motilin receptor

Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。

Motilin (26-47), human, porcine 是内源性 motilin 受体的激动剂，在中国仓鼠卵巢细胞中，Ki 值和EC50值分别为 2.3 和 0.3 nM。

[Leu13]-Motilin (KW-5139) 为motilin类似物，能够刺激家兔胃肠运动，并在体外以浓度依赖性方式引起胃窦、十二指肠、空肠、回肠以及降结肠的收缩。

[Nle13]-Motilin 是一种胃动素 (motilin) 类似物，可作为胃动素受体 motilin receptor 激动剂。

Idremcinal is a motilin receptor agonist.

Camicinal is a selective motilin receptor agonist (pEC50: 7.9).

YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).

MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 may be useful for gastrointestinal disorders associated with disturbed g