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TargetMol | Compound Library

EMA 上市药物库现货

EMA Approved Drug Library

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产品编号 L1020

EMA 上市药物库收录了 670 个欧洲药品监督管理局(EMA)批准的化合物,所有化合物通过临床验证,靶点明确,具有较好的安全性和生物利用度,是进行老药新用理想的工具,可以大大提高药物研发的成功率,能够缩短药物研发周期,节约研发成本。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1020

EMA 上市药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 680个EMA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Autophagy
Apoptosis
Antibiotic
Antibacterial
HIV Protease
5-HT Receptor
Adrenergic Receptor
c-Kit
VEGFR
PDGFR
Endogenous Metabolite
Sodium Channel
DNA/RNA Synthesis
Dopamine Receptor
SARS-CoV
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HCV Protease
COX
Potassium Channel
Reverse Transcriptase
Cytochromes P450
Antifungal
Src
Histamine Receptor
Calcium Channel
PDE
JAK
FLT
AChR
Proteasome
Bcr-Abl
Parasite
EGFR
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Glucocorticoid Receptor
Topoisomerase
FGFR
Mitophagy
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RAAS
Estrogen Receptor/ERR
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DPP-4
SGLT
Influenza Virus
ribosome
CFTR
ALK
Microtubule Associated
P2Y Receptor
Transferase
ADC Cytotoxin
Dehydrogenase
Antifolate
TRP/TRPV Channel
MAO
CDK
ROS
P-gp
Androgen Receptor
Prostaglandin Receptor
TNF
GABA Receptor
TAM Receptor
S1P Receptor
LPL Receptor
Progesterone Receptor
PARP
NMDAR
HSV
Norepinephrine
NF-κB
MEK
Monoamine Oxidase
Carbonic Anhydrase
DHFR
Proton pump
Virus Protease
Reactive Oxygen Species
Bcl-2 Family
Molecular Glues
Endothelin Receptor
Trk receptor
Ligand for E3 Ligase
Hydroxylase
Neurokinin receptor
ROS Kinase
Phosphatase
Melatonin Receptor
ATPase
PI3K
Adenosine Receptor
CETP
CaSR
iGluR
Cysteine Protease
Guanylate cyclase
Smo
MMP
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mTOR
c-Fms
Nrf2
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HIF
Chloride channel
ROR
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Ligands for Target Protein for PROTAC
Antioxidant
ROCK
IRE1
DNA gyrase
Mitochondrial Metabolism
Rho
FXR
PKC
Aryl Hydrocarbon Receptor
Drug Metabolite
MT Receptor
ABC Transporter
Antifection
Opioid Receptor
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IL Receptor
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IGF-1R
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Anti-infection
NADPH-oxidase
Sigma receptor
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
NOD-like Receptor (NLR)
Imidazoline Receptor
Kras

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