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Search Results for " corpus "

Targets Recommended: Adenosine Receptor

9

抑制剂 & 化合物

4

天然产物

3

重组蛋白

3

同位素标记化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T16136	MRS-1706	Adenosine Receptor	GPCR/G Protein; Neuroscience
	MRS-1706 是一种选择性A2B 腺苷受体的反向激动剂，对人 A2B、A2A、A1和 A3受体的Ki 值分别为 1.39、112、157 和 230 nM。
T2334	Avanafil 阿伐那非,TA1790	PDE	Metabolism
	Avanafil (TA1790) 是一种高活性PDE-5抑制剂，IC50=5.2 nM，对PDE1，PDE6和PDE11活性较低。
T4546	Dinoprost tromethamine salt Dinoprost Tromethamine,Zinoprost,Prostin F2 alpha,PGF2α THAM,Dinolytic,地诺前列素氨丁三醇,Prostaglandin F2α THAM	Apoptosis; Endogenous Metabolite; Prostaglandin Receptor; Autophagy; PROTAC Linker	Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism; PROTAC
	Dinoprost tromethamine salt (PGF2α THAM) 是一种口服有效的前列腺素 F 受体激动剂。它是在子宫内膜腔上皮和黄体中局部产生的溶酶激素，在分娩过程中起关键作用。
T1398	Tadalafil Cialis,他达那非,IC-351,西力士	Apoptosis; PDE	Apoptosis; Metabolism
	Tadalafil (IC-351) 是一种PDE5抑制剂，IC50为 1.8 nM。
T0096	Vardenafil 伐地那非,Vivanza,Levitra,Vardenafil hydrochloride	PDE	Metabolism
	Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。
T35288	Z 300 Z-300,Z300	Others	Others
	Z 300 是一种组胺 H2 受体拮抗剂。 Z 300 抑制胃酸分泌并促进胃体区域的胃粘液代谢。
T24388	LASSBio-1359 LASSBio1359,LASSBio 1359	Others	Others
	LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.
T26993	CGP 56999A CGP56999A,CGP-56999A	Others	Others
	CGP 56999A is an antagonist of GABA(B) receptor, it enhances expression of brain-derived neurotrophic factor and attenuates dopamine depletion in the rat corpus striatum.
T37919	Prostaglandin F1α PGF1α,Prostaglandin F1α	Others	Others
	Prostaglandin F1α (PGF1α) is the putative metabolite of dihomo-γ-linolenic acid (DGLA) via the cyclooxygenase (COX) pathway. Both PGF1α and PGF2α have been shown to act as priming pheromones for male Atlantic salmon with a threshold concentration of 10-11 M. [1] PGF1α binds to the ovine corpus luteum FP receptor at only 8% of the relative potency of PGF2α. [2] It is only half as active as PGF2α in inducing human respiratory smooth muscle contractions in vitro. [3]

化合物

Cat.No: T16136

Target: Adenosine Receptor

Cat.No: T2334

Synonym: 阿伐那非,TA1790

Target: PDE

Dinoprost tromethamine salt

Cat.No: T4546

Synonym: Dinoprost Tromethamine,Zinoprost,Prostin F2 alpha,PGF2α THAM,Dinolytic,地诺前列素氨丁三醇,Prostaglandin F2α THAM

Target: Apoptosis, Endogenous Metabolite, Prostaglandin Receptor, Autophagy, PROTAC Linker

Cat.No: T1398

Synonym: Cialis,他达那非,IC-351,西力士

Target: Apoptosis, PDE

Cat.No: T0096

Synonym: 伐地那非,Vivanza,Levitra,Vardenafil hydrochloride

Target: PDE

Cat.No: T35288

Synonym: Z-300,Z300

Target: Others

Cat.No: T24388

Synonym: LASSBio1359,LASSBio 1359

Target: Others

Cat.No: T26993

Synonym: CGP56999A,CGP-56999A

Target: Others

Prostaglandin F1α

Cat.No: T37919

Synonym: PGF1α,Prostaglandin F1α

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T15133	Dinoprost Prostaglandin F2a,PGF2α,地诺前列素	Endogenous Metabolite	Metabolism
	Dinoprost (Prostaglandin F2a) 是口服有效的、内源性的前列腺素 F 受体激动剂。它是在子宫内膜腔上皮和黄体中局部产生的溶酶激素。它在分娩过程中起关键作用。
T0478	Progesterone 孕酮,Pregn-4-ene-3,20-dione	Estrogen/progestogen Receptor; Progesterone Receptor; Opioid Receptor; Endogenous Metabolite	Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience; Others
	Progesterone (Pregn-4-ene-3,20-dione) 是类固醇激素，能够调节月经周期。
T6S2227	Spinosin 斯皮诺素,Flavoayamenin	Others	Others
	Spinosin (Flavoayamenin) 是一种具有神经保护作用的 C-糖苷类黄酮，从 Zizyphus jujube 种子分离得到，能够激活 Nrf2/HO-1 通路，并抑制 Aβ1-42的产生和聚合。
TN4277	Isocupressic acid	cAMP; P450; PKA	GPCR/G Protein; Metabolism; Tyrosine Kinase/Adaptors
	Isocupressic acid induces abortion in pregnant cows when ingested primarily during the last trimester, it decrease affects the angiogenesis of the female reproductive system, the decrease in blood flow and apoptosis of corpus luteum-derived endothelial ce

天然产物

Cat.No: T15133

Synonym: Prostaglandin F2a,PGF2α,地诺前列素

Target: Endogenous Metabolite

Cat.No: T0478

Synonym: 孕酮,Pregn-4-ene-3,20-dione

Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite

Cat.No: T6S2227

Synonym: 斯皮诺素,Flavoayamenin

Target: Others

Isocupressic acid

Cat.No: TN4277

Target: cAMP, P450, PKA

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPJ-00577	INSL3 Protein, Human, Recombinant (His) RLNL,Insulin-like 3,RLF,Leydig insulin-like peptide,INSL3,Re...	Human	HEK293 Cells
	Insulin-like 3 is a protein that in humans is encoded by the INSL3 gene. It is a secreted protein that belongs to the insulin family. It is expressed in prenatal and postnatal Leydig cells and found as well in the corpus luteum, trophoblast, fetal membranes and breast. It may act as a hormone to regulate growth and differentiation of gubernaculum, and thus mediating intra-abdominal testicular descent.It is a ligand for LGR8 receptor.
TMPY-03460	DCXR Protein, Human, Recombinant (His) XR,P34H,HCR2,HCRII,PNTSU,SDR20C1,DCR,dicarbonyl/L-xylulose r...	Human	E. coli
	DCXR, also known as HCR2, belongs to the short-chain dehydrogenases/reductases (SDR) family. It is highly expressed in kidney, liver and epididymis. In the epididymis, DCXR is mainly expressed in the proximal and distal sections of the corpus region. HCR2 is weakly or not expressed in brain, lung, heart, spleen and testis. DCXR catalyzes the NADPH-dependent reduction of several pentoses, tetroses, trioses, alpha-dicarbonyl compounds and L-xylulose. DCXR participates in the uronate cycle of...
TMPY-01927	ANP32A Protein, Human, Recombinant (His & GST) MAPM,PP32,I1PP2A,C15orf1,LANP,HPPCn,PHAPI,acidic (leucine-ri...	Human	E. coli
	acidic leucine-rich nuclear phosphoprotein 32 family member A, also known as acidic nuclear phosphoprotein pp32, Leucine-rich acidic nuclear protein, Mapmodulin, Potent heat-stable protein phosphatase 2A inhibitor I1PP2A, Putative HLA-DR-associated protein I, PHAPI and ANP32A, is a nucleus, cytoplasm and endoplasmic reticulum. ANP32A / LANP is expressed in all tissues tested. It is highly expressed in kidney and skeletal muscle, moderate levels of expression is in brain, placenta and panc...

重组蛋白

INSL3 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00577

Species: Human

Expression System: HEK293 Cells

DCXR Protein, Human, Recombinant (His)

Cat.No: TMPY-03460

Species: Human

Expression System: E. coli

ANP32A Protein, Human, Recombinant (His & GST)

Cat.No: TMPY-01927

Species: Human

Expression System: E. coli

Cat. No.	Product Name	Target	Signaling Pathways
TMID-0037	Tadalafil-d3
	Tadalafil-d3 是 Tadalafil 的氘代化合物。Tadalafil 的 CAS 号为 171596-29-5。Tadalafil 是一种PDE5抑制剂，IC50为 1.8 nM。
TMID-0209	Tadalafil-13C-d3
	Tadalafil-13C-d3 是 Tadalafil 的 13C 和氘代化合物。Tadalafil 的 CAS 号为 171596-29-5。Tadalafil 是一种PDE5抑制剂，IC50为 1.8 nM。
TMIJ-0114	Vardenafil-d5
	Vardenafil-d5 是 Vardenafil 的氘代化合物。Vardenafil 的 CAS 号为 224785-90-4。Vardenafil 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。

同位素标记化合物

Cat.No: TMID-0037

Tadalafil-13C-d3

Cat.No: TMID-0209

Cat.No: TMIJ-0114

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