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Search Results for " anthelmintic "
Targets Recommended: Dopamine Receptor Antibacterial Antibiotic Antifungal

67

抑制剂 & 化合物

16

天然产物

1

重组蛋白

5

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T0776 Phenothiazine

ENT 38,吩噻嗪

Dopamine Receptor; Antibacterial; Antibiotic; Antifungal GPCR/G Protein; Microbiology/Virology; Neuroscience
Phenothiazine (ENT 38) 是一种抗生素,具有杀虫,抗菌,驱虫和杀真菌活性。它也可研究神经系统疾病。
T1546 Nitazoxanide

NSC 697855,硝唑尼特

Others; Influenza Virus; Parasite; Autophagy Autophagy; Microbiology/Virology; Others
Nitazoxanide (NSC-697855) 是一种广谱驱虫剂,对感染动物和人类的各种蠕虫、原生动物和肠道细菌都具有作用活性。 它在无菌培养中抑制Giardia lamblia 滋养体增殖,IC50为 2.4 μM。它可研究寄生虫性胃肠炎,具有抗病毒特性。
T19807 Dithiazanine iodide

Delvex,Telmide,Vercidon,Abminthic,Netocyd,NSC 221154

Others Others
Dithiazanine iodide (Netocyd) 是一种苯并噻唑。它已被用作抗虫剂。它作为纳米颗粒在治疗胶质母细胞瘤方面也很有效。
T0237 Closantel

氯氰碘柳胺,R-31520,氯生太尔

Antibacterial; Parasite Microbiology/Virology
Closantel (R-31520) 是抗寄生虫活性的卤化水杨酰苯胺。它是高度特异性盘尾丝虫几丁质酶抑制剂。
T6452 Closantel Sodium

Antibacterial; Parasite Microbiology/Virology
Closantel sodium 是抗寄生虫活性的卤化水杨酰苯胺。它是高度特异性的盘尾丝虫几丁质酶抑制剂。
T7901 Emodepside

Bay 44-4400

Parasite Microbiology/Virology
Emodepside (Bay 44-4400) 是一种对多种胃肠道线虫有效的驱虫药,具有广谱驱虫活性。
T10850L CMP-5 2HCl

Others Others
CMP-5 2HCl 是一种驱虫剂。CMP-5 2HCl 体外抗H. contortus 的EC100为5μM。
T7887 8-Hydroxyquinoline hemisulfate

8-羟基喹啉硫酸盐,Oxyquinoline sulfate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
8-Hydroxyquinoline hemisulfate (Oxyquinoline sulfate) 是一种单质子双齿螯合剂,具有温和的抑菌、驱虫和杀螨作用。
T16126 Monepantel

AAD1566,PPL-1

AChR Neuroscience
Monepantel (AAD1566) 是一种有机驱虫剂,也是来自蛔虫和食管造口的烟碱乙酰胆碱受体拮抗剂,广泛用于农牧业除虫。
T1343L Crystal Violet

Methyl Violet 10B,Hexamethylpararosaniline chloride,氯化结晶紫,Basic Violet 3,结晶紫,Gentian Violet

DNA; Influenza Virus; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Crystal Violet (Hexamethylpararosaniline chloride) 是革兰氏染色染料。它对H1N1具有抗病毒作用,有显著杀菌活性。
T7605 Avermectin B1a

阿维菌素 B1a,Abamectin B1a,Avamectin B1a

Antibiotic; Parasite Microbiology/Virology
Avermectin B1a 是能够使线虫瘫痪的一种抗寄生虫剂。
T20082 Dymanthine

十八烷基二甲基叔胺,Adogen 342D,ADMA 18

Others Others
Dymanthine (ADMA 18) 是驱虫药,对多种肠道蠕虫感染具有潜在的研究价值。
T7146 Piperazine adipate

Parasite Microbiology/Virology
Piperazine adipate 是一种广谱驱虫剂,可抵抗哺乳动物中很多常见的寄生虫感染。
T30819 CGP 20376

CGP-20376,CGP20376

Others Others
CGP 20376 是一种苯并噻唑化合物,是一种驱虫剂,对嗜酸性粒细胞呼吸爆发的双重剂量依赖性调节体外作用,具有抗纤特性。
T0714 Oxfendazole

奥吩达唑,奥芬哒唑,RS-8858

Glucokinase; Microtubule Associated; Parasite Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Oxfendazole (RS-8858) 是fenbendazole 的亚砜形式,是广谱苯并咪唑驱虫剂,可保护牲畜免受蛔虫、圆线虫和蛲虫的侵害。
T15272 Febantel

Parasite Microbiology/Virology
Febantel 是一种用于家禽和家畜的蛔虫、绦虫感染的驱虫剂。
T16539 Piperazine citrate

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Piperazine citrate 是一种六元环化合物,有驱虫的作用。
T0395 Pyrantel tartrate

Banminth,酒石酸噻吩嘧啶

Antibiotic; Parasite Microbiology/Virology
Pyrantel tartrate (Banminth) 是一种四氢嘧啶类广谱牲畜驱虫剂,是烟碱乙酰胆碱受体激动剂。它能引起寄生虫的痉挛性肌肉麻痹。它可研究胃肠道线虫感染。
T5836 Eprinomectin

依普菌素,MK-397

Parasite Microbiology/Virology
Eprinomectin (MK-397) 是一种阿维菌素,具有驱虫,杀虫杀螨活性。
T6372 Albendazole sulfoxide

Ricobendazole,Albendazole Oxide,阿苯达唑亚砜

Microtubule Associated; Parasite Cytoskeletal Signaling; Microbiology/Virology
Albendazole sulfoxide (Ricobendazole) 是一种驱虫药阿苯达唑的代谢物,有抗寄生虫活性。
T30596 Brotianide

BAY-VA 4059,Dirian,BAY-VA-4059,BAY-VA4059

Parasite Microbiology/Virology
Brotianide (BAY-VA4059) 具有驱虫活性,对肝吸虫和胃吸虫侵染具有很高的效力,可用于治疗绵羊的急性、亚急性和慢性肝脏法氏囊病感染。
T77684 4-(2-Aminoethyl)amino-7-chloroquinoline

N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine

Parasite Microbiology/Virology
4-(2-Aminoethyl)amino-7-chloroquinoline (N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine) 具有潜在的抗虫和抗肿瘤活性,可用于研究疟疾。
T0955 Oxyclozanide

Oxiclozanidum,Zanil,Oxyclozanid,Zanilox,氯羟柳胺

Antibiotic; Parasite Microbiology/Virology
Oxyclozanide (Oxyclozanid) 是一种水杨酰苯胺驱虫药,用于放牧动物的片形吸虫和绦虫感染。
T77507 (-)-Benzotetramisole

Others Others
(-)-Benzotetramisole 使一种高效且具有选择性的催化剂。(-)-Benzotetramisole 是抗蠕虫化合物四咪唑3 的苯annulated 衍生物,本身也是转化的有效催化剂。
T77643 2-(Chloromethyl)Imidazo[1,2-A]Pyridine

Others Others
2-(Chloromethyl)imidazo[1,2-a]pyridine 具有潜在的抗虫活性,可用于合成有活性的化合物。
T7093 Rafoxanide

碘醚柳胺,雷复尼特

CDK; Parasite Cell Cycle/Checkpoint; Microbiology/Virology
Rafoxanide 是口服活性水杨酰苯胺类驱虫剂。它作为抗寄生虫剂,可用于控制羊和牛的 Hemonchus 种和 Fasciola 种的感染。
T62769 Tribendimidine

AChR Neuroscience
Tribendimidine 是一种广谱的、口服具有活力的驱虫剂,也是一种 L 型烟碱乙酰胆碱受体 (nAChR) 激动剂。Tribendimidine 对 A. lumbricoides 和 N. americanus 具有极高的活性。
T1420 Diethylcarbamazine citrate

Caritrol,枸橼酸乙胺嗪,Loxuran,Dicarocide

Lipoxygenase; COX; Parasite Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Diethylcarbamazine citrate (Caritrol) 是驱肠虫药,主要用作治疗丝虫病的柠檬酸盐,是丝虫微丝蚴的花生四烯酸代谢抑制剂。
T0009 Flubendazole

氟苯咪唑,Flumoxanal,Flumoxane,NSC 313680,Fluvermal

Apoptosis; Microtubule Associated; Parasite Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Flubendazole (Flumoxane) 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。
T37072 Nitroxynil

4-Hydroxy-3-iodo-5-nitrobenzonitrile,Trodax,Dovenix

Parasite Microbiology/Virology
Nitroxynil (4-Hydroxy-3-iodo-5-nitrobenzonitrile) 为一种广泛用于研究 Fasciola hepatica 感染的驱虫剂,有效作用于寄生虫的成熟及未成熟阶段。
T0066 Dichlorophen

双氯酚,DDM,Dichlorophene

Antibacterial; Parasite; Antifungal Microbiology/Virology
Dichlorophen (DDM) 是一种抗微生物剂,对绦虫,原生动物,真菌和细菌具有活性,通过增加肠道内容物的清除,消除肠道中的绦虫感染。
T4059 Selamectin

UK-124114,司拉克丁,塞拉菌素

Chloride channel; P-gp; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Selamectin (UK-124114) 是半合成的大环内酯,是一种驱虫剂,可增强线虫中谷氨酸和 GABA 门控氯离子通道的开放。它还是抗寄生虫剂,可激活神经元和咽肌中的谷氨酸门控氯离子通道,以预防恶丝虫,淋巴丝虫和线虫感染。它还是 P-糖蛋白底物和抑制剂,IC50为 120 nM。
T0124 UK-124114

UNII-A2669OWX9N,西拉菌素,Selamectin

Others Others
UK-124114 (Selamectin) 是伊维菌素的大环内酯衍生物,伊维菌素是一种驱虫剂,可增强线虫中谷氨酸和 GABA 门控氯离子通道的开放。在 H. contortus 幼虫发育试验中,赛拉菌素 (0.1 µg/ml) 显示出生长抑制作用。
T25188 Butonate

NSC17872,NSC 17872,NSC-17872

Others Others
Butonate is an Anthelmintic agent.
T0323L Oxantel

Others Others
Oxantel is a fumarate reductase inhibitor with anthelmintic activity.
T34567 Sch 18099

Sch-18099,Sch18099

Others Others
Sch 18099 showed anthelmintic activity.
T30968 Clioxanide

Tremerad,SYD-230,SYD 230,Clioxanida,Clioxanidum

Others Others
Clioxanide is an anthelmintic agent.
T21473 Naftalofos

Naftalofosum,Rawetin,Maretin,Rametin,Naphthalophos

Others Others
Naftalofos is an anthelmintic and an insecticide.
T34236 R 7-45

R 7/45,R7-45,R-7-45

Others Others
R 7-45 is an organic arsenical that acts as an anthelmintic agent.
T21476 Niclofolan

Niclofolano,Bilevon M,Menichlopholan,ME-3625,Niclofolanum

Others Others
Niclofolan, a biphenyl anthelmintic compound, is used orally towards the treatment of Fasciola hepatica infection.
T15462 Haloxon

Others Others
Haloxon is an organophosphorus anthelmintic. Haloxon is used against nematodes of the abomasum and small intestine in ruminants.
T13770 Melarsonyl

Melarsonic acid

Others Others
Melarsonyl (Melarsonic acid) can inhibit parasite potently. Melarsonyl (Melarsonic acid) is an anthelmintic agent.
T20825 Diethylcarbamazine

RP3799,Diaethylcarbamazinum,AI3-19612,RP 3799,Bitirazine,RP-3799

Others Others
Diethylcarbamazine, an anthelmintic, is used primarily as the citrate in the treatment of filariasis, particularly infestations with Loa loa or Wucheria bancrofti.
T34876 Ticarbodine

EL-974,EL 974,EL974

Others Others
Ticarbodine(EL-974)is an Anthelmintic agent.
T26679 Atelocantel

AH 353623,AH-353623,AH353623

Others Others
Atelocantel is an anthelmintic agent (veterinary drug).
T20624 Bitriben

Chloxyl,Cloxil,Fluorescent Red Mega 485 NHS-ester,Chloksil,Chloxil

Others Others
Bitriben is an agent with the anthelmintic effect.
T38729 Melarsonyl dipotassium

美拉胂钾,Melarsonic acid dipotassium

Others Others
Melarsonyl dipotassium, also known as melarsonic acid dipotassium, is a potent anthelmintic agent with the ability to effectively inhibit parasites.
T20960 Luxabendazole

HOE 216V

Others Others
Luxabendazole is a benzimidazole carbamate broad-spectrum anthelmintic agent. It has proved to be effective against immature and adult stages of the major gastrointestinal nematodes, cestodes, and trematodes.
T33690 Nitroscanate

Lopatol,CGA-23654GS,CGA 23654

Others Others
Nitroscanate is an anthelmintic found to be effective in certain strains of parasites in canines.
T21226 Albendazole sulfone

Others Others
Albendazole sulfone, a metabolite of Albendazole, is an antibiotic, anthelmintic, and antiparisitic.

化合物

Phenothiazine
Cat.No: T0776
Synonym: ENT 38,吩噻嗪
Target: Dopamine Receptor, Antibacterial, Antibiotic, Antifungal
Nitazoxanide
Cat.No: T1546
Synonym: NSC 697855,硝唑尼特
Target: Others, Influenza Virus, Parasite, Autophagy
Dithiazanine iodide
Cat.No: T19807
Synonym: Delvex,Telmide,Vercidon,Abminthic,Netocyd,NSC 221154
Target: Others
Closantel
Cat.No: T0237
Synonym: 氯氰碘柳胺,R-31520,氯生太尔
Target: Antibacterial, Parasite
Closantel Sodium
Cat.No: T6452
Synonym:
Target: Antibacterial, Parasite
Emodepside
Cat.No: T7901
Synonym: Bay 44-4400
Target: Parasite
CMP-5 2HCl
Cat.No: T10850L
Synonym:
Target: Others
8-Hydroxyquinoline hemisulfate
Cat.No: T7887
Synonym: 8-羟基喹啉硫酸盐,Oxyquinoline sulfate
Target: Others, Antibacterial, Antibiotic
Monepantel
Cat.No: T16126
Synonym: AAD1566,PPL-1
Target: AChR
Crystal Violet
Cat.No: T1343L
Synonym: Methyl Violet 10B,Hexamethylpararosaniline chloride,氯化结晶紫,Basic Violet 3,结晶紫,Gentian Violet
Target: DNA, Influenza Virus, Antibacterial
Avermectin B1a
Cat.No: T7605
Synonym: 阿维菌素 B1a,Abamectin B1a,Avamectin B1a
Target: Antibiotic, Parasite
Dymanthine
Cat.No: T20082
Synonym: 十八烷基二甲基叔胺,Adogen 342D,ADMA 18
Target: Others
Piperazine adipate
Cat.No: T7146
Synonym:
Target: Parasite
CGP 20376
Cat.No: T30819
Synonym: CGP-20376,CGP20376
Target: Others
Oxfendazole
Cat.No: T0714
Synonym: 奥吩达唑,奥芬哒唑,RS-8858
Target: Glucokinase, Microtubule Associated, Parasite
Febantel
Cat.No: T15272
Synonym:
Target: Parasite
Piperazine citrate
Cat.No: T16539
Synonym:
Target: GABA Receptor
Pyrantel tartrate
Cat.No: T0395
Synonym: Banminth,酒石酸噻吩嘧啶
Target: Antibiotic, Parasite
Eprinomectin
Cat.No: T5836
Synonym: 依普菌素,MK-397
Target: Parasite
Albendazole sulfoxide
Cat.No: T6372
Synonym: Ricobendazole,Albendazole Oxide,阿苯达唑亚砜
Target: Microtubule Associated, Parasite
Brotianide
Cat.No: T30596
Synonym: BAY-VA 4059,Dirian,BAY-VA-4059,BAY-VA4059
Target: Parasite
4-(2-Aminoethyl)amino-7-chloroquinoline
Cat.No: T77684
Synonym: N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine
Target: Parasite
Oxyclozanide
Cat.No: T0955
Synonym: Oxiclozanidum,Zanil,Oxyclozanid,Zanilox,氯羟柳胺
Target: Antibiotic, Parasite
(-)-Benzotetramisole
Cat.No: T77507
Synonym:
Target: Others
2-(Chloromethyl)Imidazo[1,2-A]Pyridine
Cat.No: T77643
Synonym:
Target: Others
Rafoxanide
Cat.No: T7093
Synonym: 碘醚柳胺,雷复尼特
Target: CDK, Parasite
Tribendimidine
Cat.No: T62769
Synonym:
Target: AChR
Diethylcarbamazine citrate
Cat.No: T1420
Synonym: Caritrol,枸橼酸乙胺嗪,Loxuran,Dicarocide
Target: Lipoxygenase, COX, Parasite
Flubendazole
Cat.No: T0009
Synonym: 氟苯咪唑,Flumoxanal,Flumoxane,NSC 313680,Fluvermal
Target: Apoptosis, Microtubule Associated, Parasite
Nitroxynil
Cat.No: T37072
Synonym: 4-Hydroxy-3-iodo-5-nitrobenzonitrile,Trodax,Dovenix
Target: Parasite
Dichlorophen
Cat.No: T0066
Synonym: 双氯酚,DDM,Dichlorophene
Target: Antibacterial, Parasite, Antifungal
Selamectin
Cat.No: T4059
Synonym: UK-124114,司拉克丁,塞拉菌素
Target: Chloride channel, P-gp, Parasite
UK-124114
Cat.No: T0124
Synonym: UNII-A2669OWX9N,西拉菌素,Selamectin
Target: Others
Butonate
Cat.No: T25188
Synonym: NSC17872,NSC 17872,NSC-17872
Target: Others
Oxantel
Cat.No: T0323L
Synonym:
Target: Others
Sch 18099
Cat.No: T34567
Synonym: Sch-18099,Sch18099
Target: Others
Clioxanide
Cat.No: T30968
Synonym: Tremerad,SYD-230,SYD 230,Clioxanida,Clioxanidum
Target: Others
Naftalofos
Cat.No: T21473
Synonym: Naftalofosum,Rawetin,Maretin,Rametin,Naphthalophos
Target: Others
R 7-45
Cat.No: T34236
Synonym: R 7/45,R7-45,R-7-45
Target: Others
Niclofolan
Cat.No: T21476
Synonym: Niclofolano,Bilevon M,Menichlopholan,ME-3625,Niclofolanum
Target: Others
Haloxon
Cat.No: T15462
Synonym:
Target: Others
Melarsonyl
Cat.No: T13770
Synonym: Melarsonic acid
Target: Others
Diethylcarbamazine
Cat.No: T20825
Synonym: RP3799,Diaethylcarbamazinum,AI3-19612,RP 3799,Bitirazine,RP-3799
Target: Others
Ticarbodine
Cat.No: T34876
Synonym: EL-974,EL 974,EL974
Target: Others
Atelocantel
Cat.No: T26679
Synonym: AH 353623,AH-353623,AH353623
Target: Others
Bitriben
Cat.No: T20624
Synonym: Chloxyl,Cloxil,Fluorescent Red Mega 485 NHS-ester,Chloksil,Chloxil
Target: Others
Melarsonyl dipotassium
Cat.No: T38729
Synonym: 美拉胂钾,Melarsonic acid dipotassium
Target: Others
Luxabendazole
Cat.No: T20960
Synonym: HOE 216V
Target: Others
Nitroscanate
Cat.No: T33690
Synonym: Lopatol,CGA-23654GS,CGA 23654
Target: Others
Albendazole sulfone
Cat.No: T21226
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T0314 Hexylresorcinol

己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol

Apoptosis; Tyrosinase; Antibacterial; Parasite Apoptosis; Microbiology/Virology; Proteases/Proteasome
Hexylresorcinol (4-Hexylresorcinol) 是在植物中发现的一种天然产物,具有抗菌、驱虫、防腐和抗肿瘤活性。它是一种可逆、非竞争性的 α-葡萄糖苷酶抑制剂,有抗 DNA 氧化损伤的保护作用。它可诱导鳞癌细胞凋亡。
T8193 α-Thujone

Thujone,ALPHA-(-)-THUJONE,α-侧柏酮,(-)-α-侧柏酮

Apoptosis; Reactive Oxygen Species; GABA Receptor; AChR; Parasite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
α-Thujone 是一种从西方金钟柏精油中分离出来的单萜,可穿透血脑屏障。它是 GABAA 受体的可逆调节剂,在抑制 GABA 诱导的电流时,它的 IC50为 21 μM。它诱导 ROS 依赖性细胞毒性,还诱导细胞凋亡和自噬。它具有抗伤害,抗肿瘤、杀虫和驱虫活性。
T0956 Avermectin B1

Avermectin B1a-Avermectin B1b mixt.,Abamectin,阿维菌素

Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Avermectin B1 是驱虫杀虫剂。
T25114 Ascaridole

NSC-406266,NSC 406266,NSC406266

Parasite Microbiology/Virology
Ascaridole (NSC-406266) 可作为驱虫化合物,能驱除人体和植物中的寄生蠕虫(蠕虫),具有较弱的抗疟活性。
TN6718 Dehydrocostuslactone

Others Others
Dehydrocostuslactone 是一种从奥克兰提取的天然产物。它具有广泛的生物作用,包括抗炎、抗癌、抗病毒、抗菌、抗真菌、抗氧化、抗糖尿病、抗溃疡和驱虫活性。
T3S0006 (E)-Ferulic acid methyl ester

Methyl ferulate,Methyl (E)-ferulate,(E)-阿魏酸甲酯

IL Receptor; p38 MAPK; TNF; COX; NO Synthase; JNK; Antifection Apoptosis; Immunology/Inflammation; MAPK; Microbiology/Virology; Neuroscience
(E)-Ferulic acid methyl ester (Methyl (E)-ferulate) 具有较强 DPPH 和 ABTS+自由基清除特性。
TN2324 Yuankanin

Antioxidant oxidation-reduction
Yuankanin 是一种是在百里香叶、Daphne gnidium 和Daphne feddei 中发现的天然化合物,是一种 genkwanin-5-bioside,具有抗虫和抗氧化活性并对o- 1葡萄糖苷酶、脂肪酶、胰蛋白酶和黄嘌呤氧化酶具有抑制作用。
T1157 Moxidectin

milbemycin B,CL301423,莫昔克丁,莫西菌素

GluCls; Antibiotic; Parasite Microbiology/Virology
Moxidectin (CL301423) 是可用于预防和控制心丝虫和蛔虫的一种驱虫剂。
T38675 Hikizimycin

Anthelmycin

Others Others
Hikizimycin is a potent anthelmintic and antibacterial natural product.
T16497 PF 1022A

Others Others
PF 1022A is an N-methylated cyclooctadepsipeptides with strong anthelmintic properties. It also acts as an ionosphere.
T38235 16-Keto Aspergillimide

Others Others
16-Keto Aspergillimide (SB202327) is a novel anthelmintic compound derived from the Aspergillus strain IMI 337664.
T35908 Paraherquamide E

Others Others
Paraherquamide E is a fungal metabolite originally isolated from P. charlesii with anthelmintic and insecticidal activities. It is lethal to C. elegans (LD50 = 6 μg/ml). Paraherquamide E is also lethal to O. fasciatus (LD50 = 0.089 μg/nymph). Oral administration of paraherquamide E (0.5-4 mg/kg) reduces T. colubriformis fecal egg count in gerbils.
T82706 Clonostachydiol

Clonostachydiol为源于真菌Clonostachys cylindrospora(菌株FH-A 6607)的大分子内酯类驱虫药。
TN4639 Neolitsine

Others Others
Neolitsine has anthelmintic activity, it exhibits EC90 values (concentration at which 90% loss of larval motility is observed) of 6.4 microg/mL.Neolitsine and dicentrine have potent vasorelaxing effects on precontracted rat aortic preparations with mean IC 50 values between 0.08 and 2.48 microM.
T75494 Shinjulactone M

Others Others
Shinjulactone M 是一种从 Ailanthus 中分离出来的一种苦木苦味素类化合物。Ailanthus 可用作退热药 (抗疟) 和驱虫药,用于慢性支气管炎、癫痫和哮喘的研究。
T37609 (rel)-Asperparaline A

Others Others
Aspergillimide is a fungal metabolite originally isolated from A. japonicus.1 It reduces nicotinic acetylcholine receptor (nAChR) peak and slowly-desensitizing amplitudes induced by acetylcholine in silkworm (B. mori) larval neurons (IC50s = 20.2 and 39.6 nM, respectively) but has no effect on chicken α3β4-, α4β2-, and α7-containing nAChRs.2 Dietary administration of aspergillimide A (10 μg/g of diet) induces paralysis in silkworm fourth instar larvae.1 Aspergillimide A (10 and 20 mg/kg) reduces...

天然产物

Hexylresorcinol
Cat.No: T0314
Synonym: 己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol
Target: Apoptosis, Tyrosinase, Antibacterial, Parasite
α-Thujone
Cat.No: T8193
Synonym: Thujone,ALPHA-(-)-THUJONE,α-侧柏酮,(-)-α-侧柏酮
Target: Apoptosis, Reactive Oxygen Species, GABA Receptor, AChR, Parasite, Autophagy
Avermectin B1
Cat.No: T0956
Synonym: Avermectin B1a-Avermectin B1b mixt.,Abamectin,阿维菌素
Target: Antibiotic, Parasite, Autophagy
Ascaridole
Cat.No: T25114
Synonym: NSC-406266,NSC 406266,NSC406266
Target: Parasite
Dehydrocostuslactone
Cat.No: TN6718
Synonym:
Target: Others
(E)-Ferulic acid methyl ester
Cat.No: T3S0006
Synonym: Methyl ferulate,Methyl (E)-ferulate,(E)-阿魏酸甲酯
Target: IL Receptor, p38 MAPK, TNF, COX, NO Synthase, JNK, Antifection
Yuankanin
Cat.No: TN2324
Synonym:
Target: Antioxidant
Moxidectin
Cat.No: T1157
Synonym: milbemycin B,CL301423,莫昔克丁,莫西菌素
Target: GluCls, Antibiotic, Parasite
Hikizimycin
Cat.No: T38675
Synonym: Anthelmycin
Target: Others
PF 1022A
Cat.No: T16497
Synonym:
Target: Others
16-Keto Aspergillimide
Cat.No: T38235
Synonym:
Target: Others
Paraherquamide E
Cat.No: T35908
Synonym:
Target: Others
Clonostachydiol
Cat.No: T82706
Synonym:
Target:
Neolitsine
Cat.No: TN4639
Synonym:
Target: Others
Shinjulactone M
Cat.No: T75494
Synonym:
Target: Others
(rel)-Asperparaline A
Cat.No: T37609
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPH-03035 M-myrmeciitoxin-Mp2b Protein, Myrmecia pilosula, Recombinant (GST & His)

DELTA-myrtoxin-Mp1a B chain,Pilosin-3 subunit b,M-myrmeciito...

Myrmecia pilosula Baculovirus Insect Cells
Heterodimer protein that may serve both defensive (pain-inducing) and predatory (insecticidal) roles. Has membrane-disrupting activity and shows induction of non-specific calcium influx into cells,. Shows broad-spectrum activity against a diverse range of bacteria, and cell lines, as well as hemolytic activity (EC(50)=2.18 uM). In vivo, shows moderate insecticidal activity against D.melanogaster and potent anthelmintic activity against the veterinary nematode H.contortus. In addition, intraplant...

重组蛋白

M-myrmeciitoxin-Mp2b Protein, Myrmecia pilosula, Recombinant (GST & His)
Cat.No: TMPH-03035
Species: Myrmecia pilosula
Expression System: Baculovirus Insect Cells
Cat. No. Product Name Target Signaling Pathways
T19527 Praziquantel D11

吡喹酮 D11

Others Others
Praziquantel D11 is the deuterium labeled Praziquantel, and is an agent of anthelmintic.
T19184 Albendazole sulfoxide D3

Albendazole oxide D3,Ricobendazole D3

Others Others
Albendazole sulfoxide D3 is deuterium-labeled Albendazole sulfoxide. Albendazole sulfoxide is a broad-spectrum anthelmintic.
TMIJ-0489 Coumaphos-d10

Coumaphos-d10 是 Coumaphos 的氘代化合物。Coumaphos 的 CAS 号为 56-72-4。
TMIJ-0295 Flubendazole-d3 (methyl-d3)

Flubendazole-d3 (methyl-d3) 是 Flubendazole 的氘代化合物。Flubendazole 的 CAS 号为 31430-15-6。Flubendazole 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。
T71055 Albendazole-d7

Albendazole-d7 is intended for use as an internal standard for the quantification of albendazole by GC- or LC-MS. Albendazole is an orally bioavailable benzimidazole anthelmintic that is active against a variety of helminths, including liver flukes, tapeworms, and roundworms. It eliminates Trichostrongylus in the fourth stomach of cattle and sheep when orally administered at doses ranging from 2.5 to 10 mg/kg as well as other species in the fourth stomach and the small and large intestine. Alben...

同位素标记化合物

Praziquantel D11
Cat.No: T19527
Synonym: 吡喹酮 D11
Target: Others
Albendazole sulfoxide D3
Cat.No: T19184
Synonym: Albendazole oxide D3,Ricobendazole D3
Target: Others
Coumaphos-d10
Cat.No: TMIJ-0489
Synonym:
Target:
Flubendazole-d3 (methyl-d3)
Cat.No: TMIJ-0295
Synonym:
Target:
Albendazole-d7
Cat.No: T71055
Synonym:
Target:
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