fiduxosin

Fiduxosin 是一种具有选择性和有效性的 α1-adrenoceptor 拮抗剂，对 α1a-adrenoceptor，α1b-adrenoceptor 和 α1d-adrenoceptor 有抑制作用，Ki 值分别为 0.160 nM，24.9 nM 和 0.920 nM。Fiduxosin 可用于治疗良性前列腺增生。

Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.

APHS is a cyclooxygenase-2 (COX-2) inhibitor with anti-inflammatory action. It also more potent than aspirin in the inhibition of COX-1.