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n6trifluoroacetylllysine

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  • 抑制剂&激动剂
    39
    TargetMol | Inhibitors_Agonists
  • 多肽产品
    3
    TargetMol | Peptide_Products
  • 染料试剂
    4
    TargetMol | Dye_Reagents
  • 天然产物
    4
    TargetMol | Natural_Products
N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- ThioureaN-[3,5-双(三氟甲基)苯基]-N′-[(9R)-6′-甲氧基-9-金鸡宁]硫脲
T7750852913-25-8
N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea 是金鸡纳生物碱衍生的双功能催化剂。
  • ¥ 142
现货
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数量
TargetMol | Inhibitor Sale
(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
T776702919211-45-1
(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid 是一种潜在的SSTR4激动剂。
  • ¥ 1300
现货
规格
数量
N-((4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methyl)-2-bromoaniline
T98371352608-94-6In house
N-((4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methyl)-2-bromoaniline 是一种有效的 ALK5 抑制剂,IC50 为 7nM。
  • ¥ 1300
现货
规格
数量
TargetMol | Inhibitor Sale
N-Biotinyl-6-aminohexanoic acidN-(+)-Biotinyl-6-aminohexanoic acid,N-生物素己酸
T1944472040-64-3
N-Biotinyl-6-aminohexanoic acid(N-(+)-Biotinyl-6-aminohexanoic acid)可用于生物素化反应。
  • ¥ 113
现货
规格
数量
TargetMol | Inhibitor Sale
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea
T1215697627-24-2
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea 是一种抗惊厥剂,对广泛强直和部分性发作挛性具有潜在的研究价值。
  • ¥ 363
现货
规格
数量
TargetMol | Inhibitor Sale
(S)-N-FMoc-2-(6'-heptenyl)alanine
T665421311933-83-1
(S)-2-((((9H-Fluoren-9-yl)methoxy)carbonyl)amino)-2-methylnon-8-enoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66542,CAS号为 1311933-83-1。
  • ¥ 148
5日内发货
规格
数量
N-(3-Chloro-4-((3-fluorobenzyl)oxy)phenyl)-6-iodoquinazolin-4-amine
T65343231278-20-9
N-(3-Chloro-4-((3-fluorobenzyl)oxy)phenyl)-6-iodoquinazolin-4-amine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65343,CAS号为 231278-20-9。
  • 询价
规格
数量
4-Chloro-N-(6-nitrobenzo[d]thiazol-2-yl)benzamide
TNU0866321943-75-3
Heterocyclic Compounds - Fused polyheterocycles; Drugs and Inhibitors; Anticancer agent
  • 询价
5日内发货
规格
数量
N-[5-[[[3-(6-Amino-4-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide
T775912757619-90-0
N-[5-[[[3-(6-Amino-4-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide在BD2 DEC-Tec实验中的IC50值为22nM。
    询价
    N-(3-Chloro-4-fluorophenyl)-7-fluoro-6-nitroquinazolin-4-amine
    T64879162012-67-1
    N-(3-Chloro-4-fluorophenyl)-7-fluoro-6-nitroquinazolin-4-amine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64879,CAS号为 162012-67-1。
    • 询价
    5日内发货
    规格
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    2-Chloro-2’-C-methyl-6-N,N-dimethyladenosine
    TNU01112095417-43-7
    2’-C-Methyl nucleoside; Halo-nucleoside; 2/6/8-Modified purine nucleoside
    • 询价
    5日内发货
    规格
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    (E)-N-(2-Chloro-6-methylphenyl)-3-ethoxyacrylamide
    T66342863127-76-8
    (E)-N-(2-Chloro-6-methylphenyl)-3-ethoxyacrylamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66342,CAS号为 863127-76-8。
    • 询价
    5日内发货
    规格
    数量
    N-[(6S)-6-Carboxy-6-(glycylamino)hexanoyl]-D-alanyl-D-alanine
    T81719306748-45-8
    N-[(6S)-6-Carboxy-6-(glycylamino)hexanoyl]-D-alanyl-D-alanine,能够干扰PAICS蛋白功能,有效降低SAICAR和SAICAr的积聚。
    • 询价
    规格
    数量
    N-[5-Bromomethyl-4-(4-fluorophenyl)-6-isopropylpyrimidine-2-yl]-N-methylmethane sulfonamide
    T66071799842-07-2
    N-[5-Bromomethyl-4-(4-fluorophenyl)-6-isopropylpyrimidine-2-yl]-N-methylmethane sulfonamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66071,CAS号为 799842-07-2。
    • 询价
    5日内发货
    规格
    数量
    N-[5-[[[3-(6-Amino-2-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide
    T775922757619-89-7
    N-[5-[[[3-(6-Amino-2-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide在BD2 DEC-Tec实验中的IC50值为94nM。
      询价
      (S)-N-(3-Chloro-4-fluorophenyl)-6-nitro-7-((tetrahydrofuran-3-yl)oxy)quinazolin-4-amine
      T66550314771-88-5
      (S)-N-(3-Chloro-4-fluorophenyl)-6-nitro-7-((tetrahydrofuran-3-yl)oxy)quinazolin-4-amine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66550,CAS号为 314771-88-5。
      • 询价
      5日内发货
      规格
      数量
      N6-Trifluoroacetyl-L-Lysine
      T67613116169-90-5
      N6-Trifluoroacetyl-L-Lysine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67613,CAS号为 116169-90-5。
      • ¥ 528
      5日内发货
      规格
      数量
      N1-(tert-Butoxycarbonylmethyl)-6-[2-(N-Cbz-amino)ethoxy)]-phenoxazine
      TNU1456476667-25-1
      N1-(tert-Butoxycarbonylmethyl)-6-[2-(N-Cbz-amino)ethoxy)]-phenoxazine is a PNA-related Derivative; Heterocyclic Compound - Fused polyheterocycle.
      • 询价
      5日内发货
      规格
      数量
      tert-Butyl 2-((4R,6S)-6-((E)-2-(4-(4-fluorophenyl)-6-isopropyl-2-(N-methylmethylsulfonamido)pyrimidin-5-yl)vinyl)-2,2-dimethyl-1,3-dioxan-4-yl)acetate
      T66277289042-12-2
      tert-Butyl 2-((4R,6S)-6-((E)-2-(4-(4-fluorophenyl)-6-isopropyl-2-(N-methylmethylsulfonamido)pyrimidin-5-yl)vinyl)-2,2-dimethyl-1,3-dioxan-4-yl)acetate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66277,CAS号为 289042-12-2。
      • 询价
      5日内发货
      规格
      数量
      4-Fluoro-N-(6-nitrobenzo[d]thiazol-2-yl)benzamide
      TNU0863313275-82-0
      4-Fluoro-N-(6-nitrobenzo[d]thiazol-2-yl)benzamide is a Heterocyclic Compound and can be used in anticancer and antimicrobial studies.
      • 询价
      5日内发货
      规格
      数量
      N-6-Furfurylguanosine
      TNU002526783-39-1
      N-6-Furfurylguanosine is a 2/6/8-modified purine nucleoside.
      • 询价
      5日内发货
      规格
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      N-(4-(4-Fluorophenyl)-5-formyl-6-isopropylpyrimidin-2-yl)-N-methylmethanesulfonamide
      T65584147118-37-4
      N-(4-(4-Fluorophenyl)-5-formyl-6-isopropylpyrimidin-2-yl)-N-methylmethanesulfonamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65584,CAS号为 147118-37-4。
      • 询价
      5日内发货
      规格
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      Canthin-6-one N-oxide
      TN358460755-87-5
      Canthin-6-one N-oxide has broad spectrum antifungal, leishmanicidal and trypanocidal activities.
      • 询价
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      数量
      7-(deoxyadenosin-N(6)-yl)aristolactam I马兜铃内酰胺 A
      TJS1226127191-86-0
      7-(deoxyadenosin-N(6)-yl)aristolactam I是一种来自马兜铃草药的天然化合物。
      • ¥ 2200
      期货
      规格
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      5-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole
      T83285611207-02-4
      5-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole 是酿酒酵母细胞色素 bc1 复合物(细胞色素c氧化还原酶)Qo位点的竞争性抑制剂。
      • 询价
      8-10周
      规格
      数量
      4-(6-Bromo-2-benzothiazolyl)-N-methylbenzenamine
      T19142566169-98-0
      4-(6-Bromo-2-benzothiazolyl)-N-methylbenzenamine is a potent amyloid imaging agent that binds to Amyloid-β (1-40) (KD: 1.7 nM).
      • 询价
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      (S)-N-(2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)propionamide
      T65667106006-84-2
      (S)-N-(2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)propionamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65667,CAS号为 106006-84-2。
      • 询价
      5日内发货
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      数量
      6-[(3R,4R)-3-(Acetyloxy)-N,4-dimethyl-6-oxo-L-norleucine]cyclosporin A
      T64488
      6-[(3R,4R)-3-(Acetyloxy)-N,4-dimethyl-6-oxo-L-norleucine]cyclosporin A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64488。
      • 询价
      5日内发货
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      9-Methoxycanthin-6-one-N-oxide
      TN3322137739-74-3
      9-Methoxycanthin-6-one-N-oxide shows cytotoxic activity against a panel of cell lines comprising a number of human cancer cell types.
      • 询价
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      (6S)-N-Benzyl-6-(4-hydroxybenzyl)-8-(naphthalen-1-ylmethyl)-4,7-dioxohexahydro-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide
      T65994868774-16-7
      Wnt signaling is required for direct multiple biological processes and also plays key roles in the pathogenesis of various diseases. Cyclic AMP response element-binding protein (CREB) is a transcription factor that is a member of the leucine zipper family of DNA binding proteins. This protein binds as a homodimer to the cAMP-responsive element, an octameric palindrome. The protein is phosphorylated by several protein kinases, and induces transcription of genes in response to hormonal stimulation of the cAMP pathway. Via generating a transcriptionally active complex with β-catenin, CREB acts as a mediator of Wnt signaling.ICG-001 is an inhibitor of β-catenin/CREB mediated transcription. The direct cellular target of ICG-001 is CREB. the inhibitory IC50of ICG-001 against β-catenin/CREB mediated transcription was 3 μM. ICG-001 treatment at the concentration of 25 μM for 24h significantly increased caspase activity in both colon cancer cell lines SW480 and HCT116 cell lines but not in normal colonic epithelial cells CCD-841Co. In a cell growth inhibition assay, the IC50s of ICG-001 against SW480 and HCT116 cells were 4.43 μM and 5.95 μM, respectively.In a SW620 nude mouse xenograft model, an water-soluble analog of ICG-001 given at the dose of 150 mg/kg i.v. once in every 2 days dramatically suppressed tumor growth. In a bleomycin-induced pulmonary fibrosis mice model, ICG-001 given at the dose of 5 mg/kg per day reversed pulmonary fibrosis. In a rat myocardial infarction model, ICG-001 was administrated subcutaneously at the dose of 50 mg/kg/day for 10 days which significantly improved cardiac contractile function after myocardial infarction in the rats.
      • ¥ 7685
      5日内发货
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      N-(5-(8-Amino-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-methylphenyl)methanesulfonamide hydrochloride
      T648372803477-07-6
      N-(5-(8-Amino-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-methylphenyl)methanesulfonamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64837。
      • ¥ 3718
      5日内发货
      规格
      数量
      2-Acetylamino-1-{3’-O-[(4,4’-dimethoxy triphenyl)methyl]-a-L-threo furanosyl}-6-(N,N-diphenylcarbamoyloxy)-9H-purine
      TNU1645325683-92-9
      2-Acetylamino-1-{3’-O-[(4,4’-dimethoxy triphenyl)methyl]-a-L-threo furanosyl}-6-(N,N-diphenylcarbamoyloxy)-9H-purine 是一种核苷类似物,在生命科学相关研究中具有广泛的应用。
      • 询价
      5日内发货
      规格
      数量
      N-(2-Bromo-6-fluorophenyl)-4,5-dihydro-1H-imidazol-2-amine hydrochloride
      T64522
      N-(2-Bromo-6-fluorophenyl)-4,5-dihydro-1H-imidazol-2-amine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64522。
      • 询价
      5日内发货
      规格
      数量
      N-(5-((Diphenylphosphoryl)methyl)-4-(4-fluorophenyl)-6-isopropylpyrimidin-2-yl)-N-methylmethanesulfonamide
      T66148289042-10-0
      N-(5-((Diphenylphosphoryl)methyl)-4-(4-fluorophenyl)-6-isopropylpyrimidin-2-yl)-N-methylmethanesulfonamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66148,CAS号为 289042-10-0。
      • 询价
      5日内发货
      规格
      数量
      tert-Butyl N-[6-(methylamino)hexyl]carbamate
      T64467
      tert-Butyl N-[6-(methylamino)hexyl]carbamate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64467。
      • ¥ 374
      5日内发货
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      N1-Carboxymethyl-6-[2-(N,N’-bis-Cbz-guanidino)   ethoxy]-phenoxazine
      TNU1457476667-27-3
      N1-Carboxymethyl-6-[2-(N,N'-bis-Cbz-guanidino) ethoxy]-phenoxazine is a PNA-related Derivative; Heterocyclic Compound - Fused polyheterocycle.
      • 询价
      5日内发货
      规格
      数量
      6-Acetonyl-N-methyl-dihydrodecarine
      TN31511253740-09-8
      6-Acetonyl- N -methyl-dihydrodecarine has mosquito larvicidal activity against the malaria vector Anopheles gambiae.
      • ¥ 3940
      期货
      规格
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      H-Lys(Tfa)-OH
      T135110009-20-8
      H-Lys(Tfa)-OH 是L-lysine cyclodeaminase 的抑制剂。
      • ¥ 108
      现货
      规格
      数量
      TargetMol | Inhibitor Sale