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TargetMol | Compound Library

药物功能重定位化合物库现货

Drug Repurposing Compound Library

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产品编号 L9200

传统的药物开发涉及从头确认和验证新分子实体,这是一个耗时且成本高昂的过程,随着对药物安全性及有效性的要求不断提高,开发新药的成本还将持续上涨。由于时间和成本大幅降低,近年来药物功能重定位受到越来越多关注,高内涵筛选、新的生物标志物发现和生物信息学的快速发展为基于靶点或细胞的药物重定位创造了机会。 TargetMol 药物功能重定位化合物库收集了4960 种已上市和进入临床期的药物,这些化合物经过大量的临床前研究实验,具有活性高、毒性低和机制明确的特点,适用于药物筛选的同时,也是细胞诱导分化的有力工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L9200

药物功能重定位化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 4960种全球上市药物和临床药物的独特集合,可用于高通量筛选和高内涵筛选,是老药新用、新的药物靶点筛选和细胞诱导的有效工具。
  • 是整个行业规模领先的药物功能重定位化合物库;
  • 所有上市化合物得到FDA、EMA、NMPA等权威部门审批或收录在USP、EP、BP、JP、CP等药典文献中;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎/免疫、神经系统药物、呼吸系统药物等;
  • 靶点多样,包括5-HT Receptor、Sodium Channel、p38 MAPK、PI3K、MEK等;
  • 详细的说明书,化合物结构、靶点信息、适应症信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Autophagy
Antibacterial
Apoptosis
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
AChR
Dopamine Receptor
Histamine Receptor
COX
HIV Protease
Parasite
DNA/RNA Synthesis
Antifungal
Sodium Channel
Potassium Channel
Calcium Channel
VEGFR
EGFR
Topoisomerase
PDE
Glucocorticoid Receptor
PI3K
Reactive Oxygen Species
SARS-CoV
Cytochromes P450
CDK
Estrogen/progestogen Receptor
Dehydrogenase
HCV Protease
FLT
Influenza Virus
Ferroptosis
PPAR
NF-κB
GABA Receptor
PDGFR
Microtubule Associated
JAK
c-Kit
HDAC
FGFR
RAAS
c-Met/HGFR
Estrogen Receptor/ERR
mTOR
HBV
Prostaglandin Receptor
Mitophagy
Nucleoside Antimetabolite/Analog
Src
Adenosine Receptor
Androgen Receptor
Reverse Transcriptase
Tyrosine Kinases
Serotonin Transporter
iGluR
Bcr-Abl
NMDAR
HSV
Cholinesterase (ChE)
GPR
TRP/TRPV Channel
Norepinephrine
Proteasome
BTK
GluR
Virus Protease
MAO
Raf
HER
ATPase
ADC Cytotoxin
Phosphatase
PARP
Antiviral
ribosome
TNF
Progesterone Receptor
Opioid Receptor
Epigenetic Reader Domain
Akt
HSP
p38 MAPK
Antioxidant
ROS
Beta Amyloid
Carbonic Anhydrase
Transferase
PKC
Aurora Kinase
ALK
IL Receptor
P-gp
HIF/HIF Prolyl-Hydroxylase
Proton pump
Antifection
MMP
MEK
Histone Methyltransferase
DPP-4
Monoamine Oxidase
Thyroid hormone receptor(THR)
DNA Alkylator/Crosslinker
Drug Metabolite
Mitochondrial Metabolism
Endothelin Receptor
TLR
c-RET
Thrombin
ERK
Interleukin
Trk receptor
Bcl-2 Family
AMPK
Phospholipase
GSK-3
P2X Receptor
CXCR
Retinoid Receptor
c-Fms
HMG-CoA Reductase
Integrin
MRP
GNRH Receptor
Caspase
ROCK
CCR
Lipoxygenase
SGLT
STAT
TAM Receptor
S1P Receptor
PKA
Gamma-secretase
Vasopressin Receptor
Chk
Neurokinin receptor
FAK
p53
NO Synthase
DNA-PK
NADPH
Factor Xa
E1/E2/E3 Enzyme
Guanylate cyclase
DNA Alkylation
HIF
Cannabinoid Receptor
Syk
CFTR
LPL Receptor
Reductase
Wnt/beta-catenin
Antifolate
DNA gyrase
TGF-beta/Smad
Nrf2
Kras
DHFR
Amino Acids and Derivatives
P2Y Receptor
Glutathione Peroxidase
Serine Protease
FXR
Hedgehog/Smoothened
IGF-1R
RSV
Sigma receptor
ROS Kinase
Histone Demethylase
IAP
CSF-1R
ATM/ATR
Hydroxylase
PLK
Tyrosinase
Mdm2
Chloride channel
NOS
CETP
Leukotriene Receptor
ABC Transporter
Glucosidase
OX Receptor
CaMK
Indoleamine 2,3-Dioxygenase (IDO)
DNA Methyltransferase
S6 Kinase
Kinesin
BACE
JNK
Cholecystokinin Receptor
Cysteine Protease
Vitamin
Smo
Xanthine Oxidase
Ligand for E3 Ligase
NOD
Glucokinase
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RIP kinase
Glucagon Receptor
DNA
Beta-Secretase
Acyltransferase
Aminopeptidase
Sirtuin
Casein Kinase
Aromatase
ROR
Pim
Monoamine Transporter
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Fatty Acid Synthase
PAK
Bradykinin Receptor
PGE Synthase
IκB/IKK
GHSR
CGRP Receptor
Gap Junction Protein
IRAK
AhR
LTR
IFNAR
Cell wall
Tie-2
IDO
MT Receptor
GlyT
FAAH
MAPK
GPCR19
Ephrin Receptor
CRFR
Melanocortin Receptor
Complement System
NADPH-oxidase
Imidazoline Receptor
PROTACs
CRM1
DprE1
YAP
Melatonin Receptor
CaSR
Serine/threonin kinase
Liver X Receptor
Annexin A
UGT
Neuropeptide Y Receptor
Somatostatin
KSP
Lipid
Wee1
OAT
STING
Decarboxylase
Neprilysin
GST
Acetyl-CoA Carboxylase
LPA Receptor
PDK
Anti-infection
Ras
Protease-activated Receptor
NOD-like Receptor (NLR)
PD-1/PD-L1
Monocarboxylate transporter
Arginase
PERK
Rho
NAMPT
PYK2
Glutaminase
Myosin
LDL
Na-K-Cl cotransporter
Hexokinase
Epoxide Hydrolase
Mucin
DUB
Telomerase
Free radical scavengers
transporter
Oxytocin Receptor
Adenosine Deaminase
Advanced Glycation End Products
Taste receptor
GSNOR
NEDD8
Ligands for Target Protein for PROTAC
Lipase
TOPK
VDA
c-Myc
Galectin
Kisspeptin
IRE1
FLAP
Phosphorylase
Integrase
HCN Channel
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Glutathione reductase
Porcupine
CD73
GluCls
PAI-1
Aquaporin
Discoidin Domain Receptor (DDR)
p97
MLK
PKM
Apelin receptor
Adenylyl Cyclase
NPC1L1
Hydrogenase
MALT
Dynamin
Na+/Ca2+ Exchanger
Arrestin
RAR/RXR 
DYRK
gp120/CD4
GTPase
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
LIM Kinase
Neurotensin Receptor
Stemness kinase
Immunology/Inflammation related
SIK
Adiponectin Receptor
PAFR
MTH1
Fas/FasL
GRK
Anion Exchanger
PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
ACK1
Angiotensin-converting Enzyme (ACE)
PAD
cAMP
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ASK
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Hippo pathway
KLF
PI4K
CRISPR/Cas9
RXFP receptor
SGK
Platelet aggregation
BMI-1