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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7586 |
trifarotene
CD5789,曲法罗汀 |
Retinoid Receptor; Autophagy | Autophagy; Metabolism |
Trifarotene (CD5789) 是一种有效的选择性 RARγ 激动剂,对 RARγ 的选择性是 RARα 和 RARβ 的 65 倍和 16 倍,EC50分别为7.7、500和125 nM。 | |||
T1093 |
Adapalene
CD271,阿达帕林 |
Apoptosis; Retinoid Receptor; Autophagy | Apoptosis; Autophagy; Metabolism |
Adapalene (CD271) 是一种合成类视黄醇,局部应用于痤疮。它以非竞争性方式抑制 GOT1的酶活性,具有抗肿瘤活性。它是一种 RAR 激动剂,对 RARβ、RARγ、RARα的AC50值分别为 2.3 nM、9.3 nM 和 22 nM。 | |||
T1142 |
Clindamycin phosphate
Clindamycin 2-phosphate,Clindamycin 2-dihydrogen phosphate,NSC 618653,U-28508,克林霉素磷酸酯 |
ribosome; Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Clindamycin phosphate (Clindamycin 2-dihydrogen phosphate) 是一种抗生素,抑制微生物的核糖体作用。可研究厌氧菌感染和原虫疾病。 | |||
T5002 |
Methyl Aminolevulinate Hydrochloride
5-Aminolevulinic acid methyl ester,Methyl δ-aminolevulinate hydrochloride,5-氨基酮戊酸甲酯盐酸盐,Methyl 5-aminolevulinate Hydrochloride,Aminolevulinic acid methyl ester Hydrochloride |
Others | Others |
Methyl Aminolevulinate Hydrochloride (5-Aminolevulinic acid methyl ester) 是增敏剂,可用于光动力疗法。Methyl aminolevulinate 是一种前药,可代谢为原卟啉 IX。 | |||
T29022 |
TU-2100
Azeloyl diethyl salicylate,Azasal-2100,TU 2100,TU2100 |
Others | Others |
TU-2100 是一种含水杨酸乙酯的化合物,具有潜在抗痤疮作用,可用于研究痤疮。 | |||
T30150 |
AS-601811
AS601811,AS 601811,UNII-LIV8A6AE5F |
Androgen Receptor | Endocrinology/Hormones |
AS-601811 是类固醇 5α还原酶抑制剂和雄激素受体调节剂,可用于研究脱发和痤疮。 | |||
T1466 |
Nadifloxacin
OPC7251,那氟沙星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Nadifloxacin (OPC7251) 是一种对粉刺有效的广谱氟喹诺酮类抗生素。 | |||
T3510 |
Olumacostat Glasaretil
|
Acetyl-CoA Carboxylase | Metabolism |
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。 | |||
TP2316 |
Myristoyl Hexapeptide-23 Acetate
|
Others | Others |
Myristoyl Hexapeptide-23 Acetate 有抗粉刺作用。 | |||
T35903 |
N-acetyl Dapsone
|
Antibacterial; Parasite | Microbiology/Virology |
N-acetyl Dapsone 是一种抗炎和抗菌化合物,广泛用于治疗麻风病、疟疾、痤疮和各种免疫疾病。 | |||
T24755 |
Salnacedin
G-201,SCY,G-201,G201,SCY,G 201 |
Others | Others |
Salnacedin (G-201) 是一种小分子化合物,可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病,可用于研究寻常痤疮、皮炎和银屑病。 | |||
T21434 |
Sulfacetamide
NSC 63871,磺胺醋酰,NSC-63871,Sebizon,Region,NSC63871,Sulphacetamide,Acetosulfamine |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Sulfacetamide (NSC-63871) 是一种抗生素,通过限制细菌生存所需的叶酸的存在来治疗睑缘炎或结膜炎,有潜力用于眼部感染的研究。 | |||
T25048 |
Algestone acetophenide
Neolutin,苯甲孕酮 |
Others | Others |
Algestone acetophenide (Neolutin) 是用于发情同步的孕酮,已被评估为与庚酸雌二醇联合使用的注射避孕药。它在治疗上也用作局部抗炎药,并在治疗痤疮时局部应用。 | |||
T38683 |
SCD1 inhibitor-3
SCD1-IN-3,SCD1 inhibitor-3,SCD1 inhibitor 17a |
Dehydrogenase | Metabolism |
SCD1 inhibitor-3 (ML-270) 是一种高效、口服的化合物,可以抑制SCD1,且安全性极高。 SCD1 inhibitor-3 显示出在代谢疾病(包括肥胖、二型糖尿病和血脂异常,以及痤疮和癌症等各种皮肤病)方面的巨大研究潜力。 | |||
T1101 |
Minocycline hydrochloride
Minocycline HCl,盐酸米诺环素,美满霉素 |
HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic | Chromatin/Epigenetic; Metabolism; Microbiology/Virology |
Minocycline hydrochloride (Minocycline HCl) 属于四环素类抗生素,具有出色的吸收和组织渗透性。Minocycline hydrochloride 是一种广谱的抗菌剂,可用于多种细菌感染以及痤疮的治疗。 | |||
T77600 |
Methyl-4-oxoretinoate
|
Apoptosis | Apoptosis |
Methyl-4-oxoretinoate 是一种合成的类视黄醇化合物,具有抗癌化合物,可可以诱导癌细胞分化和凋亡。Methyl-4-oxoretinoate 可用于治疗痤疮、牛皮癣和其他皮肤病。Methyl-4-oxoretinoate 具有治疗各种眼部疾病(如年龄相关性黄斑变性)的潜力。 | |||
T7370 |
Talarozole
R115866,他拉罗唑 |
Others; P450; Retinoid Receptor; Autophagy | Autophagy; Metabolism; Others |
Talarozole (R115866) 是一种口服性全反式维甲酸代谢阻断剂,可抑制 CYP26A1 和 CYP26B1,IC50 分别为 5.4 和 0.46 nM。它用于治疗痤疮、牛皮癣和其他角化疾病。 | |||
T25831 |
Motretinide
Ro-11-1430,Ro 11-1430,Tasmaderm,Ro11-1430 |
Others | Others |
Motretinide, an aromatic analog of retinoic acid, is an anti-acne preparation. | |||
T21016 |
Cyproterone
BAY 94-8367,Ciproterone,Androcur,SH 80881 |
Others | Others |
Cyproterone, an anti-androgen, is used in combination with estrogen for the therapy of hirsutism and severe acne in females and as a palliative in prostatic carcinoma. | |||
T29167 |
XMP-629
XOMA629,XOMA 629,XOMA-629,XMP 629 |
||
XMP-629, an endotoxin inhibitor, is used potentially for the treatment of impetigo and acne rosacea. | |||
T21394 |
Sarecycline hydrochloride
P005672,P-005672,WC-3035,WC 3035,Sarecycline HCl,WC3035,P 005672 |
Others | Others |
Sarecycline, a novel and tetracycline-derived antibiotic, is being developed for use as an oral once daily antibiotic treatment for patients suffering from moderate to severe acne vulgaris. Sarecycline has anti-inflammatory activity and the potential for | |||
T39436 |
Omiganan
|
||
Omiganan is a cationic antimicrobial peptide with activity against both gram-positive and gram-negative bacteria, as well as Candida spp. isolates. This compound, serving as an analogue of indolicidin, is utilized for research purposes related to alcohol nose and acne. | |||
T85208 |
4-epi Minocycline
4-EMC,Minocycline Impurity A |
Others | Others |
4-epiMinocycline, recognized as a primary degradation product and a probable impurity in minocycline commercial formulations, is derived from minocycline, a broad-spectrum tetracycline antibiotic notable for its extended serum half-life. Besides treating acne, especially in older patients, minocylvania exhibits significant anti-inflammatory and neuroprotective effects. | |||
T38442 |
17,17-(Ethylenedioxy)androst-4-en-3-one
|
Others | Others |
17,17-(Ethylenedioxy)androst-4-en-3-one (4- androstene- 3, 17- dione- 17- cyclic ethylene ketal) is an effective ingredient in cosmetics, which can be used for acne and promote hair growth research. 17,17-(Ethylenedioxy)androst-4-en-3-one can inhibit the reductase activity and inhibit the bond of a receptor protein and 5α-DHT. | |||
T0339 |
Resorcinol monoacetate
乙醯間二酚(1,3-苯二醇单乙酸酯 ),Resorcin monoacetate |
Others | Others |
Resorcinol monoacetate (Resorcin monoacetate) 是一种防腐剂,及消毒剂,是用于合成其他药品的化学中间体。有用于痤疮,脂溢性皮炎,湿疹,银屑病和其它皮肤病的研究潜力。 | |||
T84629 |
8,11-Eicosadiynoic acid
EDYA |
Others | Others |
8,11-Eicosadiynoic acid 是不饱和脂肪酸,兼具 steroid 5α-reductase 抑制剂功能,适用于痤疮研究。 | |||
T39436L |
Omiganan aceate( 204248-78-2 Free base )
|
||
Omiganan aceate (204248-78-2 free base) 是一种阳离子抗菌肽,对革兰氏阳性菌、革兰氏阴性菌以及念珠菌均具有活性。 Omiganan aceate (204248-78-2 Free base) 是吲哚西丁的类似物,用于与酒精鼻和痤疮相关的研究目的。 | |||
T75306 |
Clindamycin phosphate hydrochloride
|
Others | Others |
Clindamycin phosphate (Clindamycin 2-phosphate) hydrochloride 是一种广谱抑菌林可酰胺类抗生素 (antibiotic)。Clindamycin phosphate hydrochloride 是Clindamycin 的前体活性分子,在体外不具有抗菌活性 ,但在体内可通过磷酸酶酯水解迅速转化为具有活性的母体活性分子 Clindamycin。Clindamycin phosphate hydrochloride 可用于痤疮和细菌性阴道病的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1611 |
Isotretinoin
13-cis-Retinoic acid,异维A酸 |
Retinoid Receptor; Endogenous Metabolite; Autophagy | Autophagy; Metabolism |
Isotretinoin (13-cis-Retinoic acid) 是一种天然存在的维甲酸,具有潜在的抗肿瘤活性。 它结合并激活核视黄酸受体 (RAR), 活化的 RARs 作为促进细胞分化和凋亡的转录因子。它是一种类维生素A 和维生素A 衍生物,用于治疗严重的痤疮和某些形式的皮肤、头颈癌。 | |||
TN6960 |
1-Pentadecanol
pentadecan-1-ol,1-十五醇,n-Pentadecanol |
Others | Others |
1-Pentadecanol 是一种天然产物,具有抗粉刺活性。 | |||
T0978 |
Pantethine
LBF disulfide,Pantosin,Pantetina,Bis-pantethine,泛硫乙胺(维生素B5),泛硫乙胺,Pantomin,D-Pantethine |
Endogenous Metabolite | Metabolism |
D-Pantethine (Pantomin) 是泛酸的二聚体形式, 是生产辅酶 A 的中间体。D-Pantethine 能够作为膳食补充剂,用于改善血液胆固醇和研究痤疮。 | |||
TN1772 |
Isoastilbin
|
Anti-infection; Tyrosinase; Antibacterial | Microbiology/Virology; Proteases/Proteasome |
Isoastilbin 是Rhizoma Smilacis glabrae 和Astragalus membranaceus 中的二氢黄酮醇糖苷。它抑制酪氨酸酶活性,还抑制葡萄糖基转移酶,IC50值为 54.3 μg/mL。它具有神经保护、抗氧化、抗微生物和抗凋亡活性,可研究阿尔茨海默氏病。 | |||
T31766 |
Fenchone
AI300736,AI3-00736,AI3 00736 |
||
Fenchone is a Dapsone-Loaded Invasome for acne treatment. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-06476 |
CAMP Factor Protein, Cutibacterium acnes, Recombinant (His)
|
Cutibacterium acnes | Baculovirus Insect Cells |
CAMP factor is an extracellular cytolytic protein produced by Streptococcus agalactiae. CAMP factor binds the Fc fragments of IgG and is also known as protein B, in analogy to protein A of Staphylococcus aureus. |