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Targets Recommended: Sodium Channel

6

抑制剂 & 化合物

1

天然产物

1

重组蛋白

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T0378 Oxybuprocaine hydrochloride

Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐

Sodium Channel Membrane transporter/Ion channel
Oxybuprocaine hydrochloride (Oxybuprocaine HCl) 是可逆的钠通道阻断剂,可防止角膜,结膜和巩膜中疼痛神经的冲动传播。Oxybuprocaine hydrochloride 专用于眼科与耳鼻喉科。
T0924 Benzocaine

苯唑卡因,苯佐卡因

Others; MRP; Sodium Channel Immunology/Inflammation; Membrane transporter/Ion channel; Others
Benzocaine 作用电压门控 Na+通道的共同受体,+30 mV 下的 IC50为0.8 mM。
T13830 Propoxycaine hydrochloride

Propoxycaine HCl

Sodium Channel Membrane transporter/Ion channel
Propoxycaine hydrochloride 是一种酯类局部麻醉剂,抑制电压门控的钠通道,可调节神经冲动,可诱导感觉丧失。Propoxycaine hydrochloride 可调节SPMVs脂质双层的流动。
T0222 Proparacaine hydrochloride

盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride

Apoptosis; Sodium Channel Apoptosis; Membrane transporter/Ion channel
Proparacaine hydrochloride (Proparacaine HCl) 是 Lidocaine 的衍生物,具有糖皮质激素样活性和免疫调节作用。
T0802 Procaine hydrochloride

Novocaine HCl,Procaine HCl,盐酸普鲁卡因

Histone Demethylase; 5-HT Receptor; DNA/RNA Synthesis; Sodium Channel; NMDAR; AChR Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Procaine hydrochloride (Novocaine HCl) 是DNA 脱甲基剂,是一种苯甲酸衍生物,具有局部麻醉和抗心律失常特性。
T6782 Benzocaine hydrochloride

Benzocaine HCl,Ethyl p-aminobenzoate hydrochloride,Ethyl 4-aminobenzoate hydrochloride

Sodium Channel Membrane transporter/Ion channel
Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) 是一种表面麻醉剂,通过阻止脉冲沿神经纤维和神经末梢传递而起作用。

化合物

Oxybuprocaine hydrochloride
Cat.No: T0378
Synonym: Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐
Target: Sodium Channel
Benzocaine
Cat.No: T0924
Synonym: 苯唑卡因,苯佐卡因
Target: Others, MRP, Sodium Channel
Propoxycaine hydrochloride
Cat.No: T13830
Synonym: Propoxycaine HCl
Target: Sodium Channel
Proparacaine hydrochloride
Cat.No: T0222
Synonym: 盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride
Target: Apoptosis, Sodium Channel
Procaine hydrochloride
Cat.No: T0802
Synonym: Novocaine HCl,Procaine HCl,盐酸普鲁卡因
Target: Histone Demethylase, 5-HT Receptor, DNA/RNA Synthesis, Sodium Channel, NMDAR, AChR
Benzocaine hydrochloride
Cat.No: T6782
Synonym: Benzocaine HCl,Ethyl p-aminobenzoate hydrochloride,Ethyl 4-aminobenzoate hydrochloride
Target: Sodium Channel
Cat. No. Product Name Target Signaling Pathways
T0894 Thiamine hydrochloride

盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride

Apoptosis; HBV; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology
Thiamine hydrochloride (Vitamin B1) 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。

天然产物

Thiamine hydrochloride
Cat.No: T0894
Synonym: 盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride
Target: Apoptosis, HBV, Endogenous Metabolite
Cat. No. Product Name Species Expression System
TMPY-01695 CASPR2 Protein, Mouse, Recombinant (His)

5430425M22Rik,Caspr2,contactin associated protein-like 2,mKI...

Mouse HEK293 Cells
CNTNAP2/CASPR2 is a member of the neurexin family which functions in the vertebrate nervous system as cell adhesion molecules and receptors. This protein, like other neurexin proteins, contains epidermal growth factor repeats and laminin G domains. In addition, it includes an F5/8 type C domain, discoidin/neuropilin- and fibrinogen-like domains, thrombospondin N-terminal-like domains and a putative PDZ binding site. CNTNAP2/CASPR2 is localized at the juxtaparanodes of myelinated axons, and media...

重组蛋白

CASPR2 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01695
Species: Mouse
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
TMIJ-0377 Thiamine Hydrochloride-13C4

Thiamine Hydrochloride-13C4 是 Thiamine Hydrochloride 的 13C 的标记化合物。Thiamine Hydrochloride 的 CAS 号为 67-03-8。Thiamine hydrochloride 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。

同位素标记化合物

Thiamine Hydrochloride-13C4
Cat.No: TMIJ-0377
Synonym:
Target:
TargetMol Loading
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