150
42
1
2
9
Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
C0005 |
Cell Counting Kit-8 (CCK-8)
Cell Counting Kit-8 (CCK-8) |
Solution in bottle |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36587 |
APTS
8-Aminopyrene-1,3,6-trisulfonic acid trisodium |
Others | Others |
8-Aminopyrene-1,3,6-trisulfonic Acid sodium salt 是一种阴离子荧光染料,用作葡萄糖传感和检测其他糖类的报告分子。激发/发射光谱为 425/503 nm。 它可以在溶液中使用,也可以通过还原胺化连接醛官能化单体来固定,而不会显著改变荧光强度。 | |||
T19362 |
Hydroxyethyl cellulose
Cellulose hydroxyethyl ether,羟乙基纤维素,2-Hydroxyethyl cellulose |
Others | Others |
Hydroxyethyl cellulose (2-Hydroxyethyl cellulose) 是一种非离子水溶性改性纤维素聚合物,能够用作水溶性化妆品和个人护理配方中的增稠剂。 | |||
T6818 |
DEL-22379
DEL22379 |
Apoptosis; ERK | Apoptosis; MAPK |
DEL-22379 是一种水溶性 ERK 二聚化抑制剂,IC50约为 0.5 μM。 | |||
T10378 |
Artelinic acid
|
Parasite | Microbiology/Virology |
Artelinic acid 是水溶性青蒿素类似物,具有抗疟活性,用于治疗恶性疟原虫多重耐药菌株。 | |||
T5328 |
Fosfluconazole
|
Antifungal | Microbiology/Virology |
Fosfluconazole 是 fluconazole 的水溶性磷酸盐前药。 它是一种抗真菌药物。 | |||
T4449 |
LB100
LB-100,LB 100 |
Phosphatase | Metabolism |
LB100 (LB-100) 是一种水溶性蛋白磷酸酶 2A(PP2A) 抑制剂。 | |||
T34746 |
Sulfo-SANPAH Crosslinker
Sulfo-SANPAH Cross-linker,Sulfo-SANPAH Cross linker,6-[(4-叠氮-2-硝基苯基)氨基]己酸磺酸基琥珀酰亚胺酯 |
Others | Others |
Sulfo-SANPAH Crosslinker (Sulfo-SANPAH Cross linker) 是一种水溶性同双功能蛋白质交联剂。 | |||
T15025L |
CY5 triethylamine salt
CY5 triethylamine salt(146368-11-8 Free base) |
Others | Others |
CY5 triethylamine salt 是一种水溶性染料,激发光波长(nm):649,发射波长(nm):670。 | |||
T20067 |
WST-1
WST 1 |
||
WST-1 是一种具有细胞毒性的水溶性四唑盐,诱导细胞内线粒体脱氢酶进行 NADH 依赖性酶解反应,释放出水溶性甲基苯产物。WST-1 可通过检测吸收值来检测细胞增殖和细胞活性,可用于WST-1平板测定法测定超氧化物歧化酶活性。 | |||
T0294 |
6α-Methylprednisolone 21-hemisuccinate sodium salt
Asmacortone,Methylprodnisolone Sodium Succinate,甲强龙琥珀酸钠,Metypresol,Methylprednisolone sodium succinate,Corticel,6-Methylprednisolone succinate sodium |
Glucocorticoid Receptor; Glucagon Receptor | Endocrinology/Hormones; GPCR/G Protein |
6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone) 是一种糖皮质激素,是一种有效的抗炎剂,半衰期比 Prednisolone 长。 | |||
T19368 |
Hypromellose
Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose |
Others | Others |
Hypromellose (HPMC) 是一种水溶性的亲水性非离子纤维素醚。 | |||
T7551 |
Belotecan hydrochloride
CKD-602 |
Topoisomerase | DNA Damage/DNA Repair |
Belotecan hydrochloride (CKD-602) 是一种合成的水溶性喜树碱衍生物和拓扑异构酶 I 抑制剂,具有潜在的抗肿瘤活性。 | |||
T15553 |
Iganidipine
NKY 722 |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Iganidipine(NKY 722) 是一种新的水溶性 Ca2+ 拮抗剂,具有降压活性,可用于研究和神经系统相关的疾病。 | |||
T0271 |
Iodipamide
Iodipamic acid,胆影酸,Adipiodone |
Others | Others |
Iodipamide (Iodipamic acid) 是一种三碘苯甲酸酯衍生物,也是一种离子二聚剂,可用于诊断成像。 | |||
T0947L |
Dexamethasone Phosphate disodium
地塞米松磷酸二钠,EGP-437,EGP437. Dex-Phos,EGP 437 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) 是糖皮质激素受体激动剂。 | |||
T8734 |
Choline
|
Others | Others |
Choline hydroxide 是一种普遍存在的水溶性营养素,通常与 B 族维生素有关。 | |||
T13365 |
YHO-13351 free base
|
BCRP | Membrane transporter/Ion channel |
YHO-13351 free base 是 YHO-13177 的水溶性前药,YHO-13177 是 BCRP 的抑制剂。 | |||
T8459 |
DNQX disodium salt
DNQX Disodium |
NMDAR; iGluR | Membrane transporter/Ion channel; Neuroscience |
DNQX disodium salt 是一种选择性、强竞争性的非 NMDA 谷氨酸受体 (non-NMDA glutamate receptor) 拮抗剂 (对 AMPA、kainate 和 NMDA 受体的 IC50分别为 0.5、2 和 40 μM),是一种喹恶啉衍生物。 | |||
T14131 |
ADPS
N-Ethyl-N-(3-sulfopropyl)-3-methoxyaniline sodium salt,ESPAS |
Others | Others |
ADPS (N-Ethyl-N-(3-sulfopropyl)-3-methoxyaniline sodium salt) 是新型 Trinder's 试剂,是一种高水溶性苯胺衍生品,普遍用于生化试验、诊断检测。 | |||
T1254 |
Chlorophyllin sodium copper salt
Chlorophyllin copper sodium complex,Chlorophyllin,叶绿素铜钠盐,Chlorophyllin coppered trisodium salt,Sodium-copper chlorin e6 |
Others | Others |
Chlorophyllin sodium copper salt (Chlorophyllin coppered trisodium salt) 是一种由 Chlorophyll 衍生的铜钠盐的半合成混合物,常用作食品添加剂。 | |||
T22830 |
GYY4137
GYY 4137 morpholine salt |
Others | Others |
GYY4137 (GYY 4137 morpholine salt) 是一种缓释H2S 供体,具有抗炎和抗癌作用,也具有血管扩张和抗高血压活性。 | |||
T19232 |
CMC-Na (Viscosity:800-1200 mPa.s)
羧甲基纤维素钠,Sodium carboxymethyl cellulose,CMC-Na (Viscosity:800-1200 mPa.s) |
Others | Others |
Sodium carboxymethyl cellulose (CMC-Na) (Viscosity:800-1200 mPa.s) 是一种水溶性纤维素,常用作动物实验的助溶剂,对动物基本没有毒性。 | |||
T4018 |
WST-8
WST8 |
Others | Others |
WST-8 是水溶性的四唑染料,WTS-8测定法的灵敏度比常规MTS 检测高。 | |||
T4994 |
Tocofersolan
Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯 |
Others | Others |
Tocofersolan (TPGS) 是合成的 α-生育酚的聚乙二醇衍生物。 | |||
T41206 |
Poly Vinyl Alcohol
Polyvinyl alcohol |
Others | Others |
Poly Vinyl Alcohol (Polyvinyl alcohol)是一种水溶性可生物降解且可用于伤口愈合的聚合物,在生物医学领域广泛使用。Poly Vinyl Alcohol 常用于制作医用辅料。 | |||
T12042 |
Minnelide
|
Apoptosis; Virus Protease | Apoptosis; Microbiology/Virology |
Minnelide 是水溶性雷公藤内酯前药,具有抗癌症抗肿瘤活性,可诱导细胞凋亡,可预防足细胞损伤。Minnelide 通过阻断 HPV 诱导的 p53 和 pRb 变化来抑制宫颈癌的生长。 | |||
T61383 |
Diaziquone
NSC 182986 |
Others | Others |
Diaziquone (NSC-182986)是一种水溶性的合成的氮杂环苯醌,可增强对血脑屏障的渗透,具有抗肿瘤活性,可用于治疗极性肾功能衰竭。 | |||
T38367 |
CAY10640
sEH inhibitor-1 |
Epoxide Hydrolase | Metabolism |
CAY10640 (sEH inhibitor-1)一种有效的、具有口服活性、可溶于水的环氧化物水解酶 (sEH) 抑制剂,对人和鼠中的sEH 具有抑制作用,IC50s 分别为 0.4 和 5.3 nM。 | |||
T7022 |
PEG300
聚乙二醇,Polyethylene glycol 300 |
Others | Others |
PEG300 (Polyethylene glycol 300) 是一种由乙二醇重复单元形成的聚合物,具有水溶性、低免疫原性和生物相容性。PEG300 是一种分子量为300的中性聚合物。 | |||
T19271 |
DAOS
Sodium 3-((3,5-dimethoxyphenyl)(ethyl)amino)-2-hydroxypropane-1-sulfonate |
Others | Others |
DAOS (Sodium 3-((3,5-dimethoxyphenyl)(ethyl)amino)-2-hydroxypropane-1-sulfonate) 是一种 Trinder's 试剂,是新型高水溶性苯胺衍生物,普遍用于诊断检测和生化试验。 | |||
T1790 |
Fosaprepitant dimeglumine
福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt |
Neurokinin receptor | GPCR/G Protein; Neuroscience |
Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。 | |||
T11861 |
LM11A-31 dihydrochloride
|
Others | Others |
LM11A-31 dihydrochloride 是一种具有高血脑屏障通透性的氨基酸衍生物,能阻断 p75 介导的细胞死亡。它是一种 p75NTR(神经营养蛋白受体 p75) 非肽调节剂,是口服有效的 proNGF 拮抗剂。它可以逆转中晚期的阿尔茨海默氏病小鼠模型中的胆碱能神经突营养不良。 | |||
T2627 |
Nolatrexed dihydrochloride
盐酸诺拉曲塞,Thymitaq,AG 337 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Nolatrexed dihydrochloride (Thymitaq) 是一种非竞争性的胸苷酸合酶抑制剂,能够在癌细胞 S 期诱导细胞周期停滞,具有抗癌活性。它与该酶的叶酸辅因子结合位点相互作用,对人胸苷酸合酶的Ki 值为 11 nM。 | |||
T3437 |
Lys05
Lys01 trihydrochloride |
lysosomal autophagy; Autophagy | Autophagy |
Lys05 是一种有效的水溶性溶酶体自噬抑制剂,具有抗肿瘤活性。在 MTT 试验中,对1205Lu、c8161、LN229 和 HT-29细胞系的IC50值分别为3.6、3.8、6 和7.9 μM。 | |||
T22739 |
DMPO
5,5-二甲基-1-吡咯啉-N-氧化物,5,5-Dimethyl-1-pyrroline N-oxide |
Others | Others |
DMPO (5,5-Dimethyl-1-pyrroline N-oxide) 是一种亲水自旋诱捕剂,具有细胞渗透性。DMPO 可用于超氧化物检测,可检测超氧阴离子和羟自由基。 | |||
T19952 |
Sulfo-NHS-Biotin
Sulfosuccinimidobiotin,Sulfosuccinimidyl biotin,Biotin-NHS,Sulfo NHS Biotin,N-hydroxysulfosuccinimidyl biotin |
Others | Others |
Sulfo-NHS-Biotin (Biotin-NHS) 是一种水溶性生物素化试剂,用于生物素-链霉亲和素结合反应。 Sulfo-NHS-Biotin (Biotin-NHS) 特别适用于在链霉亲和素-生物素测定中靶向细胞表面蛋白。与链霉亲和素和固定化链霉亲和素一起使用时,可用于蛋白质检测或固定。 | |||
T0006 |
Methylene Blue trihydrate
碱性亚甲蓝三水合物,Methylthionine chloride,Basic blue 9,亚甲蓝三水合物,Methylene Blue |
Guanylate cyclase; Microtubule Associated; NO Synthase; Parasite; Monoamine Oxidase | Cytoskeletal Signaling; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Methylene Blue trihydrate (Basic blue 9) 是鸟苷酸环化酶,单胺氧化酶 A 和 NO 合酶抑制剂。它是血管加压药,在医疗中通常用作染料。它具有抗伤害感受,抗疟疾,抗抑郁和抗焦虑作用,可用于高铁血红蛋白血症,神经退行性疾病和异环磷酰胺引起的脑病的研究。 | |||
T19353 |
HDAOS
|
Others | Others |
HDAOS 是一种新型Trinder's 试剂,是苯胺衍生物,具有高水溶性,被广泛用于诊断检测和生化试验。 | |||
T19586 |
TOPS
|
Others | Others |
TOPS 是一种高度溶于水的苯胺衍生物,在诊断和生物实验中有广泛运用。 | |||
T1710 |
Trolox
|
Apoptosis; Antioxidant; Ferroptosis; Reactive Oxygen Species | Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
Trolox 是一种维生素 E 的衍生物,具有细胞渗透性和水溶性。Trolox 是一种膜损伤抑制剂,具有强大的抗氧化活性。 | |||
T15497 |
HOE 33187
|
Others | Others |
HOE 33187是一种DNA 染料,可渗透进入细胞。 | |||
T25511 |
Hydrocortisone-21-lysinate
|
Others | Others |
Hydrocortisone-21-lysinate is a hydrocortisone prodrug that is water soluble. | |||
T26024 |
R 87366
R87366,R-87366 |
Others | Others |
R 87366 is used as a water-soluble HIV protease inhibitor. | |||
T28332 |
PD 138142
PD-138142,PD138142 |
Others | Others |
PD 138142 is a water soluble inhibitor of ACAT. | |||
T24600 |
PC407-ws
PC407ws |
Others | Others |
PC407-ws is a water-soluble novel COX-2 inhibitor. | |||
T70519 |
Cryosim-3
|
Others | Others |
Cryosim-3 is a water-soluble, potent, and selective TRPM8 receptor agonist. | |||
T13262 |
FCE 28654
|
Others | Others |
FCE 28654 is a water-soluble acyl-CoA inhibitor. | |||
T32476 |
L 705589
L705589,L-705589 |
Others | Others |
L 705589 is a semisynthetic pneumocandin Bo derivative that is water-soluble. | |||
T19585 |
TOOS
TOOS sodium salt |
Others | Others |
TOOS is a novel highly water-soluble aniline derivative and is widely used in diagnostic tests and biochemical tests. | |||
T27023 |
Cispentacin
|
Others | Others |
Cispentacin is a β-amino acid and acts as a water-soluble antifungal antibiotic. Cispentacin is effective against Candida. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1116 |
Biotin
Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H) |
||
Biotin (Vitamin H) 属于天然产物,是一种 B 族维生素,具有水溶性。Biotin 参与脂肪酸产生、脂肪和氨基酸代谢以及细胞生长。Biotin 常被用于生物素标记。 | |||
TN2174 |
Salvianolic acid E
丹酚酸 E,丹酚酸E |
Others | Others |
Salvianolic acid E 是一种从丹参 Salvia miltiorrhiza 中分离出来的水溶性成分。 | |||
T19224 |
C-Phycocyanin
C-PC,藻蓝蛋白,C-藻蓝蛋白 |
Others | Others |
C-Phycocyanin (C-PC) 是一种蛋白质色素,常作为人类的优良营养补充剂。 | |||
T3551 |
D-Pantothenic acid hemicalcium salt
泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
D-Pantothenic acid hemicalcium salt (Calcium pantothenate) 是一种水溶性维生素,能够减少苹果汁中的棒曲霉素。 | |||
T4760 |
KSD 2405
3-羟基苯甲醇,3-Hydroxybenzyl alcohol |
Others; Endogenous Metabolite | Metabolism; Others |
KSD 2405 (3-Hydroxybenzyl alcohol) 是内源性代谢产物的一种。 | |||
T5258 |
Dodecanedioic acid diammonium salt
十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt |
Others | Others |
Dodecanedioic acid diammonium salt (1,10-Decanedicarboxylic acid diammonium salt) 是一种二元羧酸,它是水溶性的,并且参与了脂类和碳水化合物的代谢途径中间体。 | |||
T4784 |
(S)-(-)-Phenylethanol
(S)-(-)-1-Phenylethanol,右旋1-苯乙醇,(-)-Methyl phenyl carbinol,(S)-(-)-sec-Phenylethyl alcohol |
Others; Endogenous Metabolite | Metabolism; Others |
(S)-(-)-Phenylethanol ((-)-Methyl phenyl carbinol) 是内源性代谢产物的一种。 | |||
T2727 |
Salvianolic acid B
|
Others | Others |
Salvianolic acid B (Dan Shen Suan B) 是一种来自丹参提取物的水溶性抗氧化剂,具有抗血小板聚集、抗凝和抗血栓作用。它常用来研究微循环疾病。 | |||
T4107 |
4-Pyridoxic Acid
4-吡哆酸,Pyridoxic Acid,4-Pyridoxinsaeure |
Endogenous Metabolite | Metabolism |
4-Pyridoxic Acid (4-Pyridoxinsaeure) 是一种维生素B6的分解代谢产物,从尿液中分泌得到。 | |||
T5311 |
Crocin (Gardenia Fruits Extract)
藏红花,西红花苷 |
Others | Others |
Crocin (Gardenia Fruits Extract)(42553-65-1)是藏红花(Crocus sativus L.)的水溶性类胡萝卜素色素。藏红花素具有抗炎、抗氧化、抗凋亡、抗哮喘、抗癌、降血脂等作用。 | |||
T2989 |
4-Hydroxybenzoic acid
p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate |
Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology |
4-Hydroxybenzoic acid (4-hydroxybenzoate) 是苯甲酸的酚衍生物,可抑制革兰氏阳性和革兰氏阴性菌,IC50值为160 μg/mL。 | |||
T5068 |
D-Glucuronic acid sodium salt monohydrate
Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate |
Others; Endogenous Metabolite | Metabolism; Others |
D-Glucuronic acid sodium salt monohydrate (Sodium D-glucuronate) 是内源性代谢产物的一种。 | |||
T3368 |
Alpha-Hederin
α常春藤皂甙,Helixin,Tauroside E,α-Hederin,Hederoside C |
Apoptosis; Others | Apoptosis; Others |
Alpha-Hederin (Tauroside E) 是存在于黑种草种子中的一种单桥糖三萜皂苷,具有抗肿瘤作用。它可通过激活线粒体依赖性途径抑制胃癌细胞增殖,诱导凋亡,并有活性氧生成和谷胱甘肽减少。 | |||
T5725 |
Salvianolic acid B
丹酚酸B,lithospermic acid B,Dan Shen Suan B |
Sirtuin; Autophagy | Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Salvianolic acid B (Dan Shen Suan B) 是一种来自丹参的天然产物,是一种抗氧化剂,具有水溶性。Salvianolic acid B 具有抗血小板聚集、抗凝和抗血栓作用,常用来研究微循环疾病。 | |||
T2719 |
Succinic acid
Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid |
Endogenous Metabolite | Metabolism |
Succinic acid (1,2-Ethanedicarboxylic acid) 是无氧代谢的发酵产物,也是三羧酸循环的中间产物。 | |||
T2946 |
Tanshinone IIA sulfonate sodium
丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium |
CaMK; P450; Calcium Channel | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Tanshinone IIA sulfonate sodium (Tanshinone IIA sodium sulfonate) 是从丹参中提取的丹参酮IIA 的水溶性衍生物,是SOCE 抑制剂,用于心血管疾病的研究。 | |||
T0433 |
Artesunate
WR-256283,青蒿琥酯 |
Virus Protease; Ferroptosis; STAT; Parasite | Apoptosis; JAK/STAT signaling; Microbiology/Virology; Stem Cells |
Artesunate (WR-256283) 是治疗疟疾的青蒿素组药物的一部分。 它是青蒿素的半合成衍生物,具有水溶性。 | |||
T5082 |
Calcium 2-hydroxy-4-(methylthio)butanoate
羟基蛋氨酸钙,calcium hydroxymethionine,2-Hydroxy-4-(methylthio)butyric acid calcium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Calcium 2-hydroxy-4-(methylthio)butanoate (Calcium 2-hydroxy-4-(calcium hydroxymethionine)) 是内源性代谢产物的一种。 | |||
T11060 |
DMAPT
Dimethylamino Parthenolide |
NF-κB | NF-κB |
DMAPT (Dimethylamino Parthenolide) 是一种具有口服活性的NF-κB 抑制剂,是一种 Parthenolide (PTL) 的类似物,对原发性急性髓性白血病细胞的LD50值为1.7 μM。具有潜在的抗肿瘤和抗转移作用。 | |||
T6272 |
Fosbretabulin Disodium
Combretastatin A4 Phosphate,CA 4DP,CA 4P,福他布林,Combretastatin A4 disodium phosphate,Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium |
Apoptosis; Microtubule Associated | Apoptosis; Cytoskeletal Signaling |
Fosbretabulin Disodium (CA 4P) 是一种微管蛋白去稳定剂,是 Combretastatin A4 前药,可选择性靶向内皮细胞,诱导新生肿瘤新血管消退,减少肿瘤血流量并引起中央肿瘤坏死。 | |||
T4773 |
3-Ethoxy-3-oxopropanoic acid
Monoethyl malonic acid,Ethyl hydrogen malonate,丙二酸单乙酯 |
Others; Endogenous Metabolite | Metabolism; Others |
3-Ethoxy-3-oxopropanoic acid (Monoethyl malonic acid) 是内源性代谢产物的一种。 | |||
T2818 |
Methyl Vanillate
|
Reactive Oxygen Species; Wnt/beta-catenin; Endogenous Metabolite | Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells |
Methyl vanillate 是一种枳椇属植物中的提取物,是Wnt/β-catenin 信号通路活化剂,是一种香草酸的甲酯。它具有抗氧化作用。 | |||
T0879 |
Niacin
Vitamin B3,烟酸(维生素B3),Nicotinic acid |
Endogenous Metabolite; Autophagy | Autophagy; Metabolism |
Niacin (Nicotinic acid),也称为烟酸和维生素 B3,是一种水溶性必需的 B 族维生素,用于治疗维生素缺乏症以及高脂血症,血脂异常,高甘油三酯血症,并降低心肌梗塞的风险 | |||
T3947 |
Nonanoic acid
pelargonic acid,Nonoic acid,壬酸 |
Others; Antibacterial | Microbiology/Virology; Others |
Nonanoic acid (Nonoic acid) 是一种天然存在的具有九个碳原子的饱和脂肪酸。它减少细菌易位,增强抗菌活性,并增加猪 β-防御素 1 (pBD-1) 和 pBD-2 的分泌。 | |||
T6480 |
D-Pantothenic acid
vitamin B5,pantothenate,D-泛酸 |
Others | Others |
D-Pantothenic acid (vitamin B5) 是必需的微量营养素,是辅酶 A 的前体,在很多生物过程中发挥关键作用,如调节碳水化合物,脂质,蛋白和核酸代谢。 | |||
T4768 |
Diethyl oxalpropionate
草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE |
Others; Endogenous Metabolite | Metabolism; Others |
Diethyl oxalpropionate (HYL 2-METHYL-3-OXOSUCCINATE) 是一种合成 PDMMLA 的中间体。其中 PDMMLA 的衍生物可用于纳米粒子的合成和研究。 | |||
Fr13883 |
3-Methoxyphenylacetic acid
|
Others | Others |
3-Methoxyphenylacetic acid 是 m-hydroxyphenylacetic (m-OHPAA) 的衍生物,茄形假丝酵母中的一种植物毒素。它可用于针对介氧菌根腐烂的毒素介导的生物测定法的开发。 | |||
T1040 |
Vitamin B12
Cyanocobalamin,Cobalamin,维生素B12 |
Endogenous Metabolite | Metabolism |
Vitamin B12 (Cobalamin) 是一种维生素,在维持血流形成和脑、神经系统正常功能等方面发挥关键作用。 | |||
T2823 |
Crocin
西红花苷,藏红花,Gardenia Yellow,Alpha-Crocin,藏红花素 |
Others | Others |
Crocin (Gardenia Yellow) 是从Crocus sativus 柱头中分离出的主要成分,是一种营养保健品,具有抗炎,抗癌,抗抑郁和抗惊厥等强大的药理作用。 | |||
T4798 |
N-Acetyl-L-leucine
|
Others; Endogenous Metabolite | Metabolism; Others |
N-Acetyl-L-leucine 是内源性代谢产物的一种。 | |||
T1331 |
Riboflavin phosphate sodium
Riboflavin 5'-phosphate sodium,核黄素磷酸钠(维生素B2),Vitamin B2 Phosphate Sodium Salt,Flavin mononucleotide,FMN,核黄素磷酸钠,FMN-Na,riboflavin-5'-phosphate |
Endogenous Metabolite | Metabolism |
Riboflavin phosphate sodium (FMN) 是 riboflavin 的磷酸钠盐形式,riboflavin 是一种水溶性和必需的微量营养素,是自然产生的维生素B复合物的主要生长促进因子。Riboflavin phosphate sodium 转化为2种辅酶,黄素单核苷酸(FMN)和黄素腺嘌呤二核苷酸(FAD),这两种辅酶通过帮助脂肪、碳水化合物和蛋白质的代谢来产生能量,并且是红细胞形成和呼吸、抗体产生以及调节人体生长和繁殖所必需的。 | |||
T13777 |
Moniliformin sodium salt
|
Others | Others |
Moniliformin sodium salt is water-soluble mycotoxin isolate from Fusarium moniliforme. | |||
T34489 |
Salicifoline
|
||
Salicifoline is a water-soluble quaternary ammonium alkaloid. | |||
T29888 |
Aloe-emodin-glucoside
|
||
Aloe-emodin-glucoside is a stimulant-laxative which has been shown to enhance colonic membrane permeability of water-soluble and poorly permeable compounds. | |||
T0879L |
Niacin hydrochloride
|
||
Niacin hydrochloride is a water-soluble vitamin of the B complex occurring in various animal and plant tissues. It is needed by the body for the formation of coenzymes NAD and NADP. It possesses PELLAGRA-curative, vasodilating, and antilipemic properties. | |||
TN6613 |
Delphinidin-3-O-galactoside chloride
|
||
Delphinidin-3-O-galactoside chloride has anti-obesity and hypolipidemic effects. Delphinidin-3-O-galactoside (D3G) is a water-soluble anthocyanin with antioxidant activity. D3G is capable of masking the EGCG-induced cytotoxicity and ER stress, presumably | |||
TN2112 |
Przewalskinic acid A
|
Others | Others |
Przewalskinic acid A is a rare, water-soluble, and highly biologically active ingredient found, thus far, only in the Salvia przewalskii Maxim herb. | |||
T20854 |
Isethionic acid
Hydroxyethylsulfonic acid,Ethanolsulfonic acid |
Others | Others |
Isethionic acid, a major metabolite in F. cylindrus, is an organosulfur compound containing a short-chain alkane sulfonate linked to a hydroxyl group. It is a water-soluble liquid for the manufacture of mild, biodegradable, and high-foaming anionic surfac | |||
T16332 |
NKH477
Colforsin dapropate hydrochloride |
NMDAR | Neuroscience |
NKH477 is a novel water-soluble forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 shows an antiproliferative effect in vivo with an altered cytokine profile to inhibit the acute | |||
T82148 |
Hydrogenated soya phosphatidylcholines
|
Others | Others |
Hydrogenated soya phosphatidylcholines 是一种用于提升水溶性药物口服给药效果的天然产物,它能够增加药物负荷和溶解度,从而延长药物释放时间。 | |||
T35981 |
Biliverdin hydrochloride
|
Antioxidant | oxidation-reduction |
Biliverdin hydrochloride 是一种由血红素氧化形成的四吡咯水溶性化合物,具有潜在的抗氧化活性,参与胆绿素-胆红素氧化还原系统。 | |||
T35710 |
N-Acetyl-S-allyl-L-cysteine
|
Others | Others |
L-Deoxyalliin , also known as S-allyl-L-cysteine, is a water soluble organosulfur compound derived from garlic that has neuroprotective and antioxidative activities. N-Acetyl-S-allyl-L-cysteine is a principal metabolite of L-deoxyalliin in humans, mice, rats, and dogs. It is readily detected in plasma and urine. The conversion of L-deoxyalliin to N-acetyl-S-allyl-L-cysteine appears to be mediated by a family of flavin-containing monooxygenases. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-03230 |
PHB depolymerase Protein, Ralstonia pickettii, Recombinant (His)
Poly(3-hydroxybutyrate) depolymerase |
Ralstonia pickettii | E. coli |
This protein degrades water-insoluble and water-soluble PHB to monomeric D(-)-3-hydroxybutyrate. PHB depolymerase Protein, Ralstonia pickettii, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 50.9 kDa and the accession number is P12625. | |||
TMPH-01298 |
EPHX1 Protein, Human, Recombinant (His)
EPHX1,Microsomal epoxide hydrolase,Epoxide hydratase,Epoxide... |
Human | E. coli |
Biotransformation enzyme that catalyzes the hydrolysis of arene and aliphatic epoxides to less reactive and more water soluble dihydrodiols by the trans addition of water. Plays a role in the metabolism of endogenous lipids such as epoxide-containing fatty acids. Metabolizes the abundant endocannabinoid 2-arachidonoylglycerol (2-AG) to free arachidonic acid (AA) and glycerol. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T30599 |
BS3-d4 Deuterated Crosslinker
Deuterated Crosslinker BS3-d4,BS3-d4,D4-BS3 |
||
BS3-d4 Deuterated Crosslinker or Bis(Sulfosuccinimidyl) 2,2,7,7-suberate-d4, is a water-soluble and membrane impermeable protein crosslinking agent. | |||
T30598 |
BS2G-d4 Deuterated Crosslinker
D4-BS2G,BS2G-d4 |
||
BS2G-d4 or Bis(Sulfosuccinimidyl) 2,2,4,4-glutarate-d4, is a water-soluble and membrane impermeable protein crosslinking agent. | |||
TMID-0257 |
Quinoline-d7
|
||
Quinoline-d7 是 Quinoline 的氘代化合物。Quinoline 的 CAS 号为 91-22-5。Quinoline 存在于酒精饮料中。 它是一种来自包括薄荷在内的多种植物的生物碱。 也存在于可可、红茶和苏格兰威士忌中。 老化的样品,如果暴露在光线下,会变成黄色,然后变成棕色。 | |||
TMIJ-0373 |
Biotin-d2
|
||
Biotin-d2 是 Biotin 的氘代化合物。Biotin 的 CAS 号为 58-85-5。Biotin 是一种水溶性B族维生素,是细胞生长、脂肪酸产生以及脂肪和氨基酸代谢所必需的。 | |||
TMID-0029 |
Succinic-2,2,3,3-d4 Acid
|
||
Succinic-2,2,3,3-d4 Acid 是 Succinic Acid 的氘代化合物。Succinic Acid 的 CAS 号为 110-15-6。Succinic acid 是无氧代谢的发酵产物,也是三羧酸循环的中间产物。 | |||
TMIJ-0435 |
Octanoic Acid-d15
|
||
Octanoic Acid-d15 是 Octanoic Acid 的氘代化合物。Octanoic Acid 的 CAS 号为 124-07-2。Caprylic acid天然存在于椰子和母乳中。它是一种油性液体,带有些许腐臭味,能用于酯类香料和染料的生产。 | |||
TMIJ-0519 |
Fosaprepitant-d4 Dimeglumine
|
||
Fosaprepitant-d4 Dimeglumine 是 Fosaprepitant Dimeglumine 的氘代化合物。Fosaprepitant Dimeglumine 的 CAS 号为 265121-04-8。Fosaprepitant dimeglumine 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。 | |||
TMIJ-0053 |
2-Methylpropionic-d7 acid
|
||
2-Methylpropionic-d7 acid 是 2-Methylpropionic acid 的氘代化合物。2-Methylpropionic acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。 | |||
TMIJ-0047 |
Isobutyric-d6 acid
|
||
Isobutyric-d6 acid 是 Isobutyric acid 的氘代化合物。Isobutyric acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。 |