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Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).
Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 1,170 | 5日内发货 | |
5 mg | ¥ 1,980 | 5日内发货 | |
25 mg | ¥ 6,290 | 6-8周 | |
50 mg | ¥ 8,170 | 6-8周 | |
100 mg | ¥ 12,500 | 6-8周 | |
1 mL x 10 mM (in DMSO) | ¥ 2,230 | 5日内发货 |
产品描述 | Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A). |
靶点活性 | MAO-A:0.2 μM |
体外活性 | In order to assess whether the protective effect is related to the inhibition of the MAO-A or due to another mechanism, the effect of Brofaromine is determined on the activity of MAO-A in cultured cortical cells. The cultured cortical cells have significant MAO-A activity. Brofaromine inhibits the enzyme in a concentration-dependent manner (IC50: 0.19?μM). Hill coefficient is 0.96. The enzyme is almost completely inhibited at 10?μM. Brofaromine inhibits MAO-A activity of our cultured cortical cells in a concentration-dependent manner. The IC50 range of Brofaromine is 0.01?μM to 0.1?μM. |
别名 | CGP 11305A |
分子量 | 310.19 |
分子式 | C14H16BrNO2 |
CAS No. | 63638-91-5 |
密度 | 1.386 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 250 mg/mL (805.96 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
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