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Search Results for " water-soluble "
Targets Recommended: Others

150

抑制剂 & 化合物

42

天然产物

1

TargetMol 试剂盒

2

重组蛋白

9

同位素标记化合物

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Cat. No. Product Name Form Specificity Of Inhibition
C0005 Cell Counting Kit-8 (CCK-8)

Cell Counting Kit-8 (CCK-8)

Solution in bottle

TargetMol 试剂盒

Cell Counting Kit-8 (CCK-8)
Cat.No: C0005
Cat. No. Product Name Target Signaling Pathways
T36587 APTS

8-Aminopyrene-1,3,6-trisulfonic acid trisodium

Others Others
8-Aminopyrene-1,3,6-trisulfonic Acid sodium salt 是一种阴离子荧光染料,用作葡萄糖传感和检测其他糖类的报告分子。激发/发射光谱为 425/503 nm。 它可以在溶液中使用,也可以通过还原胺化连接醛官能化单体来固定,而不会显著改变荧光强度。
T19362 Hydroxyethyl cellulose

Cellulose hydroxyethyl ether,羟乙基纤维素,2-Hydroxyethyl cellulose

Others Others
Hydroxyethyl cellulose (2-Hydroxyethyl cellulose) 是一种非离子水溶性改性纤维素聚合物,能够用作水溶性化妆品和个人护理配方中的增稠剂。
T6818 DEL-22379

DEL22379

Apoptosis; ERK Apoptosis; MAPK
DEL-22379 是一种水溶性 ERK 二聚化抑制剂,IC50约为 0.5 μM。
T10378 Artelinic acid

Parasite Microbiology/Virology
Artelinic acid 是水溶性青蒿素类似物,具有抗疟活性,用于治疗恶性疟原虫多重耐药菌株。
T5328 Fosfluconazole

Antifungal Microbiology/Virology
Fosfluconazole 是 fluconazole 的水溶性磷酸盐前药。 它是一种抗真菌药物。
T4449 LB100

LB-100,LB 100

Phosphatase Metabolism
LB100 (LB-100) 是一种水溶性蛋白磷酸酶 2A(PP2A) 抑制剂。
T34746 Sulfo-SANPAH Crosslinker

Sulfo-SANPAH Cross-linker,Sulfo-SANPAH Cross linker,6-[(4-叠氮-2-硝基苯基)氨基]己酸磺酸基琥珀酰亚胺酯

Others Others
Sulfo-SANPAH Crosslinker (Sulfo-SANPAH Cross linker) 是一种水溶性同双功能蛋白质交联剂。
T15025L CY5 triethylamine salt

CY5 triethylamine salt(146368-11-8 Free base)

Others Others
CY5 triethylamine salt 是一种水溶性染料,激发光波长(nm):649,发射波长(nm):670。
T20067 WST-1

WST 1

WST-1 是一种具有细胞毒性的水溶性四唑盐,诱导细胞内线粒体脱氢酶进行 NADH 依赖性酶解反应,释放出水溶性甲基苯产物。WST-1 可通过检测吸收值来检测细胞增殖和细胞活性,可用于WST-1平板测定法测定超氧化物歧化酶活性。
T0294 6α-Methylprednisolone 21-hemisuccinate sodium salt

Asmacortone,Methylprodnisolone Sodium Succinate,甲强龙琥珀酸钠,Metypresol,Methylprednisolone sodium succinate,Corticel,6-Methylprednisolone succinate sodium

Glucocorticoid Receptor; Glucagon Receptor Endocrinology/Hormones; GPCR/G Protein
6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone) 是一种糖皮质激素,是一种有效的抗炎剂,半衰期比 Prednisolone 长。
T19368 Hypromellose

Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose

Others Others
Hypromellose (HPMC) 是一种水溶性的亲水性非离子纤维素醚。
T7551 Belotecan hydrochloride

CKD-602

Topoisomerase DNA Damage/DNA Repair
Belotecan hydrochloride (CKD-602) 是一种合成的水溶性喜树碱衍生物和拓扑异构酶 I 抑制剂,具有潜在的抗肿瘤活性。
T15553 Iganidipine

NKY 722

Calcium Channel Membrane transporter/Ion channel; Metabolism
Iganidipine(NKY 722) 是一种新的水溶性 Ca2+ 拮抗剂,具有降压活性,可用于研究和神经系统相关的疾病。
T0271 Iodipamide

Iodipamic acid,胆影酸,Adipiodone

Others Others
Iodipamide (Iodipamic acid) 是一种三碘苯甲酸酯衍生物,也是一种离子二聚剂,可用于诊断成像。
T0947L Dexamethasone Phosphate disodium

地塞米松磷酸二钠,EGP-437,EGP437. Dex-Phos,EGP 437

Glucocorticoid Receptor Endocrinology/Hormones
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) 是糖皮质激素受体激动剂。
T8734 Choline

Others Others
Choline hydroxide 是一种普遍存在的水溶性营养素,通常与 B 族维生素有关。
T13365 YHO-13351 free base

BCRP Membrane transporter/Ion channel
YHO-13351 free base 是 YHO-13177 的水溶性前药,YHO-13177 是 BCRP 的抑制剂。
T8459 DNQX disodium salt

DNQX Disodium

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
DNQX disodium salt 是一种选择性、强竞争性的非 NMDA 谷氨酸受体 (non-NMDA glutamate receptor) 拮抗剂 (对 AMPA、kainate 和 NMDA 受体的 IC50分别为 0.5、2 和 40 μM),是一种喹恶啉衍生物。
T14131 ADPS

N-Ethyl-N-(3-sulfopropyl)-3-methoxyaniline sodium salt,ESPAS

Others Others
ADPS (N-Ethyl-N-(3-sulfopropyl)-3-methoxyaniline sodium salt) 是新型 Trinder's 试剂,是一种高水溶性苯胺衍生品,普遍用于生化试验、诊断检测。
T1254 Chlorophyllin sodium copper salt

Chlorophyllin copper sodium complex,Chlorophyllin,叶绿素铜钠盐,Chlorophyllin coppered trisodium salt,Sodium-copper chlorin e6

Others Others
Chlorophyllin sodium copper salt (Chlorophyllin coppered trisodium salt) 是一种由 Chlorophyll 衍生的铜钠盐的半合成混合物,常用作食品添加剂。
T22830 GYY4137

GYY 4137 morpholine salt

Others Others
GYY4137 (GYY 4137 morpholine salt) 是一种缓释H2S 供体,具有抗炎和抗癌作用,也具有血管扩张和抗高血压活性。
T19232 CMC-Na (Viscosity:800-1200 mPa.s)

羧甲基纤维素钠,Sodium carboxymethyl cellulose,CMC-Na (Viscosity:800-1200 mPa.s)

Others Others
Sodium carboxymethyl cellulose (CMC-Na) (Viscosity:800-1200 mPa.s) 是一种水溶性纤维素,常用作动物实验的助溶剂,对动物基本没有毒性。
T4018 WST-8

WST8

Others Others
WST-8 是水溶性的四唑染料,WTS-8测定法的灵敏度比常规MTS 检测高。
T4994 Tocofersolan

Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯

Others Others
Tocofersolan (TPGS) 是合成的 α-生育酚的聚乙二醇衍生物。
T41206 Poly Vinyl Alcohol

Polyvinyl alcohol

Others Others
Poly Vinyl Alcohol (Polyvinyl alcohol)是一种水溶性可生物降解且可用于伤口愈合的聚合物,在生物医学领域广泛使用。Poly Vinyl Alcohol 常用于制作医用辅料。
T12042 Minnelide

Apoptosis; Virus Protease Apoptosis; Microbiology/Virology
Minnelide 是水溶性雷公藤内酯前药,具有抗癌症抗肿瘤活性,可诱导细胞凋亡,可预防足细胞损伤。Minnelide 通过阻断 HPV 诱导的 p53 和 pRb 变化来抑制宫颈癌的生长。
T61383 Diaziquone

NSC 182986

Others Others
Diaziquone (NSC-182986)是一种水溶性的合成的氮杂环苯醌,可增强对血脑屏障的渗透,具有抗肿瘤活性,可用于治疗极性肾功能衰竭。
T38367 CAY10640

sEH inhibitor-1

Epoxide Hydrolase Metabolism
CAY10640 (sEH inhibitor-1)一种有效的、具有口服活性、可溶于水的环氧化物水解酶 (sEH) 抑制剂,对人和鼠中的sEH 具有抑制作用,IC50s 分别为 0.4 和 5.3 nM。
T7022 PEG300

聚乙二醇,Polyethylene glycol 300

Others Others
PEG300 (Polyethylene glycol 300) 是一种由乙二醇重复单元形成的聚合物,具有水溶性、低免疫原性和生物相容性。PEG300 是一种分子量为300的中性聚合物。
T19271 DAOS

Sodium 3-((3,5-dimethoxyphenyl)(ethyl)amino)-2-hydroxypropane-1-sulfonate

Others Others
DAOS (Sodium 3-((3,5-dimethoxyphenyl)(ethyl)amino)-2-hydroxypropane-1-sulfonate) 是一种 Trinder's 试剂,是新型高水溶性苯胺衍生物,普遍用于诊断检测和生化试验。
T1790 Fosaprepitant dimeglumine

福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt

Neurokinin receptor GPCR/G Protein; Neuroscience
Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
T11861 LM11A-31 dihydrochloride

Others Others
LM11A-31 dihydrochloride 是一种具有高血脑屏障通透性的氨基酸衍生物,能阻断 p75 介导的细胞死亡。它是一种 p75NTR(神经营养蛋白受体 p75) 非肽调节剂,是口服有效的 proNGF 拮抗剂。它可以逆转中晚期的阿尔茨海默氏病小鼠模型中的胆碱能神经突营养不良。
T2627 Nolatrexed dihydrochloride

盐酸诺拉曲塞,Thymitaq,AG 337

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Nolatrexed dihydrochloride (Thymitaq) 是一种非竞争性的胸苷酸合酶抑制剂,能够在癌细胞 S 期诱导细胞周期停滞,具有抗癌活性。它与该酶的叶酸辅因子结合位点相互作用,对人胸苷酸合酶的Ki 值为 11 nM。
T3437 Lys05

Lys01 trihydrochloride

lysosomal autophagy; Autophagy Autophagy
Lys05 是一种有效的水溶性溶酶体自噬抑制剂,具有抗肿瘤活性。在 MTT 试验中,对1205Lu、c8161、LN229 和 HT-29细胞系的IC50值分别为3.6、3.8、6 和7.9 μM。
T22739 DMPO

5,5-二甲基-1-吡咯啉-N-氧化物,5,5-Dimethyl-1-pyrroline N-oxide

Others Others
DMPO (5,5-Dimethyl-1-pyrroline N-oxide) 是一种亲水自旋诱捕剂,具有细胞渗透性。DMPO 可用于超氧化物检测,可检测超氧阴离子和羟自由基。
T19952 Sulfo-NHS-Biotin

Sulfosuccinimidobiotin,Sulfosuccinimidyl biotin,Biotin-NHS,Sulfo NHS Biotin,N-hydroxysulfosuccinimidyl biotin

Others Others
Sulfo-NHS-Biotin (Biotin-NHS) 是一种水溶性生物素化试剂,用于生物素-链霉亲和素结合反应。 Sulfo-NHS-Biotin (Biotin-NHS) 特别适用于在链霉亲和素-生物素测定中靶向细胞表面蛋白。与链霉亲和素和固定化链霉亲和素一起使用时,可用于蛋白质检测或固定。
T0006 Methylene Blue trihydrate

碱性亚甲蓝三水合物,Methylthionine chloride,Basic blue 9,亚甲蓝三水合物,Methylene Blue

Guanylate cyclase; Microtubule Associated; NO Synthase; Parasite; Monoamine Oxidase Cytoskeletal Signaling; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Methylene Blue trihydrate (Basic blue 9) 是鸟苷酸环化酶,单胺氧化酶 A 和 NO 合酶抑制剂。它是血管加压药,在医疗中通常用作染料。它具有抗伤害感受,抗疟疾,抗抑郁和抗焦虑作用,可用于高铁血红蛋白血症,神经退行性疾病和异环磷酰胺引起的脑病的研究。
T19353 HDAOS

Others Others
HDAOS 是一种新型Trinder's 试剂,是苯胺衍生物,具有高水溶性,被广泛用于诊断检测和生化试验。
T19586 TOPS

Others Others
TOPS 是一种高度溶于水的苯胺衍生物,在诊断和生物实验中有广泛运用。
T1710 Trolox

Apoptosis; Antioxidant; Ferroptosis; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Trolox 是一种维生素 E 的衍生物,具有细胞渗透性和水溶性。Trolox 是一种膜损伤抑制剂,具有强大的抗氧化活性。
T15497 HOE 33187

Others Others
HOE 33187是一种DNA 染料,可渗透进入细胞。
T25511 Hydrocortisone-21-lysinate

Others Others
Hydrocortisone-21-lysinate is a hydrocortisone prodrug that is water soluble.
T26024 R 87366

R87366,R-87366

Others Others
R 87366 is used as a water-soluble HIV protease inhibitor.
T28332 PD 138142

PD-138142,PD138142

Others Others
PD 138142 is a water soluble inhibitor of ACAT.
T24600 PC407-ws

PC407ws

Others Others
PC407-ws is a water-soluble novel COX-2 inhibitor.
T70519 Cryosim-3

Others Others
Cryosim-3 is a water-soluble, potent, and selective TRPM8 receptor agonist.
T13262 FCE 28654

Others Others
FCE 28654 is a water-soluble acyl-CoA inhibitor.
T32476 L 705589

L705589,L-705589

Others Others
L 705589 is a semisynthetic pneumocandin Bo derivative that is water-soluble.
T19585 TOOS

TOOS sodium salt

Others Others
TOOS is a novel highly water-soluble aniline derivative and is widely used in diagnostic tests and biochemical tests.
T27023 Cispentacin

Others Others
Cispentacin is a β-amino acid and acts as a water-soluble antifungal antibiotic. Cispentacin is effective against Candida.

化合物

APTS
Cat.No: T36587
Synonym: 8-Aminopyrene-1,3,6-trisulfonic acid trisodium
Target: Others
Hydroxyethyl cellulose
Cat.No: T19362
Synonym: Cellulose hydroxyethyl ether,羟乙基纤维素,2-Hydroxyethyl cellulose
Target: Others
DEL-22379
Cat.No: T6818
Synonym: DEL22379
Target: Apoptosis, ERK
Artelinic acid
Cat.No: T10378
Synonym:
Target: Parasite
Fosfluconazole
Cat.No: T5328
Synonym:
Target: Antifungal
LB100
Cat.No: T4449
Synonym: LB-100,LB 100
Target: Phosphatase
Sulfo-SANPAH Crosslinker
Cat.No: T34746
Synonym: Sulfo-SANPAH Cross-linker,Sulfo-SANPAH Cross linker,6-[(4-叠氮-2-硝基苯基)氨基]己酸磺酸基琥珀酰亚胺酯
Target: Others
CY5 triethylamine salt
Cat.No: T15025L
Synonym: CY5 triethylamine salt(146368-11-8 Free base)
Target: Others
WST-1
Cat.No: T20067
Synonym: WST 1
Target:
6α-Methylprednisolone 21-hemisuccinate sodium salt
Cat.No: T0294
Synonym: Asmacortone,Methylprodnisolone Sodium Succinate,甲强龙琥珀酸钠,Metypresol,Methylprednisolone sodium succinate,Corticel,6-Methylprednisolone succinate sodium
Target: Glucocorticoid Receptor, Glucagon Receptor
Hypromellose
Cat.No: T19368
Synonym: Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose
Target: Others
Belotecan hydrochloride
Cat.No: T7551
Synonym: CKD-602
Target: Topoisomerase
Iganidipine
Cat.No: T15553
Synonym: NKY 722
Target: Calcium Channel
Iodipamide
Cat.No: T0271
Synonym: Iodipamic acid,胆影酸,Adipiodone
Target: Others
Dexamethasone Phosphate disodium
Cat.No: T0947L
Synonym: 地塞米松磷酸二钠,EGP-437,EGP437. Dex-Phos,EGP 437
Target: Glucocorticoid Receptor
Choline
Cat.No: T8734
Synonym:
Target: Others
YHO-13351 free base
Cat.No: T13365
Synonym:
Target: BCRP
DNQX disodium salt
Cat.No: T8459
Synonym: DNQX Disodium
Target: NMDAR, iGluR
ADPS
Cat.No: T14131
Synonym: N-Ethyl-N-(3-sulfopropyl)-3-methoxyaniline sodium salt,ESPAS
Target: Others
Chlorophyllin sodium copper salt
Cat.No: T1254
Synonym: Chlorophyllin copper sodium complex,Chlorophyllin,叶绿素铜钠盐,Chlorophyllin coppered trisodium salt,Sodium-copper chlorin e6
Target: Others
GYY4137
Cat.No: T22830
Synonym: GYY 4137 morpholine salt
Target: Others
CMC-Na (Viscosity:800-1200 mPa.s)
Cat.No: T19232
Synonym: 羧甲基纤维素钠,Sodium carboxymethyl cellulose,CMC-Na (Viscosity:800-1200 mPa.s)
Target: Others
WST-8
Cat.No: T4018
Synonym: WST8
Target: Others
Tocofersolan
Cat.No: T4994
Synonym: Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯
Target: Others
Poly Vinyl Alcohol
Cat.No: T41206
Synonym: Polyvinyl alcohol
Target: Others
Minnelide
Cat.No: T12042
Synonym:
Target: Apoptosis, Virus Protease
Diaziquone
Cat.No: T61383
Synonym: NSC 182986
Target: Others
CAY10640
Cat.No: T38367
Synonym: sEH inhibitor-1
Target: Epoxide Hydrolase
PEG300
Cat.No: T7022
Synonym: 聚乙二醇,Polyethylene glycol 300
Target: Others
DAOS
Cat.No: T19271
Synonym: Sodium 3-((3,5-dimethoxyphenyl)(ethyl)amino)-2-hydroxypropane-1-sulfonate
Target: Others
Fosaprepitant dimeglumine
Cat.No: T1790
Synonym: 福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
LM11A-31 dihydrochloride
Cat.No: T11861
Synonym:
Target: Others
Nolatrexed dihydrochloride
Cat.No: T2627
Synonym: 盐酸诺拉曲塞,Thymitaq,AG 337
Target: DNA/RNA Synthesis
Lys05
Cat.No: T3437
Synonym: Lys01 trihydrochloride
Target: lysosomal autophagy, Autophagy
DMPO
Cat.No: T22739
Synonym: 5,5-二甲基-1-吡咯啉-N-氧化物,5,5-Dimethyl-1-pyrroline N-oxide
Target: Others
Sulfo-NHS-Biotin
Cat.No: T19952
Synonym: Sulfosuccinimidobiotin,Sulfosuccinimidyl biotin,Biotin-NHS,Sulfo NHS Biotin,N-hydroxysulfosuccinimidyl biotin
Target: Others
Methylene Blue trihydrate
Cat.No: T0006
Synonym: 碱性亚甲蓝三水合物,Methylthionine chloride,Basic blue 9,亚甲蓝三水合物,Methylene Blue
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
HDAOS
Cat.No: T19353
Synonym:
Target: Others
TOPS
Cat.No: T19586
Synonym:
Target: Others
Trolox
Cat.No: T1710
Synonym:
Target: Apoptosis, Antioxidant, Ferroptosis, Reactive Oxygen Species
HOE 33187
Cat.No: T15497
Synonym:
Target: Others
Hydrocortisone-21-lysinate
Cat.No: T25511
Synonym:
Target: Others
R 87366
Cat.No: T26024
Synonym: R87366,R-87366
Target: Others
PD 138142
Cat.No: T28332
Synonym: PD-138142,PD138142
Target: Others
PC407-ws
Cat.No: T24600
Synonym: PC407ws
Target: Others
Cryosim-3
Cat.No: T70519
Synonym:
Target: Others
FCE 28654
Cat.No: T13262
Synonym:
Target: Others
L 705589
Cat.No: T32476
Synonym: L705589,L-705589
Target: Others
TOOS
Cat.No: T19585
Synonym: TOOS sodium salt
Target: Others
Cispentacin
Cat.No: T27023
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1116 Biotin

Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H)

Biotin (Vitamin H) 属于天然产物,是一种 B 族维生素,具有水溶性。Biotin 参与脂肪酸产生、脂肪和氨基酸代谢以及细胞生长。Biotin 常被用于生物素标记。
TN2174 Salvianolic acid E

丹酚酸 E,丹酚酸E

Others Others
Salvianolic acid E 是一种从丹参 Salvia miltiorrhiza 中分离出来的水溶性成分。
T19224 C-Phycocyanin

C-PC,藻蓝蛋白,C-藻蓝蛋白

Others Others
C-Phycocyanin (C-PC) 是一种蛋白质色素,常作为人类的优良营养补充剂。
T3551 D-Pantothenic acid hemicalcium salt

泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
D-Pantothenic acid hemicalcium salt (Calcium pantothenate) 是一种水溶性维生素,能够减少苹果汁中的棒曲霉素。
T4760 KSD 2405

3-羟基苯甲醇,3-Hydroxybenzyl alcohol

Others; Endogenous Metabolite Metabolism; Others
KSD 2405 (3-Hydroxybenzyl alcohol) 是内源性代谢产物的一种。
T5258 Dodecanedioic acid diammonium salt

十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt

Others Others
Dodecanedioic acid diammonium salt (1,10-Decanedicarboxylic acid diammonium salt) 是一种二元羧酸,它是水溶性的,并且参与了脂类和碳水化合物的代谢途径中间体。
T4784 (S)-(-)-Phenylethanol

(S)-(-)-1-Phenylethanol,右旋1-苯乙醇,(-)-Methyl phenyl carbinol,(S)-(-)-sec-Phenylethyl alcohol

Others; Endogenous Metabolite Metabolism; Others
(S)-(-)-Phenylethanol ((-)-Methyl phenyl carbinol) 是内源性代谢产物的一种。
T2727 Salvianolic acid B

Others Others
Salvianolic acid B (Dan Shen Suan B) 是一种来自丹参提取物的水溶性抗氧化剂,具有抗血小板聚集、抗凝和抗血栓作用。它常用来研究微循环疾病。
T4107 4-Pyridoxic Acid

4-吡哆酸,Pyridoxic Acid,4-Pyridoxinsaeure

Endogenous Metabolite Metabolism
4-Pyridoxic Acid (4-Pyridoxinsaeure) 是一种维生素B6的分解代谢产物,从尿液中分泌得到。
T5311 Crocin (Gardenia Fruits Extract)

藏红花,西红花苷

Others Others
Crocin (Gardenia Fruits Extract)(42553-65-1)是藏红花(Crocus sativus L.)的水溶性类胡萝卜素色素。藏红花素具有抗炎、抗氧化、抗凋亡、抗哮喘、抗癌、降血脂等作用。
T2989 4-Hydroxybenzoic acid

p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
4-Hydroxybenzoic acid (4-hydroxybenzoate) 是苯甲酸的酚衍生物,可抑制革兰氏阳性和革兰氏阴性菌,IC50值为160 μg/mL。
T5068 D-Glucuronic acid sodium salt monohydrate

Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate

Others; Endogenous Metabolite Metabolism; Others
D-Glucuronic acid sodium salt monohydrate (Sodium D-glucuronate) 是内源性代谢产物的一种。
T3368 Alpha-Hederin

α常春藤皂甙,Helixin,Tauroside E,α-Hederin,Hederoside C

Apoptosis; Others Apoptosis; Others
Alpha-Hederin (Tauroside E) 是存在于黑种草种子中的一种单桥糖三萜皂苷,具有抗肿瘤作用。它可通过激活线粒体依赖性途径抑制胃癌细胞增殖,诱导凋亡,并有活性氧生成和谷胱甘肽减少。
T5725 Salvianolic acid B

丹酚酸B,lithospermic acid B,Dan Shen Suan B

Sirtuin; Autophagy Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair
Salvianolic acid B (Dan Shen Suan B) 是一种来自丹参的天然产物,是一种抗氧化剂,具有水溶性。Salvianolic acid B 具有抗血小板聚集、抗凝和抗血栓作用,常用来研究微循环疾病。
T2719 Succinic acid

Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid

Endogenous Metabolite Metabolism
Succinic acid (1,2-Ethanedicarboxylic acid) 是无氧代谢的发酵产物,也是三羧酸循环的中间产物。
T2946 Tanshinone IIA sulfonate sodium

丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium

CaMK; P450; Calcium Channel Membrane transporter/Ion channel; Metabolism; Neuroscience
Tanshinone IIA sulfonate sodium (Tanshinone IIA sodium sulfonate) 是从丹参中提取的丹参酮IIA 的水溶性衍生物,是SOCE 抑制剂,用于心血管疾病的研究。
T0433 Artesunate

WR-256283,青蒿琥酯

Virus Protease; Ferroptosis; STAT; Parasite Apoptosis; JAK/STAT signaling; Microbiology/Virology; Stem Cells
Artesunate (WR-256283) 是治疗疟疾的青蒿素组药物的一部分。 它是青蒿素的半合成衍生物,具有水溶性。
T5082 Calcium 2-hydroxy-4-(methylthio)butanoate

羟基蛋氨酸钙,calcium hydroxymethionine,2-Hydroxy-4-(methylthio)butyric acid calcium salt

Others; Endogenous Metabolite Metabolism; Others
Calcium 2-hydroxy-4-(methylthio)butanoate (Calcium 2-hydroxy-4-(calcium hydroxymethionine)) 是内源性代谢产物的一种。
T11060 DMAPT

Dimethylamino Parthenolide

NF-κB NF-κB
DMAPT (Dimethylamino Parthenolide) 是一种具有口服活性的NF-κB 抑制剂,是一种 Parthenolide (PTL) 的类似物,对原发性急性髓性白血病细胞的LD50值为1.7 μM。具有潜在的抗肿瘤和抗转移作用。
T6272 Fosbretabulin Disodium

Combretastatin A4 Phosphate,CA 4DP,CA 4P,福他布林,Combretastatin A4 disodium phosphate,Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Fosbretabulin Disodium (CA 4P) 是一种微管蛋白去稳定剂,是 Combretastatin A4 前药,可选择性靶向内皮细胞,诱导新生肿瘤新血管消退,减少肿瘤血流量并引起中央肿瘤坏死。
T4773 3-Ethoxy-3-oxopropanoic acid

Monoethyl malonic acid,Ethyl hydrogen malonate,丙二酸单乙酯

Others; Endogenous Metabolite Metabolism; Others
3-Ethoxy-3-oxopropanoic acid (Monoethyl malonic acid) 是内源性代谢产物的一种。
T2818 Methyl Vanillate

Reactive Oxygen Species; Wnt/beta-catenin; Endogenous Metabolite Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells
Methyl vanillate 是一种枳椇属植物中的提取物,是Wnt/β-catenin 信号通路活化剂,是一种香草酸的甲酯。它具有抗氧化作用。
T0879 Niacin

Vitamin B3,烟酸(维生素B3),Nicotinic acid

Endogenous Metabolite; Autophagy Autophagy; Metabolism
Niacin (Nicotinic acid),也称为烟酸和维生素 B3,是一种水溶性必需的 B 族维生素,用于治疗维生素缺乏症以及高脂血症,血脂异常,高甘油三酯血症,并降低心肌梗塞的风险
T3947 Nonanoic acid

pelargonic acid,Nonoic acid,壬酸

Others; Antibacterial Microbiology/Virology; Others
Nonanoic acid (Nonoic acid) 是一种天然存在的具有九个碳原子的饱和脂肪酸。它减少细菌易位,增强抗菌活性,并增加猪 β-防御素 1 (pBD-1) 和 pBD-2 的分泌。
T6480 D-Pantothenic acid

vitamin B5,pantothenate,D-泛酸

Others Others
D-Pantothenic acid (vitamin B5) 是必需的微量营养素,是辅酶 A 的前体,在很多生物过程中发挥关键作用,如调节碳水化合物,脂质,蛋白和核酸代谢。
T4768 Diethyl oxalpropionate

草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE

Others; Endogenous Metabolite Metabolism; Others
Diethyl oxalpropionate (HYL 2-METHYL-3-OXOSUCCINATE) 是一种合成 PDMMLA 的中间体。其中 PDMMLA 的衍生物可用于纳米粒子的合成和研究。
Fr13883 3-Methoxyphenylacetic acid

Others Others
3-Methoxyphenylacetic acid 是 m-hydroxyphenylacetic (m-OHPAA) 的衍生物,茄形假丝酵母中的一种植物毒素。它可用于针对介氧菌根腐烂的毒素介导的生物测定法的开发。
T1040 Vitamin B12

Cyanocobalamin,Cobalamin,维生素B12

Endogenous Metabolite Metabolism
Vitamin B12 (Cobalamin) 是一种维生素,在维持血流形成和脑、神经系统正常功能等方面发挥关键作用。
T2823 Crocin

西红花苷,藏红花,Gardenia Yellow,Alpha-Crocin,藏红花素

Others Others
Crocin (Gardenia Yellow) 是从Crocus sativus 柱头中分离出的主要成分,是一种营养保健品,具有抗炎,抗癌,抗抑郁和抗惊厥等强大的药理作用。
T4798 N-Acetyl-L-leucine

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-leucine 是内源性代谢产物的一种。
T1331 Riboflavin phosphate sodium

Riboflavin 5'-phosphate sodium,核黄素磷酸钠(维生素B2),Vitamin B2 Phosphate Sodium Salt,Flavin mononucleotide,FMN,核黄素磷酸钠,FMN-Na,riboflavin-5'-phosphate

Endogenous Metabolite Metabolism
Riboflavin phosphate sodium (FMN) 是 riboflavin 的磷酸钠盐形式,riboflavin 是一种水溶性和必需的微量营养素,是自然产生的维生素B复合物的主要生长促进因子。Riboflavin phosphate sodium 转化为2种辅酶,黄素单核苷酸(FMN)和黄素腺嘌呤二核苷酸(FAD),这两种辅酶通过帮助脂肪、碳水化合物和蛋白质的代谢来产生能量,并且是红细胞形成和呼吸、抗体产生以及调节人体生长和繁殖所必需的。
T13777 Moniliformin sodium salt

Others Others
Moniliformin sodium salt is water-soluble mycotoxin isolate from Fusarium moniliforme.
T34489 Salicifoline

Salicifoline is a water-soluble quaternary ammonium alkaloid.
T29888 Aloe-emodin-glucoside

Aloe-emodin-glucoside is a stimulant-laxative which has been shown to enhance colonic membrane permeability of water-soluble and poorly permeable compounds.
T0879L Niacin hydrochloride

Niacin hydrochloride is a water-soluble vitamin of the B complex occurring in various animal and plant tissues. It is needed by the body for the formation of coenzymes NAD and NADP. It possesses PELLAGRA-curative, vasodilating, and antilipemic properties.
TN6613 Delphinidin-3-O-galactoside chloride

Delphinidin-3-O-galactoside chloride has anti-obesity and hypolipidemic effects. Delphinidin-3-O-galactoside (D3G) is a water-soluble anthocyanin with antioxidant activity. D3G is capable of masking the EGCG-induced cytotoxicity and ER stress, presumably
TN2112 Przewalskinic acid A

Others Others
Przewalskinic acid A is a rare, water-soluble, and highly biologically active ingredient found, thus far, only in the Salvia przewalskii Maxim herb.
T20854 Isethionic acid

Hydroxyethylsulfonic acid,Ethanolsulfonic acid

Others Others
Isethionic acid, a major metabolite in F. cylindrus, is an organosulfur compound containing a short-chain alkane sulfonate linked to a hydroxyl group. It is a water-soluble liquid for the manufacture of mild, biodegradable, and high-foaming anionic surfac
T16332 NKH477

Colforsin dapropate hydrochloride

NMDAR Neuroscience
NKH477 is a novel water-soluble forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 shows an antiproliferative effect in vivo with an altered cytokine profile to inhibit the acute
T82148 Hydrogenated soya phosphatidylcholines

Others Others
Hydrogenated soya phosphatidylcholines 是一种用于提升水溶性药物口服给药效果的天然产物,它能够增加药物负荷和溶解度,从而延长药物释放时间。
T35981 Biliverdin hydrochloride

Antioxidant oxidation-reduction
Biliverdin hydrochloride 是一种由血红素氧化形成的四吡咯水溶性化合物,具有潜在的抗氧化活性,参与胆绿素-胆红素氧化还原系统。
T35710 N-Acetyl-S-allyl-L-cysteine

Others Others
L-Deoxyalliin , also known as S-allyl-L-cysteine, is a water soluble organosulfur compound derived from garlic that has neuroprotective and antioxidative activities. N-Acetyl-S-allyl-L-cysteine is a principal metabolite of L-deoxyalliin in humans, mice, rats, and dogs. It is readily detected in plasma and urine. The conversion of L-deoxyalliin to N-acetyl-S-allyl-L-cysteine appears to be mediated by a family of flavin-containing monooxygenases.

天然产物

Biotin
Cat.No: T1116
Synonym: Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H)
Target:
Salvianolic acid E
Cat.No: TN2174
Synonym: 丹酚酸 E,丹酚酸E
Target: Others
C-Phycocyanin
Cat.No: T19224
Synonym: C-PC,藻蓝蛋白,C-藻蓝蛋白
Target: Others
D-Pantothenic acid hemicalcium salt
Cat.No: T3551
Synonym: 泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate
Target: Apoptosis, Endogenous Metabolite
KSD 2405
Cat.No: T4760
Synonym: 3-羟基苯甲醇,3-Hydroxybenzyl alcohol
Target: Others, Endogenous Metabolite
Dodecanedioic acid diammonium salt
Cat.No: T5258
Synonym: 十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt
Target: Others
(S)-(-)-Phenylethanol
Cat.No: T4784
Synonym: (S)-(-)-1-Phenylethanol,右旋1-苯乙醇,(-)-Methyl phenyl carbinol,(S)-(-)-sec-Phenylethyl alcohol
Target: Others, Endogenous Metabolite
Salvianolic acid B
Cat.No: T2727
Synonym:
Target: Others
4-Pyridoxic Acid
Cat.No: T4107
Synonym: 4-吡哆酸,Pyridoxic Acid,4-Pyridoxinsaeure
Target: Endogenous Metabolite
Crocin (Gardenia Fruits Extract)
Cat.No: T5311
Synonym: 藏红花,西红花苷
Target: Others
4-Hydroxybenzoic acid
Cat.No: T2989
Synonym: p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate
Target: Endogenous Metabolite, Antibacterial
D-Glucuronic acid sodium salt monohydrate
Cat.No: T5068
Synonym: Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate
Target: Others, Endogenous Metabolite
Alpha-Hederin
Cat.No: T3368
Synonym: α常春藤皂甙,Helixin,Tauroside E,α-Hederin,Hederoside C
Target: Apoptosis, Others
Salvianolic acid B
Cat.No: T5725
Synonym: 丹酚酸B,lithospermic acid B,Dan Shen Suan B
Target: Sirtuin, Autophagy
Succinic acid
Cat.No: T2719
Synonym: Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid
Target: Endogenous Metabolite
Tanshinone IIA sulfonate sodium
Cat.No: T2946
Synonym: 丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium
Target: CaMK, P450, Calcium Channel
Artesunate
Cat.No: T0433
Synonym: WR-256283,青蒿琥酯
Target: Virus Protease, Ferroptosis, STAT, Parasite
Calcium 2-hydroxy-4-(methylthio)butanoate
Cat.No: T5082
Synonym: 羟基蛋氨酸钙,calcium hydroxymethionine,2-Hydroxy-4-(methylthio)butyric acid calcium salt
Target: Others, Endogenous Metabolite
DMAPT
Cat.No: T11060
Synonym: Dimethylamino Parthenolide
Target: NF-κB
Fosbretabulin Disodium
Cat.No: T6272
Synonym: Combretastatin A4 Phosphate,CA 4DP,CA 4P,福他布林,Combretastatin A4 disodium phosphate,Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium
Target: Apoptosis, Microtubule Associated
3-Ethoxy-3-oxopropanoic acid
Cat.No: T4773
Synonym: Monoethyl malonic acid,Ethyl hydrogen malonate,丙二酸单乙酯
Target: Others, Endogenous Metabolite
Methyl Vanillate
Cat.No: T2818
Synonym:
Target: Reactive Oxygen Species, Wnt/beta-catenin, Endogenous Metabolite
Niacin
Cat.No: T0879
Synonym: Vitamin B3,烟酸(维生素B3),Nicotinic acid
Target: Endogenous Metabolite, Autophagy
Nonanoic acid
Cat.No: T3947
Synonym: pelargonic acid,Nonoic acid,壬酸
Target: Others, Antibacterial
D-Pantothenic acid
Cat.No: T6480
Synonym: vitamin B5,pantothenate,D-泛酸
Target: Others
Diethyl oxalpropionate
Cat.No: T4768
Synonym: 草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE
Target: Others, Endogenous Metabolite
3-Methoxyphenylacetic acid
Cat.No: Fr13883
Synonym:
Target: Others
Vitamin B12
Cat.No: T1040
Synonym: Cyanocobalamin,Cobalamin,维生素B12
Target: Endogenous Metabolite
Crocin
Cat.No: T2823
Synonym: 西红花苷,藏红花,Gardenia Yellow,Alpha-Crocin,藏红花素
Target: Others
N-Acetyl-L-leucine
Cat.No: T4798
Synonym:
Target: Others, Endogenous Metabolite
Riboflavin phosphate sodium
Cat.No: T1331
Synonym: Riboflavin 5'-phosphate sodium,核黄素磷酸钠(维生素B2),Vitamin B2 Phosphate Sodium Salt,Flavin mononucleotide,FMN,核黄素磷酸钠,FMN-Na,riboflavin-5'-phosphate
Target: Endogenous Metabolite
Moniliformin sodium salt
Cat.No: T13777
Synonym:
Target: Others
Salicifoline
Cat.No: T34489
Synonym:
Target:
Aloe-emodin-glucoside
Cat.No: T29888
Synonym:
Target:
Niacin hydrochloride
Cat.No: T0879L
Synonym:
Target:
Delphinidin-3-O-galactoside chloride
Cat.No: TN6613
Synonym:
Target:
Przewalskinic acid A
Cat.No: TN2112
Synonym:
Target: Others
Isethionic acid
Cat.No: T20854
Synonym: Hydroxyethylsulfonic acid,Ethanolsulfonic acid
Target: Others
NKH477
Cat.No: T16332
Synonym: Colforsin dapropate hydrochloride
Target: NMDAR
Hydrogenated soya phosphatidylcholines
Cat.No: T82148
Synonym:
Target: Others
Biliverdin hydrochloride
Cat.No: T35981
Synonym:
Target: Antioxidant
N-Acetyl-S-allyl-L-cysteine
Cat.No: T35710
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPH-03230 PHB depolymerase Protein, Ralstonia pickettii, Recombinant (His)

Poly(3-hydroxybutyrate) depolymerase

Ralstonia pickettii E. coli
This protein degrades water-insoluble and water-soluble PHB to monomeric D(-)-3-hydroxybutyrate. PHB depolymerase Protein, Ralstonia pickettii, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 50.9 kDa and the accession number is P12625.
TMPH-01298 EPHX1 Protein, Human, Recombinant (His)

EPHX1,Microsomal epoxide hydrolase,Epoxide hydratase,Epoxide...

Human E. coli
Biotransformation enzyme that catalyzes the hydrolysis of arene and aliphatic epoxides to less reactive and more water soluble dihydrodiols by the trans addition of water. Plays a role in the metabolism of endogenous lipids such as epoxide-containing fatty acids. Metabolizes the abundant endocannabinoid 2-arachidonoylglycerol (2-AG) to free arachidonic acid (AA) and glycerol.

重组蛋白

PHB depolymerase Protein, Ralstonia pickettii, Recombinant (His)
Cat.No: TMPH-03230
Species: Ralstonia pickettii
Expression System: E. coli
EPHX1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01298
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
T30599 BS3-d4 Deuterated Crosslinker

Deuterated Crosslinker BS3-d4,BS3-d4,D4-BS3

BS3-d4 Deuterated Crosslinker or Bis(Sulfosuccinimidyl) 2,2,7,7-suberate-d4, is a water-soluble and membrane impermeable protein crosslinking agent.
T30598 BS2G-d4 Deuterated Crosslinker

D4-BS2G,BS2G-d4

BS2G-d4 or Bis(Sulfosuccinimidyl) 2,2,4,4-glutarate-d4, is a water-soluble and membrane impermeable protein crosslinking agent.
TMID-0257 Quinoline-d7

Quinoline-d7 是 Quinoline 的氘代化合物。Quinoline 的 CAS 号为 91-22-5。Quinoline 存在于酒精饮料中。 它是一种来自包括薄荷在内的多种植物的生物碱。 也存在于可可、红茶和苏格兰威士忌中。 老化的样品,如果暴露在光线下,会变成黄色,然后变成棕色。
TMIJ-0373 Biotin-d2

Biotin-d2 是 Biotin 的氘代化合物。Biotin 的 CAS 号为 58-85-5。Biotin 是一种水溶性B族维生素,是细胞生长、脂肪酸产生以及脂肪和氨基酸代谢所必需的。
TMID-0029 Succinic-2,2,3,3-d4 Acid

Succinic-2,2,3,3-d4 Acid 是 Succinic Acid 的氘代化合物。Succinic Acid 的 CAS 号为 110-15-6。Succinic acid 是无氧代谢的发酵产物,也是三羧酸循环的中间产物。
TMIJ-0435 Octanoic Acid-d15

Octanoic Acid-d15 是 Octanoic Acid 的氘代化合物。Octanoic Acid 的 CAS 号为 124-07-2。Caprylic acid天然存在于椰子和母乳中。它是一种油性液体,带有些许腐臭味,能用于酯类香料和染料的生产。
TMIJ-0519 Fosaprepitant-d4 Dimeglumine

Fosaprepitant-d4 Dimeglumine 是 Fosaprepitant Dimeglumine 的氘代化合物。Fosaprepitant Dimeglumine 的 CAS 号为 265121-04-8。Fosaprepitant dimeglumine 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
TMIJ-0053 2-Methylpropionic-d7 acid

2-Methylpropionic-d7 acid 是 2-Methylpropionic acid 的氘代化合物。2-Methylpropionic acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。
TMIJ-0047 Isobutyric-d6 acid

Isobutyric-d6 acid 是 Isobutyric acid 的氘代化合物。Isobutyric acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。

同位素标记化合物

BS3-d4 Deuterated Crosslinker
Cat.No: T30599
Synonym: Deuterated Crosslinker BS3-d4,BS3-d4,D4-BS3
Target:
BS2G-d4 Deuterated Crosslinker
Cat.No: T30598
Synonym: D4-BS2G,BS2G-d4
Target:
Quinoline-d7
Cat.No: TMID-0257
Synonym:
Target:
Biotin-d2
Cat.No: TMIJ-0373
Synonym:
Target:
Succinic-2,2,3,3-d4 Acid
Cat.No: TMID-0029
Synonym:
Target:
Octanoic Acid-d15
Cat.No: TMIJ-0435
Synonym:
Target:
Fosaprepitant-d4 Dimeglumine
Cat.No: TMIJ-0519
Synonym:
Target:
2-Methylpropionic-d7 acid
Cat.No: TMIJ-0053
Synonym:
Target:
Isobutyric-d6 acid
Cat.No: TMIJ-0047
Synonym:
Target:
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