3
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1069 |
Metoclopramide hydrochloride
盐酸甲氧氯普胺,Maxolon,Metoclopramide HCl |
Dopamine Receptor; 5-HT Receptor; AChR | GPCR/G Protein; Neuroscience |
Metoclopramide hydrochloride (Metoclopramide HCl) 是可口服的5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,用于恶心呕吐、胃食管反流和胃轻瘫的研究。 | |||
T4616 |
Metoclopramide
甲氧氯普胺,胃复安,5-Chloro-2-methoxyprocainamide |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Metoclopramide (5-Chloro-2-methoxyprocainamide) 是5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,可用于恶心呕吐、胃食管反流和胃轻瘫的研究。 | |||
T8385 |
Metoclopramide hydrochloride hydrate
盐酸甲氧氯普胺,甲氧氯普胺盐酸水合物,Metoclopramide monohydrochloride monohydrate |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) 是5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,可用于恶心呕吐、胃食管反流和胃轻瘫的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3605 |
Gastrodenol
Bismuth tripotassium dicitrate,枸橼酸铋钾,Bismuth subcitrate |
Others | Others |
Gastrodenol (Bismuth tripotassium dicitrate) 是一种对溃疡和胃不适具有潜在的应用价值的药物。 | |||
TN3495 |
Benzyl ferulate
|
TNF; Antifection | Apoptosis; Microbiology/Virology |
Benzyl ferulate has antimicrobial activity. It also shows good anti-proliferative against three gastro-intestinal cancer cell lines(HCT-116 colon carcinoma, KYSE-30 oesophageal squamous cancer, and NCI-N87 gastric carcinoma). |