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Search Results for " cleavable "
Targets Recommended: Others

616

抑制剂 & 化合物

2

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2

重组蛋白

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T18866 UV Cleavable Biotin-PEG2-Azide

Others Others
UV Cleavable Biotin-PEG2-Azide, a PEG-based PROTAC linker, enables the synthesis of PROTACs[1].
T17475 Azido-C3-UV-biotin

UV Cleavable Biotin-PEG2-alkyne

Others Others
Azido-C3-UV-biotin is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T15175 DSP Crosslinker

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DSP Crosslinker 是一种可降解的 ADC 连接剂,用于合成可用于合成抗体偶联药物。
T15171 DSG Crosslinker

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DSG Crosslinker 是用于合成抗体偶联药物的 linker,可降解。
T15058 DBCO-amine

ADC Linker Antibody-drug Conjugate/ADC Related
DBCO-amine 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T22334 FMOC-3VVD-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-3VVD-OH 是一种可降解的 ADC 连接剂,用于合成抗体-药物偶联物。
T17950 Fmoc-Asp-NH2

FMOC-L-异天冬酰胺

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Asp-NH2 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T16218 N-Boc-PEG5-bromide

Others; PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; Others; PROTAC
N-Boc-PEG5-bromide 是 PROTAC 的 linker,属于 PEG 类和 Alkyl/ether 类.它也是可降解的 ADC 连接桥,用于抗体药物结合物的合成。
T18143 m-PEG12-OH

Dodecaethylene Glycol Monomethyl Ether

Others; PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; Others; PROTAC
m-PEG12-OH (Dodecaethylene Glycol Monomethyl Ether) 是一种基于 PEG 的 PROTAC 接头,可用于 PROTAC 的合成。它也是一种不可切割的 12 单元 PEG ADC 接头,用于合成抗体-药物偶联物。
T18408 N-Butanoyl-L-homoserine lactone

N-丁酰基-L-高丝氨酸内酯,N-Butyryl-L-homoserine lactone,C4-HSL

Antibacterial; ADC Linker Antibody-drug Conjugate/ADC Related; Microbiology/Virology
N-Butanoyl-L-homoserine lactone 是一种可降解的ADClinker,用于抗体偶联药物的合成。它可用于抗菌生物膜,具有抗菌活性。它的适配体抑制铜绿假单胞菌生物膜的形成,可用于阻止群体感应。
T17213 Val-cit-PAB-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Val-cit-PAB-OH 是可降解ADC 连接剂。
T17946 Fmoc-Ala-Ala-Asn(Trt)-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Ala-Ala-Asn(Trt)-OH 是一种可切割的 ADC 接头,用于抗体-药物偶联物。
T17372 Ald-Ph-NHS ester

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Ald-Ph-NHS ester 是用于抗体-药物偶联的不可切割接头。
T17977 Fmoc-PEA

ADC Linker Antibody-drug Conjugate/ADC Related
Fmoc-PEA 是一种可降解的抗体偶联药物 (ADC)的linker。
T17691 Boc-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-OH 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T15179 DTSSP Crosslinker

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DTSSP Crosslinker 是一种可降解的 ADC linker,可用于合成抗体-药物偶联物 (ADCs)。
T14271 Aminooxy-PEG4-alcohol

Others; PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; Others; PROTAC
Aminooxy-PEG4-alcohol 既是不可裂解的 4 单元 PEG ADC linker,也是基于 PEG 的 PROTAC linker。
T18868 Val-Cit

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Val-Cit 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T18308 MC-Gly-Gly-Phe

ADC Linker Antibody-drug Conjugate/ADC Related
MC-Gly-Gly-Phe 是一种用于抗体-药物偶联物的可切割接头。
T22278 BOC-Dap-NE

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Dap-NE 是一种二肽,用作一种可降解的 ADC 连接剂,可用于合成抗体偶联药物。
T17654 Boc-NH-C6-Br

N-BOC-6-溴代己胺

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-NH-C6-Br 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T38953 Azido-C6-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Azido-C6-OH 是可降解的 ADC linker,可用于合成抗体偶联药物。
T17953 Fmoc-Gly-Gly-Phe-OtBu

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Gly-Gly-Phe-OtBu 是一种用于合成抗体偶联药物的 linker,可降解。
T16437 PC Biotin-PEG3-alkyne

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
PC Biotin-PEG3-alkyne 是一种 ADC 连接剂,可裂解的 3 单元 PEG,还可以用于合成抗体药物共轭物 (ADC)。
T14392 Azide-C2-SS-C2-biotin

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Azide-C2-SS-C2-biotin 是一种可裂解的生物素化试剂 ,是可用于合成抗体偶联活性分子的 ADC linker。
T39222 Mc-VC-PAB-SN38

Mc-VC-PAB-SN38

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Mc-VC-PAB-SN38 由可降解 (cleavable) 的 ADC linker (Mc-VC-PAB) 和 SN38 组成,属于抗体偶联活性分子的一部分,常用来合成靶向作用位点的抗体偶联活性分子 (ADC)。
T17952 Fmoc-Gly-Gly-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Gly-Gly-OH 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T9783 Boc-C16-COOH

PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
Boc-C16-COOH 可以作为 ADC linker 或 PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T9781 Boc-C14-COOH

十六烷基二酸单叔丁酯

PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
Boc-C14-COOH 可以作为 ADC linker 或PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T16225 N-Hydroxysulfosuccinimide sodium

ADC Linker Antibody-drug Conjugate/ADC Related
N-Hydroxysulfosuccinimide sodium 是一种不可降解的 ADC 连接剂,用于合成抗体-药物偶联物。
T14833L BS3 Crosslinker disodium

双琥珀酰亚胺辛二酸酯钠盐

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
BS3 Crosslinker disodium 是一种不可切割的 ADC 接头,用于合成抗体-药物偶联物。
T17692 Boc-Val-Cit-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-PAB-PNP 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
FL0195 N-Boc-4-hydroxy-L-proline methyl ester

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
N-Boc-cis-4-hydroxy-L-proline methyl ester为不可降解(non-cleavable)的ADC linker,用于抗体药物偶联体(ADCs)合成。该化合物同时作为基于烷基链(alkyl chain)的PROTAC linker,适用于PROTAC合成。
T17679 Boc-NH-PEG4-CH2CH2NH2

Others; PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; Others; PROTAC
Boc-NH-PEG4-CH2CH2NH2 是一种可切割的 5 单元 PEG ADC 接头,用于合成抗体-药物偶联物。它也是一种基于 PEG 的 PROTAC 连接剂,可用于 PROTAC 的合成。
T17693 Boc-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-PAB 是一种可切割的 ADC 接头,用于抗体-药物偶联物的合成。
T5149 MC-Val-Cit-PAB

N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺

Others; AChR; ADC Linker Antibody-drug Conjugate/ADC Related; Neuroscience; Others
MC-Val-Cit-PAB 是一种组织蛋白酶可裂解的 ADC 接头,用于制备抗体-药物偶联物。
T61156 L-Lysyl-L-lysine dihydrochloride

Lysyllysine dihydrochloride

Others Others
L-Lysyl-L-lysine dihydrochloride (Lysyllysine dihydrochloride) 是一种酶可裂解的接头。L-Lysyl-L-lysine dihydrochloride 可用作递送多种生物活性肽的简单接头。
T18719 SPP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
SPP 是一种可裂解的连接体,可用于形成对癌症有治疗作用的抗体偶联化合物。
T18467 N3-C4-NHS ester

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
N3-C4-NHS ester 是一种不可切割的 ADC 接头,用于合成抗体-药物偶联物。
T17576 Biotin-PEG3-SS-azide

Biotin-PEG3-amido-SS-amido-azide

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Biotin-PEG3-SS-azide (Biotin-PEG3-amido-SS-amido-azide) 是一种可裂解的ADC 连接物,含有3个单位的PEG,可用于合成抗体-药物结合物。
T14746 Boc-NH-PEG4-CH2COOH

N-叔丁氧羰基-四聚乙二醇-乙酸

PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
Boc-NH-PEG4-CH2COOH 是一种可切割的 ADC 接头,用作抗体-药物偶联物的接头。它也是基于 PEG 的 PROTAC 接头,可用于 PROTAC 的合成。
T18529 PDEC-NB

4-Nitrophenyl 2-(Pyridin-2-Yldisulfanyl)Ethyl Carbonate

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
PDEC-NB (4-Nitrophenyl 2-(Pyridin-2-Yldisulfanyl)Ethyl Carbonate) 是用于抗体-药物偶联物的二硫键可切割接头。
T17017 TCO-PEG4-NHS ester

PROTACs; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
TCO-PEG4-NHS ester 是一种属于 PEG 类的 PROTAC 连接桥。TCO-PEG4-NHS ester 可用于合成一系列 PROTAC 分子。TCO-PEG4-NHS ester 是一种可降解 (cleavable) 且可用于抗体活性分子结合物 (ADCs) 的合成 ADC 连接桥。
T18540 Phe-Lys(Trt)-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Phe-Lys(Trt)-PAB 是一种组织蛋白酶可裂解的 ADC 接头,用于合成抗体-药物偶联物。
T9785 20-(tert-Butoxy)-20-oxoicosanoic acid

PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
20-(tert-Butoxy)-20-oxoicosanoic acid 可以作为 ADC linker 或 PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T18318 MC-Val-Ala-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
MC-Val-Ala-PAB-PNP 是一种用于合成抗体偶联药物的 linker,可降解。
T15067 DBCO-NHS ester

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DBCO-NHS ester 是一种 ADC 连接剂,可裂解的 3 单元 PEG,还可以用于合成抗体药物共轭物 (ADC)。
T18267 Mal-PEG1-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mal-PEG1-Val-Cit-OH是一种在抗体药物偶联体(ADCs)[1]合成中使用的可裂解单元聚乙二醇(PEG)连接器。
T15839 m-PEG12-amine

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
m-PEG12-amine是一种基于PEG的PROTAC连接器,同时也是一种在PROTACs[1]和抗体药物偶联物(ADCs)[2]的合成中使用的不可切割的12单位PEG ADC连接器。
TP1535L GPLGIAGQ acetate

GPLGIAGQ acetate(109053-09-0 Free base)

MMP Proteases/Proteasome
GPLGIAGQ acetate 是一种 MMP2 可切割的多肽。GPLGIAGQ acetate 可用作脂质体和胶束纳米载体中的刺激敏感接头,以在光动力治疗中合成独特的 MMP2 靶向光敏剂。

化合物

UV Cleavable Biotin-PEG2-Azide
Cat.No: T18866
Synonym:
Target: Others
Azido-C3-UV-biotin
Cat.No: T17475
Synonym: UV Cleavable Biotin-PEG2-alkyne
Target: Others
DSP Crosslinker
Cat.No: T15175
Synonym:
Target: Others, ADC Linker
DSG Crosslinker
Cat.No: T15171
Synonym:
Target: Others, ADC Linker
DBCO-amine
Cat.No: T15058
Synonym:
Target: ADC Linker
FMOC-3VVD-OH
Cat.No: T22334
Synonym:
Target: Others, ADC Linker
Fmoc-Asp-NH2
Cat.No: T17950
Synonym: FMOC-L-异天冬酰胺
Target: Others, ADC Linker
N-Boc-PEG5-bromide
Cat.No: T16218
Synonym:
Target: Others, PROTAC Linker, ADC Linker
m-PEG12-OH
Cat.No: T18143
Synonym: Dodecaethylene Glycol Monomethyl Ether
Target: Others, PROTAC Linker, ADC Linker
N-Butanoyl-L-homoserine lactone
Cat.No: T18408
Synonym: N-丁酰基-L-高丝氨酸内酯,N-Butyryl-L-homoserine lactone,C4-HSL
Target: Antibacterial, ADC Linker
Val-cit-PAB-OH
Cat.No: T17213
Synonym:
Target: Others, ADC Linker
Fmoc-Ala-Ala-Asn(Trt)-OH
Cat.No: T17946
Synonym:
Target: Others, ADC Linker
Ald-Ph-NHS ester
Cat.No: T17372
Synonym:
Target: Others, ADC Linker
Fmoc-PEA
Cat.No: T17977
Synonym:
Target: ADC Linker
Boc-Val-Cit-OH
Cat.No: T17691
Synonym:
Target: Others, ADC Linker
DTSSP Crosslinker
Cat.No: T15179
Synonym:
Target: Others, ADC Linker
Aminooxy-PEG4-alcohol
Cat.No: T14271
Synonym:
Target: Others, PROTAC Linker, ADC Linker
Val-Cit
Cat.No: T18868
Synonym:
Target: Others, ADC Linker
MC-Gly-Gly-Phe
Cat.No: T18308
Synonym:
Target: ADC Linker
BOC-Dap-NE
Cat.No: T22278
Synonym:
Target: Others, ADC Linker
Boc-NH-C6-Br
Cat.No: T17654
Synonym: N-BOC-6-溴代己胺
Target: Others, ADC Linker
Azido-C6-OH
Cat.No: T38953
Synonym:
Target: Others, ADC Linker
Fmoc-Gly-Gly-Phe-OtBu
Cat.No: T17953
Synonym:
Target: Others, ADC Linker
PC Biotin-PEG3-alkyne
Cat.No: T16437
Synonym:
Target: Others, ADC Linker
Azide-C2-SS-C2-biotin
Cat.No: T14392
Synonym:
Target: Others, ADC Linker
Mc-VC-PAB-SN38
Cat.No: T39222
Synonym: Mc-VC-PAB-SN38
Target: Others, Drug-Linker Conjugates for ADC
Fmoc-Gly-Gly-OH
Cat.No: T17952
Synonym:
Target: Others, ADC Linker
Boc-C16-COOH
Cat.No: T9783
Synonym:
Target: PROTAC Linker, ADC Linker
Boc-C14-COOH
Cat.No: T9781
Synonym: 十六烷基二酸单叔丁酯
Target: PROTAC Linker, ADC Linker
N-Hydroxysulfosuccinimide sodium
Cat.No: T16225
Synonym:
Target: ADC Linker
BS3 Crosslinker disodium
Cat.No: T14833L
Synonym: 双琥珀酰亚胺辛二酸酯钠盐
Target: Others, ADC Linker
Boc-Val-Cit-PAB-PNP
Cat.No: T17692
Synonym:
Target: Others, ADC Linker
N-Boc-4-hydroxy-L-proline methyl ester
Cat.No: FL0195
Synonym:
Target: Others, ADC Linker
Boc-NH-PEG4-CH2CH2NH2
Cat.No: T17679
Synonym:
Target: Others, PROTAC Linker, ADC Linker
Boc-Val-Cit-PAB
Cat.No: T17693
Synonym:
Target: Others, ADC Linker
MC-Val-Cit-PAB
Cat.No: T5149
Synonym: N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺
Target: Others, AChR, ADC Linker
L-Lysyl-L-lysine dihydrochloride
Cat.No: T61156
Synonym: Lysyllysine dihydrochloride
Target: Others
SPP
Cat.No: T18719
Synonym:
Target: Others, ADC Linker
N3-C4-NHS ester
Cat.No: T18467
Synonym:
Target: Others, ADC Linker
Biotin-PEG3-SS-azide
Cat.No: T17576
Synonym: Biotin-PEG3-amido-SS-amido-azide
Target: Others, ADC Linker
Boc-NH-PEG4-CH2COOH
Cat.No: T14746
Synonym: N-叔丁氧羰基-四聚乙二醇-乙酸
Target: PROTAC Linker, ADC Linker
PDEC-NB
Cat.No: T18529
Synonym: 4-Nitrophenyl 2-(Pyridin-2-Yldisulfanyl)Ethyl Carbonate
Target: Others, ADC Linker
TCO-PEG4-NHS ester
Cat.No: T17017
Synonym:
Target: PROTACs, ADC Linker
Phe-Lys(Trt)-PAB
Cat.No: T18540
Synonym:
Target: Others, ADC Linker
20-(tert-Butoxy)-20-oxoicosanoic acid
Cat.No: T9785
Synonym:
Target: PROTAC Linker, ADC Linker
MC-Val-Ala-PAB-PNP
Cat.No: T18318
Synonym:
Target: Others, ADC Linker
DBCO-NHS ester
Cat.No: T15067
Synonym:
Target: Others, ADC Linker
Mal-PEG1-Val-Cit-OH
Cat.No: T18267
Synonym:
Target: Others, ADC Linker
m-PEG12-amine
Cat.No: T15839
Synonym:
Target: Others, ADC Linker
GPLGIAGQ acetate
Cat.No: TP1535L
Synonym: GPLGIAGQ acetate(109053-09-0 Free base)
Target: MMP
Cat. No. Product Name Target Signaling Pathways
T9784 Docosanedioic acid 

PROTAC Linker; ADC Linker Antibody-drug Conjugate/ADC Related; PROTAC
Docosanedioic acid 可以作为ADC linker 或PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。

天然产物

Docosanedioic acid 
Cat.No: T9784
Synonym:
Target: PROTAC Linker, ADC Linker
Irinotecan Hydrochloride
Cat.No: T0486L
Synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
Cat. No. Product Name Species Expression System
TMPJ-01092 MGAT2 Protein, Human, Recombinant (His)

Alpha-1,Mannoside Acetylglucosaminyltransferase 2,6-Mannosyl...

Human HEK293 Cells
Mannoside Acetylglucosaminyltransferase 2 (MGAT2) is a single-pass type II membrane protein that contains the typical glycosyltransferase domains: a short N-terminal cytoplasmic domain, a hydrophobic non-cleavable signal-anchor domain and a C-terminal catalytic domain. MGAT2 catalyzes an essential step in the conversion of oligo-mannose to complex N-glycans. Defects in MGAT2 are the cause of congenital disorder of glycosylation type 2A.
TMPY-01217 ANGPTL5 Protein, Human, Recombinant (GST)

angiopoietin like 5,ANGPTL5

Human Baculovirus Insect Cells
The angiopoietins are protein growth factors that promote angiogenesis, the formation of blood vessels from pre-existing blood vessels. There are now four identified angiopoietins: Ang1, Ang2, Ang3, Ang4. In addition, there are a number of proteins that are closely related to angiopoietins (ANGPTL2, ANGPTL3, ANGPTL4, ANGPTL5, ANGPTL6, ANGPTL7). Angiopoietin-like 5 (ANGPTL5) is mainly expressed in adult heart. Like other members of the angiopoietin family, ANGPTL5-deduced protein also has an N-te...

重组蛋白

MGAT2 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01092
Species: Human
Expression System: HEK293 Cells
ANGPTL5 Protein, Human, Recombinant (GST)
Cat.No: TMPY-01217
Species: Human
Expression System: Baculovirus Insect Cells
Cat. No. Product Name Target Signaling Pathways
TMID-0078 Irinotecan-d10 Hydrochloride

Irinotecan-d10 Hydrochloride 是 Irinotecan Hydrochloride 的氘代化合物。Irinotecan Hydrochloride 的 CAS 号为 100286-90-6。Irinotecan Hydrochloride 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。

同位素标记化合物

Irinotecan-d10 Hydrochloride
Cat.No: TMID-0078
Synonym:
Target:
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