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Search Results for " congener "

Targets Recommended: Adenosine Receptor

17

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T23535L	Xanthine amine congener trihydrochloride Xanthine amine congener trihydrochloride (96865-92-8 Free base)	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Xanthine amine congener trihydrochloride 是一种有效的腺苷拮抗剂，可逆转由腺苷激动剂 N6-环己基腺苷产生的尿流量、钠排泄和心率的减少。
T7683	Adenosine amine congener ADAC	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Adenosine amine congener (ADAC) 是一种选择性的 A1 腺苷受体激动剂，具有神经保护作用，可以改善噪音和顺铂引起的耳蜗损伤。
T39387	Xanthine amine congener dihydrochloride XAC dihydrochloride,Xanthine amine congener dihydrochloride	Others	Others
	Xanthine amine congener dihydrochloride (XAC dihydrochloride), a potent antagonist for both Adenosine A1 and A2 receptors, exhibits IC50 values of 1.8 nM for A1 and 114 nM for A2 receptors. Additionally, it functions as a convulsant agent in mouse models.
T23535	Xanthine amine congener	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Xanthine amine congener 是非选择性的腺苷受体拮抗剂，在小鼠中具有诱发惊厥的作用。
T62963	Xanthine amine congener hydrochloride	Others	Others
	Xanthine amine congener (XAC) hydrochloride 是一种非选择性腺苷受体拮抗剂，在小鼠中能够诱发惊厥。
T0797	Cimetidine 西米替汀,SKF-92334,西咪替丁	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Cimetidine (SKF-92334) 是一种可口服的可逆组胺H2受体拮抗剂，Ki 为 0.6 μM。它抑制胃酸分泌，以及胃蛋白酶和胃泌素的输出，具有抗癌和抗炎活性。
T1378	Tegafur Fluorafur,替加氟,FT-207,NSC 148958,FT 207	Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	Tegafur (FT 207) 是一种前药，在肝脏中被细胞色素 P-450 酶逐渐转化为氟尿嘧啶。它是抗代谢物氟尿嘧啶的同源物，具有抗肿瘤活性。
T21161	Ancitabine	Others	Others
	Ancitabine, a congener of cyterabine, is metabolized to cytarabine, thereby maintains a more constant antineoplastic action.
T72682	Lankacyclinone C	Others	Others
	Lankacyclinone C 是一种缺乏 δ-内酯部分的 lankacidin C 同源物，具有抗肿瘤活性。
T36162	8-iso Prostaglandin F1α 8-iso Prostaglandin F1α	Others	Others
	8-iso PGF1α is an isoprostane that was first identified in human semen. It is a member of the isoprostane family, which are eicosanoids of non-cyclooxygenase origin. 8-iso PGF1α is present along with its 19-hydroxy congener at 5-10 μg/ml of seminal plasma.
T37216	N-Arachidonoyl-L-Alanine
	Several different arachidonoyl amino acids, including N-arachidonoyl-L-alanine (NALA), have been isolated and characterized from bovine brain. The glycine congener (NAGly) was further characterized and found to suppress formalin-induced pain in rats. NALA may have activity at cannabinoid receptor and/or VR1, but has not been fully characterized to date.
T61409	CXCR4 antagonist 3	Others	Others
	CXCR4 antagonist 3 (compound 12a), an effective antagonist of CXCR4, exhibits an IC50 of 11 nM. It is a congener of TIQ15, showcasing exceptional properties such as CXCR4 antagonism, CYP 2D6 inhibition, metabolic stability, and permeability. With its potential for research on the human immunodeficiency virus, CXCR4 antagonist 3 holds great promise [1].
T37731	TPU-0037A	Others	Others
	TPU-0037A is an antibiotic and a congener of lydicamycin . It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs = 1.56-12.5 μg/ml), but not Gram-negative E. coli, P. mirabilis, P. vulgaris, or P. aeruginosa strains (MICs = >50 μg/ml).
T74722	Demethyl bleomycin A2	Others	Others
	Demethyl bleomycin A2 是Bleomycin 的同源物。Demethyl bleomycin A2 的 DNA 裂解对5-Methylcytidine 不敏感。
T84648	2-Linoleoyl Glycerol 2-LG	Others	Others
	2-Arachidonoyl glycerol (2-AG), a natural endocannabinoid ligand for the CB1 receptor, was isolated from porcine brain and characterized. Its congener, 2-linoleoyl glycerol (2-LG), which has a linoleoyl group instead of an arachidonoyl group, also exists alongside 2-AG in vivo. While 2-LG exhibits low intrinsic activity, it enhances the activity of 2-AG and other endocannabinoids through an "entourage" effect, attributed to the inhibition of breakdown and reuptake pathways that typically decreas...
T60728	M1 ligand 1	Others	Others
	M1 ligand 1 (compound 3b-b) 是槟榔碱衍生物的 N- 去甲基同源物，是毒蕈碱乙酰胆碱受体 M1 的配体。M1 ligand 1 用作正电子发射断层扫描(PET)的放射性示踪剂。
T38225	N-Arachidonoyl-3-hydroxy-γ-Aminobutyric Acid
	Several different arachidonoyl amino acids, including N-arachidonoyl-3-hydroxy-γ-aminobutyric acid (NAG-3H-ABA), have been isolated and characterized from bovine brain. The glycine congener was further characterized and found to suppress formalin-induced pain in rats. NAG-3H-ABA was also found in rat brain by LC-MS techniques, but has not been fully characterized to date. Most arachidonoyl amino acids are poor ligands for the CB1 receptor.

化合物

Xanthine amine congener trihydrochloride

Cat.No: T23535L

Synonym: Xanthine amine congener trihydrochloride (96865-92-8 Free base)

Target: Adenosine Receptor

Adenosine amine congener

Cat.No: T7683

Synonym: ADAC

Target: Adenosine Receptor

Xanthine amine congener dihydrochloride

Cat.No: T39387

Synonym: XAC dihydrochloride,Xanthine amine congener dihydrochloride

Target: Others

Xanthine amine congener

Cat.No: T23535

Target: Adenosine Receptor

Xanthine amine congener hydrochloride

Cat.No: T62963

Target: Others

Cat.No: T0797

Synonym: 西米替汀,SKF-92334,西咪替丁

Target: Histamine Receptor

Cat.No: T1378

Synonym: Fluorafur,替加氟,FT-207,NSC 148958,FT 207

Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis

Cat.No: T21161

Target: Others

Lankacyclinone C

Cat.No: T72682

Target: Others

8-iso Prostaglandin F1α

Cat.No: T36162

Synonym: 8-iso Prostaglandin F1α

Target: Others

N-Arachidonoyl-L-Alanine

Cat.No: T37216

CXCR4 antagonist 3

Cat.No: T61409

Target: Others

Cat.No: T37731

Target: Others

Demethyl bleomycin A2

Cat.No: T74722

Target: Others

2-Linoleoyl Glycerol

Cat.No: T84648

Synonym: 2-LG

Target: Others

Cat.No: T60728

Target: Others

N-Arachidonoyl-3-hydroxy-γ-Aminobutyric Acid

Cat.No: T38225

Cat. No.	Product Name	Target	Signaling Pathways
T3421	Nordihydrocapsaicin	Others	Others
	Nordihydrocapsaicin(诺地氢辣椒碱)是Capsaicin(辣椒素)的模拟物和同源物，属于在Capsicum(辣椒)中发现的Capsaicinoid(辣椒素类)化合物。
T1591	Ancitabine hydrochloride NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C	Others; DNA/RNA Synthesis; Autophagy	Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
	Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。

天然产物

Nordihydrocapsaicin

Cat.No: T3421

Target: Others

Ancitabine hydrochloride

Cat.No: T1591

Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Target: Others, DNA/RNA Synthesis, Autophagy

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