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Search Results for " oxytocin "

Targets Recommended: Oxytocin Receptor Others

73

抑制剂 & 化合物

4

天然产物

3

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T21534L	Oxytocin C-terminal tripeptide Acetate Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base)	Others	Others
	Oxytocin C-terminal tripeptide Acetate 是 Oxytocin 的 C-末端三肽。Oxytocin 是哺乳动物的神经垂体激素，催产素受体的配体。
T40756	[Asp5]-Oxytocin [Asp5]-Oxytocin
	[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity.
T40534	[Leu3]-Oxytocin [Leu3]-Oxytocin
	[Leu3]-Oxytocin, an oxytocin analogue, is a derivative of oxytocin wherein the leucine amino acid (Leu) has been substituted at the 3rd position in the sequence.
T40536	[Glu4]-Oxytocin [Glu4]-Oxytocin
	[Glu4]-Oxytocin is a suitable derivative of oxytocin for conducting a thorough investigation, utilizing various methods, into the conformation of "oxytocin-like" molecules in aqueous solution.
T40658	[D-Asn5]-Oxytocin [D-Asn5]-Oxytocin
	[D-Asn5]-Oxytocin exhibits minimal specific oxytocic and vasodepressor effects. Comparative cumulative dose-response investigations reveal that [D-Asn5]-Oxytocin demonstrates a similar intrinsic activity to oxytocin in terms of oxytocic activity.
T33850	Oxytocin, deamino-6-carba- Deamino-6-carbaoxytocin,beta-Deaminocystathionine-oxytocin	Others	Others
	Deamino-6-carba-oxytoxin (dC60), a potent oxytocin analog considered to be resistant to some of the physiologically significant enzymic systems.
T39388	Oxytocin parallel dimer
	Oxytocin parallel dimer is the disulfide-bridged homo peptide dimer.
T39420	Oxytocin antiparallel dimer
	Oxytocin antiparallel dimer is the disulfide-bridged homo peptide dimer.
T40528	Oxytocin free acid 9-Deamidooxytocin
	Oxytocin free acid, also known as 9-Deamidooxytocin, is an analog of oxytocin where the glycinamide residue at position 9 has been substituted with a glycine residue. Oxytocin, a pleiotropic peptide hormone, has wide-ranging implications for general health, adaptation, development, reproduction, and social behavior.
T33849	Oxytocin, deamino-1-carba- Deamino-1-carbaoxytocin	Others	Others
	Oxytocin, deamino-1-carba- is a biochemical.
T80136	Val9-Oxytocin	Vasopressin Receptor	GPCR/G Protein
	Val9-Oxytocin为完全抗拮抗加压素(1a)受体的化合物，其结构上是Oxytocin的衍生物，特点在于Gly9位点被Val9取代。
T76624	(Ile8)-Oxytocin
	(Ile8)-Oxytocin 是一种神经垂体激素间催产素，在有袋动物中产生。
T80133	Pro8-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Pro8-Oxytocin是一种改良的OXT配体。在灵长类动物OXTR中，Pro8-Oxytocin比标准哺乳动物OXT配体Leu8-Oxytocin诱发更强效的反应和显著的行为影响。相较于Vasopressin (AVP)，Pro8-Oxytocin对人类AVPR1a的活性较低，但对狨猴AVPR1a的激活作用则高于AVP。
T12331	OT-R antagonist 2 Oxytocin receptor antagonist 2	Others	Others
	OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .
T12331L	OT-R antagonist 1 Oxytocin receptor antagonist 1	Others	Others
	OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM). OT-R antagonist 1 is a new effective and selective nonpeptide low molecular weight OT-R antagonist.
T76211	[Asp5]-Oxytocin acetate
	[Asp5]-Oxytocin acetate 是一款功能强大的5位 (5-position) 神经垂体激素类似物，能引发体外大鼠子宫收缩，其效果可被 Mg2+ 增强。此化合物展现出在大鼠子宫收缩、禽血管抑制及大鼠抗利尿作用方面的活性。
T76629	(Phe2,Orn8)-Oxytocin
	'(Phe2,Orn8)-Oxytocin' 作为选择性 V1 加压素激动剂，具有引发兔附睾持续收缩的功能，其EC50值达280 nM。
T80134	Pro8-Oxytocin TFA	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Pro8-Oxytocin TFA 作为一种优化的OXT配体，在灵长类动物OXTR上展现出较Leu8-Oxytocin更强的功能反应和行为效应。相对于AVP，在人类AVPR1a上的活性较低，但在狨猴AVPR1a上则显示出更高的活性。
T76265	(Thr4,Gly7)-Oxytocin
	(Thr4,Gly7)-Oxytocin，一种Oxytocin类似物，特异性激活OT受体。通过激活TRPV1通道及抑制K+通道，诱导眼下神经元兴奋。
T80140	(Val3,Pro8)-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	"(Val3,Pro8)-Oxytocin"为Gq依赖性途径的激动剂，同时作为β-arrestin结合及催产素受体（OXTR）内化作用的次级激动剂。
T78021	Oxytocin parallel dimer TFA
	Oxytocin parallel dimer TFA为具有催产素和加压素样活性的二硫键桥连同肽二聚体，其毒性低于催产素。
T81583	Oxytocin antiparallel dimer TFA
	Oxytocin antiparallel dimer TFA为一种通过二硫键桥联形成的同肽二聚体。该化合物展现出催产素和加压素样的生物活性，同时具有低于催产素的毒性。
T76630	(Phe2,Orn8)-Oxytocin acetate
	(Phe2,Orn8)-Oxytocin acetate 是一种选择性 V1 加压素 (V1 vasopressin) 激动剂，能诱导兔附睾持续收缩，其EC50值为 280 nM。
T5148	Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban acetate (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T11857	LIT-001	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	LIT-001 是非肽类催产素受体激动剂，EC50为55 nM，Ki 为226 nM。它可改善孤独症小鼠模型的社交互动。
T80126	(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	'(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin (OVT)' 是催产素受体的一种拮抗剂，主要应用于神经系统疾病的研究领域。
T4996	Atosiban 阿托西班,RWJ22164,RW22164	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T7601L	Carbetocin acetate 醋酸卡贝缩宫素,Carbetocin acetate(37025-55-1 free base),卡贝缩宫素醋酸盐	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Carbetocin acetate 是催产素类似物，是催产素受体激动剂，Ki 是 7.1 nM。它对催产素受体的嵌合 N 末端具有高亲和力，Ki 为 1.17 μM。它能透过血脑屏障，可以通过激活 CNS 中的催产素受体而具有类抗抑郁活性，具有用于产后出血的研究潜力。
T7601	Carbetocin 卡贝缩宫素,醋酸卡贝缩宫素	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Carbetocin 是催产素类似物，是催产素受体激动剂，Ki 是 7.1 nM。它对催产素受体的嵌合 N 末端具有高亲和力，Ki 为 1.17 μM。它能透过血脑屏障，可以通过激活 CNS 中的催产素受体而具有类抗抑郁活性，具有用于产后出血的研究潜力。
T76049	Demoxytocin
	Demoxytocin为一种异源性环肽，属于催产素类似物。其通过影响细胞膜通透性，提升平滑肌细胞内钙离子含量，进而加强平滑肌细胞收缩力，具备刺激子宫平滑肌收缩的能力，发挥催产素功能。此外，Demoxytocin在研究早产破裂引发的分娩刺激中有应用。
T37694	N-Acetyloxytocin
	N-Acetyloxytocin, a chemical compound, has been identified and analyzed in the neurointermediate lobe of the rat pituitary (NIL). Furthermore, its presence has also been detected in various brain regions of the rat[1].
T3347	PF3274167 PF 3274167,Cligosiban,PF-3274167	OX Receptor	GPCR/G Protein; Neuroscience
	PF3274167 (Cligosiban) 是一种有效的、选择性的、高亲和力的非肽催产素受体拮抗剂。
T11794	L-368,899 hydrochloride L-368899 hydrochloride,L-368,899 HCl	OX Receptor	GPCR/G Protein; Neuroscience
	L-368,899 hydrochloride 是一种可口服且具有选择性的非肽类催产素受体(OXTR)拮抗剂，可用于预防早产。L-368,899 hydrochloride 可预防催产素诱导的抗异常性疼痛和抗厌恶，可用于研究抑郁症。
TP1400L	[Arg8]-Vasotocin acetate（113-80-4 free base)	Others	Others
	[Arg8]-Vasotocin acetate（113-80-4 free base) 是一种存在于非哺乳动物脊椎动物神经垂体中的激素，与加压素和催产素有关。
T28855	SSR126768A SSR-126768A,SSR 126768A	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	SSR126768A 是一种新型且具有选择性、口服活性和有效性的催产素(OT)受体拮抗剂，对子宫收缩有抑制作用，可用于预防早产。
T15682	L-371,257	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	L-371,257 是催产素受体的竞争性拮抗剂，pA2 为 8.4，Ki 为 19 nM。 L-371,257 对加压素受体 1a 的 Ki 值为 3.7 nM。
TP2082L	d[Cha4]-AVP acetate(500170-27-4 free base)	Vasopressin Receptor	GPCR/G Protein
	d[Cha4]-AVP acetate(500170-27-4 free base) 是一种有效的选择性人血管加压素 V1B 受体激动剂（V1B、V1A、催产素和 V2 受体的 Ki 值分别为 1.2、151、240 和 750 nM）。刺激 ACTH 和皮质酮分泌，并在体内表现出微不足道的血管加压活性。
T16736	Retosiban GSK 221149,GSK 221149A	Others	Others
	Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).
T23441	TC OT 39	Others	Others
	oxytocin receptor partial agonist
T24286	L 364918 L364,918,L-364918,L-364,918,L 364,918,L364918	Others	Others
	L 364918 is an oxytocin antagonist.
T27763	L-366509 L 366,509,L 366509,L366,509,L-366,509	Others	Others
	L-366,509 is an antagonist of oxytocin.
T23528	WAY-267464	Others	Others
	oxytocin receptor (OTR) agonist
T11502	Epelsiban GSK 557296	Others	Others
	Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).
T24291	L 366811 L 366,811,L-366,811,L366811,L366,811,L-366811	Others	Others
	L 366811 is a potent oxytocin antagonist.
T24288	L 365209 L365,209,L365209,L 365,209,L-365,209,L-365209	Others	Others
	L 365209 is an oxytocin antagonist.
T24289	L 366682 L366,682,L-66,682,L 366,682,L-366682,L366682	Others	Others
	L 366682 is an oxytocin antagonist.
T12334	OT antagonist 3	Others	Others
	OT antagonist 3 is an antagonist of oxytocin (OT).
T24292	L 366948 L366,948,L-366948,L-366,948,L 366,948,L366948	Others	Others
	L 366948 is an antagonist of the oxytocin receptor.
T28018	Merotocin FE202767,FE 202767,FE-202767	Others	Others
	Merotocin is a potent and highly selective peptidic agonist of the oxytocin receptor.
T24278	L 156373 L-156373,L156373	Others	Others
	L 156373 is an oxytocin antagonist.

化合物

Oxytocin C-terminal tripeptide Acetate

Cat.No: T21534L

Synonym: Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base)

Target: Others

[Asp5]-Oxytocin

Cat.No: T40756

Synonym: [Asp5]-Oxytocin

[Leu3]-Oxytocin

Cat.No: T40534

Synonym: [Leu3]-Oxytocin

[Glu4]-Oxytocin

Cat.No: T40536

Synonym: [Glu4]-Oxytocin

[D-Asn5]-Oxytocin

Cat.No: T40658

Synonym: [D-Asn5]-Oxytocin

Oxytocin, deamino-6-carba-

Cat.No: T33850

Synonym: Deamino-6-carbaoxytocin,beta-Deaminocystathionine-oxytocin

Target: Others

Oxytocin parallel dimer

Cat.No: T39388

Oxytocin antiparallel dimer

Cat.No: T39420

Oxytocin free acid

Cat.No: T40528

Synonym: 9-Deamidooxytocin

Oxytocin, deamino-1-carba-

Cat.No: T33849

Synonym: Deamino-1-carbaoxytocin

Target: Others

Val9-Oxytocin

Cat.No: T80136

Target: Vasopressin Receptor

(Ile8)-Oxytocin

Cat.No: T76624

Pro8-Oxytocin

Cat.No: T80133

Target: Oxytocin Receptor

OT-R antagonist 2

Cat.No: T12331

Synonym: Oxytocin receptor antagonist 2

Target: Others

OT-R antagonist 1

Cat.No: T12331L

Synonym: Oxytocin receptor antagonist 1

Target: Others

[Asp5]-Oxytocin acetate

Cat.No: T76211

(Phe2,Orn8)-Oxytocin

Cat.No: T76629

Pro8-Oxytocin TFA

Cat.No: T80134

Target: Oxytocin Receptor

(Thr4,Gly7)-Oxytocin

Cat.No: T76265

(Val3,Pro8)-Oxytocin

Cat.No: T80140

Target: Oxytocin Receptor

Oxytocin parallel dimer TFA

Cat.No: T78021

Oxytocin antiparallel dimer TFA

Cat.No: T81583

(Phe2,Orn8)-Oxytocin acetate

Cat.No: T76630

Atosiban acetate

Cat.No: T5148

Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班

Target: Oxytocin Receptor, Vasopressin Receptor

Cat.No: T11857

Target: Oxytocin Receptor

(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin

Cat.No: T80126

Target: Oxytocin Receptor

Cat.No: T4996

Synonym: 阿托西班,RWJ22164,RW22164

Target: Oxytocin Receptor, Vasopressin Receptor

Carbetocin acetate

Cat.No: T7601L

Synonym: 醋酸卡贝缩宫素,Carbetocin acetate(37025-55-1 free base),卡贝缩宫素醋酸盐

Target: Oxytocin Receptor

Cat.No: T7601

Synonym: 卡贝缩宫素,醋酸卡贝缩宫素

Target: Oxytocin Receptor

Cat.No: T76049

N-Acetyloxytocin

Cat.No: T37694

Cat.No: T3347

Synonym: PF 3274167,Cligosiban,PF-3274167

Target: OX Receptor

L-368,899 hydrochloride

Cat.No: T11794

Synonym: L-368899 hydrochloride,L-368,899 HCl

Target: OX Receptor

[Arg8]-Vasotocin acetate（113-80-4 free base)

Cat.No: TP1400L

Target: Others

Cat.No: T28855

Synonym: SSR-126768A,SSR 126768A

Target: Oxytocin Receptor

Cat.No: T15682

Target: Oxytocin Receptor, Vasopressin Receptor

d[Cha4]-AVP acetate(500170-27-4 free base)

Cat.No: TP2082L

Target: Vasopressin Receptor

Cat.No: T16736

Synonym: GSK 221149,GSK 221149A

Target: Others

Cat.No: T23441

Target: Others

Cat.No: T24286

Synonym: L364,918,L-364918,L-364,918,L 364,918,L364918

Target: Others

Cat.No: T27763

Synonym: L 366,509,L 366509,L366,509,L-366,509

Target: Others

Cat.No: T23528

Target: Others

Cat.No: T11502

Synonym: GSK 557296

Target: Others

Cat.No: T24291

Synonym: L 366,811,L-366,811,L366811,L366,811,L-366811

Target: Others

Cat.No: T24288

Synonym: L365,209,L365209,L 365,209,L-365,209,L-365209

Target: Others

Cat.No: T24289

Synonym: L366,682,L-66,682,L 366,682,L-366682,L366682

Target: Others

OT antagonist 3

Cat.No: T12334

Target: Others

Cat.No: T24292

Synonym: L366,948,L-366948,L-366,948,L 366,948,L366948

Target: Others

Cat.No: T28018

Synonym: FE202767,FE 202767,FE-202767

Target: Others

Cat.No: T24278

Synonym: L-156373,L156373

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T5026	Oxytocin 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Oxytocin (Oxytocin (Syntocinon)) 是哺乳动物的神经垂体激素，是多效的下丘脑肽，是催产素受体的配体，有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子，具有抗炎、抗氧化剂和保护作用。
T5145	Oxytocin acetate Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素，是多效的下丘脑肽，是催产素受体的配体，有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子，具有抗炎、抗氧化剂和保护作用。
T5065	GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP	PKA	Tyrosine Kinase/Adaptors
	GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) 也称为 cGMP，是一种细胞调节剂，被描述为第二信使。它的水平随着各种激素的增加而增加，包括乙酰胆碱、胰岛素和催产素。 cGMP 激活蛋白激酶 G(PKG) 并调节离子通道电导，信号传导影响多种过程，包括平滑肌松弛和增殖、光转导和能量稳态。
T36931	Penicillide	Others	Others
	Penicillide is a fungal metabolite originally isolated from Penicillium that has diverse biological activities. It is an inhibitor of calpain 2/m-calpain (IC50 = 7.1 μM) and acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 22.9 μM). It is also an antagonist of oxytocin receptors (IC50 = 67 μM). Penicillide inhibits RNA synthesis in P388 murine leukemia cells.

天然产物

Cat.No: T5026

Synonym: 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)

Target: Oxytocin Receptor

Oxytocin acetate

Cat.No: T5145

Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素

Target: Oxytocin Receptor

GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD

Cat.No: T5065

Synonym: Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP

Target: PKA

Cat.No: T36931

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-01820	OXT Protein, Human, Recombinant (His) OXT,Oxytocin-neurophysin 1	Human	P. pastoris (Yeast)
	Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR). OXT Protein, Human, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 11.6 kDa and the accession number is P01178.
TMPH-01821	OXT Protein, Human, Recombinant (His & Myc & SUMO) OXT,Oxytocin-neurophysin 1	Human	E. coli
	Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR). OXT Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 29.6 kDa and the accession number is P01178.
TMPY-03269	Prolyl Endopeptidase Protein, Mouse, Recombinant (His) PEP,AI450383,AI047692,D10Wsu136e,prolyl endopeptidase,Pop	Mouse	Baculovirus Insect Cells
	Prolyl endopeptidase, also known as PREP, belongs to a distinct class of serine peptidases. It is a large cytosolic enzyme which was first described in the cytosol of rabbit brain as an oligopeptidase. Prolyl endopeptidase degrades the nonapeptide bradykinin at the Pro-Phe bond. It is involved in the maturation and degradation of peptide hormones and neuropeptides such as alpha-melanocyte-stimulating hormone, luteinizing hormone-releasing hormone (LH-RH), thyrotropin-releasing hormone, angiotens...

重组蛋白

OXT Protein, Human, Recombinant (His)

Cat.No: TMPH-01820

Species: Human

Expression System: P. pastoris (Yeast)

OXT Protein, Human, Recombinant (His & Myc & SUMO)

Cat.No: TMPH-01821

Species: Human

Expression System: E. coli

Prolyl Endopeptidase Protein, Mouse, Recombinant (His)

Cat.No: TMPY-03269

Species: Mouse

Expression System: Baculovirus Insect Cells

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