8
2
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7839 |
Lasofoxifene Tartrate
CP-336156,酒石酸拉索昔芬 |
Estrogen Receptor/ERR | Endocrinology/Hormones |
Lasofoxifene Tartrate (CP-336156) 是一种非甾体类的雌激素受体选择性调节剂 (SERM)。 | |||
T1536 |
Promestriene
3-propyl ethyl,舒经劳,17B-methyl estradiol,Promestriano |
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Promestriene (3-propyl ethyl) 是局部有效的雌激素,是合成的雌二醇二乙醚。它对阴道萎缩有作用,但吸收量小。 | |||
T40598 |
Norethindrone acetate
19-Norethindroneacetate |
Estrogen Receptor/ERR; Progesterone Receptor | Endocrinology/Hormones; Others |
Norethindrone acetate (19-Norethindroneacetate) 是一种雌性激素,对青少年月经和肝腺瘤有抑制作用,常与孕激素联合使用,可用于研究子宫内膜异位症。 | |||
T7313 |
Enclomiphene citrate
恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate |
Estrogen Receptor/ERR | Endocrinology/Hormones |
Enclomiphene citrate (trans-Clomiphene citrate) 是口服具有活力的 oestrogen receptor 拮抗剂,具有抗雌激素活性。 | |||
T19170 |
Carbazole derivative 1
2-Fluoro-7-[(3-pyridinyl)methyl]-9H-carbazole |
Others | Others |
Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals. | |||
T30259 |
AZD-4992
|
Others | Others |
AZD-4992 是一种选择性雌激素受体下调剂。 | |||
T20419 |
Raloxifene
Pharoxifene,雷洛昔芬,Raloxifenum,Keoxifene,LY-139481 |
Estrogen Receptor/ERR; Others | Endocrinology/Hormones; Others |
Raloxifene (LY-139481) 是一种苯并噻吩类化合物,是一种选择性雌激素受体 (estrogen receptor) 调节剂 (SERM),对骨、血脂有雌激素激动作用,对乳腺和子宫有雌激素拮抗作用。它用于乳腺癌和骨质疏松症研究。 | |||
T62108 |
ErSO-DFP
|
Others | Others |
ErSO-DFP 是一种预期的未折叠蛋白反应 (a-UPR) 激活剂。ErSO-DFP 能够提高对雌激素受体α+ (ERα+) 癌细胞的选择性,选择性高于 ErSO。ErSO-DFP 具有抗肿瘤作用,能够明显消除小鼠模型中 MCF-7 肿瘤。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPJ-00050 |
AG-3 Protein, Human, Recombinant (His)
BCMP11,hAG-3,AG-3,AG3,Anterior Gradient Protein 3 Homolog,Br... |
Human | HEK293 Cells |
Anterior Gradient Protein 2(AG-2) and Anterior Gradient Protein 3 (AG-3) are human homologues of genes involved in differentiation, are associated with oestrogen receptor-positive breast tumours and interact with metastasis gene C4.4a and dystroglycan (hAG-3 protein). AG-3 could serve as a prognostic marker for survival in patients with low grade and high grade serous ovarian carcinomas. | |||
TMPY-01383 |
PRMT6 Protein, Human, Recombinant (His & Flag)
protein arginine methyltransferase 6,HRMT1L6 |
Human | HEK293 Cells |
Protein arginine N-methyltransferase 6, also known as Histone-arginine N-methyltransferase PRMT6, PRMT6, and HRMT1L6, is a member of the protein arginine N-methyltransferase family and PRMT6 subfamily. PRMT6 is highly expressed in kidney and testes. PRMT6 is known to catalyze the generation of asymmetric dimethylarginine in polypeptides. It has been implicated in human immunodeficiency virus pathogenesis, DNA repair, and transcriptional regulation. PRMT6 is known to methylate histone H3 Arg-2 (H... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11197 |
Enclomiphene D4 hydrochloride
(E)-Clomiphene D4 hydrochloride,Enclomifene D4 hydrochloride,trans-Clomiphene D4 hydrochloride |
Others | Others |
Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property.Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a deuterium labeled Enclomiphene. | |||
TMIJ-0039 |
Norethindrone Acetate-2,2,4,6,6,10-d6
|
||
Norethindrone Acetate-2,2,4,6,6,10-d6 是 Norethindrone Acetate 的氘代化合物。Norethindrone Acetate 的 CAS 号为 51-98-9。Norethindrone acetate 是一种雌性激素,对青少年月经和肝腺瘤有抑制作用,常与孕激素联合使用,可用于研究子宫内膜异位症。 |