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Targets Recommended: Apoptosis Estrogen Receptor/ERR Others

2

抑制剂 & 化合物

2

天然产物

4

化合物库

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Cat. No. Product Name
LF9100 丝氨酸靶向共价抑制剂库

2700 compounds
Over 2,700 small-molecule screening compounds in the library.
L8800 药物片段库

1119 compounds
1119 种药物片段分子,是FBDD 方法新药筛选的有力工具;
L4020 NO PAINS 化合物库

9384 compounds
TargetMol NO PAINS 化合物库包含 9384 个剔除了PAINS 的小分子活性化合物,可用于新药研发,信号通路研究,老药新用等研究。
DF4500 多样性核心库Part1

50000 compounds
绝大部分分子量<500,主要集中于250-450之间,方便后续的改造优化;

化合物库

丝氨酸靶向共价抑制剂库
Cat.No: LF9100
Compounds: 2700
药物片段库
Cat.No: L8800
Compounds: 1119
NO PAINS 化合物库
Cat.No: L4020
Compounds: 9384
多样性核心库Part1
Cat.No: DF4500
Compounds: 50000
Cat. No. Product Name Target Signaling Pathways
T0695 Avobenzone

阿伏苯宗,Butyl methoxydibenzoylmethane,BF2AVB

Apoptosis; Estrogen Receptor/ERR; Others Apoptosis; Endocrinology/Hormones; Others
Avobenzone 是一种二苯甲酰甲烷内分泌干扰物,可直接与雌激素受体 β 结合,起到雌激素激动剂的作用。它是紫外线波段皮肤光防护防晒霜中应用最广泛的滤光剂之一。
T78400 4-Di-16-ASP

DiA

4-Di-16-ASP为膜染料,属亲脂性氨基苯乙烯基探针,发射光谱宽(适用绿色、橙色或红色滤光片检测)。适应于神经元膜追踪,扩散速度优于DiO。

化合物

Avobenzone
Cat.No: T0695
Synonym: 阿伏苯宗,Butyl methoxydibenzoylmethane,BF2AVB
Target: Apoptosis, Estrogen Receptor/ERR, Others
4-Di-16-ASP
Cat.No: T78400
Synonym: DiA
Target:
Cat. No. Product Name Target Signaling Pathways
T19278 Dicaprylyl carbonate

碳酸二辛酯,Dimethyl carbonate

Others Others
Dicaprylyl carbonate (Dimethyl carbonate) 是植物来源的固体脂肪,是干燥润肤剂。它具有强大的皮肤相容性和全面的性能,如防晒滤光片的增溶和分散能力。
TN4178 Gyrophoric acid

cAMP GPCR/G Protein
Vulpinic and gyrophoric acids are known as ultraviolet filters for natural lichen populations, they can effectively prevent cytotoxic, apoptotic and cytoskeleton alterative activities of 2.5 J/cm(2) UVB in a dose-dependent manner, suggest that vulpinic and gyrophoric acids can be promising cosmetic ingredients to photo-protect human skin cells. Gyrophoric acid also has anti-proliferative/cytotoxic effect.

天然产物

Dicaprylyl carbonate
Cat.No: T19278
Synonym: 碳酸二辛酯,Dimethyl carbonate
Target: Others
Gyrophoric acid
Cat.No: TN4178
Synonym:
Target: cAMP
TargetMol Loading
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