K+电流 (Isus) (IC50: 8.6 nM) ，具有抗心律失常的作用。它能够诱导线粒体功能障碍及诱导细胞凋亡，从而抑制食管癌增殖。
T6707	Tiotropium Bromide hydrate BA-679 BR hydrate,BA 679BR,噻托溴铵一水合物	AChR	Neuroscience
	Tiotropium Bromide hydrate (BA-679 BR hydrate) 是长效的毒蕈碱受体拮抗剂，可用于治疗慢性阻塞性气道疾病 (COPD)。
T22662	Chromanol 293B	Others	Others
	slow delayed rectifier K+ current (IKs) blocker
T71836	2-FPBA	Others	Others
	2-FPBA is a potent, reversible and slow-onset inhibitor of mandelate racemase (MR).
T35323	ZYZ-803 ZYZ 803	Others	Others
	ZYZ-803 is a slow H2S-NO-releasing hybrid, attenuating cardiac dysfunction after heart failure.
T28798	SL-25.1188 SL25.1188	Others	Others
	SL-25.1188 is a monoamine oxidase B (MAO-B) inhibitor. SL-25.1188 is characterized by reversible binding, high brain uptake, and very slow plasma metabolism in vivo.
T38730	Ara-F-NAD+	Others	Others
	Ara-F-NAD+, an arabino analogue of NAD + , is a potent, slow-binding CD38 NADase inhibitor, with a K i of 169 nM.
T23710	Watanidipine dihydrochloride	Others	Others
	Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.
T38456	Tribenuron	Others	Others
	Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.
T69375	Oxarbazole	Others	Others
	Oxarbazole is an antagonist of slow-reacting substance of anaphylaxis.
T37494	11-trans Leukotriene E4 11-trans Leukotriene E4	Others	Others
	Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans LTE4 is equipotent to LTE4 in contracting guinea pig ileum.
T34750	Sut 8701 Sut8701,Sut-8701	Others	Others
	Sut 8701 is a cholecystokinin analog that prevents cholinergic degeneration in the rat cerebral cortex following basal forebrain lesioning and can slow down the degenerative processes in Alzheimer's disease.
T24348	L 708286 L708286,L-708286,DFKi	Others	Others
	L 708286 is an agent of peptide-based phenethylcarbamoyldifluoromethylene. It is a slow-binding inhibitor of human leucocyte elastase (HLE).
T15285	FK706	Serine Protease	Proteases/Proteasome
	FK706 is a slow-binding and competitive human neutrophil elastase inhibitor (IC50: 83 nM; Ki: 4.2 nM). FK706 also inhibits mouse neutrophil elastase and porcine pancreatic elastase (IC50s: 22 nM and 100 nM, respectively). FK706 has an anti-inflammatory ef
T28392	Pfn1-IN-C1 Pfn1INC1,Pfn1 IN C1,Pfn1 inhibitor C1	Others	Others
	Pfn1-IN-C1, an inhibitor of Profilin1 (Pfn1), has been shown to reduce the overall level of cellular filamentous (F)-actin, slow EC migration and proliferation, and inhibit the angiogenic ability of EC both in vitro and ex vivo.
T28245	ONO-0300302 ONO 0300302	Others	Others
	ONO-0300302 is a slow tight binding LPA1 antagonist (IC50: 0.16 nM) used to treat Benign Prostatic Hyperplasia. ONO-0300302 inhibits significantly an LPA-induced increase of intraurethral pressure (IUP) in rat (3 mg/kg, p.o.) and dog (1 mg/kg, p.o.) over
T38050	CP-609754	Transferase	Metabolism
	CP-609754 是高效的、可逆的法尼基转移酶抑制剂，对重组人 H-Ras 和重组 K-Ras 法尼基化的 IC50分别为 0.57 ng/mL 和 46 ng/mL。CP-609754有潜在的抗癌作用。
T81586	Oxonol V
	Oxonol V是一种对测量细胞膜电位反应缓慢的敏感探针。

化合物

Cat.No: T12909

Target: Cysteine Protease, Parasite

Cat.No: T11831

Target: Others

Cat.No: T24421

Synonym: DB-7,LY2624803,HY-10275,LY 2624803

Target: 5-HT Receptor, Histamine Receptor

Cat.No: T24932

Synonym: AE-0047,AE 0047,AE0047

Target: Calcium Channel

Cat.No: T9597

Synonym: N-(苯甲酰基硫基)苯甲酰胺

Target: Endogenous Metabolite

Cat.No: T20206

Synonym: CSI Paste,1'3-双羟甲基脲,Carbamol,Caurite,Dimethylolurea

Target: Others

Cat.No: T70470L

Synonym: isomer-1542205-83-3

Target: MMP

Cat.No: T28748

Synonym: RG14202,DTI0009,DTI-0009,RG-14202,DT-009,DT009

Target: Adenosine Receptor

Cat.No: T25372

Synonym: EMD-57033,(+)-EMD 57033,EMD 57033

Target: Calcium Channel, Carbonic Anhydrase

FFAGLDD amine salt

Cat.No: TP1545L1

Target: Others

Cat.No: T11805

Target: NOS

β-Pompilidotoxin Acetate

Cat.No: T21769L

Synonym: β-Pompilidotoxin Acetate(216064-36-7 Free base)

Target: Sodium Channel

Bisaramil hydrochloride

Cat.No: T26822

Synonym: RGH-2957,NK 1556,NK1556,Bisaramil,NK-1556,RGH 2957

Target: Potassium Channel, Adrenergic Receptor

Cat.No: T30188L

Synonym: PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base）

Target: Calcium Channel

Cat.No: T22830

Synonym: GYY 4137 morpholine salt

Target: Others

Cat.No: T0377

Synonym: NSC-141046,氯法齐明,氯苯吩嗪

Target: DNA, Antibacterial, Antibiotic

Cat.No: T7502L

Synonym: PF-05089771,PF05089771

Target: Sodium Channel

Pimelic diphenylamide 106

Cat.No: T3193

Synonym: Histone Deacetylase Inhibitor VII,TC-H 106,RGFA-8

Target: HDAC

Cat.No: T15673

Synonym: KU-59403,KU59403

Target: ATM/ATR

Cat.No: T0029

Synonym: Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因

Target: Histone Demethylase, DNA/RNA Synthesis, Sodium Channel

Cat.No: T1439

Synonym: SN-305,拉西地平,GX-1048,GR-43659X

Target: Apoptosis, Calcium Channel, Reactive Oxygen Species

Cat.No: T40870

Synonym: LTE4

Target: Endogenous Metabolite

Cat.No: T5117

Target: Others

Cat.No: T61111

Target: TNF

Cat.No: T24415

Synonym: Privaprol,L-12717,DL 717-IT,L 12717,L12717,Canocenta

Target: Others

Cat.No: T4440

Target: GABA Receptor

Ibutilide Fumarate

Cat.No: T6541

Synonym: Corvert Fumarate,U70226E,富马酸伊布利特

Target: Calcium Channel, Sodium Channel

PF-06424439 methanesulfonate

Cat.No: T12425

Target: Acyltransferase, Transferase

Cat.No: T17197

Target: Others

Cat.No: T15257

Synonym: MSP-2017,(-)-MSP-2017

Target: Calcium Channel

Zatebradine hydrochloride

Cat.No: T13387L

Synonym: UL-FS-49CL,UL-FS-49

Target: Others, HCN Channel

Strontium ranelate

Cat.No: T1641

Synonym: Distrontium renelate,S12911,雷尼酸锶

Target: Calcium Channel, CaSR

Cat.No: T0866

Synonym: Rythmol,普罗帕酮,Propafenonum

Target: Potassium Channel, MRP, Sodium Channel

Tiotropium Bromide hydrate

Cat.No: T6707

Synonym: BA-679 BR hydrate,BA 679BR,噻托溴铵一水合物

Target: AChR

Cat.No: T22662

Target: Others

Cat.No: T71836

Target: Others

Cat.No: T35323

Synonym: ZYZ 803

Target: Others

Cat.No: T28798

Synonym: SL25.1188

Target: Others

Cat.No: T38730

Target: Others

Watanidipine dihydrochloride

Cat.No: T23710

Target: Others

Cat.No: T38456

Target: Others

Cat.No: T69375

Target: Others

11-trans Leukotriene E4

Cat.No: T37494

Synonym: 11-trans Leukotriene E4

Target: Others

Cat.No: T34750

Synonym: Sut8701,Sut-8701

Target: Others

Cat.No: T24348

Synonym: L708286,L-708286,DFKi

Target: Others

Cat.No: T15285

Target: Serine Protease

Cat.No: T28392

Synonym: Pfn1INC1,Pfn1 IN C1,Pfn1 inhibitor C1

Target: Others

Cat.No: T28245

Synonym: ONO 0300302

Target: Others

Cat.No: T38050

Target: Transferase

Cat.No: T81586

Cat. No.	Product Name	Target	Signaling Pathways
T8195	Lotusine	Others	Others
	Lotusine 是一种提取自Nelumbo nucifera Gaertn 的绿色种胚中的纯生物碱。它能够作用于心肌中动作电位及心脏浦肯野纤维缓慢内向电流。
TMS2182	trans-Zeatinriboside Ribosylzeatin,Zeatin Riboside,Trans-Zeatin Riboside,玉米素核苷	Others	Others
	trans-Zeatinriboside (Ribosylzeatin) 是一种细胞分裂素前体，是木质素导管中主要的长距离信号形式，能够调节叶片大小和分生组织活性相关形状。
T3606	γ-Oryzanol 谷维素,Gamma-Oryzanol,Oliver,γ-谷维素,Gammariza	DNA Methyltransferase	Chromatin/Epigenetic
	γ-Oryzanol (Gamma-Oryzanol) 是一种从米糠油中分离出来的营养提取物，是含有甾醇和阿魏酸的混合物，有助于破坏皮肤中的自由基。它有效抑制小鼠纹状体中的 DNA 甲基转移酶(DNMTs)。它抑制DNMT1和DNMT3a，IC50分别为 3.2 和 22.3 μM。
T1591	Ancitabine hydrochloride NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C	Others; DNA/RNA Synthesis; Autophagy	Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
	Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
TN4368	Kaempferol-3,7-di-O-β-glucoside Kaempferol 3,7-di-O-glucoside	Glucosidase; Amylase	Metabolism
	Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) 是一种来自 Morettia philaena 的黄酮醇，对 α-淀粉酶 (α-amylase)、α-葡萄糖苷酶 (α-glucosidase) 和乙酰胆碱酯酶 (Acetylcholinesterase) 具有抑制作用。Kaempferol-3,7-di-O-β-glucoside 具有神经保护活性，可减缓分化神经元细胞 SH-SY5Y 免受 Amyloid β 肽诱导的损伤。Kaempferol-3,7-di-O-β-glucoside 可用于研究阿尔茨海默氏症类的神经系统疾病。
TN3540	Broussonin C	Tyrosinase; Antifection	Microbiology/Virology; Proteases/Proteasome
	Broussonin C and broussin are antifungal compounds. Broussonin C exerts simple reversible slow-binding inhibition against diphenolase.
T78489	Lotusine hydroxide	Others	Others
	Lotusine (hydroxide)为纯生物碱，源自Nelumbo nucifera Gaertn绿色种胚提取。该化合物能够影响心肌动作电位和心脏浦肯野纤维的缓慢内向电流。

天然产物

Cat.No: T8195

Target: Others

trans-Zeatinriboside

Cat.No: TMS2182

Synonym: Ribosylzeatin,Zeatin Riboside,Trans-Zeatin Riboside,玉米素核苷

Target: Others

Cat.No: T3606

Synonym: 谷维素,Gamma-Oryzanol,Oliver,γ-谷维素,Gammariza

Target: DNA Methyltransferase

Ancitabine hydrochloride

Cat.No: T1591

Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Target: Others, DNA/RNA Synthesis, Autophagy

Kaempferol-3,7-di-O-β-glucoside

Cat.No: TN4368

Synonym: Kaempferol 3,7-di-O-glucoside

Target: Glucosidase, Amylase

Cat.No: TN3540

Target: Tyrosinase, Antifection

Lotusine hydroxide

Cat.No: T78489

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-02956	TNNI1 Protein, Mouse, Recombinant (Flag & His & Myc) Troponin I, slow skeletal muscle,Tnni1,Troponin I, ...	Mouse	E. coli
	Troponin I is the inhibitory subunit of troponin, the thin filament regulatory complex which confers calcium-sensitivity to striated muscle actomyosin ATPase activity. TNNI1 Protein, Mouse, Recombinant (Flag & His & Myc) is expressed in E. coli expression system with N-10xHis-Flag and C-Myc tag. The predicted molecular weight is 29.6 kDa and the accession number is Q9WUZ5.
TMPY-03957	Troponin C Protein, Human, Recombinant TN-C,CMD1Z,TNNC,TNC,CMH13,troponin C type 1 (slow)	Human	E. coli
	Troponin I, also known as TNNC1, is part of the troponin complex. This complex contains 3 subunits: troponin I (TnI), troponin T (TnT) and troponin C (TnC). Troponin I is the inhibitory subunit, blocking actin-myosin interactions and thereby mediating striated muscle relaxation. It binds to actin in thin myofilaments to hold the actin-tropomyosin complex in place. Because of it myosin cannot bind actin in relaxed muscle. When calcium binds to the Troponin C it causes conformational changes which...
TMPH-01725	MYL3 Protein, Human, Recombinant (GST) Ventricular myosin alkali light chain,Ventricular/slow	Human	E. coli
	Regulatory light chain of myosin. Does not bind calcium. MYL3 Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 48.8 kDa and the accession number is P08590.
TMPY-02219	Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His) NS1 Protein	H1N1	E. coli
	The NS1 Influenza protein is created by the internal protein-encoding, linear negative-sense, single-stranded RNA, NS gene segment and which also codes for the nuclear export protein or NEP, formerly referred to as the NS2 protein, which mediates the export of vRNPs. The non-structural (NS1) protein is found in Influenzavirus A, Influenzavirus B, and Influenzavirus C. The non-structural (NS1) protein of the highly pathogenic avian H5N1 viruses circulating in poultry and waterfowl in Southeast As...
TMPH-03070	TAP Protein, Ornithodoros moubata, Recombinant (His) Tick anticoagulant peptide	Ornithodoros moubata	P. pastoris (Yeast)
	TAP is a slow, tight-binding inhibitor of blood coagulation, specific for factor Xa.
TMPH-03071	TAP Protein, Ornithodoros moubata, Recombinant (His & Myc & SUMO) Tick anticoagulant peptide	Ornithodoros moubata	E. coli
	TAP is a slow, tight-binding inhibitor of blood coagulation, specific for factor Xa.
TMPH-00782	OMP P5 Protein, Haemophilus influenzae, Recombinant (His & Myc & SUMO) Outer membrane porin A,Outer membrane protein P5,Outer membr...	Haemophilus influenzae	E. coli
	Acts as a fimbriae subunit, allowing adhesion to host cells.; With TolR probably plays a role in maintaining the position of the peptidoglycan cell wall in the periplasm. Acts as a porin with low permeability that allows slow penetration of small solutes; an internal gate slows down solute passage.
TMPH-02377	OmpA Protein, Klebsiella pneumoniae, Recombinant (His & Myc) Outer membrane protein 3A,Outer membrane protein A,ompA,Oute...	Klebsiella pneumoniae	E. coli
	With TolR probably plays a role in maintaining the position of the peptidoglycan cell wall in the periplasm. Acts as a porin with low permeability that allows slow penetration of small solutes; an internal gate slows down solute passage.; Required for conjugation with F-type plasmids; probably serves as the mating receptor on recipient cells.
TMPH-03472	OmpA Protein, Salmonella typhi, Recombinant (His) Outer membrane porin A,Outer membrane protein A,ompA	Salmonella typhi	E. coli
	With TolR probably plays a role in maintaining the position of the peptidoglycan cell wall in the periplasm. Acts as a porin with low permeability that allows slow penetration of small solutes; an internal gate slows down solute passage.; Required for conjugation with F-type plasmids; probably serves as the mating receptor on recipient cells. OmpA Protein, Salmonella typhi, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 38.9 kDa an...
TMPY-03603	AHSP Protein, Human, Recombinant ERAF,alpha hemoglobin stabilizing protein,α hemoglobin stabi...	Human	E. coli
	AHSP, also known as ERAF, is a conserved mammalian erythroid protein which belongs to the AHSP family. It is expressed in blood and bone marrow. AHSP facilitates the production of Hemoglobin A by stabilizing free α-globin. It rapidly binds to ferrous α with association (k'(AHSP)) and dissociation (k(AHSP)) rate constants of ≈1 μm(-1) s(-1) and .2 s(-1), respectively, at pH 7.4 at 22 ℃. A small slow phase was observed when AHSP binds to excess ferrous αCO. This slow phase appears to be due to cis...
TMPH-00674	OmpA Protein, E. coli O157:H7, Recombinant (His & SUMO) ompA,Outer membrane protein A,Outer membrane porin A	E. coli	E. coli
	With TolR probably plays a role in maintaining the position of the peptidoglycan cell wall in the periplasm. Acts as a porin with low permeability that allows slow penetration of small solutes; an internal gate slows down solute passage.; Required for conjugation with F-type plasmids; probably serves as the mating receptor on recipient cells. OmpA Protein, E. coli O157:H7, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is ...
TMPH-00056	Delta-AITX-Avd1c Protein, Anemonia sulcata, Recombinant (His) ATX II,Delta-AITX-Avd1c,Toxin II,Delta-actitoxin-Avd1c,Neuro...	Anemonia sulcata	P. pastoris (Yeast)
	Binds specifically to voltage-gated sodium channels (Nav) (site 3), thereby delaying their inactivation. Has a strong effect on crustaceans and insects (DmNav1) and a weaker effect on mammals. This toxin is highly potent at mammalian Nav1.1/SCN1A (EC(50)=6.01 nM) and Nav1.2/SCN2A (EC(50)=7.88 nM). It has also great activity on Nav1.5/SCN5A (EC(50)=49.05 nM), Nav1.4/SCN4A (EC(50)=109.49 nM) and Nav1.6/SCN8A (EC(50)=about 180 nM) and is less potent on Nav1.3/SCN3A (EC(50)=759.22 nM) (when measured...
TMPY-01479	SPG3A Protein, Human, Recombinant (GST) HSN1D,atlastin GTPase 1,FSP1,atlastin1,GBP3,SPG3,SPG3A,AD-FS...	Human	Baculovirus Insect Cells
	Atlastin-1, also known as Spastic paraplegia 3 protein A, Guanine nucleotide-binding protein 3, GTP-binding protein 3, GBP3, ATL1 and SPG3A, is a multi-pass membrane protein which belongs to theGBP family and atlastin subfamily. ATL1 / SPG3A is expressed predominantly in the adult and fetal central nervous system. Expression of ATL1 / SPG3A in adult brain is at least 5-fold higher than in other tissues. ATL1 / SPG3A is detected predominantly in pyramidal neurons in the cerebral cortex and...

重组蛋白

TNNI1 Protein, Mouse, Recombinant (Flag & His & Myc)

Cat.No: TMPH-02956

Species: Mouse

Expression System: E. coli

Troponin C Protein, Human, Recombinant

Cat.No: TMPY-03957

Species: Human

Expression System: E. coli

MYL3 Protein, Human, Recombinant (GST)

Cat.No: TMPH-01725

Species: Human

Expression System: E. coli

Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His)

Cat.No: TMPY-02219

Species: H1N1

Expression System: E. coli

TAP Protein, Ornithodoros moubata, Recombinant (His)

Cat.No: TMPH-03070

Species: Ornithodoros moubata

Expression System: P. pastoris (Yeast)

TAP Protein, Ornithodoros moubata, Recombinant (His & Myc & SUMO)

Cat.No: TMPH-03071

Species: Ornithodoros moubata

Expression System: E. coli

OMP P5 Protein, Haemophilus influenzae, Recombinant (His & Myc & SUMO)

Cat.No: TMPH-00782

Species: Haemophilus influenzae

Expression System: E. coli

OmpA Protein, Klebsiella pneumoniae, Recombinant (His & Myc)

Cat.No: TMPH-02377

Species: Klebsiella pneumoniae

Expression System: E. coli

OmpA Protein, Salmonella typhi, Recombinant (His)

Cat.No: TMPH-03472

Species: Salmonella typhi

Expression System: E. coli

AHSP Protein, Human, Recombinant

Cat.No: TMPY-03603

Species: Human

Expression System: E. coli

OmpA Protein, E. coli O157:H7, Recombinant (His & SUMO)

Cat.No: TMPH-00674

Species: E. coli

Expression System: E. coli

Delta-AITX-Avd1c Protein, Anemonia sulcata, Recombinant (His)

Cat.No: TMPH-00056

Species: Anemonia sulcata

Expression System: P. pastoris (Yeast)

SPG3A Protein, Human, Recombinant (GST)

Cat.No: TMPY-01479

Species: Human

Expression System: Baculovirus Insect Cells

Cat. No.	Product Name	Target	Signaling Pathways
TMIJ-0497	Lacidipine-d10
	Lacidipine-d10 是 Lacidipine 的氘代化合物。Lacidipine 的 CAS 号为 103890-78-4。Lacidipine 是一种L型钙离子通道阻断剂。
TMIJ-0240	Lacosamide-d3 (Acetyl-d3)
	Lacosamide-d3 (Acetyl-d3) 是 Lacosamide 的氘代化合物。Lacosamide 的 CAS 号为 175481-36-4。Lacosamide是一种功能化氨基酸。Lacosamide以一种新的方式调节钠通道：它选择性地增强钠通道缓慢失活，而对快速失活没有影响Lacosamine在不同的啮齿类动物癫痫发作模型中显示出抗癫痫作用，在反映神经性疼痛和慢性炎性疼痛的不同类型和症状的实验动物模型中显示了抗伤害潜力。
TMID-0247	LacosaMide-d3
	LacosaMide-d3 是 LacosaMide 的氘代化合物。LacosaMide 的 CAS 号为 175481-36-4。Lacosamide是一种功能化氨基酸。Lacosamide以一种新的方式调节钠通道：它选择性地增强钠通道缓慢失活，而对快速失活没有影响Lacosamine在不同的啮齿类动物癫痫发作模型中显示出抗癫痫作用，在反映神经性疼痛和慢性炎性疼痛的不同类型和症状的实验动物模型中显示了抗伤害潜力。

同位素标记化合物

Cat.No: TMIJ-0497

Lacosamide-d3 (Acetyl-d3)

Cat.No: TMIJ-0240

Cat.No: TMID-0247

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