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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0930 |
Sulfadiazine
Sulphadiazine,磺胺嘧啶 |
Antibacterial; Antibiotic; Parasite; Autophagy | Autophagy; Microbiology/Virology |
Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。 | |||
T37688 |
Cyfluthrin
|
Reactive Oxygen Species; Sodium Channel | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB |
Cyfluthrin 属于 II 型拟除虫菊酯,对多种昆虫都有杀灭效果。Cyfluthrin 是Nav1.8钠通道调节剂。它可应用于农业、兽医、杀虫剂、拟除虫菊酯和贮存产品等领域。 | |||
T0668 |
1-Aminohydantoin hydrochloride
|
Others | Others |
1-Aminohydantoin hydrochloride 是一种呋喃妥因在动物组织中的主要代谢物。它与组织蛋白共价结合,在微酸性条件下从组织中释放出来,与 2-硝基苯甲醛衍生形成 AHD 的硝基苯基衍生物可被检测。它可作为测定肉、奶等兽药残留的测定指标。 | |||
T6114 |
Nifursol
硝呋索尔,尼呋索尔 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Nifursol 是一种具有口服活性的兽用抗生素,用于预防组织口炎。它快速代谢形成代谢标记物 3,5-二硝基水杨酸环肼,并能持续很长时间。它可研究沙门氏菌感染的家禽、家禽和水生动物的大肠杆菌肠胃病。 | |||
T1550 |
Thiamphenicol
甲砜霉素,Dextrosulphenidol,Thiophenicol |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。 | |||
T0456 |
Cinchophen
2-苯基-4-喹啉羧酸,辛可芬,Cinconal |
COX | Immunology/Inflammation; Neuroscience |
Cinchophen (Cinconal) 是口服具有活性的非甾体抗炎试剂,具有抗菌活性。它可用于研究关节炎和某些肝脏疾病。 | |||
T1647 |
Ronidazole
洛硝哒唑,Ronidazol,罗硝唑,Ridzol |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Ronidazole (Ronidazol) 是一种口服有效的抗原虫和抗菌试剂。它在猫模型中对胎儿三毛滴虫有效,还可研究组织口癣和猪痢疾。 | |||
T1177 |
Sulfaquinoxaline
磺胺喹恶啉,Avicocid,磺胺喹噁啉,Sulphaquinoxaline,Sulfabenzpyrazine |
Others; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Others |
Sulfaquinoxaline (Sulfabenzpyrazine) 是一种兽用抗菌剂,对革兰氏阴性菌和革兰氏阳性菌均有活性。它能用于预防球虫病和细菌感染。 | |||
T22228 |
Tylvalosin tartrate
酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) 是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。 | |||
T13633 |
D-Phenothrin
(-)-trans-Phenothrin,右旋苯醚菊酯 |
Parasite | Microbiology/Virology |
D-Phenothrin ((-)-trans-Phenothrin) 是一种口服有效的 II 型合成拟除虫菊酯,广泛用于杀死昆虫,蚊子和人类虱子。它还用于兽医,保护农作物和控制动物上的害虫。 | |||
T6992 |
Sulfadiazine sodium
Sulfadiazin-natrium,磺胺嘧啶钠,Sodium sulfadiazine |
Others; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Others |
Sulfadiazine sodium (Sulfadiazin-natrium) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。 | |||
T0917 |
Sulfaquinoxaline sodium salt
SQ-Na,磺胺喹恶啉钠盐,Sulfaquinoxaline sodium,磺胺喹啉钠 |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Sulfaquinoxaline sodium salt (SQ-Na) 是一种兽用广谱抗菌剂,有抗革兰氏阴性菌和革兰氏阳性菌活性。Sulfaquinoxaline 能用于预防球虫病和细菌感染。 | |||
T20702 |
Ormetoprim
Ro5-9754,奥美普林,Ro 5-9754,Ro-5-9754 |
Antibiotic | Microbiology/Virology |
Ormetoprim (Ro 5-9754) 是一种兽用抗菌剂,通常用于水产养殖和家禽行业,可以预防疾病在淡水水产养殖中的传播,促进家畜的生长。 | |||
T1141 |
Fenbendazole
Fenbendazol,苯硫咪唑,芬苯达唑,Phenbendasol,Panacur |
Others; HIF/HIF Prolyl-Hydroxylase; Antibiotic; Parasite | Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Others |
Fenbendazole (Fenbendazol) 是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。 | |||
T38724 |
Modoflaner
|
Parasite | Microbiology/Virology |
Modoflaner 是一种抗寄生虫剂 (兽医用)。 | |||
T1251 |
Dicloralurea
双(三氯乙醛基)脲,Dichlorolurea,双 (三氯乙醛基) 脲,DCU |
Others | Others |
Dicloralurea (DCU) 是一种兽用的食品添加剂,可用作生长刺激剂。 | |||
T20082 |
Dymanthine
十八烷基二甲基叔胺,Adogen 342D,ADMA 18 |
Others | Others |
Dymanthine (ADMA 18) 是驱虫药,对多种肠道蠕虫感染具有潜在的研究价值。 | |||
T1617 |
Enrofloxacin
恩诺沙星,BAY-Vp2674,PD160788 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Enrofloxacin (BAY-Vp2674) 是一种作用于支原体的抗生素,MIC90为 0.312 μg/mL。 | |||
T0198 |
Ceftiofur sodium
Naxcel,头孢噻呋钠,Sodium ceftiofur |
Antibacterial; Antibiotic | Microbiology/Virology |
Ceftiofur sodium (Naxcel) 是一种兽用头孢菌素类抗生素。 | |||
T7096 |
Tildipirosin
|
Antibacterial; Antibiotic | Microbiology/Virology |
Tildipirosin 是一种具有长效抗菌作用的大环内酯抗生素。 | |||
T6398 |
Azaperone
R-1929,Fluoperidol,阿扎哌隆,Stresnil,NSC 170976,Suicalm |
Others; Dopamine Receptor | GPCR/G Protein; Neuroscience; Others |
Azaperone (Fluoperidol) 是多巴胺拮抗剂,具有一些抗组胺和抗胆碱特性,具有止吐活性。 | |||
T0870 |
Altrenogest
R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素 |
Estrogen/progestogen Receptor; Progesterone Receptor | Endocrinology/Hormones; Others |
Altrenogest (Allyltrenbolone) 是一种结构与trenbolone 相关的孕激素,能作用于孕激素受体。 | |||
T2184 |
Sulfachloropyridazine
Sulfachlorpyridazine,磺胺二甲基嘧啶 |
Antibacterial; Antibiotic | Microbiology/Virology |
Sulfachloropyridazine (Sulfachlorpyridazine) 是一种广谱磺酰胺,抑制革兰氏阳性和革兰氏阴性好氧细菌的生长。 | |||
T0777 |
Tilmicosin
LY-177370,替米考星,EL-870 |
Antibacterial; Antibiotic | Microbiology/Virology |
Tilmicosin (EL-870) 是一种抗生素,可研究曼氏杆菌和巴氏杆菌相关的牛羊呼吸系统疾病。 | |||
T15272 |
Febantel
|
Parasite | Microbiology/Virology |
Febantel 是一种用于家禽和家畜的蛔虫、绦虫感染的驱虫剂。 | |||
T0770 |
Carbadox
Getroxel,卡巴多,Mecadox |
Antibacterial; Antibiotic | Microbiology/Virology |
Carbadox (Mecadox) 是一种喹喔啉二氧化氮抗生素,用于育龄期的猪,治疗猪痢疾和肠炎,促进成长。 | |||
T13823 |
Polyvinylpyrrolidone
PVP,Povidone,Polyvidone,聚乙烯吡咯烷酮 |
Others | Others |
Polyvinylpyrrolidone (Polyvidone) 与碘和其他化合物结合后,可用作人类和兽医学中有效的伤口愈合促进剂和消毒剂。 | |||
T6607 |
Nitenpyram
烯啶虫胺,Niterndipoine,烯啶蟲胺,Bestguard,Capstar |
AChR | Neuroscience |
Nitenpyram (Capstar) 是一种烟碱型乙酰胆碱受体 (AchR) 激动剂,IC50为 14 nM,用作治疗牲畜和宠物寄生虫的兽药。 | |||
T36020 |
Florfenicol amine hydrochloride
|
Antibiotic | Microbiology/Virology |
Florfenicol amine hydrochloride 是一种人工合成的兽用抗生素,具有抗菌活性。Florfenicol amine hydrochloride 在水产养殖业和牧业养殖业中应用广泛,可以用来研究巴氏杆菌、爱德华氏菌、大肠杆菌和沙门氏杆菌引起的疾病。 | |||
T0066 |
Dichlorophen
双氯酚,DDM,Dichlorophene |
Antibacterial; Parasite; Antifungal | Microbiology/Virology |
Dichlorophen (DDM) 是一种抗微生物剂,对绦虫,原生动物,真菌和细菌具有活性,通过增加肠道内容物的清除,消除肠道中的绦虫感染。 | |||
T7865 |
Danofloxacin
达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine |
Others; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。 | |||
T31928 |
Giminabant
|
Others | Others |
Giminabant is an antagonist of cannabinoid receptor antagonist (veterinary use). | |||
T39425 |
Umifoxolaner
|
Others | Others |
Umifoxolaner is an anti-parasitic agent (veterinary). | |||
T26679 |
Atelocantel
AH 353623,AH-353623,AH353623 |
Others | Others |
Atelocantel is an anthelmintic agent (veterinary drug). | |||
T32539L |
Laidlomycin propionate potassium
RS11988,RS 11988,RS-11988,Cattlyst |
Others | Others |
Laidlomycin propionate potassium is a growth stimulant (Veterinary). | |||
T19744 |
Isometamidium chloride
A-4180,A4180,A 4180 |
Others | Others |
Isometamidium chloride is an antiprotozoal agent. It is also used in veterinary medicine. | |||
T38840 |
Mivorilaner
|
Others | Others |
Mivorilaner is an antineoplastic compound that has shown potential for application in veterinary medicine research (WO2012155676, Example 245). | |||
T13027 |
Sulfaethoxypyridazine
|
Antibacterial | Microbiology/Virology |
Sulfaethoxypyridazine is an agent of sulfonamide antibacterial. Sulfaethoxypyridazine is a sulfonamide that is used in veterinary medicine as feedstuffs. | |||
T31377 |
Demiditraz
PF 3814927,PF-3814927,PF3814927 |
Others | Others |
Demiditraz(PF-3814927) is an acaricide (veterinary use). | |||
T30964 |
Clamoxyquin hydrochloride
Clamoxyquin HCl,Clamoxyquin dihydrochloride,CN-17,900-2B,Clamoxyquine hydrochloride,CN 17900-2 B |
Others | Others |
Clamoxyquin hydrochloride is an anti ameba and antidiarrheal drug. It has been used as a veterinary drug to treat salmon infected with brain armyworm. | |||
T28976 |
Tigolaner
|
Others | Others |
Tigolaner is a antiparasitic drug candidate for veterinary use. | |||
T39627 |
Ocarocoxib
|
Others | Others |
Ocarocoxib, a potent COX- 2 (cyclooxygenase- 2) inhibitor, is a non-steroidal anti-inflammatory for veterinary use. | |||
T32915 |
Lubabegron
LY 488756,LY488756,LY-488756 |
Others | Others |
Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary. | |||
T84389 |
Valnemulin
|
Others | Others |
Valnemulin, a broad-spectrum pleuromutilin antibiotic, targets peptidyl transferase within the 50S ribosomal subunit, effectively used in veterinary medicine to address swine diseases such as B. hyodysenteriae and M. hyopneumoniae. | |||
T0872 |
Amprolium
氨丙啉,安普罗林 |
Others; Parasite | Microbiology/Virology; Others |
Amprolium 是一种干扰硫胺素代谢的兽用球虫抑制剂。 | |||
T19697 |
Norgestomet
SC21009,Norprogesterone, Syncro-Mate B,SC-21009,SC 21009 |
Others | Others |
Norgestomet is a steroidal progestin of the 19-norprogesterone group used in veterinary medicine to control estrus and ovulation in cattle. In addition to the progesterone receptor, norgestomet possesses a weak (micromolar) affinity for the glucocorticoid | |||
T62200 |
Bunamidine hydrochloride
|
Others | Others |
Bunamidine hydrochloride 是一种兽用抗扁形虫剂,能够作用于细粒棘球绦虫和带状绦虫。 | |||
T39154 |
Demethyl linezolid
|
Others | Others |
Demethyl linezolid is an impurity observed in linezolid, an antimicrobial compound. It exhibits effective antimicrobial properties against various human and veterinary pathogens. | |||
T12742 |
Ro 20-0657/000
|
Others | Others |
Ro 20-0657/000 is a Trimethoprim metabolite. Trimethoprim is an inhibitor of dihydrofolate reductase, used as an antibacterial agent in human and veterinary medicine. | |||
T2214 |
Flumethrin
|
Others | Others |
Flumethrin 是一种拟除虫菊酯类杀虫剂。外用在兽药中,用于防治牛、绵羊、山羊、马和狗身上的寄生虫和蜱,以及治疗蜜蜂群中的寄生虫。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8065 |
Tiamulin
Thiamutilin,泰妙菌素 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Tiamulin (Thiamutilin) 是一类二萜,广泛用于控制猪的传染疾病,包括猪痢疾和地方性肺炎等。 | |||
T0861 |
Tylosin tartrate
酒石酸泰洛星,酒石酸泰乐菌素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。 | |||
T1003 |
Tylosin
Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylosin (Tylosine) 是一种兽医用大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。 | |||
T2769 |
3-Aminopropionitrile fumarate (2:1)
Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,3-氨基丙腈,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate |
Others | Others |
3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) 是一种能抑制胶原蛋白(collagen)交联的山黧豆素。 | |||
T5040 |
Medroxyprogesterone
甲羟孕酮,甲孕酮 |
Estrogen/progestogen Receptor; Progesterone Receptor | Endocrinology/Hormones; Others |
Medroxyprogesterone 是一种合成的人孕酮变体,是孕酮受体激动剂,用于治疗肾癌。在兽医实践中用作发情调节剂。 | |||
T1381 |
Milbemycin oxime
|
Others; Antibiotic; Parasite | Microbiology/Virology; Others |
Milbemycin oxime 是一种大环内酯,具有广谱抗寄生虫活性。它由 Milbemycin A4 和 A3 组成。它可结合谷氨酸门控的氯离子通道,可作用于肠道线虫,肺和心脏蠕虫。 | |||
T1679 |
Thiostrepton
Thiactin,Bryamycin,Alaninamide,硫链丝菌素 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。 | |||
TN6564 |
Palustrol
|
||
Palustrol exhibits acaricidal, insecticidal, 'pesticidal' and/or arthropod repellent properties, may be useful sources of chemicals for the control of arthropods of medical, veterinary or agricultural importance. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-03035 |
M-myrmeciitoxin-Mp2b Protein, Myrmecia pilosula, Recombinant (GST & His)
DELTA-myrtoxin-Mp1a B chain,Pilosin-3 subunit b,M-myrmeciito... |
Myrmecia pilosula | Baculovirus Insect Cells |
Heterodimer protein that may serve both defensive (pain-inducing) and predatory (insecticidal) roles. Has membrane-disrupting activity and shows induction of non-specific calcium influx into cells,. Shows broad-spectrum activity against a diverse range of bacteria, and cell lines, as well as hemolytic activity (EC(50)=2.18 uM). In vivo, shows moderate insecticidal activity against D.melanogaster and potent anthelmintic activity against the veterinary nematode H.contortus. In addition, intraplant... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIJ-0307 |
Fenbendazole-d3
|
||
Fenbendazole-d3 是 Fenbendazole 的氘代化合物。Fenbendazole 的 CAS 号为 43210-67-9。Fenbendazole是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。 | |||
TMID-0008 |
Boldenone-d3
|
||
Boldenone-d3 是 Boldenone 的氘代化合物。Boldenone 的 CAS 号为 846-48-0。Boldenone 是一种为兽医开发的合成代谢类固醇。 | |||
TMIH-0532 |
Sulfachloropyridazine-d4
|
||
Sulfachloropyridazine-d4 是 Sulfachloropyridazine 的氘代化合物。Sulfachloropyridazine 的 CAS 号为 80-32-0。Sulfachloropyridazine 是一种广谱磺酰胺,抑制革兰氏阳性和革兰氏阴性好氧细菌的生长。 | |||
TMIJ-0288 |
Danofloxacin-d3
|
||
Danofloxacin-d3 是 Danofloxacin 的氘代化合物。Danofloxacin 的 CAS 号为 112398-08-0。Danofloxacin free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。 | |||
TMID-0133 |
Medroxyprogesterone-d3
|
||
Medroxyprogesterone-d3 是 Medroxyprogesterone 的氘代化合物。Medroxyprogesterone 的 CAS 号为 520-85-4。Medroxyprogesterone 是一种合成的人孕酮变体,是孕酮受体激动剂,用于治疗肾癌。在兽医实践中用作发情调节剂。 | |||
TMIJ-0520 |
(1E,13E) Tilmicosin-d3
|
||
(1E,13E) Tilmicosin-d3 是 Tilmicosin 的氘代化合物。Tilmicosin 的 CAS 号为 108050-54-0。Tilmicosin是一种抗生素,可研究曼氏杆菌和巴氏杆菌相关的牛羊呼吸系统疾病。 | |||
T71984 |
Enrofloxacin-d5
|
||
Enrofloxacin-d5 is intended for use as an internal standard for the quantification of enrofloxacin by GC- or LC-MS. Enrofloxacin is a fluoroquinolone antibiotic. It is active against panels of Campylobacter, E. coli, and Salmonella isolates (mean MIC50s = 0.06, 0.5, and 0.03 µg/ml, respectively). It is also active against equine isolates of L. intracellularis (MICs = 0.125-0.5 µg/ml). Enrofloxacin inhibits bacterial DNA gyrase. In vivo, enrofloxacin (10 mg/kg) increases survival in a mouse model... | |||
TMIJ-0009 |
1-Amino Hydantoin-13C3
|
||
1-Amino Hydantoin-13C3 是 1-Amino Hydantoin 的 13C 的标记化合物。1-Amino Hydantoin 的 CAS 号为 6301-02-6。1-Aminohydantoin 是一种呋喃妥因在动物组织中的主要代谢物。1-Aminohydantoin 与组织蛋白共价结合,在微酸性条件下从组织中释放出来,与 2-硝基苯甲醛衍生形成 AHD 的硝基苯基衍生物可被检测。1-Aminohydantoin 可作为测定肉、奶等兽药残留的测定指标。 | |||
T36021 |
Flumequine-13C3
Flumequine-13C3 |
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Flumequine-13C3is intended for use as an internal standard for the quantification of flumequine by GC- or LC-MS. Flumequine is a fluoroquinolone antibiotic.1It is active againstS. aureus, S. pyogenes, B. subtilis, E. coli, P. aeruginosa, S. faecalis, andK. pneumoniae(MICs = 1-100 μg/ml). Flumequine is also active against field isolates of B. hyodysenteriae (MICs = 6.25-200 μg/ml).2It inhibits DNA gyrase, disrupting supercoiling of bacterial DNA to block transcription and replication.3In vivo, fl... |