73
7
6
6
3
Cat. No. | Product Name | ||
---|---|---|---|
L4660 | 神经疾病库Plus | 1246 compounds | |
1246 种神经系统相关、结构新颖的化合物; | |||
L2600 | 神经信号分子库 | 2540 compounds | |
2540 种CNS 相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
L7400 | 钠通道分子库 | 118 compounds | |
118 种钠通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L9840 | 抗阿尔茨海默症化合物库 | 986 compounds | |
986 种阿尔茨海默症相关的化合物集合,可用于高通量和高内涵筛选; | |||
L2630 | 神经元分化化合物库 | 672 compounds | |
672 种与神经元分化相关的化合物,可以用于神经系统疾病药物研发 | |||
L2610 | 神经递质受体化合物库 | 1513 compounds | |
1513 种与神经递质受体相关的化合物,用于高通量、高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9989 |
AChE-IN-27
|
Others | Others |
AChE-IN-27是一种用于高通量测定的小分子。 | |||
T35878 |
N-(3-Aminopropyl)cyclohexylamine
|
Others | Others |
N-(3-Aminopropyl)cyclohexylamine, a derivative of cyclohexylamine, functions as a selective and competitive inhibitor of spermine synthase, making it suitable for research on neurological diseases[1]. | |||
TP1856 |
Colivelin
|
Beta Amyloid; STAT | JAK/STAT signaling; Neuroscience; Stem Cells |
Colivelin 是一种神经保护肽和 STAT3 的激活剂,是一种合成的杂合肽,可增强 humanin (HN) 的神经保护作用。它通过激活 STAT3 在体外抑制神经元死亡,具有潜力用于阿尔茨海默病和缺血性脑损伤的相关研究。 | |||
T1594 |
Vecuronium bromide
ORG NC 45,维库溴铵 |
AChR | Neuroscience |
Vecuronium bromide (ORG NC 45) 是一种合成的中效单季铵盐类固醇和非去极化神经肌肉阻滞剂,具有肌肉松弛活性。 | |||
T1476 |
Pramipexole
SND 919,普拉克索 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Pramipexole (SND 919) 是能够透过血脑屏障的 D2 型多巴胺受体的选择性激动剂,对 D2 型受体、D2、D3、D4亚型受体的Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM。它可用于研究帕金森综合症和腿多动综合征。 | |||
T4497 |
Amifampridine
3,4-Pyridinediamine,Pyridine-3,4-Diamine,阿米吡啶,3,4-Diaminopyridine |
Others | Others |
Amifampridine (3,4-Diaminopyridine) 可用于罕见肌肉疾病的研究。 | |||
T3198L |
PRE-084 hydrochloride
|
Sigma receptor | GPCR/G Protein |
PRE-084 hydrochloride 是 σ1 的选择性激动剂在sigma 受体检测中,IC50值为44 nM。 | |||
T7805 |
GW791343 dihydrochloride
GW791343 (HCl) |
P2X Receptor | Membrane transporter/Ion channel; Neuroscience |
GW791343 dihydrochloride (GW791343 (HCl)) 是有种属特异性的 P2X7变构调节剂,对人 P2X7的 pIC50为6.9-7.2。 | |||
T3217 |
PF-CBP1 hydrochloride
PF-CBP1 HCl |
Epigenetic Reader Domain; Histone Acetyltransferase | Chromatin/Epigenetic |
PF-CBP1 hydrochloride (PF-CBP1 HCl) 是 CREB 结合蛋白溴结构域的一种高选择性抑制剂,抑制 CREBBP 和 EP300溴结构域的 IC50分别为 125 和 363 nM。它降低 LPS 诱导的巨噬细胞中炎症因子的表达,也可下调皮质神经元 RGS4 的表达,可用于癫痫和帕金森病等神经疾病的研究。 | |||
T6951 |
Pramipexole dihydrochloride hydrate
Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Pramipexole dihydrochloride hydrate (Mirapex) 是选择性的,具有血脑屏障 (BBB) 渗透性的 D2 型多巴胺受体激动剂,对 D2 型受体、D2、D3、D4亚型受体的 Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM,可用于研究帕金森综合症和腿多动综合征。 | |||
T6526 |
GW791343 trihydrochloride
GW791343 3HCl |
P2X Receptor | Membrane transporter/Ion channel; Neuroscience |
GW791343 trihydrochloride (GW791343 3HCl) 是 P2X7变构调节剂,有种属特异性,对人 P2X7的pIC50为6.9-7.2。 | |||
T27143 |
Delucemine Hydrochloride
NPS 1506,Delucemine,Delucemine HCl,NPS1506,NPS-1506 |
NMDAR | Neuroscience |
Delucemine Hydrochloride (Delucemine) 是一种多胺NMDA受体拮抗剂,可用于研究抑郁症和阿尔茨海默症等神经系统疾病。 | |||
T28441 |
PPI-1019
PPI1019,Apan |
Beta Amyloid | Neuroscience |
PPI-1019 是一种 APP( β -淀粉状蛋白 A4 )抑制剂,可用于治疗神经系统疾病和研究阿尔茨海默病(AD)。 | |||
T31079 |
CP-810123
CP 810123,UNII-E6G4550EC4,CP810123 |
AChR | Neuroscience |
CP-810123 是一种新的α 7 nAChR 激动剂,可用于治疗与精神分裂症和阿尔茨海默病等精神或神经疾病相关的认知障碍。 | |||
T74031 |
Cardiolipin (Heart, Bovine) (sodium)
|
||
Cardiolipin (Heart, Bovine) sodium,一种线粒体专有磷脂,展现出在神经系统疾病研究中的应用潜力。 | |||
TP1195 |
Cibinetide
ARA290 |
Others | Others |
Cibinetide (ARA290) 是特异性的 erythropoietin/CD131 heteroreceptor 的激动剂,是一种 EPO 衍生物,常用于神经系统疾病研究。 | |||
T13047 |
Synta66
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Synta66 是一种钙池操纵钙离子通道 Orai 抑制剂,用于神经系统疾病的研究。 | |||
T64344 |
N-Methyl-DL-aspartic acid
|
NMDAR | Neuroscience |
N-Methyl-DL-aspartic acid 是谷氨酸类似物,是一种 NMDA receptor 激动剂,可用于神经疾病的研究。 | |||
T23649 |
AF-710B
ANAVEX 3-71,AF 710B,AF710B |
Sigma receptor; AChR | GPCR/G Protein; Neuroscience |
AF-710B 是一种特异性变构 M1 毒蕈碱和 Sigma-1 受体激动剂,可用于研究阿尔茨海默病痴呆和神经分裂等神经系统疾病。 | |||
TP1866L |
β-amyloid 1-11 acetate(190436-05-6 free base)
|
Beta Amyloid | Neuroscience |
β-amyloid 1-11 acetate(190436-05-6 free base) 是 Amyloid-β 肽的片段,可用于神经系统疾病的研究。 | |||
T81633 |
Nurr1 agonist 7
|
Others | Others |
Nurr1 agonist 7 是 Nurr1 的激动剂(EC50:0.12 μM),可用于研究帕金森等神经系统疾病。 | |||
T11949 |
Masupirdine mesylate
SUVN-502 mesylate,SVN-502 mesylate |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Masupirdine mesylate (SUVN-502 mesylate) 是一种具有选择性且可穿越血脑屏障的 5-HT6 受体拮抗剂。Masupirdine mesylate 可用于研究阿尔茨海默病和痴呆等神经系统疾病。 | |||
TQ0238 |
Lanabecestat
LY3314814,AZD3293 |
BACE | Neuroscience |
Lanabecestat (AZD3293) 是一种具有高效性和高渗透性、口服活性且可穿过血脑屏障的 BACE1 抑制剂(Ki:0.4 nM),Lanabecestat 可用于研究像阿尔茨海默症类的神经系统疾病。 | |||
T32368 |
KB-74935
KB 74935 |
Others | Others |
KB-74935是一种酶抑制剂,是一种矿物皮质激素受体拮抗剂,可用于治疗 胆固醇、低血脂、神经系统疾病和阿尔茨海默病。 | |||
T68084 |
Icopezil
|
AChE | Neuroscience |
Icopezil是一种小分子乙酰胆碱酯酶在(AChE)抑制剂,可用于治疗神经系统疾病,可用于研究阿尔茨海默病。 | |||
TP1214L |
β-Amyloid 15-21 acetate
Beta-Amyloid (15-21) acetate |
Beta Amyloid | Neuroscience |
β-Amyloid 15-21 acetate (Beta-Amyloid(15-21) acetate) 是 Amyloid-β 肽的片段,可用于神经系统疾病的研究。该片段参与β折叠形成。 | |||
T77509 |
hBChE-IN-2
|
AChR | Neuroscience |
hBChE-IN-2 是一种丁酰胆碱酯酶 (BChE) 抑制剂和大麻素受体 2 BChE) 抑制剂,具有神经保护活性,可用于研究阿尔茨海默症类的神经系统疾病。 | |||
T26551 |
Acetyl-L-carnitine
RO 447190,L-Acetylcarnitine,LAC,L-O-Acetylcarnitine,ALCAR,Acetyl L carnitine |
Endogenous Metabolite | Metabolism |
Acetyl-L-carnitine(RO 447190) 是一种可透过血脑屏障的氨基酸左旋肉碱,常作为膳食补充剂,对神经炎症有益。Acetyl-L-carnitine 具有神经保护作用,可用以研究像阿尔茨海默病类的神经疾病。 | |||
T27795L |
(Iso)-Landipirdine
(Iso)-SYN120,(Iso)-RO5025181,(Iso)-Landipirdine(Iso-1000308-25-7) |
5-HT Receptor | GPCR/G Protein; Neuroscience |
(Iso)-Landipirdine((Iso)-RO5025181) 是一种具有选择性和有效性的 5-HT6R 拮抗剂。(Iso)-Landipirdine 对 hERG 药效团有明显影响,可用于研究阿尔茨海默病类的神经系统疾病。 | |||
T76726 |
Zagotenemab
LY33003560 |
Microtubule Associated | Cytoskeletal Signaling |
Zagotenemab 是一种人源化抗微管相关蛋白 tau 抗体,能选择性地调节大脑中的 tau 沉积物。Zagotenemab 可用于研究阿尔兹海默症等神经系统疾病。 | |||
T80622 |
Trontinemab
RO-7126209,RG6102 |
Beta Amyloid | Neuroscience |
Trontinemab (RG6102) 是一种选择性靶向Aβ前体蛋白(APP)与转铁蛋白受体p90, CD71 (TFRC)的人源IgG1-κ抗体,抑制淀粉样蛋白产生,可用于研究阿兹海默症等神经系统疾病。 | |||
T9340 |
1-phenyl-3,4-dihydroisochinoline
3,4-Dihydro-1-phenylisoquinoline,1-苯基-3,4-二氢异喹啉 |
Others | Others |
1-phenyl-3,4-dihydroisochinoline (3,4-Dihydro-1-phenylisoquinoline) 是神经递质多巴胺的结构类似物,与中枢神经系统中的多巴胺受体相互作用。它已被研究为治疗帕金森病、阿尔茨海默病和亨廷顿舞蹈症等神经疾病的潜在治疗剂。 | |||
T68492 |
AM 374
HDSF,Hexadecanesulfonyl fluoride |
FAAH | Metabolism; Neuroscience |
AM 374 (HDSF) 是一种脂肪酸酰胺水解酶(FAAH)抑制剂。AM 374 对氨基酶活性的抑制作用的IC50为 13 nM。AM 374 可用于神经系统疾病的研究。 | |||
T69726 |
Oditrasertib
DNL-788 |
RIP kinase | Apoptosis; NF-κB |
Oditrasertib (DNL-788) 是一种高效的 RIPKl 抑制剂,其 IC50 值低于 100 nM。Oditrasertib 可用于研究多发性硬化症和阿尔茨海默症等免疫系统疾病与神经系统疾病。 | |||
T50046 |
L-Valyl-L-phenylalanine HCl
Valylphenylalanine HCl; H-VAL-PHE-OH HCl |
Others | Others |
2-(2-amino-3-methylbutanamido)-3-phenylpropanoic acid hydrochloride 是一种氨基酸类化合物,是谷氨酸的合成类似物,谷氨酸是中枢神经系统中的一种重要神经递质。它已被研究其在各种神经疾病中的潜在治疗应用,包括阿尔茨海默病、帕金森病和癫痫。 | |||
T111959 |
IFB-088 acetate
|
Others | Others |
IFB-088 acetate 是一种苄基胍衍生物,可用于治疗与PPP1R15A 途径相关并与蛋白质错误折叠应激相关的疾病和癌症,如tau 病、突触核蛋白病、多谷氨酰胺和多丙氨酸疾病、白质营养不良、囊性纤维化、多发性硬化症、溶酶体储存障碍、淀粉样变性疾病、炎症、代谢障碍、心血管疾病、骨质疏松症、神经系统创伤等等。 | |||
T50003 |
Debrisoquin hydriodide
1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide |
Others | Others |
Debrisoquin hydriodide (1,2,3,4-tetrahydroisoquinoline-2-carboximidamide hydroiodide) 具有抗氧化、抗炎和神经保护特性,也被发现可以调节某些神经递质的活性,包括多巴胺和血清素,使其成为治疗帕金森病和抑郁症等神经疾病的有前途的候选药物。 | |||
T50090 |
3-(2-phenylethynyl)pyridine
|
Others | Others |
3-(2-phenylethynyl)pyridine 是一种吡啶衍生物,是人体中各种受体的配体,包括多巴胺 D2受体、sigma-1受体和5-HT6受体,已被研究用于治疗各种神经疾病,包括精神分裂症、抑郁症和阿尔茨海默病。 | |||
T11948 |
Masupirdine free base
Masupirdine,SUVN-502 free base |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Masupirdine free base(SUVN-502 free base)是一种可口服且可穿过血脑屏障的 5-HT6 受体拮抗剂,对人类 5-HT6 受体的 Ki 值为 2.04 nM。Masupirdine free base 具有高效性和选择性且对多种靶点都具有抑制作用。Masupirdine free base 可用于研究像阿尔茨海默病类的神经系统疾病。 | |||
T77342 |
GSK-3 inhibitor 3
|
GSK-3; Microtubule Associated | Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Stem Cells |
GSK-3 inhibitor 3 是一种具有选择性、具有口服活性和脑渗透性的 GSK-3 抑制剂,对 GSK-3α 和 GSK-3β 具有抑制作用, IC50s 分别为 0.35 nM 和 0.25 nM。GSK-3 inhibitor 3 在三重转基因小鼠阿尔茨海默病模型中降低 Tau 蛋白 (tau protein) S396 磷酸化水平,IC50为 10 nM。GSK-3 inhibitor 3 可用于研究神经系统疾病。 | |||
T39218 |
(S)-CVN424
(S)-CVN424 |
Others | Others |
(S)-CVN424 is a powerful modulator of G-Protein-Coupled Receptor 6 (GPR6), known for its involvement in neurological and psychiatric disorders research, such as Parkinson's disease. | |||
TP1214 |
β-Amyloid 15-21
Beta-Amyloid (15-21) |
||
β-amyloid (15-21) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease. This fragment is involved in beta sheet formation. | |||
T7352L |
Pridopidine hydrochloride
ASP2314 HCl,Pridopidine HCl,FR310826,ASP-2314 hydrochloride |
Others | Others |
Pridopidine Hydrochloride is a dopaminergic stabilizer that has been shown to improve a variety of neurological and psychiatric disorders, including Huntington's disease. Pridopidine Hydrochloride stabilizes psychomotor activity in a state-dependent way t | |||
T81520 |
Penta-alanine
Penta-L-alanine |
||
Penta-alanine (Penta-L-alanine)为一种具有研究价值的肽,常用于探究神经系统疾病。 | |||
T79191 |
AMPA receptor modulator-5
|
iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptormodulator-5 (Example 217) 为一种AMPA receptor调节剂,适用于神经系统疾病研究。 | |||
T75969 |
β-Amyloid (15-21)
|
Others | Others |
β-amyloid (15-21) 是 β 淀粉样肽的一个片段,在神经领域具有潜在的作用。 | |||
T40701 |
Ezeprogind
AZP-2006 |
Others | Others |
Ezeprogind (AZP-2006) is an orally active neurotrophic inducer that effectively addresses the underlying factors contributing to neurodegeneration, with a broad scope extending beyond the conventional targets like Abeta protein and tau protein. Exhibiting potent neuroprotective properties, Ezeprogind is a valuable tool for studying a range of neurological disorders, including progressive supranuclear palsy (PSP), tauopathies, Alzheimer's disease, Parkinson's disease, and others. | |||
T78111 |
NCS-382 sodium
|
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
NCS-382 (sodium) 为一种高效GABA受体拮抗剂,具备抗镇静及抗催眠特性,适用于神经系统疾病研究。 | |||
T80468 |
δ-Dendrotoxin
|
Potassium Channel | Membrane transporter/Ion channel |
δ-Dendrotoxin,作为一种K+通道阻滞剂,来源于黑曼巴蛇的毒液,常用于研究神经系统疾病。 | |||
T80484 |
Aa1 toxin
|
Potassium Channel | Membrane transporter/Ion channel |
Aa1 toxin 是从 Androctonus australis Garzoni 毒液中提取的神经毒性肽,特异性阻断钾通道(potassium channel)。它在神经系统疾病研究中有应用。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1045 |
Trimipramine maleate
Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐 |
Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂,对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。 | |||
T8790 |
1-Methylhistamine dihydrochloride
|
Endogenous Metabolite | Metabolism |
1-Methylhistamine dihydrochloride 是组胺代谢物。 | |||
T32614 |
L-Clausenamide
(-)-Clausenamide |
Microtubule Associated | Cytoskeletal Signaling |
L-Clausenamide 是从黄皮 (Clausena lansium (Lour) skeels) 的树叶中提取出来的生物碱,可用于提高认知功能。L-Clausenamide 对β-淀粉样蛋白 (Aβ) 毒性有抑制作用,通过抑制 tau 蛋白磷酸化阻止神经纤维缠结的形成。L-Clausenamide 具有神经保护活性,可用于调节 Aβ25-35 引发的刺激。L-Clausenamide 可用于研究阿尔兹海默症类的神经系统疾病。 | |||
T7984 |
2-Hydroxyflavanone
|
Others | Others |
2-Hydroxyflavanone 是一种天然存在的黄酮类化合物,存在于许多植物和水果中。它具有抗氧化、抗炎和抗肿瘤的活性,可以清除自由基,减少炎症,并抑制肿瘤细胞的生长,还具有治疗糖尿病、肥胖症、心血管疾病和神经系统疾病等多种疾病的潜力。 | |||
TN4368 |
Kaempferol-3,7-di-O-β-glucoside
Kaempferol 3,7-di-O-glucoside |
Glucosidase; Amylase | Metabolism |
Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) 是一种来自 Morettia philaena 的黄酮醇,对 α-淀粉酶 (α-amylase)、α-葡萄糖苷酶 (α-glucosidase) 和乙酰胆碱酯酶 (Acetylcholinesterase) 具有抑制作用。Kaempferol-3,7-di-O-β-glucoside 具有神经保护活性,可减缓分化神经元细胞 SH-SY5Y 免受 Amyloid β 肽诱导的损伤。Kaempferol-3,7-di-O-β-glucoside 可用于研究阿尔茨海默氏症类的神经系统疾病。 | |||
T4S2126 |
Ginkgetin
银杏双黄酮,银杏素 |
Apoptosis; Wnt/beta-catenin; COX; STAT; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells |
Ginkgetin 是从银杏叶中分离得到的一种双黄酮,具有抗肿瘤、抗炎、神经保护、抗真菌的作用。它也是 Wnt 信号抑制剂,IC50值为 5.92 μM。 | |||
T82341 |
Ganglioside GM1
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Ganglioside GM1,一种神经节苷脂家族成员,用于神经系统疾病研究。同时,它作为霍乱毒素 1 的功能性组织受体。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-06802 |
HSV 2 (strain 333) Glycoprotein D/gD Protein (His)
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HSV2 | HEK293 Cells |
Herpes simplex viruses (human herpesviruses types 1 and 2) commonly cause recurrent infection affecting the skin, mouth, lips, eyes, and genitals. Herpes simplex virus type 2 (HSV-2) infection is responsible for significant neurological morbidity, perhaps more than any other virus. Herpes simplex virus type 2–associated neurological disease may result from primary infection or reactivation of latent HSV-2. Common severe infections include encephalitis, meningitis, neonatal herpes, and, in immun... | |||
TMPJ-01022 |
SUMO3 Protein, Human, Recombinant (HEK293, His)
SMT3 homolog 1,Smt3A,Small ubiquitin-related modifier 3,Ubiq... |
Human | HEK293 Cells |
Small ubiquitin-like modifier (SUMO), also known as SUMO homologue and SMT3, is a member of the superfamily of ubiquitin-like polypeptides that become covalently attached to various intracellular target proteins as a way to alter their function, location, and/or half-life. Small ubiquitin-like modifiers include SUMO1, SUMO2, SUMO3, and SUMO4. Except for SUMO4, all other SUMOs are ubiquitously expressed, including in the brain. In human, SUMO2 and SUMO3 are two highly homologous proteins, collect... | |||
TMPJ-01002 |
SGSH Protein, Human, Recombinant (His)
SGSH,N-Sulphoglucosamine Sulphohydrolase,Sulfoglucosamine Su... |
Human | HEK293 Cells |
N-Sulphoglucosamine Sulphohydrolase (SGSH) is an important member of the sulfatase family which is involved in the degradation of heparin sulfate. SGSH binds one calcium ion per subunit as a cofactor. SGSH catalyzes N-sulfo-D-glucosamine and H2O to D-glucosamine and sulfate. SGSH deficiency is result in mucopolysaccharidosis type 3A (MPS3A), a recessive lysosomal storage disease characterized by neurological dysfunction but relatively mild somatic manifestations. | |||
TMPY-03332 |
PRTFDC1 Protein, Human, Recombinant (His)
HHGP,PRTFDC1,phosphoribosyl transferase domain containing 1 |
Human | E. coli |
PRTFDC1 is a member of the purine/pyrimidine phosphoribosyltransferase family. It can bind GMP, IMP and alpha-D-5-phosphoribosyl 1-pyrophosphate (PRPP). The epigenetic silencing of PRTFDC1 by hypermethylation of the CpG island leads to a loss of PRTFDC1 function, which might be involved in squamous cell oral carcinogenesis. PRTFDC1 is a genetic modifier of HPRT-deficiency in the mouse and has important implications for unraveling the molecular etiology of lesch-Nyhan disease(LND). LND is a sever... | |||
TMPY-01290 |
CHIT1 Protein, Human, Recombinant (His)
chitinase 1 (chitotriosidase),CHITD,CHI3,CHIT |
Human | HEK293 Cells |
Chitotriosidase, also known as Chitinase-1 and CHIT1, is a member of the glycosyl hydrolase 18 family and Chitinase class II subfamily. It is a member of the mammalian chitinase family, structurally homologous to chitinases from other species, is synthesized and secreted by specifically activated macrophages. Chitotriosidase is a polymer of N-acetylglucosamine. Serum and plasma chitotriosidase activity is usually measured as the first step in diagnosis of Gaucher disease. Monitoring chitotriosid... | |||
TMPJ-00495 |
ISG15 Protein, Human, Recombinant (His)
ISG15,Ubiquitin Cross-Reactive Protein,G1P2,Interferon-Induc... |
Human | E. coli |
Ubiquitin-Like Protein ISG15 (ISG15) is a ubiquitin-like protein that becomes conjugated to many cellular proteins upon activation by interferon-alpha and -beta. Several functions have been ascribed to the encoded protein, including chemotactic activity towards neutrophils, direction of ligated target proteins to intermediate filaments, cell-to-cell signaling, and antiviral activity during viral infections. While conjugates of this protein have been found to be noncovalently attached to intermed... |
Cat. No. | Product Name | Target | Signaling Pathways |
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TMIH-0028 |
2-(1-(methyl-d3)-1H-imidazol-4-yl)ethan-1-amine 2HCl
1-Methylhistamine-d3 Dihydrochloride |
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2-(1-(methyl-d3)-1H-imidazol-4-yl)ethan-1-amine 2HCl 是 2-(1-(methyl)-1H-imidazol-4-yl)ethan-1-amine 2HCl 的氘代化合物。2-(1-(methyl)-1H-imidazol-4-yl)ethan-1-amine 2HCl 的 CAS 号为 6481-48-7。1-Methylhistamine dihydrochloride 是组胺代谢物。 | |||
TMIJ-0054 |
Propionic-2,2-d2 acid
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Propionic-2,2-d2 acid 是 Propionic acid 的氘代化合物。Propionic acid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。 | |||
TMIJ-0052 |
Propionicacid-d5
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Propionicacid-d5 是 Propionicacid 的氘代化合物。Propionicacid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。 |