36
23
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4
3
Cat. No. | Product Name | ||
---|---|---|---|
L2195 | 抗前列腺癌化合物库 | 2070 compounds | |
2070 种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6400 |
AZD3514
|
Androgen Receptor | Endocrinology/Hormones |
AZD3514 是一种口服雄激素受体下调剂(Ki :2.2 μM),能够减少 AR 蛋白表达。 | |||
T0380 |
Bicalutamide
比卡鲁胺,ICI-176334 |
Androgen Receptor; Autophagy | Autophagy; Endocrinology/Hormones |
Bicalutamide (ICI-176334) 是一种具有口服活性的非甾体雄激素受体拮抗剂,可研究前列腺癌。 | |||
T2275 |
YK-4-279
4,7-二氯-1,3-二氢-3-羟基-3-[2-(4-甲氧基苯基)-2-氧代乙基]-2H-吲哚-2-酮 |
Apoptosis; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
YK 4-279是一种RNA 解旋酶A 与致癌转录因子EWS-FLI1结合抑制剂,能抑制ESFT 细胞增长,诱导凋亡。 | |||
T4102 |
Goserelin acetate
醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex |
Apoptosis; GNRH Receptor | Apoptosis; GPCR/G Protein |
Goserelin acetate (Fertilan) 是一种促性腺激素释放激素 (GnRH/LHRH) 十肽类似物,能作为GnRH 激动剂。它可研究乳腺癌、上皮性卵巢癌和前列腺癌。 | |||
T0487 |
Metoprolol tartrate
酒石酸美托洛尔,CGP 2175E |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Metoprolol tartrate 是一种心脏选择性β1肾上腺素阻断剂。 | |||
T11340 |
Furprofen
|
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Furprofen 是一种非甾体类抗炎剂,抑制前列腺 (PGE) 合成,可用于研究类风湿关节炎和骨关节炎。 | |||
T23647 |
Zindoxifene
D 16726 |
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Zindoxifene (D 16726) 是一种抗雌激素化合物,具有抗肿瘤活性,可用于研究乳腺癌和前列腺癌。 | |||
T69564 |
YK-2-69
|
DYRK | Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors |
YK-2-69 是一种高选择性的DYRK2 抑制剂,具有抗前列腺癌作用。 | |||
T39189 |
3,4,5-Trihydroxycinnamic acid decyl ester
|
Apoptosis | Apoptosis |
3,4,5-Trihydroxycinnamic acid decyl ester 是一种胰腺脂肪酶抑制剂,具有抗癌活性,可诱导细胞凋亡。3,4,5-Trihydroxycinnamic acid decyl ester 具有抗肥胖作用,抑制脂质吸收和积累,可用于研究乳腺癌和前列腺癌。 | |||
T0740 |
Metformin hydrochloride
Metformin HCl,盐酸二甲双胍,1, 1-Dimethylbiguanide hydrochloride,1,1-Dimethylbiguanide hydrochloride |
Mitophagy; AMPK; Autophagy | Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling |
Metformin hydrochloride (1,1-Dimethylbiguanide hydrochloride) 是一种抗糖尿病药物,抑制结肠、前列腺等多种 Y 细胞的增殖,具有作为抗 Y 药物的潜在功能。它可以透过血脑屏障,诱导自噬。 | |||
T29110 |
VPC-13163
2,3-dihydro-2,3'-Bi-1H-indole,VPC13163,NSC52361,NSC 52361,VPC 13163 |
Others | Others |
VPC-13163 (NSC-52361) 对 LNCaP 和耐恩杂鲁胺的前列腺癌细胞系 (MR49F) 具有很强的抗增殖活性,而它不影响 AR 独立 PC3 细胞系的生长。它还抑制 LNCaP 和 MR49F 中的前列腺特异性抗原 (PSA) 并降低 AR 靶基因 PSA 和 TMPRSS2 的表达。这些发现表明 VPC-13566 表现出 AR BF3 特定的作用机制。 | |||
T0272 |
Nilutamide
尼鲁米特,RU23908 |
Androgen Receptor | Endocrinology/Hormones |
Nilutamide (RU23908) 是一种非甾体抗雄激素药物,有用于转移性前列腺癌的潜力。 | |||
T60967 |
Atg4B-IN-2
|
Phospholipase; Autophagy | Autophagy; Metabolism |
Atg4B-IN-2 是一种具有有效性的选择性的Atg4B 抑制剂,具有抗癌活性,对 Atg4B 和 PLA2 的活性有抑制作用。Atg4B-IN-2 通过细胞自噬 (autophagy) 来抵抗抗去势抗性前列腺癌药物的抗癌活性。 | |||
T13273 |
UT-34
|
Androgen Receptor | Endocrinology/Hormones |
UT-34 是选择性的、具有口服活性的泛雄激素受体拮抗剂和降解剂,能够作用于野生型 AR (IC50:211.7 nM)、F876L-AR (IC50:262.4 nM)、W741L-AR (IC50:215.7 nM)。它与配体结合结构域和功能 1结构域结合,并需要泛素蛋白酶体途径来降解AR。它有抗前列腺癌的能力。 | |||
T74485 |
STC314
|
Others | Others |
STC314 具有抗感染作用,通过中和胞外组蛋白和中性粒细胞诱捕网来逆转机体过度免疫反应造成的器官损伤,可用于研究脓毒症和急性呼吸窘迫综合征(ARDS)。STC314 可保护脂质双层的稳定性,抑制血小板活化和红细胞损伤。 | |||
T41070 |
LP-184
|
Others | Others |
LP-184 (Compound 6), referred to as an acylfulvene analog, demonstrates the ability to inhibit tumor growth with noteworthy anti-cancer efficacy observed across multiple cell lines, including ovarian, colon, prostate, and pancreatic. | |||
T75057 |
RLA-4842
|
Others | Others |
RLA-4842,含有抗雄激素性质的铁活化剂,表现出对于转移性去势抵抗性前列腺癌(mCRPC)细胞系的抗增殖活性。 | |||
T76955 | Voxalatamab | ||
Voxalatamab (JNJ-63898081) 是一种可结合 PSMA 和 CD3的双特异性 IgG4抗体,具有抗癌活性,可用于前列腺癌研究。 | |||
T75058 |
RLA-5331
|
Others | Others |
RLA-5331,一种含有抗雄激素的铁活化剂,针对(mCRPC)细胞系显示出抗增殖活性。 | |||
T61139 |
HDAC6-IN-3
|
Others | Others |
HDAC6-IN-3 (Compound 14) is a potent anti-prostate cancer agent that acts as an orally active inhibitor of HDAC6. It has IC50 values ranging from 0.02-1.54 μM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, and HDAC10. Additionally, HDAC6-IN-3 also demonstrates effective inhibition of MAO-A (IC50 = 0.79 μM) and LSD1 [1]. | |||
T72785 |
PRMT5:MEP50 PPI
|
Others | Others |
PRMT5:MEP50 PPI是一款新型的抑制剂,专门针对PRMT5:MEP50蛋白-蛋白相互作用,展现了抗肿瘤活性,并对肺癌及前列腺癌细胞具有显著的抗增殖效果。 | |||
T64209 |
Anticancer agent 55
|
Others | Others |
Anticancer Agent 是一种有效的抗癌剂。Anticancer Agent 能够以剂量依赖性方式抑制细胞活力和细胞迁移,诱导细胞凋亡 (apoptosis),表现出抗癌效果。Anticancer Agent 具有潜力进行前列腺癌和乳腺癌的研究。 | |||
T76736 | Abituzumab | ||
Abituzumab (DI17E6) 是一种人源化抗integrinαV 单克隆抗体 (IgG2 型)。Abituzumab 能有效减少FAK、Akt 和ERK 的磷酸化。Abituzumab 可用于癌症,尤其是前列腺癌的研究。 | |||
T68406 |
A-849519
|
Others | Others |
A-849519 is a reversible inhibitor of MetAP2 that has demonstrated anti-angiogenesis and anticancer activity in a number of in vitro and in vivo models. In this study, we evaluated the anticancer activity of A-849519 in a modified Dunning model of androgen-independent prostate cancer and compared its efficacy with TNP-470, an established MetAP2 inhibitor. | |||
T63109 |
Y08284
|
Others | Others |
Y08284 是一种选择性的、高效的、口服具有活力的 CBP bromodomain 抑制剂 (IC50: 4.21 nM)。Y08284 能够抑制前列腺癌细胞系 LNCaP、C4-2B 和 22Rv1 的增殖,并具有抗肿瘤效果。 | |||
T78793 |
MAOA-IN-1
|
Monoamine Oxidase | Neuroscience |
MAOA-IN-1(化合物15)是一种口服有效的MAOA抑制剂,对前列腺癌细胞显示出细胞毒性。该化合物表现出Caco-2渗透性,同时具有较低的CNS渗透性。MAOA-IN-1可以用于研究抗癌和抗炎适应症。 | |||
T79494 |
VEGFR-2-IN-31
|
VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
VEGFR-2-IN-31(compound 3i)是一款针对VEGFR-2的高效抑制剂(IC50=8.93 nM),具有抗前列腺癌的活性。该化合物能够导致细胞周期在S期停滞,并诱导细胞发生凋亡(apoptosis)。 | |||
T63168 |
VEGFR-2-IN-26
|
Others | Others |
VEGFR-2-IN-26 (compound 5h) 是一种 VEGFR-2 的高效抑制剂 (IC50: 15.5 nM)。VEGFR-2-IN-26 对白血病、中枢神经系统、非小肺、卵巢、肾、前列腺和乳腺癌细胞表现出良好的抗增殖作用。 | |||
T79495 |
VEGFR-2-IN-32
|
VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
VEGFR-2-IN-32(Comp 3a)作为一种VEGFR-2的抑制剂,其IC50值为8.93 nM。该化合物对PC-3细胞表现出细胞毒性,IC50为1.22 μM,适用于前列腺癌研究。 | |||
T79668 |
PIK5-12d
|
Autophagy; PROTACs | Autophagy; PROTAC |
PIK5-12d为一种高效的PROTAC PIKfyve降解剂,具有显著的DC50值为1.48 nM。该化合物在多种前列腺癌细胞系中有效诱导细胞质空泡化,同时阻碍自噬流的进行,有效抑制前列腺癌细胞的增殖,并展现出抗肿瘤活性。 | |||
T79674 |
HDAC-IN-64
|
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
HDAC-IN-64 (Compound 13) 为HDAC抑制剂,对HDAC4/6的IC50值为24 nM及85 nM。其对前列腺癌(PCA)细胞表现出抗增殖与抗迁移效果,并能抑制LNCaP和RWPE-1细胞的生长,GI50值分别达到0.32 μM与1.1 μM。 | |||
T61935 |
B-Raf IN 9
|
Others | Others |
B-Raf IN 9 (compound 8b) 是有效的B-Raf 抑制剂(IC50= 24.79 nM)。B-Raf IN 9 将细胞周期阻滞于 G2/M 期,诱导凋亡。B-Raf IN 9 对人前列腺癌 PC-3 细胞表现出较强的抗肿瘤活性(IC50= 7.83 μM)。 | |||
T78801 |
BRD7-IN-2
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
BRD7-IN-2(化合物2-77)是针对前列腺癌细胞的有效BRD7抑制剂,具有对BRD7的选择性但不选择性抑制BRD9,IC50分别为5.4 μM和>300 μM。 | |||
T63391 |
Calpain Inhibitor-2
|
Others | Others |
Calpain Inhibitor-2 是具有亲脂性的钙蛋白酶抑制剂,与黑色素瘤细胞系(A-375和B-16F1)和PC-3前列腺癌细胞相比,他们在体外具有中等到良好的抗增殖效果。Calpain Inhibitor-2 中的化合物3,在基质胶细胞侵袭测定中以2μM 浓度能够抑制了80%的DU-145细胞侵袭。 | |||
T74557 |
α1A-AR Degrader 9c
|
PROTACs | PROTAC |
α1A-AR Degrader 9c(化合物 9c)是一种高效、选择性且可逆的α1A-AR PROTAC降解剂,DC50值为2.86 μM。它通过蛋白酶体途径诱导α1A-AR的降解,并且在抑制PC-3细胞增殖方面表现出活性,IC50为6.12 μM。此外,α1A-AR Degrader 9c展现出在前列腺癌研究中的抗肿瘤潜力。 | |||
T75142 |
Acid Ceramidase-IN-2
|
Others | Others |
Acid Ceramidase-IN-2(compound 1)是一款针对酸性神经酰胺酶(ceramidase)的抑制剂,显示出抗增殖及细胞活性抑制的潜力。有研究表明,该化合物在前列腺癌细胞中可阻止人酸性神经酰胺酶的过度表达,从而揭示了其潜在的抗肿瘤能力。此外,Acid Ceramidase-IN-2被三种α-酮酰胺:GT85、GT98和GT99在体外有效抑制其水解作用。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN7020 |
Astragenol
|
Others | Others |
Astragenol 是合成黄芪醇衍生物的中间体。它的衍生物具有抗炎作用,可用于前列腺癌的研究。 | |||
T2895 |
Lupeol
Fagarasterol,羽扇豆醇,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol |
Apoptosis; Androgen Receptor; Akt | Apoptosis; Cytoskeletal Signaling; Endocrinology/Hormones; PI3K/Akt/mTOR signaling |
Lupeol (Monogynol B) 是一个活跃的五环三萜,具有抗氧化剂、抗肿瘤和抗炎活性。它是一种雄激素受体抑制剂,可研究癌症,特别是雄激素依赖表型和去势抵抗表型的前列腺癌。 | |||
T3324 |
Lycorine
Galanthidine,Narcissine,石蒜碱,Amarylline,Belamarine,Licorine,番石榴碱 |
Apoptosis; Virus Protease; Antibacterial; AChR; Fatty Acid Synthase | Apoptosis; Metabolism; Microbiology/Virology; Neuroscience |
Lycorine (Narcissine) 是从金眼科植物科中提取的一种天然生物碱。它是一种具有口服活性的SCAP 抑制剂,Kd 值 15.24 nM。它也是黑色素瘤血管生成抑制剂,有用于前列腺癌和代谢疾病的研究潜力。 | |||
T2S1158 |
4,5-Dicaffeoylquinic acid
3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C |
Others; HBV; Endogenous Metabolite | Metabolism; Microbiology/Virology; Others |
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。 | |||
T4S1173 |
Agrimol B
仙鹤草酚B,仙鹤草酚 B |
Sirtuin; PPAR | Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism |
Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物,可抑制脂肪形成,降低PPARγ的表达,诱导SIRT1易位和表达。 | |||
T6S1255 |
Ophiopogonin-D
麦冬皂苷D |
ROS | Immunology/Inflammation |
Ophiopogonin-D 通过 RIPK1 显着抑制前列腺细胞的体外和体内生长,OPD 可能被开发为潜在的抗前列腺癌药物。 | |||
T4869 |
D-Allose
阿洛糖,β-D-Allopyranose,D-(+)-ALLOSE |
Others; Endogenous Metabolite | Metabolism; Others |
D-Allose (β-D-Allopyranose) 是内源性代谢产物的一种。 | |||
T14008 |
2,2,5,7,8-Pentamethyl-6-Chromanol
PMC |
Androgen Receptor | Endocrinology/Hormones |
2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) 是维生素 E (α-tocopherol) 的抗氧化部分,能够有效的调节雄激素受体 (androgen receptor) 信号,及抗前列腺癌细胞系的抗癌活性。 | |||
T7990 |
9-hydroxy-4-androstene-3,17-dione
|
Others | Others |
9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。 | |||
T4S2157 |
Campesterol
菜油甾醇,(24R)-5-Ergosten-3β-ol |
Endogenous Metabolite | Metabolism |
Campesterol ((24R)-5-Ergosten-3β-ol) 是一种植物甾醇,具有降胆固醇和抗癌的活性。 | |||
TN1805 |
Isosilybin B
|
Apoptosis; Androgen Receptor | Apoptosis; Endocrinology/Hormones |
Isosilybin B 是一种从水飞蓟中提取的黄酮木脂素,具有抗前列腺癌 (PCA) 活性,对癌细胞增殖有抑制作用,促使 G1 期阻滞和凋亡。Isosilybin B 诱导雄激素受体降解。 | |||
TN1804 |
Isosilybin A
异水飞蓟素 A,异水飞蓟宾A,水飞蓟素 B2 |
Apoptosis; Tyrosinase; PPAR; ABC | Apoptosis; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome |
Isosilybin A 是从水飞蓟中分离出来的一种黄酮木脂素,可抑制癌细胞增殖并诱导 G1 期停滞和凋亡,通过靶向 Akt-NF-κB-雄激素受体轴激活前列腺癌细胞的凋亡机制,具有抗前列腺癌活性。 | |||
T2795 |
Amygdalin
苦杏仁苷,Laetrile |
Others | Others |
Amygdalin (Laetrile) 是一种植物葡萄糖苷,分离自蔷薇果实的果核中,如杏,桃,杏仁,樱桃和李子。 | |||
T3851 |
Vicenin 2
Vicenin -2,维采宁 2,新西兰牡荆苷 |
RAAS | Endocrinology/Hormones |
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。 | |||
T4S2126 |
Ginkgetin
银杏双黄酮,银杏素 |
Apoptosis; Wnt/beta-catenin; COX; STAT; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells |
Ginkgetin 是从银杏叶中分离得到的一种双黄酮,具有抗肿瘤、抗炎、神经保护、抗真菌的作用。它也是 Wnt 信号抑制剂,IC50值为 5.92 μM。 | |||
T1660 |
Silibinin
水飞蓟宾 A,水飞蓟宾,Silibinin A,Silybin,Silymarin I |
Reactive Oxygen Species; Autophagy | Autophagy; Immunology/Inflammation; Metabolism; NF-κB |
Silibinin (Silybin) 是水飞蓟的主要活性成分,具有抗癌和化疗预防作用,能抑制细胞增殖和迁移。 | |||
T6S0735 |
Flavokawain B
黄卡瓦胡椒素B,Flavokavain B,Flavokawin B,2'-Hydroxy-4',6'-Dimethoxychalcone |
Apoptosis; Others | Apoptosis; Others |
Flavokawain B (Flavokavain B) 是从卡瓦醉椒的根提取物中,分离出的查尔酮。它是一种凋亡诱导剂,可抑制各种癌细胞株生长。它以极低的无毒浓度抑制人脑内皮细胞的迁移和血管形成,具有抗血管生成活性。 | |||
T4S0797 |
Berberine
小檗碱,Berberin,Umbellatine,黄连素 |
Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic; Autophagy | Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Berberine (Umbellatine) 属于生物碱类天然产物,可以激活 AMPK、抑制 DNA 拓扑异构酶、诱导 ROS 生成。Berberine 具有抗肿瘤、抗菌、降血糖、降血脂等生物学活性。 | |||
TN6638 |
(E)-6-O-(p-coumaroyl)scandoside methyl ester
|
||
(E)-6-O-(p-coumaroyl)scandoside methyl ester shows moderate anti-proliferation effect on PC3 human androgen-independent prostate cancer cells. | |||
TN1867 |
Licoricidin
|
MMP; VEGFR; ROS | Angiogenesis; Immunology/Inflammation; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
Licoricidin, is a potent anti-metastatic agent, which can markedly inhibit the metastatic and invasive capacity of malignant prostate cancer cells. | |||
TN3737 |
Cycloartane-3,24,25-triol
|
ATPase | Membrane transporter/Ion channel |
Cycloartane-3,24,25-triol has potential for development as an anti-cancer agent against prostate cancer. It reduces the viability of PC-3 and DU145 cell lines with IC50 values of 2.226 ± 0.28 μM and 1.67 ± 0.18 μM respectively. | |||
TN4774 |
Physalin A
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ERK; BCL; p38 MAPK; NF-κB; Androgen Receptor; ROS; JAK; JNK; STAT; p53; Autophagy | Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Endocrinology/Hormones; Immunology/Inflammation; JAK/STAT signaling; MAPK; NF-κB; Stem Cells |
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate cancer cell growth through activation of cell apoptosis and downregulation of androgen receptor ex | |||
T82326 |
Genkwadaphnin
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Genkwadaphnin是一种瑞香烷二萜,能够靶向内输蛋白importin-β1,减少CRPC核心驱动因子在细胞核内的积累,并关闭其下游致癌信号通路。此外,Genkwadaphnin在小鼠体内显现出能显著抑制去势抵抗性前列腺癌(CRPC)发展的抗癌活性。 |
Cat. No. | Product Name | Species | Expression System |
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TMPK-00906 |
PSCA Protein, Mouse, Recombinant (hFc)
UNQ206,PSCA,PRO232 |
Mouse | HEK293 Cells |
Gastric cancer is a deadly malignancy and is a prognostically unfavorable entity with restricted therapeutic strategies available. Prostate stem cell antigen (PSCA) is a glycosylphosphatidylinositol (GPI)-anchored cell surface protein widely expressed in bladder, prostate, and pancreatic cancers. Existing studies have thoroughly recognized the availability of utilizing anti-PSCA CAR-T cells in the treatment of metastatic prostate cancer and non-small-cell lung cancer. PSCA Protein, Mouse, Recomb... | |||
TMPK-00728 |
PSCA Protein, Human, Recombinant (hFc)
UNQ206,PRO232,PSCA |
Human | HEK293 Cells |
Gastric cancer is a deadly malignancy and is a prognostically unfavorable entity with restricted therapeutic strategies available. Prostate stem cell antigen (PSCA) is a glycosylphosphatidylinositol (GPI)-anchored cell surface protein widely expressed in bladder, prostate, and pancreatic cancers. Existing studies have thoroughly recognized the availability of utilizing anti-PSCA CAR-T cells in the treatment of metastatic prostate cancer and non-small-cell lung cancer. PSCA Protein, Human, Recomb... | |||
TMPY-03416 |
TNFAIP8 Protein, Human, Recombinant (His)
GG2-1,tumor necrosis factor, alpha-induced protein 8,SCCS2,S... |
Human | E. coli |
Tumor necrosis factor (TNF)-alpha-induced protein 8 (TNFAIP8) family is a newly identified protein with vital roles in maintaining immune homeostasis. Tumor necrosis factor-alpha-inducible protein 8 (TNFAIP8) is a TNF-alpha inducible anti-apoptotic protein with multiple roles in tumor growth and survival. by the creation of cellular autophagy events, TNFAIP8 promotes cell survival and drug resistance in prostate cancer cells. TNFAIP8 regulates Hippo pathway through interacting with LATS1 to prom... | |||
TMPY-02965 |
MMP-19 Protein, Human, Recombinant
MMP18,matrix metallopeptidase 19,RASI-1 |
Human | E. coli |
MMP19, also known as RASI-1, is a member of the peptidase M1A family. It contains 4 hemopexin-like domains and is expressed in the mammary gland, placenta, lung, pancreas, ovary, small intestine, spleen, thymus, prostate, testis colon, heart, and blood vessel walls. It is a matrix metalloproteinase (MMP). Proteins of the MMP family are involved in the breakdown of extracellular matrix in normal physiological processes, such as embryonic development, reproduction, and tissue remodeling, as well a... |
Cat. No. | Product Name | Target | Signaling Pathways |
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TMIH-0089 |
Androstenedione-d7
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Androstenedione-d7 是 Androstenedione 的氘代化合物。Androstenedione 的 CAS 号为 560-62-3。9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。 | |||
TMIJ-0337 |
(24Rac)-Campesterol-d7
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(24Rac)-Campesterol-d7 是 (24Rac)-Campesterol 的氘代化合物。(24Rac)-Campesterol 的 CAS 号为 474-62-4。Campesterol是一种植物甾醇,具有降胆固醇和抗癌的活性。 | |||
TMIH-0521 |
Silibinin-d3
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Silibinin-d3 是 Silibinin 的氘代化合物。Silibinin 的 CAS 号为 22888-70-6。Silibinin 是水飞蓟的主要活性成分,具有抗癌和化疗预防作用,能抑制细胞增殖和迁移。 |