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Targets Recommended: Others

49

抑制剂 & 化合物

47

天然产物

2

化合物库

6

重组蛋白

1

同位素标记化合物

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Cat. No.	Product Name
L9410	共价抑制剂库		1920 compounds
	1920 种小分子的独特集合，包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子，如氯乙酰基，2-氯丙酰基，丙烯酰基，1-丙-2-炔基，1-丁-2-炔基，酮羰基，二硫键等，可以用于共价抑制剂药物研发；
L7700	神经再生化合物库		524 compounds
	524 种神经再生相关化合物的独特集合，可用于高通量筛选和高内涵筛选；

化合物库

共价抑制剂库

Cat.No: L9410

Compounds: 1920

神经再生化合物库

Cat.No: L7700

Compounds: 524

Cat. No.	Product Name	Target	Signaling Pathways
T22426	Sodium carbonate 碳酸钠,Soda Ash,Disodium carbonate,Carbonic acid disodium salt	Others	Others
	Sodium carbonate (Soda Ash) 又称碳酸二钠、纯碱、碳酸二钠盐，是具有碱化性能的碳酸二钠盐。
T1371	1H-1,2,4-Triazole-3-carboxylic acid	Others	Others
	1H-1,2,4-Triazole-3-carboxylic acid，具有 isoprenyl transferases 抑制蛋白质的特性。
T8520	Tetrazole 1H-TETRAZOLE,1H-四唑	Antibacterial	Microbiology/Virology
	Tetrazole (1H-TETRAZOLE) 是羧酸的生物等排体，具有相当的抗菌性能。
T1144L	Lidocaine Hydrochloride hydrate	EGFR; Sodium Channel	Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
	Lidocaine Hydrochloride hydrate 是一种酰胺类局部麻醉剂，具有抗炎作用。
T7313	Enclomiphene citrate 恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate	Estrogen Receptor/ERR	Endocrinology/Hormones
	Enclomiphene citrate (trans-Clomiphene citrate) 是口服具有活力的 oestrogen receptor 拮抗剂，具有抗雌激素活性。
T65133	3-Hydroxybutyric acid sodium β-Hydroxybutyric acid sodium	Others	Others
	3-Hydroxybutyric acid sodium (β-Hydroxybutyric acid sodium) 是一种存在 I 型糖尿病患者体内的一种代谢物，具有调节膜脂的性质。
T12950	Sodium laureth sulfate Sodium lauryl polyoxyethylene ether sulfate,月桂醇聚氧乙烯醚硫酸酯钠盐	Others	Others
	Sodium laureth sulfate (Sodium lauryl polyoxyethylene ether sulfate) 是一种阴离子活性剂，具有优良的去污，分散，乳化，润湿等性能。
T18890	5-ROX 5-羧基-X-罗丹明,5-Carboxy-X-rhodamine	Others	Others
	5-ROX (5-Carboxy-X-rhodamine) 是罗丹明染料的一种，λexit 为 580 nm (ε=3.6×104M-1cm-1)，λemit 为 604 nm (ϕ=0.94)。
TP1554L	HPV16 E7 (86-93) acetate HPV16 E7 (86-93) acetate(160212-93-1 Free base)	Others	Others
	HPV16 E7 (86-93) acetate 是人源白细胞抗原 A2.1 限制性 HPV16 E7 的衍生肽，在宫颈癌中具有免疫原性。
T1425	Pemirolast potassium BMY 26517,TWT-8152,吡嘧司特钾	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Pemirolast potassium (TWT-8152) 是 H1组胺受体拮抗剂和肥大细胞稳定剂，是一种具有抗过敏特性的嘧啶酮衍生物。
T10239	Acolbifene 阿考比芬,EM-652,SCH 57068	Estrogen Receptor/ERR	Endocrinology/Hormones
	Acolbifene (SCH 57068) 是一种选择性雌激素受体拮抗剂，对雌二醇诱导的 ERα 和 ERβ 转录活性的 IC50 分别为 2 nM 和 0.4 nM。 Acolbifene 显示出抗癌特性。
T7000	Tiagabine hydrochloride NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Tiagabine hydrochloride (NO050328 hydrochloride) 是具有抗惊厥特性的选择性GABA 再摄取抑制剂，在突触体、神经元和神经胶质中，能够抑制 [3H]GABA 的重摄取，IC50值分别为 67、446 和 182 nM。
T2592	Ropinirole hydrochloride SKF 101468 hydrochloride,SKF-101468A,Ropinirole HCl,盐酸罗匹尼罗	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Ropinirole hydrochloride (SKF-101468A) 是D3/D2受体激动剂，对 D2受体的Ki=29 nM。它对 hD2，hD3和 hD4受体的pEC50分别为 7.4、8.4 和 6.8。它对 D1受体没有亲和力。它对帕金森氏病具有潜在的研究价值。
T29457L	5-Hydroxydecanoate sodium	Potassium Channel	Membrane transporter/Ion channel
	5-Hydroxydecanoate sodium 是一种选择性 ATP 敏感的 K+ (KATP) 通道阻滞剂，IC50 约为 30 μM。它是线粒体外膜酰基辅酶A 合成酶的底物，具有抗氧化性。
T9560	MAO-B-IN-2	Others	Others
	MAO-B-IN-2 是一种选择性和竞争性的MAO-B 和 BChE 抑制剂，其IC50值分别为 0.51 和 7.00 μM。MAO-B-IN-2 通过良好的 ROS 清除特性减轻 H2O2 诱导的细胞损伤。
T0018	Procainamide hydrochloride Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺	DNA Methyltransferase; Sodium Channel; AChR; Autophagy	Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Neuroscience
	Procainamide hydrochloride (Procapan) 是一种用于研究心律失常的抗心律失常制剂。
T0222	Proparacaine hydrochloride 盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride	Apoptosis; Sodium Channel	Apoptosis; Membrane transporter/Ion channel
	Proparacaine hydrochloride (Proparacaine HCl) 是 Lidocaine 的衍生物，具有糖皮质激素样活性和免疫调节作用。
T1435	Praziquantel 吡喹酮,Pyquiton,Droncit,Biltricide	Calcium Channel; Antibiotic; Parasite	Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
	Praziquantel (Droncit) 是一种外消旋混合物，由 (R)-Praziquantel 和 (S)-Praziquantel 组成。它可研究血吸虫病。
T2546	Pimozide R6238,匹莫奇特,匹莫齐特	Potassium Channel; Dopamine Receptor; Adrenergic Receptor; STAT	GPCR/G Protein; JAK/STAT signaling; Membrane transporter/Ion channel; Neuroscience; Stem Cells
	Pimozide (R6238) 是多巴胺受体拮抗剂，对多巴胺 D1、D2 和 D3 受体的 Ki 值分别为 588、1.4 和 2.5 nM。它也是STAT3和STAT5的抑制剂，对 α1 肾上腺素受体也有较高亲和性，Ki 值为 39 nM。
T1281	Tropicamide Ro 1-7683,托吡卡胺	AChR	Neuroscience
	Tropicamide (Ro 1-7683) 是一种选择性的 M4毒蕈碱乙酰胆碱受体拮抗剂，作为滴眼剂使用时，会产生短效瞳孔扩张和睫状肌麻痹。
T6686	Sulconazole mononitrate Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑	Antibacterial; Antibiotic; Antifungal	Microbiology/Virology
	Sulconazole mononitrate (Exelderm) 是一种咪唑类广谱杀菌剂。它可研究皮肤真菌病，花斑糠疹病，皮肤念珠菌病。
T0893	Tinidazole 替硝唑,CP12574	Antibacterial; Antibiotic	Microbiology/Virology
	Tinidazole (CP12574) 是一种对厌氧菌和原生动物具有选择性抗菌活性的 5-硝基咪唑，是一种具有口服活性的抗菌剂。
T6602	Naratriptan hydrochloride Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride	5-HT Receptor	GPCR/G Protein; Neuroscience
	Naratriptan hydrochloride (GR-85548A hydrochloride) 是一种5-HT1受体激动剂，有抗偏头疼特性。它还可以通过刺激三叉神经系统感觉神经末梢上的 5-HT1D/1B 受体来发挥其作用，从而减少促炎神经肽的释放。
T27183	Diproteverine	Others	Others
	Diproteverine is a calcium antagonist, it has antianginal property.
T27276	Epeleuton	Others	Others
	Epeleuton has anti-inflammatory property.
T0149	Pheneticillin	Others	Others
	Pheneticillin 是一种具有抗菌性的抗生素。
T16268	Namitecan ST-1968	Others	Others
	Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.
T39190	ATX-002	Others	Others
	ATX-002 is a property-tunable lipid for RNA drug delivery.
T15166	DPM-1001	Phosphatase	Metabolism
	DPM-1001 is an orally bioavailable and non-competitive protein-tyrosine phosphatase (PTP1B) inhibitor (IC50: 100 nM) with the anti-diabetic property.
T18932	Calcein tetraethyl ester 钙黄绿素四乙酯,Fluorexon tetraethyl ester	Others	Others
	Calcein tetraethyl ester, a fluorescent dye, is utilized in biological studies for its ability to penetrate cellular membranes into living cells. This property renders it valuable for assessing cell viability and short-term cell labeling.
T68937	Carbidopa hydrochloride	Others	Others
	Carbidopa hydrochloride is a drug given to people with Parkinson's disease in order to inhibit peripheral metabolism of levodopa. This property is significant in that it allows a greater proportion of peripheral levodopa to cross the blood–brain barrier for central nervous system effect.
T39128	Pro-Phe-Phe
	Pro-Phe-Phe, a highly aggregation-prone tripeptide composed of natural amino acids, exhibits the formation of distinctive helical-like sheets that engage in aromatic dry interfaces. This property makes Pro-Phe-Phe an excellent candidate for the development of modular super-helical self-assembling nanostructures.
T25170	Botryodiplodin Cytostipin,Antibiotic PSX 1	Others	Others
	Botryodiplodin, an antibiotic, has antileukemic activity from Botryodiplodia theobromae. It has the property of turning the skin of the individual in various shades of pink 2-3 hrs after application. It is a toxic metabolite of Penicillium carneo-lutescen
T28618	RS-93522 RS 93522	Others	Others
	RS-93522 is an antagonist of calcium channel. RS-93522 had the additional property of inhibiting phosphodiesterase activity in myocardial homogenates (IC50 = 1.6 x 10(-5)M), the potency and efficacy of phosphodiesterase inhibition was similar to that for
T79086	MC4171	Histone Acetyltransferase	Chromatin/Epigenetic
	MC4171（化合物34）作为KAT8选择性抑制剂，IC50值为8.1 µM。该化合物在多种癌症细胞系中（包括NSCLC和AML）展现中等微摩尔级别抗增殖效果，显示出其研究治疗癌症的可能性。
T77280	DSPE-succinic acid	Others	Others
	DSPE-succinic acid是一种具有羧酸末端的磷脂，能够通过其羧酸部分与胺发生反应，形成稳定的酰胺键。该化合物常用于纳米颗粒或脂质体的制备，用作活性分子的纳米载体。
T81403	Priliximab cM-T412,CEN 000029
	Priliximab (CEN 000029) 是一种针对CD4的人源化单克隆抗体。其与T细胞表面CD4的结合作用可引起循环中CD4+T细胞的显著并持久的减少，适用于类风湿性关节炎 (RA) 研究。
T77158	Diridavumab
	Diridavumab为一种针对HA茎的单克隆抗体。它能稳定HA的融合前结构，阻断细胞膜与病毒膜在核内体内因pH变化引起的融合。此抗体主要用于H2流感病毒研究。
T0204	Protriptyline hydrochloride 盐酸普罗替林,Protriptyline HCl	5-HT Receptor; AChE	GPCR/G Protein; Neuroscience
	Protriptyline hydrochloride (Protriptyline HCl) 是一种含有一个仲胺的三环结构抗抑郁试剂，可以用于抑郁和 ADHD 的相关研究。它使动物精力充沛起激励作用，并且有时用于嗜睡症的相关研究。
T76497	KRFK
	KRFK是一种源自TSP-1的多肽，具备激活TGF-β的能力。通过独立于TSP受体（例如CD47和CD36）的方式，KRFK能够促进TGF-β介导的信号传递以及其下游效应的发生，可作为慢性眼表炎症疾病研究的工具。
T80487	MmTx2 toxin Micrurotoxin 2	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	MmTx2 toxin作为一种GABAA受体调节剂，具有提升GABAA受体对激动剂反应敏感性的作用。该毒素来源于珊瑚蛇的毒液，并在神经系统相关疾病（例如癫痫、精神分裂症及慢性疼痛）的研究中发挥重要用途。
T70897	Zotiraciclib HCl	Others	Others
	Zotiraciclib, also known as TG02 and SB1317, is a novel small molecule potent CDK/JAK2/FLT3 inhibitor. Zotiraciclib may be useful for the treatment of cancer that crosses the blood brain barrier and acts by depleting Myc through the inhibition of cyclin-dependent kinase 9 (CDK9). It is one of a number of CDK inhibitors under investigation; others targeting CDK9 for the treatment of acute myeloid leukemia include alvocidib and atuveciclib. Myc overexpression is a known factor in many cancers, w...
T81305	ReAsH-EDT2
	ReAsH-EDT2为膜透性红色荧光染料，专用于蛋白质标记。作为二砷化合物，其通过共价结合至四半胱氨酸序列实现蛋白质成像，并可监测其定位与转运。(λex=530 nm，λem=592 nm)。
T84851	O-Phthalimide-C3-acid 4-Phthalimidobutyric acid	Others	Others
	4-(N-Phthalimidoyl)butanoic acid (化合物 FB) 是半抗原，其间隔臂末端具有羧基，便于与蛋白质游离胺基发生反应。此化合物适用于载体蛋白结合，用于抗原设计。
T78391	DAUDA
	DAUDA (11-(dansylamino) undecanoic acid)是一种荧光脂肪酸类似物，对环境变化敏感。该分子通过调整其发射强度和荧光光谱与结合蛋白发生相互作用。在研究中，DAUDA用于评估天然脂肪酸与曼氏血吸虫Sm14脂肪酸结合蛋白多晶型的相对亲和力。
T77252	Dihydrorhodamine 6G	Others	Others
	Dihydrorhodamine 6G (DHR 6G) 为 Rhodamine 6G 的还原型，作为线粒体荧光染料而被广泛应用。该化合物在原状态下无荧光性，但能轻易渗透大部分细胞，并由氧化物或细胞的氧化还原系统氧化为具有荧光的 Rhodamine 6G，进而在线粒体膜中累积。Dihydrorhodamine 6G 主要用于活性氧 (ROS) 的检测，包括超氧化物。
T60782	THK-5470	Others	Others
	THK-5470 是具有高选择性和高亲和力的单胺氧化酶B 的成像探针，可用于研究神经系统疾病。THK-5470 对MAO-B 表现出显著的高结合亲和力，IC50值为 4.2 nM，其对tau 的结合亲和力较低，IC50值为 4462 nM。
T64640	Melanin probe-2	Others	Others
	Melanoma is a lethal skin cancer. The early detection of melanoma using positron emission tomography (PET) probes is critical for improving the survival of melanoma patients. Melanin probe-2 is a non-radioactive bromo-picolinamide precursor that has been used for the synthesis of18F-picolinamides based PET probe (melanin probe-1). The tumor-targeting efficacy and imaging property of three melanin probes were evaluated in B16F10 tumor-bearing mice.18F-1 and18F-3 had much lower tumor uptake compar...
T76255	Certepetide
	Certepetide (CEND-1)，即双功能环肽（a.k.a. iRGD），是一种具有穿透肿瘤功能的多肽。通过与α-V整联蛋白（alphav-integrins）的RGD motif相互作用，以及激活神经纤毛蛋白1（NRP-1），Certepetide能够将实体瘤微环境转化成临时的活性分子通道，从而在肿瘤中累积。该化合物在胰腺癌和其他实体瘤的研究中具有应用潜力。

化合物

Sodium carbonate

Cat.No: T22426

Synonym: 碳酸钠,Soda Ash,Disodium carbonate,Carbonic acid disodium salt

Target: Others

1H-1,2,4-Triazole-3-carboxylic acid

Cat.No: T1371

Target: Others

Cat.No: T8520

Synonym: 1H-TETRAZOLE,1H-四唑

Target: Antibacterial

Lidocaine Hydrochloride hydrate

Cat.No: T1144L

Target: EGFR, Sodium Channel

Enclomiphene citrate

Cat.No: T7313

Synonym: 恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate

Target: Estrogen Receptor/ERR

3-Hydroxybutyric acid sodium

Cat.No: T65133

Synonym: β-Hydroxybutyric acid sodium

Target: Others

Sodium laureth sulfate

Cat.No: T12950

Synonym: Sodium lauryl polyoxyethylene ether sulfate,月桂醇聚氧乙烯醚硫酸酯钠盐

Target: Others

Cat.No: T18890

Synonym: 5-羧基-X-罗丹明,5-Carboxy-X-rhodamine

Target: Others

HPV16 E7 (86-93) acetate

Cat.No: TP1554L

Synonym: HPV16 E7 (86-93) acetate(160212-93-1 Free base)

Target: Others

Pemirolast potassium

Cat.No: T1425

Synonym: BMY 26517,TWT-8152,吡嘧司特钾

Target: Histamine Receptor

Cat.No: T10239

Synonym: 阿考比芬,EM-652,SCH 57068

Target: Estrogen Receptor/ERR

Tiagabine hydrochloride

Cat.No: T7000

Synonym: NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride

Target: GABA Receptor

Ropinirole hydrochloride

Cat.No: T2592

Synonym: SKF 101468 hydrochloride,SKF-101468A,Ropinirole HCl,盐酸罗匹尼罗

Target: Dopamine Receptor

5-Hydroxydecanoate sodium

Cat.No: T29457L

Target: Potassium Channel

Cat.No: T9560

Target: Others

Procainamide hydrochloride

Cat.No: T0018

Synonym: Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺

Target: DNA Methyltransferase, Sodium Channel, AChR, Autophagy

Proparacaine hydrochloride

Cat.No: T0222

Synonym: 盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride

Target: Apoptosis, Sodium Channel

Cat.No: T1435

Synonym: 吡喹酮,Pyquiton,Droncit,Biltricide

Target: Calcium Channel, Antibiotic, Parasite

Cat.No: T2546

Synonym: R6238,匹莫奇特,匹莫齐特

Target: Potassium Channel, Dopamine Receptor, Adrenergic Receptor, STAT

Cat.No: T1281

Synonym: Ro 1-7683,托吡卡胺

Target: AChR

Sulconazole mononitrate

Cat.No: T6686

Synonym: Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑

Target: Antibacterial, Antibiotic, Antifungal

Cat.No: T0893

Synonym: 替硝唑,CP12574

Target: Antibacterial, Antibiotic

Naratriptan hydrochloride

Cat.No: T6602

Synonym: Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride

Target: 5-HT Receptor

Cat.No: T27183

Target: Others

Cat.No: T27276

Target: Others

Cat.No: T0149

Target: Others

Cat.No: T16268

Synonym: ST-1968

Target: Others

Cat.No: T39190

Target: Others

Cat.No: T15166

Target: Phosphatase

Calcein tetraethyl ester

Cat.No: T18932

Synonym: 钙黄绿素四乙酯,Fluorexon tetraethyl ester

Target: Others

Carbidopa hydrochloride

Cat.No: T68937

Target: Others

Cat.No: T39128

Cat.No: T25170

Synonym: Cytostipin,Antibiotic PSX 1

Target: Others

Cat.No: T28618

Synonym: RS 93522

Target: Others

Cat.No: T79086

Target: Histone Acetyltransferase

DSPE-succinic acid

Cat.No: T77280

Target: Others

Cat.No: T81403

Synonym: cM-T412,CEN 000029

Cat.No: T77158

Protriptyline hydrochloride

Cat.No: T0204

Synonym: 盐酸普罗替林,Protriptyline HCl

Target: 5-HT Receptor, AChE

Cat.No: T76497

Cat.No: T80487

Synonym: Micrurotoxin 2

Target: GABA Receptor

Zotiraciclib HCl

Cat.No: T70897

Target: Others

Cat.No: T81305

O-Phthalimide-C3-acid

Cat.No: T84851

Synonym: 4-Phthalimidobutyric acid

Target: Others

Cat.No: T78391

Dihydrorhodamine 6G

Cat.No: T77252

Target: Others

Cat.No: T60782

Target: Others

Melanin probe-2

Cat.No: T64640

Target: Others

Cat.No: T76255

Cat. No.	Product Name	Target	Signaling Pathways
TN1353	N-Benzyllinoleamide (9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺	Others	Others
	N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) 是一种分离自 Lepidium meyeniiWalp，能够抗运动性疲劳的药物。
T0144	Ftaxilide Histanorm,安息香酸,伏保克西里	Antibacterial	Microbiology/Virology
	Ftaxilide (Histanorm) 是新型抗结核剂。
TN7113	Methacrylamide	Others	Others
	Methacrylamide 是一种具有染色性的天然产物。
T0938	Thiabendazole 2-(4-Thiazolyl)benzimidazole,噻菌灵	Microtubule Associated; Mitochondrial Metabolism; Parasite	Cytoskeletal Signaling; Metabolism; Microbiology/Virology
	Thiabendazole (2-(4-Thiazolyl)benzimidazole) 是具有驱虫特性的苯并咪唑衍生物。
TN1005	Parishin E 巴利森苷E,巴利森苷 E	Others	Others
	Parishin E 是一种分离自天麻的 Parishin 衍生物，可能具有抗氧化活性。
T4S2164	Narirutin Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷	Others; Antibacterial	Microbiology/Virology; Others
	Narirutin (Naringenin-7-O-rutinoside) 是从Citrus unshiu 中分离的活性成分之一，具有抗氧化和抗炎活性。它是一种具有抗结核效力的shikimate 激酶抑制剂。
TN1432	Bacopasaponin C (-)-假马齿苋皂苷 C,假马齿苋皂苷C	Anti-infection; GABA Receptor; NMDAR	Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
	Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷，具有抗肿瘤和抗利什曼原虫作用。
T0416	Gluconate sodium Sodium D-gluconate,Sodium gluconate,葡萄糖酸钠,D-Gluconic acid sodium salt,D-Gluconate sodium salt	Others; Endogenous Metabolite	Metabolism; Others
	Gluconate sodium (Sodium D-gluconate) 是一种阻垢缓蚀剂。
TMA1603	Parishin C 巴利森苷 C,巴利森苷C	Antioxidant	oxidation-reduction
	Parishin C 是一种从天麻中分离出的 Parishin 衍生物，可能具有抗氧化作用。
TN1513	Clitorin 碟豆宁,碟豆素	PKC; Antifection	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
	Clitorin 是一种山奈酚糖苷，分离自 Acalypha indica 的花和叶，表现出抗氧化活性。
T4241	Rubiadin 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素	Free radical scavengers; PARP; Caspase	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; oxidation-reduction; Proteases/Proteasome
	Rubiadin (1,3-Dihydroxy-2-Methylanthracene-9,10-Dione) 是一种二羟基蒽醌，提取自茜草，具有抗氧化剂作用。
T13350	Wushanicaritin	Others	Others
	Wushanicaritin 在 DPPH 自由基清除活性测试中显示出显著的抗氧化活性，其IC50值为35.3 μM，具有抗肿瘤作用和抗炎活性。
TN1644	Flavanomarein	Others	Others
	Flavanomarein 是Coreopsis tinctoria Nutt 的主要黄酮类化合物，对糖尿病性肾病具有保护作用。它具有很好的抗氧化，降糖，降压和降血脂作用。
Fr14298	2'-Hydroxy-4'-methylacetophenone 2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮	Anti-infection	Microbiology/Virology
	2'-Hydroxy-4'-methylacetophenone 是一种分离自韩国当归根部得到的酚类，可用于合成 4’-methyl-2’-[(p-tolylsulfonyl) oxy] acetophenone，具有杀螨作用。
T3948	Undecanoic acid Hendecanoic acid,十一烷酸,Undecylic acid	Others; Endogenous Metabolite; Antifungal	Metabolism; Microbiology/Virology; Others
	Undecanoic acid (Hendecanoic acid) 是一种具有抗真菌特性的一元羧酸，可抑制红色葡萄球菌中细胞外角蛋白酶、脂肪酶的产生和几种磷脂的生物合成。
T3787	Didymin Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙	Apoptosis; Others	Apoptosis; Others
	Didymin (Neoponcirin) 从柑橘类水果中提取的一种膳食类黄酮苷，具有抗氧化特性。它通过抑制 N-Myc 和上调 RKIP 诱导凋亡。
T3S0218	Thonningianin A	Apoptosis; Others	Apoptosis; Others
	Thonningianin A 是从非洲草药通宁宁的甲醇提取物中，分离得到的一种鞣花素，具有抗癌和抗氧化性，涉及自由基清除、抗超氧化物形成和金属螯合。
T1045	Trimipramine maleate Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐	Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
	Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂，对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。
TN1892	Lusianthridin	Others; c-Myc	Cell Cycle/Checkpoint; Others
	Lusianthridin 是来自石斛 Dendrobium venustum 的天然产物。 Lusianthridin 在无毒浓度下表现出抗迁移特性。 Lusianthridin 通过抑制 Src-STAT3 信号传导增强 c-Myc 降解。
T3771	Methyl protodioscin 山药,Smilax saponin B,NSC-698790	Apoptosis	Apoptosis
	Methyl protodioscin (Smilax saponin B) 是一种甾二糖苷，能诱导细胞周期阻滞，具有抗肿瘤活性。
TJS0314	5,7-Dihydroxy-4-methylcoumarin Methyl-2H-Chromen-2-One,5,7-二羟基-4-甲基香豆素,4-Methyllimetol,4-Methyl-5,7-Dihydroxycoumarin	Others; Antibacterial; Antifungal	Microbiology/Virology; Others
	5,7-Dihydroxy-4-methylcoumarin (Methyl-2H-Chromen-2-One) 是墨西哥龙蒿中的一种香豆素衍生物。它抑制人类中性粒细胞氧化代谢和弹性蛋白酶活性，有抗真菌和抗细菌活性。
T3816	Velutin	NF-κB; HIF/HIF Prolyl-Hydroxylase	Chromatin/Epigenetic; Metabolism; NF-κB
	Velutin 是一种苷元，提取自槲寄生中，能够抑制黑色素生物合成。它利用 NF-κB 途径减少破骨细胞分化和下调 HIF-1α。
T1468	Lornoxicam Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康	COX; Endogenous Metabolite	Immunology/Inflammation; Metabolism; Neuroscience
	Lornoxicam (Chlortenoxicam) 是一种新型非甾体抗炎药，是高活性 COX-1 和 COX-2 抑制剂，IC50 分别为 5 和 8 nM。
T6480	D-Pantothenic acid vitamin B5,pantothenate,D-泛酸	Others	Others
	D-Pantothenic acid (vitamin B5) 是必需的微量营养素，是辅酶 A 的前体，在很多生物过程中发挥关键作用，如调节碳水化合物，脂质，蛋白和核酸代谢。
T7032	Eupatorin	Others; P450	Metabolism; Others
	Eupatorin 是天然存在的黄酮，可捕获 G2-M 细胞周期，激活多个 caspase、细胞色素 C 的释放、多聚 (ADP-核糖) 聚合酶的裂解，促使凋亡细胞死亡。
T4S0867	Pogostone DHELWANGIN,广藿香酮	Apoptosis; Antibacterial; Autophagy	Apoptosis; Autophagy; Microbiology/Virology
	Pogostone (DHELWANGIN) 是从薄荷中分离出，对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T6S1784	Brazilin Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素	Apoptosis; Others; AMPK; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Others; PI3K/Akt/mTOR signaling
	Brazilin (Braziletto) 是来自几种热带硬木的心材的一种红色染料前体，有软骨保护和抗炎活性。它抑制细胞增殖，促进细胞凋亡并通过 AMPK/mTOR 途径诱导自噬。
T3795	Corilagin	Apoptosis; TLR; Reverse Transcriptase; Antibacterial; Autophagy	Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology
	Corilagin 是一种鞣酸，有抑制 RNA 肿瘤病毒逆转录酶的活性。它抑制金黄色葡萄球菌的生长，MIC 为 25 μg/mL。它有抗肿瘤活性，可用于肝癌和卵巢癌。
T6S1917	Schisandrol B Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B	P450; Reactive Oxygen Species; Autophagy	Autophagy; Immunology/Inflammation; Metabolism; NF-κB
	Schisandrol B (Besigomsin) 是华中五味子的主要活性成分，具有保肝、抗炎、抗糖尿病和抗氧化的作用。它抑制活性氧的产生，也抑制 P-糖蛋白和CYP3A 的活性。
T6S1699	Shogaol [6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol	Lipoxygenase; Autophagy	Autophagy; Metabolism
	6-Shogaol (6-Shogaol) 是从生姜中分离的一种天然产物，具有抗癌、抗炎和抗氧化的多种生物活性。
TN6456	N-trans-caffeoyloctopamine
	N-trans-Caffeoyltyramine has both arginase inhibitory property and antioxidant capacity.
TN4777	Physalin G	Others	Others
	Physalin G has antinociceptive property.
TN4414	Laricitrin 3-O-glucoside	Others	Others
	Laricitrin 3-O-glucoside has antioxidant property.
T72794	Millmerranone A	Others	Others
	Millmerranone A 具有抑制乙酰胆碱酯酶的特性。
TN3113	5-Heptadecylresorcinol 芒果	Others	Others
	5-Heptadecylresorcinol has strong inhibitory property against the growth of PC3 cells.
TN1931	Methyllinderone	Antifection	Microbiology/Virology
	Methyllinderone is a human chymase inhibitor, it has antioxidant property, it also shows moderate to weak antifungal activities against various pathogenic fungi.
TN1811	Jionoside D	Others	Others
	Jionoside D exhibits antioxidant property.
TN1760	Icariside E5 淫羊藿次甙E5,淫羊藿次甙 E5	Others	Others
	Icariside E5 may have antioxidant property that strengthen the importance of peppers in the Mediterranean diet.
T28834	Spirolaxine	Others	Others
	Spirolaxine, a natural product isolated from Sporotrichum laxum ATCC 15155, has shown a variety of biological activities including promising anti-Helicobacter pylori property.
TN3133	5-O-Methylgenistein	Others	Others
	5-O-Methylgenistein may show free radical scavenging activity, it also may have hepatoprotective property on the model of toxic hepatitis induced by carbon tetrachloride damage.
TN1484	Cheilanthifoline	NF-κB; Antifection	Microbiology/Virology; NF-κB
	Cheilanthifoline has anti-osteoclastogenic property, it gives significant inhibitions on receptor activator of nuclear factor-κB ligand-induced differentiation of mouse bone marrow-derived macrophages into multinucleated osteoclasts.
TN3836	Desacetylmatricarin	Others	Others
	Desacetylmatricarin has anti-allergic property, it shows a potent inhibitory activity upon the beta-hexosaminidase release from RBL-2H3 cells in a dose-dependent manner and the IC50 of 7.5 microM.
T5S0313	Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷	Others; TNF	Apoptosis; Others
	Liquiritin apioside has antioxidant property by inducing glutathione (GSH) biosynthesis via the inhibition of cytokines and protected lung epithelial cells against cigarette smoke-mediated oxidative stress, might be as protective agent against epithelial
T69369	Cladosporin	Others	Others
	Cladosporin 是一种真菌代谢物，在 Cladosporium cladosporioid 的菌丝体中产生。含浓度 75 μg/mL Cladosporin 的琼脂培养基可完全抑制多种皮肤癣菌的生长。
TN4223	Homopterocarpin	Antifection	Microbiology/Virology
	Homopterocarpin and Pterocarpus extract offer gastroprotection against indomethacin- induced ulcer by antioxidative mechanism and the modulation of gastric homeostasis, homopterocarpin may be responsible for, or contribute to the antiulcerogenic property
TN3525	Boehmenan	ERK; Phosphatase; EGFR; PARP; MEK; Wnt/beta-catenin; Akt; Caspase; STAT; p53	Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; JAK/STAT signaling; MAPK; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
	(±)-Boehmenan shows potent protein-tyrosine phosphatase 1B (PTP1B) inhibitory activity in vitro with the IC(50) values of 43.5 uM, it inhibits PTP1B activity in a competitive manner. Boehmenan exhibits the potent cytotoxic effects against many cancer cell
T35751	Violacein	Others	Others
	Violacein is a bacterial metabolite originally isolated from C. violaceum that has antibacterial and antiprotozoal activities.[1] [2] It is produced by C. violaceum as a purple pigment in response to N-hexanoyl homoserine lactone , a property that has been modified to create a strain of C. violaceum used in detecting quorum-sensing molecules.[3] Violacein is active against Gram-positive bacteria, including B. subtilis and S. aureus (MICs = 0.8 and 1.6 &#181M, respectively). It is also active aga...

天然产物

N-Benzyllinoleamide

Cat.No: TN1353

Synonym: (9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺

Target: Others

Cat.No: T0144

Synonym: Histanorm,安息香酸,伏保克西里

Target: Antibacterial

Cat.No: TN7113

Target: Others

Cat.No: T0938

Synonym: 2-(4-Thiazolyl)benzimidazole,噻菌灵

Target: Microtubule Associated, Mitochondrial Metabolism, Parasite

Cat.No: TN1005

Synonym: 巴利森苷E,巴利森苷 E

Target: Others

Cat.No: T4S2164

Synonym: Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷

Target: Others, Antibacterial

Bacopasaponin C

Cat.No: TN1432

Synonym: (-)-假马齿苋皂苷 C,假马齿苋皂苷C

Target: Anti-infection, GABA Receptor, NMDAR

Gluconate sodium

Cat.No: T0416

Synonym: Sodium D-gluconate,Sodium gluconate,葡萄糖酸钠,D-Gluconic acid sodium salt,D-Gluconate sodium salt

Target: Others, Endogenous Metabolite

Cat.No: TMA1603

Synonym: 巴利森苷 C,巴利森苷C

Target: Antioxidant

Cat.No: TN1513

Synonym: 碟豆宁,碟豆素

Target: PKC, Antifection

Cat.No: T4241

Synonym: 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素

Target: Free radical scavengers, PARP, Caspase

Cat.No: T13350

Target: Others

Cat.No: TN1644

Target: Others

2'-Hydroxy-4'-methylacetophenone

Cat.No: Fr14298

Synonym: 2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮

Target: Anti-infection

Undecanoic acid

Cat.No: T3948

Synonym: Hendecanoic acid,十一烷酸,Undecylic acid

Target: Others, Endogenous Metabolite, Antifungal

Cat.No: T3787

Synonym: Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙

Target: Apoptosis, Others

Thonningianin A

Cat.No: T3S0218

Target: Apoptosis, Others

Trimipramine maleate

Cat.No: T1045

Synonym: Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐

Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor

Cat.No: TN1892

Target: Others, c-Myc

Methyl protodioscin

Cat.No: T3771

Synonym: 山药,Smilax saponin B,NSC-698790

Target: Apoptosis

5,7-Dihydroxy-4-methylcoumarin

Cat.No: TJS0314

Synonym: Methyl-2H-Chromen-2-One,5,7-二羟基-4-甲基香豆素,4-Methyllimetol,4-Methyl-5,7-Dihydroxycoumarin

Target: Others, Antibacterial, Antifungal

Cat.No: T3816

Target: NF-κB, HIF/HIF Prolyl-Hydroxylase

Cat.No: T1468

Synonym: Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康

Target: COX, Endogenous Metabolite

D-Pantothenic acid

Cat.No: T6480

Synonym: vitamin B5,pantothenate,D-泛酸

Target: Others

Cat.No: T7032

Target: Others, P450

Cat.No: T4S0867

Synonym: DHELWANGIN,广藿香酮

Target: Apoptosis, Antibacterial, Autophagy

Cat.No: T6S1784

Synonym: Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素

Target: Apoptosis, Others, AMPK, Autophagy

Cat.No: T3795

Target: Apoptosis, TLR, Reverse Transcriptase, Antibacterial, Autophagy

Cat.No: T6S1917

Synonym: Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B

Target: P450, Reactive Oxygen Species, Autophagy

Cat.No: T6S1699

Synonym: [6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol

Target: Lipoxygenase, Autophagy

N-trans-caffeoyloctopamine

Cat.No: TN6456

Cat.No: TN4777

Target: Others

Laricitrin 3-O-glucoside

Cat.No: TN4414

Target: Others

Millmerranone A

Cat.No: T72794

Target: Others

5-Heptadecylresorcinol

Cat.No: TN3113

Synonym: 芒果

Target: Others

Methyllinderone

Cat.No: TN1931

Target: Antifection

Cat.No: TN1811

Target: Others

Cat.No: TN1760

Synonym: 淫羊藿次甙E5,淫羊藿次甙 E5

Target: Others

Cat.No: T28834

Target: Others

5-O-Methylgenistein

Cat.No: TN3133

Target: Others

Cheilanthifoline

Cat.No: TN1484

Target: NF-κB, Antifection

Desacetylmatricarin

Cat.No: TN3836

Target: Others

Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside

Cat.No: T5S0313

Synonym: Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷

Target: Others, TNF

Cat.No: T69369

Target: Others

Homopterocarpin

Cat.No: TN4223

Target: Antifection

Cat.No: TN3525

Target: ERK, Phosphatase, EGFR, PARP, MEK, Wnt/beta-catenin, Akt, Caspase, STAT, p53

Cat.No: T35751

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-03617	Miraculin Protein, Synsepalum dulcificum, Recombinant (His) Miraculin	Synsepalum dulcificum	P. pastoris (Yeast)
	Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 23.4 kDa and the accession number is P13087.
TMPH-03616	Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His) Miraculin	Synsepalum dulcificum	E. coli
	Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 24.9 kDa and the accession number is P13087.
TMPJ-01138	UBE2S Protein, Human, Recombinant (GST) UBE2S,Ubiquitin-Conjugating Enzyme E2-24 kDa,E2-EPF,E2EPF,Ub...	Human	E. coli
	Ubiquitin-Conjugating Enzyme E2 S (UBE2S) is a member of the Ubiquitin-Conjugating Enzyme family. UBE2S interacts with CDC20, FZR1/CDH1 and VHL. UBE2S can form a thiol ester linkage with Ubiquitin in an Ubiquitin Activating Enzyme-Dependent manner, a characteristic property of Ubiquitin Carrier Proteins. UBE2S acts as an essential factor of the Anaphase Promoting Complex/Cyclosome, a cell cycle-regulated Ubiquitin ligase that controls progression through mitosis. UBE2S is also involved in ubiqui...
TMPY-04075	CLIC1 Protein, Human, Recombinant (His) NCC27,G6,chloride intracellular channel 1	Human	E. coli
	Members of the CLIC family are largely soluble proteins that possess the intriguing property of spontaneous insertion into phospholipid bilayers to form integral membrane ion channels. Chloride intracellular channel 1 (CLIC1), a newly discovered member of the chloride channel protein family, has been implicated in multiple human cancers. CLIC1 is a Chloride Intracellular Ion Channel protein that exists either in a soluble state in the cytoplasm or as a membrane bound protein. CLIC1 acts as a put...
TMPY-01910	TIE1 Protein, Human, Recombinant (His) tyrosine kinase with immunoglobulin-like and EGF-like domain...	Human	HEK293 Cells
	Tyrosine kinase with immunoglobulin-like and EGF-like domains 1 also known as Tie1 is an angiopoietin receptor and is an orphan receptor tyrosine kinase that is expressed almost exclusively in endothelial cells and that is required for normal embryonic vascular development. The receptor tyrosine kinase Tie1 is expressed primarily in vascular endothelial cells. The receptor has also been detected in epithelial tumours in breast, thyroid and gastric cancers and in tumour cell lines where it appear...
TMPY-01416	OLFM4 Protein, Human, Recombinant (His) hGC-1,GC1,OLM4,bA209J19.1,GW112,olfactomedin 4,OlfD,hOLfD,UN...	Human	HEK293 Cells
	Olfactomedin-4, also known as G-CSF-stimulated clone 1 protein, Antiapoptotic protein GW112, and OLFM4, is a secreted protein that contains one olfactomedin-like domain. The OLFM4 gene was recently reported to inhibit various apoptotic pathways and promote the proliferation of cancer cells, suggesting that OLFM4 might serve as a diagnostic marker for human cancers. Thus, OLFM4 mRNA might be a useful tool to support the diagnosis of cancer, irrespective of the clinical stages. It is overexpressed...

重组蛋白

Miraculin Protein, Synsepalum dulcificum, Recombinant (His)

Cat.No: TMPH-03617

Species: Synsepalum dulcificum

Expression System: P. pastoris (Yeast)

Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His)

Cat.No: TMPH-03616

Species: Synsepalum dulcificum

Expression System: E. coli

UBE2S Protein, Human, Recombinant (GST)

Cat.No: TMPJ-01138

Species: Human

Expression System: E. coli

CLIC1 Protein, Human, Recombinant (His)

Cat.No: TMPY-04075

Species: Human

Expression System: E. coli

TIE1 Protein, Human, Recombinant (His)

Cat.No: TMPY-01910

Species: Human

Expression System: HEK293 Cells

OLFM4 Protein, Human, Recombinant (His)

Cat.No: TMPY-01416

Species: Human

Expression System: HEK293 Cells

Cat. No.	Product Name	Target	Signaling Pathways
TMIJ-0484	Thiabendazole NH-d6
	Thiabendazole NH-d6 是 Thiabendazole NH 的氘代化合物。Thiabendazole NH 的 CAS 号为 148-79-8。Thiabendazole 是具有驱虫特性的苯并咪唑衍生物。

同位素标记化合物

Thiabendazole NH-d6

Cat.No: TMIJ-0484

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