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Search Results for " bactericidal "
Targets Recommended: Antibacterial DprE1

106

抑制剂 & 化合物

18

天然产物

15

重组蛋白

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T3583 Macozinone

PBTZ169

Antibacterial; DprE1 Microbiology/Virology; Others
Macozinone (PBTZ169) 是具有杀菌作用的苯并噻嗪酮,也有抗结核作用。它也是一种 DprE1有效抑制剂,可通过与活性位点 Cys387 残基形成共价键来抑制必需的黄素蛋白 DprE1。
T7872 Monolaurin

Others Others
Monolaurin 是椰子油中的一种表面活性剂和乳化剂。它抑制葡萄球菌、链球菌、加德纳菌、念珠菌和嗜血杆菌的生长,并减少促炎细胞因子的产生。
T1312 Nafcillin sodium monohydrate

CL 8491,萘夫西林钠,nafcillin sodium

Antibacterial; Antibiotic Microbiology/Virology
Nafcillin sodium monohydrate (CL 8491) 是一种抗生素,是可逆的β-lactamase 抑制剂。它用于治疗由耐青霉素的葡萄球菌菌株引起的感染。
T16073 Micronomicin

小诺霉素,Gentamicin C2b,Antibiotic XK-62-2,Sagamicin

Others; Antibacterial Microbiology/Virology; Others
Micronomicin (Gentamicin C2b) 是一种具有抗菌和杀菌能力的抗生素。
T40417 Ethylhydrocupreine hydrochloride

Optochin hydrochloride,乙氢去甲奎宁盐酸盐;奥普托欣盐酸盐

Antibacterial; Parasite Microbiology/Virology
Ethylhydrocupreine hydrochloride (Optochin hydrochloride) 是奎宁的一种衍生物,具有抗菌作用,可抑制肺炎链球菌的活性。Ethylhydrocupreine hydrochloride 具有抗疟活性,对 Plasmodium falciparum 的IC50为 25.75 nM。Ethylhydrocupreine hydrochloride 是Gallus gallus2 受体 (ggTas2r1,ggTas2r2和ggTas2r7) 激动剂。
T1495 Cefaclor monohydrate

Cefaclor,头孢克洛一水物,头孢克洛一水合物,Cefaclorum,Cefachlor

Antibacterial; Antibiotic Microbiology/Virology
Cefaclor monohydrate (Cefaclorum) 是一种抗生素,可特异性地结合青霉素结合蛋白。
T7735 5-Nitro-1,10-phenanthroline

5-NP,5-硝基-1,10-菲咯啉

Antibacterial Microbiology/Virology
5-Nitro-1,10-phenanthroline (5-NP) 是一种有效的杀菌剂,可抑制艰难梭菌。
T1143 Carbenicillin disodium

BRL-2064,羧苄青霉素钠,Sodium carbenicillin

Cell wall; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Carbenicillin disodium (BRL-2064) 作用于细菌细胞壁合成的最后阶段,是β-内酰胺青霉素衍生物。
T3247 Lysozyme from chicken egg white

鸡蛋清溶菌酶,溶菌酶,Lysozyme

Others; Antibacterial Microbiology/Virology; Others
Lysozyme from chicken egg white (Lysozyme) 是一种存在于鸡蛋清中的杀菌酶,它溶解革兰氏阳性菌。
T64346 DDAC

Quaternium 12

Antibacterial Microbiology/Virology
DDAC (Quaternium 12), also known as Didecyldimethylammonium chloride, is a dialkyl-quaternary ammonium compound widely utilized in various products due to its bactericidal, virucidal, and fungicidal characteristics.
T0328 Hexetidine

NSC-17764,海克替啶

Antibacterial; Antifungal Microbiology/Virology
Hexetidine (NSC-17764) 是一种口服活性的抗菌抗真菌试剂,可用于口腔感染的相关研究。
T16071 MGB-BP-3

DNA/RNA Synthesis; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
MGB-BP-3 是一种合成抗生素,具有杀菌活性,抑制细菌 DNA 复制,可用于研究复发性艰难梭菌感染。
T3263 (6R,7S)-Cefminox sodium heptahydrate

Meicelin,头孢米诺钠,Cefminox Sodium,Alteporina,Tencef

Antibiotic Microbiology/Virology
(6R,7S)-Cefminox sodium heptahydrate (Meicelin) 是一种 Cefminox sodium heptahydrate 的异构体。它也是一种具有广谱抗菌活性的 β-内酰胺头孢菌素抗生素。
T72030 6,6'-Dimethyl-2,2'-dipyridyl

6,6'-Bi-2-picoline

Others Others
6,6'-Dimethyl-2,2'-dipyridyl (6,6'-Bi-2-picoline) 是一种新型的时间分辨荧光免疫分析(TRFIA)螯合物,具有较好的杀菌效果,可用于研究酒渣鼻。
T7533 Taurolidine

Apoptosis; Others; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Others
Taurolidine 是一种广谱抗菌剂,用于预防中心静脉导管相关感染。它具有抗真菌和抗肿瘤作用。
T3582 BTZ043

Antibacterial; Antibiotic; DprE1 Microbiology/Virology; Others
BTZ043 是一种 DprE1 的抑制剂,它对结核分枝杆菌 H37Rv 和耻垢分枝杆菌具有纳摩尔杀菌活性,MIC 值分别为 2.3 nM 和 9.2 nM。
T1405 Cefditoren pivoxil

头孢妥仑匹酯,ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl

Antibacterial; Antibiotic Microbiology/Virology
Cefditoren pivoxil (ME 1207) 是一种半合成、广谱、β-内酰胺酶耐药的第三代头孢菌素抗生素,具有杀菌活性。
T12593 Pyrithione

1-hydroxyl-1H-pyridine-2-thione,吡啶硫酮

Others Others
Pyrithione (1-hydroxyl-1H-pyridine-2-thione) 是一种锌离子载体,过渡金属配合物,可引起哺乳动物细胞内锌水平的升高,有杀菌和抗真菌作用。
T2211 Dihydrostreptomycin sulfate

Dihydrostreptomycin sesquisulfate,双氢链霉索

Antibacterial; Antibiotic Microbiology/Virology
Dihydrostreptomycin sulfate (Dihydrostreptomycin sesquisulfate) 是一种氨基糖苷类抗生素,可研究牛、猪和羊的细菌性疾病。
T28229 Olanexidine hydrochloride

OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045

Antibacterial Microbiology/Virology
Olanexidine hydrochloride (OPB-2045 HCl) 对革兰氏阳性菌和革兰氏阴性菌具有杀菌活性。 Olanexidine hydrochloride 破坏金黄色葡萄球菌的膜完整性。
T5022 Ceforanide

Antibacterial; Antibiotic Microbiology/Virology
Ceforanide 是一种头孢菌素,可静脉或肌肉给药。它在体外具有一系列抗菌活性。
T79468 Antimicrobial agent-22

THI 6c

Antibacterial Microbiology/Virology
Antimicrobial agent-22 (THI 6c) 是一种抗菌剂,具有低细胞毒性、抗生物膜活性和快速杀菌的作用。
T6706 Ticarcillin sodium

Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。
T0199 Cephradine

Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定

TOPK; Antibacterial; Antibiotic MAPK; Microbiology/Virology
Cephradine (Anspor) 是广谱口服活性头孢菌素。它对革兰氏阳性和革兰氏阴性病原体都有活性。它已用于泌尿生殖系统、胃肠道和呼吸道感染以及皮肤和软组织感染的研究。它通过直接抑制TOPK 抑制太阳紫外线诱导的皮肤炎症。
T7191 Diphenyleneiodonium chloride

二苯基氯化碘盐,DPI

NOS; Reactive Oxygen Species; NADPH; TRP/TRPV Channel Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
Diphenyleneiodonium chloride (DPI) 是 NADPH 氧化酶抑制剂,也是 TRPA1激活剂,EC50为 1 - 3 μM 。它选择性抑制胞内活性氧。
T1305 Ceftazidime

GR20263,头孢他啶

Antibacterial; Antibiotic Microbiology/Virology
Ceftazidime (GR20263) 是可静脉内或肌肉给药的第头孢菌素。它对革兰氏阳性和革兰氏阴性需氧细菌有体外活性。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。
T0868 Cefepime Dihydrochloride Monohydrate

Cefepime HCl,头孢吡肟二盐酸盐一水合物

Antibacterial; Antibiotic; Antifection Microbiology/Virology
Cefepime Dihydrochloride Monohydrate (Cefepime HCl) 是一种广谱头孢菌素,对革兰氏阳性菌和革兰氏阴性菌有更高的覆盖率。
T1005L Amoxicillin trihydrate

Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。
T0377 Clofazimine

NSC-141046,氯法齐明,氯苯吩嗪

DNA; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料,与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。
T11348 G907

Antibiotic Microbiology/Virology
G907 是一种具有选择性和有效性的小分子ATP 结合盒 (ABC) 转运蛋白 MsbA 的拮抗剂,具有杀菌活性,可将 MsbA 捕获在朝内的脂多糖中。 G907 对大肠杆菌 MsbA 有抑制作用, IC50 值为 18 nM。
TP1341L Polymyxin B nonapeptide acetate

Polymyxin B nonapeptide acetate(86408-36-8 free base)

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B nonapeptide acetate(86408-36-8 free base) 是一种阳离子环肽。 Polyxin B 九肽是 polyxin B 经酶解产生的衍生物。与 polyxin B 相比,polyxin B 九肽毒性低,缺乏杀菌活性,仍具有破坏革兰氏阴性菌外膜的能力。
T0953 Cefazolin sodium

Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin sodium (cephazolin sodium) salt 是一种头孢类抗生素, 可研究多种细菌感染。
T76662 Ac-Pro-Gly-Pro-OH

Apoptosis; CXCR; Antibiotic Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology
Ac-Pro-Gly-Pro-OH 是乙酰基修饰的三肽化合物,可用作 CXCR2 激动剂。Ac-Pro-Gly-Pro-OH 具有杀菌和抗炎活性,抑制免疫细胞凋亡,抑制促炎细胞因子的产生。Ac-Pro-Gly-Pro-OH 可用于研究脓毒症和肺部炎症。
T1213 Piperacillin sodium

哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt

Antibacterial; Antibiotic Microbiology/Virology
Piperacillin sodium salt(CL227193) )是一种β-内酰胺类广谱抗生素。
T41275 PF-04753299

Others Others
PF-04753299 是一种有效的、选择性的LpxC 抑制剂。PF-04753299 对淋球菌分离株具有杀菌作用,对大肠杆菌、铜绿假单胞菌和肺炎菌株的抑制的MIC90值分别为 2 μg/ml、4 μg/ml 和 16 μg/ml。PF-04753299 用于革兰氏阴性菌感染的研究。
T77574 ROS inducer 1

ROS; Antibiotic Immunology/Inflammation; Microbiology/Virology
ROS inducer 1 是一种具有杀菌作用的小分子化合物,对 Xanthomonas axonopodis pv. citri (Xac)、Xanthomonas oryzae pv. oryzae (Xoo)和 Pseudomonas syringae pv. actinidiae (Psa) 具有抑制作用。ROS inducer 1 诱 Xanthomonas 细胞内 ROS 的产生可用于研究农作物细菌感染。
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T1224 Cefuroxime sodium

Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin

Antibacterial; Antibiotic Microbiology/Virology
Cefuroxime sodium (Cefuroxime sodium salt) 是一种具有口服活性的头孢菌素抗生素,增加了对 β-内酰胺酶的稳定性。
T1122 Cephalothin sodium

头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性,抑制革兰氏阳性和阴性菌。
T1063 Ticarcillin disodium

Ticarpen,Ticarcillin disodium salt,替卡西林二钠

Antibacterial; Antibiotic Microbiology/Virology
Ticarcillin disodium (Ticarpen) 主要用于抗革兰氏阴性菌, 特别是绿脓杆菌, 也是少数可研究嗜麦芽感染的抗生素。
T35976 6-Formylpterin

Pterin-6-aldehyde,6 Formylpterin

Apoptosis; NOS; Xanthine Oxidase; Antibacterial Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology
6-Formylpterin (Pterin-6-aldehyde) 是 Xanthine Oxidase 的抑制剂(Ki约为0.6 nM),对沙鼠的短暂性IRI具有强大的神经保护作用。6-Formylpterin 诱导 HL-60 细胞内ROS 生成以及细胞凋亡 (apoptosis)。6-Formylpterin 抑制iNOS的表达,可在细胞内产生过氧化氢并恢复人中性粒细胞杀菌活性受损。
T22390 Olanexidine Hydrochloride semihydrate

OPB-2045,OPB-2045G,奥兰西丁标准品HCL

Others Others
Olanexidine is a monobiguanide compound with the activity of bactericidal.
T29505 A039

A-039,A 039

Others Others
A039 is a highly active bactericidal agent against M. tuberculosis.
T23613 ACH-702

Others Others
ACH-702 is an agent of anti-tubercular. ACH-702 is an effective, bactericidal compound with activity against many antibiotic-resistant pathogens.
T13326 SPR719

VXc-486

Others Others
SPR719 is an inhibitor of gyrase B, has bactericidal activity.
T38801 Fobrepodacin

SPR720,pVXc-486

Others Others
Fobrepodacin (SPR720) is an orally active and potent phosphate prodrug of SPR719 (VXc-486). Fobrepodacin has potent bactericidal activities in vivo.
T68809 Trichomonacid

Others Others
Trichomonacid is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro.
T69488 CB5255829

Others Others
CB5255829 is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro.
T71846 CB6513745

Others Others
CB6513745 is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro.
T61951 Oxacillin

Others Others
Oxacillin 是口服有效的合成青霉素。Oxacillin 对葡萄球菌和其他革兰氏阳性病原体具有良好的杀菌 (bactericidal) 活性。

化合物

Macozinone
Cat.No: T3583
Synonym: PBTZ169
Target: Antibacterial, DprE1
Monolaurin
Cat.No: T7872
Synonym:
Target: Others
Nafcillin sodium monohydrate
Cat.No: T1312
Synonym: CL 8491,萘夫西林钠,nafcillin sodium
Target: Antibacterial, Antibiotic
Micronomicin
Cat.No: T16073
Synonym: 小诺霉素,Gentamicin C2b,Antibiotic XK-62-2,Sagamicin
Target: Others, Antibacterial
Ethylhydrocupreine hydrochloride
Cat.No: T40417
Synonym: Optochin hydrochloride,乙氢去甲奎宁盐酸盐;奥普托欣盐酸盐
Target: Antibacterial, Parasite
Cefaclor monohydrate
Cat.No: T1495
Synonym: Cefaclor,头孢克洛一水物,头孢克洛一水合物,Cefaclorum,Cefachlor
Target: Antibacterial, Antibiotic
5-Nitro-1,10-phenanthroline
Cat.No: T7735
Synonym: 5-NP,5-硝基-1,10-菲咯啉
Target: Antibacterial
Carbenicillin disodium
Cat.No: T1143
Synonym: BRL-2064,羧苄青霉素钠,Sodium carbenicillin
Target: Cell wall, Antibacterial, Antibiotic
Lysozyme from chicken egg white
Cat.No: T3247
Synonym: 鸡蛋清溶菌酶,溶菌酶,Lysozyme
Target: Others, Antibacterial
DDAC
Cat.No: T64346
Synonym: Quaternium 12
Target: Antibacterial
Hexetidine
Cat.No: T0328
Synonym: NSC-17764,海克替啶
Target: Antibacterial, Antifungal
MGB-BP-3
Cat.No: T16071
Synonym:
Target: DNA/RNA Synthesis, Antibiotic
(6R,7S)-Cefminox sodium heptahydrate
Cat.No: T3263
Synonym: Meicelin,头孢米诺钠,Cefminox Sodium,Alteporina,Tencef
Target: Antibiotic
6,6'-Dimethyl-2,2'-dipyridyl
Cat.No: T72030
Synonym: 6,6'-Bi-2-picoline
Target: Others
Taurolidine
Cat.No: T7533
Synonym:
Target: Apoptosis, Others, Antibacterial, Antibiotic
BTZ043
Cat.No: T3582
Synonym:
Target: Antibacterial, Antibiotic, DprE1
Cefditoren pivoxil
Cat.No: T1405
Synonym: 头孢妥仑匹酯,ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl
Target: Antibacterial, Antibiotic
Pyrithione
Cat.No: T12593
Synonym: 1-hydroxyl-1H-pyridine-2-thione,吡啶硫酮
Target: Others
Dihydrostreptomycin sulfate
Cat.No: T2211
Synonym: Dihydrostreptomycin sesquisulfate,双氢链霉索
Target: Antibacterial, Antibiotic
Olanexidine hydrochloride
Cat.No: T28229
Synonym: OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045
Target: Antibacterial
Ceforanide
Cat.No: T5022
Synonym:
Target: Antibacterial, Antibiotic
Antimicrobial agent-22
Cat.No: T79468
Synonym: THI 6c
Target: Antibacterial
Ticarcillin sodium
Cat.No: T6706
Synonym: Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen
Target: Others, Antibacterial, Antibiotic
Cephradine
Cat.No: T0199
Synonym: Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定
Target: TOPK, Antibacterial, Antibiotic
Diphenyleneiodonium chloride
Cat.No: T7191
Synonym: 二苯基氯化碘盐,DPI
Target: NOS, Reactive Oxygen Species, NADPH, TRP/TRPV Channel
Ceftazidime
Cat.No: T1305
Synonym: GR20263,头孢他啶
Target: Antibacterial, Antibiotic
Cefepime Dihydrochloride Monohydrate
Cat.No: T0868
Synonym: Cefepime HCl,头孢吡肟二盐酸盐一水合物
Target: Antibacterial, Antibiotic, Antifection
Amoxicillin trihydrate
Cat.No: T1005L
Synonym: Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate
Target: Antibacterial, Antibiotic
Clofazimine
Cat.No: T0377
Synonym: NSC-141046,氯法齐明,氯苯吩嗪
Target: DNA, Antibacterial, Antibiotic
G907
Cat.No: T11348
Synonym:
Target: Antibiotic
Polymyxin B nonapeptide acetate
Cat.No: TP1341L
Synonym: Polymyxin B nonapeptide acetate(86408-36-8 free base)
Target: Antibacterial, Antibiotic
Cefazolin sodium
Cat.No: T0953
Synonym: Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin
Target: Others, Antibacterial, Antibiotic
Ac-Pro-Gly-Pro-OH
Cat.No: T76662
Synonym:
Target: Apoptosis, CXCR, Antibiotic
Piperacillin sodium
Cat.No: T1213
Synonym: 哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt
Target: Antibacterial, Antibiotic
PF-04753299
Cat.No: T41275
Synonym:
Target: Others
ROS inducer 1
Cat.No: T77574
Synonym:
Target: ROS, Antibiotic
Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
Cefuroxime sodium
Cat.No: T1224
Synonym: Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin
Target: Antibacterial, Antibiotic
Cephalothin sodium
Cat.No: T1122
Synonym: 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin
Target: Antibacterial, Antibiotic
Ticarcillin disodium
Cat.No: T1063
Synonym: Ticarpen,Ticarcillin disodium salt,替卡西林二钠
Target: Antibacterial, Antibiotic
6-Formylpterin
Cat.No: T35976
Synonym: Pterin-6-aldehyde,6 Formylpterin
Target: Apoptosis, NOS, Xanthine Oxidase, Antibacterial
Olanexidine Hydrochloride semihydrate
Cat.No: T22390
Synonym: OPB-2045,OPB-2045G,奥兰西丁标准品HCL
Target: Others
A039
Cat.No: T29505
Synonym: A-039,A 039
Target: Others
ACH-702
Cat.No: T23613
Synonym:
Target: Others
SPR719
Cat.No: T13326
Synonym: VXc-486
Target: Others
Fobrepodacin
Cat.No: T38801
Synonym: SPR720,pVXc-486
Target: Others
Trichomonacid
Cat.No: T68809
Synonym:
Target: Others
CB5255829
Cat.No: T69488
Synonym:
Target: Others
CB6513745
Cat.No: T71846
Synonym:
Target: Others
Oxacillin
Cat.No: T61951
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T20198 Potassium gluconate

Kalium-beta,Kalium Gluconate,Kaon elixir,Kaon,Potassium D-gluconate,HSDB 3165,K-Iao

Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology
Potassium gluconate (Potassium D-gluconate) 是一种具有口服活性和螯合性质的氧化型羧酸,具有杀菌活性。
T1029 Aztreonam

SQ-26,776,氨曲南

Antibacterial; Antibiotic Microbiology/Virology
Aztreonam (SQ-26,776) 是单环β-内酰胺抗生素,与青霉素结合蛋白3有较高亲和力。
T0832 Vancomycin hydrochloride

盐酸万古霉素,Vancomycin HCl

Cell wall; Antibacterial; Antibiotic; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Vancomycin hydrochloride (Vancomycin HCl) 是Vancomycin 的盐酸盐,是一种支链三环糖基化肽,对大多数生物体具有杀菌活性,对肠球菌具有抑菌作用。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
T0814L Ampicillin

Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin (Aminobenzylpenicillin) 属于 β-内酰胺类抗生素,是一种半合成的青霉素。Ampicillin 具有杀菌活性,对各种革兰氏阳性细菌和革兰氏阴性细菌均有抑制活性。
T1104 Paromomycin Sulfate

Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Paromomycin Sulfate (Aminosidine sulfate) 是一种广谱氨基糖苷类抗生素 ,是具有杀螨杀菌作用的新霉素衍生物。它通过与细菌 30S 核糖体 A 位点的 RNA 寡核苷酸特异性结合,使 mRNA 的翻译提前终止,并抑制蛋白质合成。它可研究细菌和寄生虫感染。
T1165 Ethionamide

Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide

Dehydrogenase; CAT; Antibacterial; Antibiotic Metabolism; Microbiology/Virology; oxidation-reduction
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。
T3123 Allicin

ERK; IL Receptor; Others; IκB/IKK; p38 MAPK; TNF; ROS; Caspase; Antifection Apoptosis; Immunology/Inflammation; MAPK; Microbiology/Virology; NF-κB; Others; Proteases/Proteasome
Allicin 具有抗氧化、杀菌、抗癌、抗炎活性,对肠上皮细胞具有抑制性免疫调节作用。 Allicin 能显着抑制胰岛素诱导的血管平滑肌细胞的增殖和迁移,这可能与抑制 ERK 信号通路的激活有关。 Allicin 有利于降低高胆固醇血症大鼠的血液胆固醇、甘油三酯水平和收缩压,它可能有益于影响动脉粥样硬化的两个危险因素——高脂血症和高血压。
T40797 Essential oils, Melaleuca alternifolia

Others Others
Melaleuca alternifolia essential oil, derived from the leaves of Melaleuca alternifolia, exhibits bactericidal and anti-inflammatory properties.
TN2760 2-Hydroxy-1,8-cineole

Antifection Microbiology/Virology
1. 2-endo-Hydroxy-1,8-cineole shows antimicrobial and bactericidal activities against against test bacteria (Staphylococcus aureus, Escherichia coli, and Pseudomonas fluorescens) .<BR/>
TN3177 6-Methyl-5,6-dihydropyran-2-one

Antifection Microbiology/Virology
6-Methyl-5,6-dihydropyran-2-on is bactericidal,and antiprotozoal agents.
TN4944 Santamarine

Caspase Apoptosis; Proteases/Proteasome
Santamarine has significant anticancer activity, can inhibit L1210 cells because of its cytotoxic,cytostatic and blocking mitosis and reducing uptake of thymidine. Santamarine and reynosin show bactericidal activity against clinical strains of Mycobacterium tuberculosis.
T10928 Cytochalasin A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), inhibits actin polymerization and interferes with microtubule assembly by reacting with sulfhy
T13970 Xinjiachalcone A

Others Others
Xinjiachalcone A is a natural product isolated from Glycyrrhiza inflata Batalin. Xinjiachalcone A shows both a low MIC and a strong bactericidal activity against H. pylori(MIC : 12.5 to 50 µM, seventeen H. pylori strains).
T80357 Bombinin H7

Others Others
Bombinin H7 是一种抗菌肽,提取自铃蟾Bombina的皮肤分泌物。该化合物对Bacillus megateriumBm11显示出高效活性,其致死浓度达到25.2 μM。
TN1407 Artocarpin

Antibiotic Microbiology/Virology
Artocarpin 是一种从 Artocarpus heterophyllus 的木材中分离出来的黄酮类化合物,具有杀菌活性,抑制耐多药金黄色葡萄球菌和肠球菌属细菌。Artocarpin 可抑制 B16 黑色素瘤细胞中黑色素的生物合成,诱导快速细胞裂解。Artocarpin 可用于研究皮肤病。
T80360 Bombinin H4

Others Others
Bombinin H4,蛾Bombina variegata皮肤中的抗菌肽,其对大肠杆菌D21和金黄色葡萄球菌Cowan 1的致死浓度分别为4.8 μM和3.3 μM。
TN4437 Licorisoflavan A

MMP; IL Receptor; NF-κB; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; NF-κB; Proteases/Proteasome
Licorisoflavan A shows weak scavenging activity against superoxide anion radical, it and licoricidin have potential for the development of novel host-modulating strategies for the treatment of cytokine and/or MMP-mediated disorders such as periodontitis.L

天然产物

Potassium gluconate
Cat.No: T20198
Synonym: Kalium-beta,Kalium Gluconate,Kaon elixir,Kaon,Potassium D-gluconate,HSDB 3165,K-Iao
Target: Endogenous Metabolite, Antifungal
Aztreonam
Cat.No: T1029
Synonym: SQ-26,776,氨曲南
Target: Antibacterial, Antibiotic
Vancomycin hydrochloride
Cat.No: T0832
Synonym: 盐酸万古霉素,Vancomycin HCl
Target: Cell wall, Antibacterial, Antibiotic, Autophagy
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Ampicillin
Cat.No: T0814L
Synonym: Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid
Target: Antibacterial, Antibiotic
Paromomycin Sulfate
Cat.No: T1104
Synonym: Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐
Target: Antibacterial, Antibiotic, Parasite
Ethionamide
Cat.No: T1165
Synonym: Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide
Target: Dehydrogenase, CAT, Antibacterial, Antibiotic
Allicin
Cat.No: T3123
Synonym:
Target: ERK, IL Receptor, Others, IκB/IKK, p38 MAPK, TNF, ROS, Caspase, Antifection
Essential oils, Melaleuca alternifolia
Cat.No: T40797
Synonym:
Target: Others
2-Hydroxy-1,8-cineole
Cat.No: TN2760
Synonym:
Target: Antifection
6-Methyl-5,6-dihydropyran-2-one
Cat.No: TN3177
Synonym:
Target: Antifection
Santamarine
Cat.No: TN4944
Synonym:
Target: Caspase
Cytochalasin A
Cat.No: T10928
Synonym:
Target: HIV Protease
Xinjiachalcone A
Cat.No: T13970
Synonym:
Target: Others
Bombinin H7
Cat.No: T80357
Synonym:
Target: Others
Artocarpin
Cat.No: TN1407
Synonym:
Target: Antibiotic
Bombinin H4
Cat.No: T80360
Synonym:
Target: Others
Licorisoflavan A
Cat.No: TN4437
Synonym:
Target: MMP, IL Receptor, NF-κB, DNA/RNA Synthesis
Cat. No. Product Name Species Expression System
TMPY-02908 BPI Protein, Human, Recombinant (His)

BPIFD1,bactericidal/permeability-increasing protein...

Human HEK293 Cells
Bactericidal/permeability-increasing protein is a member of the BPI/LBP/Plunc superfamily and BPI/LBP family. It is a cationic protein which can be detected in the azurophilic granule and on the surface of polymorphonuclear leukocytes. Bactericidal/permeability-increasing protein also is a lipopolysaccharide binding protein. It is associated with human neutrophil granules and has bactericidal activity on gram-negative organisms. Bactericidal/permeability-increasing protein contains two domains t...
TMPH-03101 DEFB1 Protein, Pig, Recombinant (GST)

DEFB1,Defensin, beta 1,Beta-defensin 1,BD-1

Sus scrofa (Pig) E. coli
Has bactericidal activity. May act as a ligand for C-C chemokine receptor CCR6. Positively regulates the sperm motility and bactericidal activity in a CCR6-dependent manner. Binds to CCR6 and triggers Ca2+ mobilization in the sperm which is important for its motility. DEFB1 Protein, Pig, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 31.1 kDa and the accession number is O62697.
TMPH-02879 REG3G Protein, Mouse, Recombinant (His)

Regenerating islet-derived protein III-gamma,Reg3g,Pancreati...

Mouse P. pastoris (Yeast)
Bactericidal C-type lectin which acts exclusively against Gram-positive bacteria and mediates bacterial killing by binding to surface-exposed carbohydrate moieties of peptidoglycan. Restricts bacterial colonization of the intestinal epithelial surface and consequently limits activation of adaptive immune responses by the microbiota. The uncleaved form has bacteriostatic activity, whereas the cleaved form has bactericidal activity against L.monocytogenes and methicillin-resistant S.aureus. Regula...
TMPH-02541 Beta Defensin 1/DEFB1 Protein, Mouse, Recombinant (His & SUMO)

Beta-defensin 1,BD-1,mBD-1,Defensin, beta 1,Defb1

Mouse E. coli
Has bactericidal activity. May act as a ligand for C-C chemokine receptor CCR6. Positively regulates the sperm motility and bactericidal activity in a CCR6-dependent manner. Binds to CCR6 and triggers Ca2+ mobilization in the sperm which is important for its motility.
TMPH-00314 Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI)

Lingual antimicrobial peptide

Bubalus bubalis E. coli
Has bactericidal activity. Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 19.8 kDa and the accession number is A3RJ36.
TMPK-01201 BPIFA1/LUNX Protein, Human, Recombinant

Lung-specific protein X,BPI fold-containing family A member ...

Human E. coli
Bactericidal/permeability-increasing fold containing family A, member 1 (BPIFA1) is a secretory protein found in human upper aerodigestive tract mucosa. This innate material is secreted in mucosal fluid or found in submucosal tissue in the human soft palate, lung, uvula, and nasal cavity. BPIFA1 is a critical component of the innate immune response that prevents upper airway diseases.
TMPH-03365 REG3A Protein, Rat, Recombinant (E.coli, His)

Lithostathine 3,Reg3a,RegIII,Regenerating islet-derived prot...

Rat E. coli
Bactericidal C-type lectin. Regulates keratinocyte proliferation and differentiation after skin injury via activation of EXTL3-PI3K-AKT signaling pathway. REG3A Protein, Rat, Recombinant (E.coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 20.5 kDa and the accession number is P35231.
TMPH-02507 Angiogenin-4 Protein, Mouse, Recombinant (His & Myc & SUMO)

EC:3.1.27.-,Angiogenin-4,Ang4

Mouse E. coli
Has bactericidal activity against E.faecalis and L.monocytogenes, but not against L.innocua and E.coli. Promotes angiogenesis (in vitro). Has low ribonuclease activity (in vitro). Promotes proliferation of melanoma cells, but not of endothelial cells or fibroblasts (in vitro). Angiogenin-4 Protein, Mouse, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO and C-Myc tag. The predicted molecular weight is 31.4 kDa and the accession number is Q3TMQ6.
TMPH-02019 REG3A Protein, Human, Recombinant (GST)

Regenerating islet-derived protein 3-alpha,REG3A,Regeneratin...

Human E. coli
Bactericidal C-type lectin which acts exclusively against Gram-positive bacteria and mediates bacterial killing by binding to surface-exposed carbohydrate moieties of peptidoglycan. Regulates keratinocyte proliferation and differentiation after skin injury via activation of EXTL3-PI3K-AKT signaling pathway. REG3A Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 43.6 kDa and the accession number is Q06141.
TMPH-02508 Angiogenin-4 Protein, Mouse, Recombinant (His & SUMOstar)

Ang4,Angiogenin-4,EC:3.1.27.-

Mouse P. pastoris (Yeast)
Has bactericidal activity against E.faecalis and L.monocytogenes, but not against L.innocua and E.coli. Promotes angiogenesis (in vitro). Has low ribonuclease activity (in vitro). Promotes proliferation of melanoma cells, but not of endothelial cells or fibroblasts (in vitro). Angiogenin-4 Protein, Mouse, Recombinant (His & SUMOstar) is expressed in yeast with N-6xHis-sumostar tag. The predicted molecular weight is 29.9 kDa and the accession number is Q3TMQ6.
TMPH-02046 Ribonuclease 7 Protein, Human, Recombinant (His)

RNASE7,Skin-derived antimicrobial protein 2,Ribonuclease 7

Human E. coli
Exhibits a potent RNase activity. Has broad-spectrum antimicrobial activity against many pathogenic microorganisms and remarkably potent activity (lethal dose of 90% < 30 nM) against a vancomycin resistant Enterococcus faecium. Causes loss of bacterial membrane integrity. Probably contributes to urinary tract sterility. Bactericidal activity is independent of RNase activity. Ribonuclease 7 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted...
TMPH-02670 Gasdermin-A3 Protein, Mouse, Recombinant (His)

Gsdma3,Gasdermin-3,Gasdermin-A3

Mouse E. coli
Precursor of a pore-forming protein involved in the transition from catagen to telogen at the end of hair follicle morphogenesis. This form constitutes the precursor of the pore: upon cleavage, the released N-terminal moiety (Gasdermin-A3, N-terminal) binds to membranes and forms pores, triggering cell death.; Pore-forming protein that causes membrane permeabilization and pyroptosis. Released upon cleavage in vitro of genetically engineered Gsdma3, and binds to membrane inner leaflet lipids. Hom...
TMPY-02163 PGLYRP1 Protein, Mouse, Recombinant (His)

Tnfsf3l,peptidoglycan recognition protein 1,PGRP,Tasg7,Tag7,...

Mouse HEK293 Cells
Peptidoglycan recognition protein 1, also known as Peptidoglycan recognition protein short, PGRP-S, PGLYRP1, PGLYRP, PGRP and TNFSF3L, is a secreted protein that belongs to the N-acetylmuramoyl-L-alanine amidase 2 family. PGLYRP1 / PGLYRP is highly expressed in bone marrow. It is weakly expressed in kidney, liver, small intestine, spleen, thymus, peripheral leukocyte, lung, fetal spleen and neutrophils. PGLYRP1 / PGLYRP is a pattern receptor that binds to murein peptidoglycans (PGN) of Gram-posi...
TMPH-02671 Gasdermin-D Protein, Mouse, Recombinant (His & Myc)

Gasdermin-D,Gasdermin domain-containing protein 1,Gsdmd

Mouse E. coli
Precursor of a pore-forming protein that plays a key role in host defense against pathogen infection and danger signals. This form constitutes the precursor of the pore-forming protein: upon cleavage, the released N-terminal moiety (Gasdermin-D, N-terminal) binds to membranes and forms pores, triggering pyroptosis.; Promotes pyroptosis in response to microbial infection and danger signals. Produced by the cleavage of gasdermin-D by inflammatory caspases CASP1 or CASP4/CASP11 in response to canon...
TMPH-02690 PLA2G10 Protein, Mouse, Recombinant (His & Myc)

Pla2g10,Group X secretory phospholipase A2,Phosphatidylcholi...

Mouse E. coli
Secretory calcium-dependent phospholipase A2 that primarily targets extracellular phospholipids. Hydrolyzes the ester bond of the fatty acyl group attached at sn-2 position of phospholipids with preference for phosphatidylcholines and phosphatidylglycerols over phosphatidylethanolamines. Preferentially releases sn-2 omega-6 and omega-3 polyunsaturated fatty acyl (PUFA) chains over saturated fatty acyls. Contributes to phospholipid remodeling of very low-density lipoprotein (VLDL), low-density li...

重组蛋白

BPI Protein, Human, Recombinant (His)
Cat.No: TMPY-02908
Species: Human
Expression System: HEK293 Cells
DEFB1 Protein, Pig, Recombinant (GST)
Cat.No: TMPH-03101
Species: Sus scrofa (Pig)
Expression System: E. coli
REG3G Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02879
Species: Mouse
Expression System: P. pastoris (Yeast)
Beta Defensin 1/DEFB1 Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02541
Species: Mouse
Expression System: E. coli
Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI)
Cat.No: TMPH-00314
Species: Bubalus bubalis
Expression System: E. coli
BPIFA1/LUNX Protein, Human, Recombinant
Cat.No: TMPK-01201
Species: Human
Expression System: E. coli
REG3A Protein, Rat, Recombinant (E.coli, His)
Cat.No: TMPH-03365
Species: Rat
Expression System: E. coli
Angiogenin-4 Protein, Mouse, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-02507
Species: Mouse
Expression System: E. coli
REG3A Protein, Human, Recombinant (GST)
Cat.No: TMPH-02019
Species: Human
Expression System: E. coli
Angiogenin-4 Protein, Mouse, Recombinant (His & SUMOstar)
Cat.No: TMPH-02508
Species: Mouse
Expression System: P. pastoris (Yeast)
Ribonuclease 7 Protein, Human, Recombinant (His)
Cat.No: TMPH-02046
Species: Human
Expression System: E. coli
Gasdermin-A3 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02670
Species: Mouse
Expression System: E. coli
PGLYRP1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02163
Species: Mouse
Expression System: HEK293 Cells
Gasdermin-D Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02671
Species: Mouse
Expression System: E. coli
PLA2G10 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02690
Species: Mouse
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMID-0004 Ampicillin-d5

Ampicillin-d5 是 Ampicillin 的氘代化合物。Ampicillin 的 CAS 号为 69-53-4。Ampicillin是一种广谱、半合成的β-内酰胺类青霉素抗生素,具有杀菌活性。

同位素标记化合物

Ampicillin-d5
Cat.No: TMID-0004
Synonym:
Target:
TargetMol Loading
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