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Search Results for " first-generation "

Targets Recommended: Antibacterial Antibiotic

51

抑制剂 & 化合物

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天然产物

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化合物库

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重组蛋白

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同位素标记化合物

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Cat. No.	Product Name
L9410	共价抑制剂库		1920 compounds
	1920 种小分子的独特集合，包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子，如氯乙酰基，2-氯丙酰基，丙烯酰基，1-丙-2-炔基，1-丁-2-炔基，酮羰基，二硫键等，可以用于共价抑制剂药物研发；

化合物库

共价抑制剂库

Cat.No: L9410

Compounds: 1920

Cat. No.	Product Name	Target	Signaling Pathways
T8134	Cefathiamidine	Antibacterial; Antibiotic	Microbiology/Virology
	Cefathiamidine 是一种头孢菌素抗菌剂，可研究由易感细菌引起的感染，还可用于呼吸道、肝脏、五官感觉、尿路感染以及心内膜炎和败血症的研究。
T8345	Carbutamide	Others	Others
	Carbutamide 是一代磺酰脲，口服具有活性，具有降血糖作用。
T6451	Clodronic acid disodium salt Loron,Clodronate Disodium,氯屈膦酸二钠,Lodronate	Others	Others
	Clodronic acid disodium salt (Lodronate) 是一种口服具有活力的破骨细胞骨吸收 (osteoclastic bone resorption) 的抑制剂，是一代双磷酸盐。它可用于高骨转换状态、Paget’s 病和溶骨性骨转移中。
T0370	Pheniramine maleate Daneral,Inhiston,Trimetose,马来酸非尼拉敏	5-HT Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Pheniramine maleate (Trimetose) 是一种具有抗组胺和血管扩张特性的烷基胺衍生物，可与组胺 H1 受体结合，从而抑制磷脂酶 A2 和内皮源性松弛因子一氧化氮的产生。
T0141	Cephalonium 头孢洛宁,Cefalonium	Others	Others
	Cephalonium (Cefalonium) 是第一代头孢菌素类抗生素。
T0141L	Cefalonium Dihydrate(5575-21-3 free base) Cefalonium Dihydrate	Others	Others
	Cefalonium Dihydrate(5575-21-3 free base) 是第一代头孢菌素类抗生素。
T0371	Gliquidone AR-DF 26,格列喹酮,Glurenorm	Potassium Channel	Membrane transporter/Ion channel
	Gliquidone (AR-DF 26) 是一种磺酰脲类的抗糖尿病药物，可用于2型糖尿病的研究。
T9225	Vebicorvir ABI-H0731	HBV	Microbiology/Virology
	Vebicorvir (ABI-H0731) 是一种乙型肝炎病毒核心蛋白的抑制剂，有抗病毒活性。
T8457	NPS2390	GluR	Neuroscience
	NPS2390 是钙敏感受体抑制剂，也是 mGluR1 和 mGluR5 的非竞争性拮抗剂。
T0092	Antazoline hydrochloride 盐酸安他唑啉,Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Antazoline hydrochloride (Phenazoline hydrochloride) 是一种抗组胺药，可与组胺H1受体结合，阻断内源性组胺的作用。它也具有抗胆碱能特性，可缓解鼻塞，也可用作眼药水。
T21419	Diphenhydramine 苯海拉明,Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Diphenhydramine (Syntedril) 是第一代具有抗胆碱能作用的H1 受体拮抗剂，它能透过血脑屏障。
T0199	Cephradine Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定	TOPK; Antibacterial; Antibiotic	MAPK; Microbiology/Virology
	Cephradine (Anspor) 是广谱口服活性头孢菌素。它对革兰氏阳性和革兰氏阴性病原体都有活性。它已用于泌尿生殖系统、胃肠道和呼吸道感染以及皮肤和软组织感染的研究。它通过直接抑制TOPK 抑制太阳紫外线诱导的皮肤炎症。
T7941	Imipramine hydrochloride 盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine	Serotonin Transporter	Neuroscience
	Imipramine hydrochloride (Imipramine HCl) 可抑制血清素转运蛋白，IC50=32 nM。它可阻止胰酶的易位，阻碍 MV 和外泌体的分泌。
T0445L	Promethazine hydrochloride 盐酸异丙嗪,Promethazine HCl,Phenergan	Adrenergic Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Promethazine hydrochloride (Promethazine HCl) 是抗组胺药物，是 H1 受体的强拮抗剂和 mACh 受体的中度拮抗剂，对 5-HT2A、5-HT2C、D2 和 α1-肾上腺素能受体具有中等亲和力。
T0059	Diphenylpyraline hydrochloride 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂，抑制多巴胺的吸收。它是可口服的抗组胺试剂，具有抗胆碱和抗过敏作用，可用于缓解过敏性疾病，如鼻炎、花粉热和瘙痒性皮肤疾病等。
T2551	Etravirine TMC125,依曲韦林,R165335	HIV Protease; Reverse Transcriptase	Microbiology/Virology; Proteases/Proteasome
	Etravirine (R165335) 是一种非核苷逆转录酶抑制剂，具有抗 HIV 的作用。
T16472	Pericyazine Propericiazine,氰噻嗪,RP 8909	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Pericyazine (Propericiazine) 是第一代抗精神病药物，是一种选择性的 D2 多巴胺受体 (D2-dopamine receptor) 拮抗剂，具有肾上腺溶解、抗胆碱能和锥体外系作用，被用作短期管理严重焦虑状态和精神病的辅助药物。
T21390	Fexofenadine Carboxyterfenadine,Telfast,非索非那定,MDL 16.455,Allegra	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Fexofenadine (Carboxyterfenadine) 是一种抗组胺药物，用于治疗过敏症状，如鼻塞、花粉热和荨麻疹。与第一代抗组胺药相比，它通过血脑屏障并引起镇静的能力较差。
T0816	Acetohexamide Acetohexamid,醋磺环已脲,Dymelor,醋磺己脲,Gamadiabet	Potassium Channel; NADPH	Membrane transporter/Ion channel; Metabolism
	Acetohexamide (Acetohexamid) 是磺脲类试剂，可刺激胰腺分泌胰岛素，能够用于 2 型糖尿病的相关研究。
T0953	Cefazolin sodium Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Cefazolin sodium (cephazolin sodium) salt 是一种头孢类抗生素, 可研究多种细菌感染。
T1122	Cephalothin sodium 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin	Antibacterial; Antibiotic	Microbiology/Virology
	Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性，抑制革兰氏阳性和阴性菌。
T0373	Erlotinib OSI-744,NSC 718781,CP358774,埃罗替尼,R1415	EGFR; Autophagy	Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Erlotinib (CP358774) 是一种 EGFR 一代抑制剂，抑制 EGFR 19 Del 和 L858R 突变。Erlotinib 具有抗肿瘤活性，用于治疗 EGFR 突变的非小细胞肺癌。Erlotinib 用药会产生 EGFR C797S 耐药突变。
T68967	AFG206	Others	Others
	AFG206 is the novel first-generation type II" FLT3 inhibitor."
T0059L	Diphenylpyraline Difenilpiralina,AN 1041,AN1041,Dayfen,AN-1041,二苯拉林	Others	Others
	Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.
T33319	Methdilazine Hydrochloride Bristaline,Dilosyn,Methdilazine Hcl,Tacaryl hydrochloride,Disyncran	Others	Others
	Methdilazine Hydrochloride is a first-generation phenothiazine class antihistamine with anticholinergic properties.
T14929	Cephradine monohydrate 头孢拉定一水合物,Cefradine monohydrate	Antibacterial	Microbiology/Virology
	Cephradine monohydrate, a first-generation cephalosporin, is active against a wide range of Gram-positive and Gram-negative bacteria.
T0445L1	Promethazine hibenzate D-08768,D08768,D 08768	Others	Others
	Promethazine is a neuroleptic medication and first-generation antihistamine of the phenothiazine family.
T32233	Isothipendyl Udantol,Isothipendylum,Odantol,Andanton,Nilergex	Others	Others
	Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.
T20616	Coumachlor G-23133,Ratilan,G23133,Tomorin,G 23133	Others	Others
	Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.
T70308	PLX7683	Others	Others
	PLX7683 is a paradox breaker. Paradox breakers overcame several known mechanisms of resistance to first-generation RAF inhibitors. Dissociating MAPK pathway inhibition from paradoxical activation might yield both improved safety and more durable efficacy than first-generation RAF inhibitors
T69702	AFG210	Others	Others
	AFG210 is a novel first-generation “type II” FLT3 inhibitor.
T71117	AZD5248	Others	Others
	AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).
T38918	Revusiran ALN-TTRSC	Others	Others
	Revusiran (ALN-TTRSC) is a first-generation short interfering RNA (siRNA) that specifically targets transthyretin (TTR) mRNA. It is utilized in TTR-mediated amyloidosis research.
T40591	Verapamil EP Impurity C hydrochloride NSC-609249 hydrochloride	Others	Others
	NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.
T38972	Cefalonium hydrate	Others	Others
	Cefalonium hydrate is a first-generation β-lactam cephalosporin antibiotic commonly employed in the study of bovine mastitis induced by Gram-positive bacteria, particularly staphylococci. It demonstrates significant effectiveness in this research area.
T32700	Levocabastine Livostin,Bilina	Others	Others
	Levocarbastine is a second-generation H1 receptor antagonist for allergic conjunctivitis. It also acts as a potent selective antagonist for the neurotensin receptor NTS2 and is the first drug to be used to characterize different neurotensin subtypes.
T14040	4-Hydroxytolbutamide Hydroxytolbutamide	Potassium Channel	Membrane transporter/Ion channel
	4-Hydroxytolbutamide(Hydroxytolbutamide), a metabolite of Tolbutamide, which is metabolized by CYP2C8 and CYP2C9. Tolbutamide is a first generation potassium channel blocker and a sulfonylurea oral antidiabetic[1][2].
T19979	Saccharin sodium hydrate O-benzoic sulfimide sodium salt,糖精钠,Saccharin, sodium salt hydrate	Others	Others
	Saccharin, sodium salt hydrate is used in the food industry and for sweetening diabetes diet. It is also used as a synthetic sweet ignorance agent. Saccharin, sodium salt hydrate is the first generation′ synthetic sugar alternative that has been studied f
T19678	Cefaloridine Cephaloridine,Sch 11527	Others	Others
	Cefaloridine is a first-generation semisynthetic derivative of cephalosporin C. It is unique among cephalosporins in that it exists as a zwitterion. Cephaloridine was very effective to cure pneumococcal pneumonia. It has a high clinical and bacteriologica
T36211	16(R)-Iloprost	Others	Others
	Iloprost is a second generation structural analog of prostacyclin (PGI2) with about ten-fold greater potency than the first generation stable analogs, typified by carbaprostacyclin. Iloprost binds with equal affinity to the recombinant human IP and EP1 receptors with a Ki value of 11 nM. Most preparations of iloprost contain 16(S) and 16(R) stereoisomers. 16(R)-Iloprost inhibits platelet aggregation with an IC50 value of 65 nM.
T36212	16(S)-Iloprost	Others	Others
	Iloprost is a second generation structural analog of prostacyclin (PGI2) with about ten-fold greater potency than the first generation stable analogs, typified by carbaprostacyclin. Iloprost binds with equal affinity to the recombinant human IP and EP1 receptors with a Ki value of 11 nM. Most preparations of iloprost contain 16(S) and 16(R) stereoisomers. 16(S)-Iloprost potently inhibits platelet aggregation with an IC50 value of 3.5 nM.
TP2288	Rapalink-1	Others	Others
	RapaLink-1 is the third-generation mTOR inhibitor exploiting the unique juxtaposition of two drugs (first- and second-generation mTOR kinase inhibitors) -binding pockets to create a bivalent interaction that allows inhibition of the mutants which has resi
T71577	KOS-1584	Others	Others
	KOS-1584 is a second-generation epothilone with potential antineoplastic activity. Epothilone KOS-1584 binds to tubulin and induces microtubule polymerization and stabilizes microtubules against depolymerization, which may result in the inhibition of cell division, the induction of G2/M arrest, and apoptosis. Compared to first-generation epothilones, this agent exhibits greater safety and efficacy with an enhanced pharmaceutical profile, including enhanced water solubility and tumor penetration,...
T75300	Cefazolin sodium pentahydrate	Others	Others
	Cefazolin sodium pentahydrate 是一代头孢菌素类抗生素，可用于多种细菌感染的研究。Cefazolin sodium pentahydrate 具有抗炎作用，可以减轻术后认知功能障碍 (POCD)。
T35619	Dapagliflozin-3-O-β-D-Glucuronide	Others	Others
	Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin . Dapagliflozin is a first generation selective sodium glucose cotransporter (SGLT) 2 inhibitor that blocks glucose transport.[1] Dapagliflozin is metabolized by uridine diphosphate glucuronosyltransferase (UGT) 1A9 to dapagliflozin-3-O-β-D-glucuronide, which is 2,600-fold less potent than the parent compound with regard to SGLT2 inhibition.[2]
T0366L	Cefadroxil (hydrate)	Others	Others
	Cefadroxil is a first generation aminocephalosporin with good patient compliance, a long-acting therapeutic effect, high solubility and relatively broad spectrum of anti-bacterial activity. Cefadroxil is also a substrate of the intestinal peptide transporter PepT1, which is primarily responsible for the drug's uptake across the apical membrane of small intestine.
T71110	Nanatinostat TFA	Others	Others
	Nanatinostat, also known as Tractinostat, CHR-3996 and VRx-3996, is an orally bioavailable, second-generation hydroxamic acid-based inhibitor of histone deacetylase (HDAC) with potential antineoplastic activity. HDAC inhibitor CHR-3996 inhibits HDAC, resulting in an accumulation of highly acetylated histones, the induction of chromatin remodeling, and the selective transcription of tumor suppressor genes; these events may result in the inhibition of tumor cell division and the induction of tumor...
T69925	NVR3-778 hydrate	Others	Others
	NVR 3-778 is the first capsid assembly modulator (CAM) that has demonstrated antiviral activity in hepatitis B virus (HBV)-infected patients. NVR 3-778 inhibited the generation of infectious HBV DNA-containing virus particles with a mean antiviral 50% effective concentration (EC50) of 0.40 µM in HepG2.2.15 cells. The antiviral profile of NVR 3-778 indicates pan-genotypic antiviral activity and a lack of cross-resistance with nucleos(t)ide inhibitors of HBV replication.
T70287	BMS-186511	Others	Others
	BMS-186511 is a Farnesyltransferase (FT) inhibitor with potential anticancer activity. BMS-186511 is a bisubstrate analogue inhibitor of FT, would inhibit the malignant growth properties of a cell line established from malignant schwannoma of an NF1 patient. Following treatment with BMS-186511 , ST88-14 cells became flat, nonrefractile, were contact-inhibited, and lost their ability to grow in soft agar. BMS-186511 was found to specifically inhibit FT, but not geranylgeranyltransferase I, a clos...
T36175	AAPH	Others	Others
	AAPH is a water-soluble azo compound which is used extensively as a free radical generator, often in the study of lipid peroxidation and the characterization of antioxidants.[1],[2],[3],[4] Decomposition of AAPH produces molecular nitrogen and 2 carbon radicals. The carbon radicals may combine to produce stable products or react with molecular oxygen to give peroxyl radicals. The half-life of AAPH is about 175 hours (37°C at neutral pH), making the rate of free radical generation essentially con...

化合物

Cat.No: T8134

Target: Antibacterial, Antibiotic

Cat.No: T8345

Target: Others

Clodronic acid disodium salt

Cat.No: T6451

Synonym: Loron,Clodronate Disodium,氯屈膦酸二钠,Lodronate

Target: Others

Pheniramine maleate

Cat.No: T0370

Synonym: Daneral,Inhiston,Trimetose,马来酸非尼拉敏

Target: 5-HT Receptor, Histamine Receptor

Cat.No: T0141

Synonym: 头孢洛宁,Cefalonium

Target: Others

Cefalonium Dihydrate(5575-21-3 free base)

Cat.No: T0141L

Synonym: Cefalonium Dihydrate

Target: Others

Cat.No: T0371

Synonym: AR-DF 26,格列喹酮,Glurenorm

Target: Potassium Channel

Cat.No: T9225

Synonym: ABI-H0731

Target: HBV

Cat.No: T8457

Target: GluR

Antazoline hydrochloride

Cat.No: T0092

Synonym: 盐酸安他唑啉,Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl

Target: Histamine Receptor

Diphenhydramine

Cat.No: T21419

Synonym: 苯海拉明,Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255

Target: Histamine Receptor

Cat.No: T0199

Synonym: Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定

Target: TOPK, Antibacterial, Antibiotic

Imipramine hydrochloride

Cat.No: T7941

Synonym: 盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine

Target: Serotonin Transporter

Promethazine hydrochloride

Cat.No: T0445L

Synonym: 盐酸异丙嗪,Promethazine HCl,Phenergan

Target: Adrenergic Receptor, Histamine Receptor

Diphenylpyraline hydrochloride

Cat.No: T0059

Synonym: 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride

Target: Histamine Receptor

Cat.No: T2551

Synonym: TMC125,依曲韦林,R165335

Target: HIV Protease, Reverse Transcriptase

Cat.No: T16472

Synonym: Propericiazine,氰噻嗪,RP 8909

Target: Dopamine Receptor

Cat.No: T21390

Synonym: Carboxyterfenadine,Telfast,非索非那定,MDL 16.455,Allegra

Target: Histamine Receptor

Cat.No: T0816

Synonym: Acetohexamid,醋磺环已脲,Dymelor,醋磺己脲,Gamadiabet

Target: Potassium Channel, NADPH

Cefazolin sodium

Cat.No: T0953

Synonym: Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin

Target: Others, Antibacterial, Antibiotic

Cephalothin sodium

Cat.No: T1122

Synonym: 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin

Target: Antibacterial, Antibiotic

Cat.No: T0373

Synonym: OSI-744,NSC 718781,CP358774,埃罗替尼,R1415

Target: EGFR, Autophagy

Cat.No: T68967

Target: Others

Diphenylpyraline

Cat.No: T0059L

Synonym: Difenilpiralina,AN 1041,AN1041,Dayfen,AN-1041,二苯拉林

Target: Others

Methdilazine Hydrochloride

Cat.No: T33319

Synonym: Bristaline,Dilosyn,Methdilazine Hcl,Tacaryl hydrochloride,Disyncran

Target: Others

Cephradine monohydrate

Cat.No: T14929

Synonym: 头孢拉定一水合物,Cefradine monohydrate

Target: Antibacterial

Promethazine hibenzate

Cat.No: T0445L1

Synonym: D-08768,D08768,D 08768

Target: Others

Cat.No: T32233

Synonym: Udantol,Isothipendylum,Odantol,Andanton,Nilergex

Target: Others

Cat.No: T20616

Synonym: G-23133,Ratilan,G23133,Tomorin,G 23133

Target: Others

Cat.No: T70308

Target: Others

Cat.No: T69702

Target: Others

Cat.No: T71117

Target: Others

Cat.No: T38918

Synonym: ALN-TTRSC

Target: Others

Verapamil EP Impurity C hydrochloride

Cat.No: T40591

Synonym: NSC-609249 hydrochloride

Target: Others

Cefalonium hydrate

Cat.No: T38972

Target: Others

Cat.No: T32700

Synonym: Livostin,Bilina

Target: Others

4-Hydroxytolbutamide

Cat.No: T14040

Synonym: Hydroxytolbutamide

Target: Potassium Channel

Saccharin sodium hydrate

Cat.No: T19979

Synonym: O-benzoic sulfimide sodium salt,糖精钠,Saccharin, sodium salt hydrate

Target: Others

Cat.No: T19678

Synonym: Cephaloridine,Sch 11527

Target: Others

Cat.No: T36211

Target: Others

Cat.No: T36212

Target: Others

Cat.No: TP2288

Target: Others

Cat.No: T71577

Target: Others

Cefazolin sodium pentahydrate

Cat.No: T75300

Target: Others

Dapagliflozin-3-O-β-D-Glucuronide

Cat.No: T35619

Target: Others

Cefadroxil (hydrate)

Cat.No: T0366L

Target: Others

Nanatinostat TFA

Cat.No: T71110

Target: Others

NVR3-778 hydrate

Cat.No: T69925

Target: Others

Cat.No: T70287

Target: Others

Cat.No: T36175

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T8063	Cephapirin Benzathine	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式，是一种广谱抗生素。
T8062	Cefazedone Refosporen,头孢西酮	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。
T1004	6-Benzylaminopurine 6-苄氨基嘌呤,6-BAP,N6-Benzyladenine,BA,Benzyladenine	Others	Others
	6-Benzylaminopurine (6-BAP) 是一种细胞分裂素，能够通过刺激细胞分裂引起植物生长和发育，抑制呼吸激酶，从而延长绿色蔬菜的保鲜。
T1181	Gefitinib ZD1839,吉非替尼	EGFR; Tyrosine Kinases; Autophagy	Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Gefitinib (ZD1839) 是一种 EGFR 一代抑制剂，具有口服活性，抑制 EGFR 19 Del 和 L858R 突变。Gefitinib 具有抗肿瘤活性，用于治疗 EGFR 突变的非小细胞肺癌。Gefitinib 用药会产生 EGFR C797S 耐药突变。

天然产物

Cephapirin Benzathine

Cat.No: T8063

Target: Others, Antibacterial, Antibiotic

Cat.No: T8062

Synonym: Refosporen,头孢西酮

Target: Others, Antibacterial, Antibiotic

6-Benzylaminopurine

Cat.No: T1004

Synonym: 6-苄氨基嘌呤,6-BAP,N6-Benzyladenine,BA,Benzyladenine

Target: Others

Cat.No: T1181

Synonym: ZD1839,吉非替尼

Target: EGFR, Tyrosine Kinases, Autophagy

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-00585	Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (Yeast, His) Beta-lactamase MEN-1,Cefotaximase 1,bla,men1,Beta-lactamase ...	E. coli	P. pastoris (Yeast)
	Broad spectrum beta-lactamase which confers resistance to penicillins, as well as first, second and third-generation cephalosporins.
TMPH-00584	Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (His) men1,Beta-lactamase MEN-1,Cefotaximase 1,Beta-lactamase CTX-...	E. coli	E. coli
	Broad spectrum beta-lactamase which confers resistance to penicillins, as well as first, second and third-generation cephalosporins.
TMPH-03106	Coagulation factor XII Protein, Pig, Recombinant (His) HAF,Hageman factor,F12,Coagulation factor XII	Sus scrofa (Pig)	E. coli
	Factor XII is a serum glycoprotein that participates in the initiation of blood coagulation, fibrinolysis, and the generation of bradykinin and angiotensin. Prekallikrein is cleaved by factor XII to form kallikrein, which then cleaves factor XII first to alpha-factor XIIa and then trypsin cleaves it to beta-factor XIIa. Alpha-factor XIIa activates factor XI to factor XIa. Coagulation factor XII Protein, Pig, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predic...

重组蛋白

Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (Yeast, His)

Cat.No: TMPH-00585

Species: E. coli

Expression System: P. pastoris (Yeast)

Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (His)

Cat.No: TMPH-00584

Species: E. coli

Expression System: E. coli

Coagulation factor XII Protein, Pig, Recombinant (His)

Cat.No: TMPH-03106

Species: Sus scrofa (Pig)

Expression System: E. coli

Cat. No.	Product Name	Target	Signaling Pathways
TMIJ-0523	Gliquidone-d6
	Gliquidone-d6 是 Gliquidone 的氘代化合物。Gliquidone 的 CAS 号为 33342-05-1。Gliquidone 是一种磺酰脲类的抗糖尿病药物，可用于2型糖尿病的研究。

同位素标记化合物

Cat.No: TMIJ-0523

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