92
1
9
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10335 |
Antihistamine-1
|
P450 | Metabolism |
Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂,其 IC50 值分别为 5.4 和 0.8 μM。 | |||
T25180 |
Bromodiphenhydramine hydrochloride
|
Others | Others |
Bromodiphenhydramine hydrochloride 是一种控制皮肤的新型抗组胺药。 | |||
T9353 |
OXOMEMAZINE
|
AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Oxomemazine 是毒菌碱 M1 受体的选择性拮抗剂,具有明显的抗毒蕈碱活性。它是基于吩噻嗪的组胺 H1 受体阻滞剂,是抗组胺和抗胆碱能试剂,可用于咳嗽相关研究。 | |||
T0211 |
Azelastine
Azelastina,Astelin,Azelastinum,氮卓斯汀 |
SARS-CoV; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。 | |||
T1030 |
Triprolidine hydrochloride monohydrate
盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Triprolidine hydrochloride monohydrate 是一种组胺 H1 拮抗剂,用于过敏性鼻炎、哮喘。 | |||
T0211L |
Azelastine hydrochloride
Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin |
SARS-CoV; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。 | |||
T0118 |
Mizolastine
SL 850324,咪唑司汀,咪唑斯汀 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mizolastine (SL 850324) 是组胺 H1 受体拮抗剂,IC50为 47 nM。它用于治疗过敏反应,如花粉热和荨麻疹等。 | |||
T1278 |
Astemizole
Laridal,Histaminos,Paralergin,阿司咪唑 |
Potassium Channel; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience |
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。 | |||
T6488 |
Epinastine hydrochloride
Alesion,Epinastine HCl,WAL-801CL HCl,依匹斯汀盐酸盐,Elestat |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Epinastine hydrochloride (WAL-801CL HCl) 是抗组胺剂和肥大细胞稳定剂,是一种可口服的选择性组胺 H1 受体拮抗剂,可抑制 IL-8 释放,具有抗过敏作用。 | |||
T1110 |
Meclizine dihydrochloride
Meclozine dihydrochloride,NSC28728,Meclizine 2HCl,盐酸美克洛嗪 |
Apoptosis; Histamine Receptor | Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Meclizine dihydrochloride (NSC28728) 是一种组胺 H1 拮抗剂,用于治疗妊娠期间的晕动病、眩晕和恶心以及放射病。它是小鼠组成型雄甾烷受体激动剂,是人 CAR 的反向激动剂。它可透过血脑屏障,可用于多聚谷氨酰胺毒性障碍方面的研究。 | |||
T6426 |
Buclizine dihydrochloride
盐酸安其敏,Longifene,Buclina,Buclizine HCl,UCB-4445 |
5-HT Receptor; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Buclizine dihydrochloride (Buclina) 是可口服的一种哌嗪组胺 H1 受体拮抗剂,主要具有止吐和抗眩晕活性。 | |||
T6814 |
Cyproheptadine hydrochloride
Periactin hydrochloride,Anarexol,盐酸赛庚啶,Cyproheptadine HCl,Nuran |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Cyproheptadine hydrochloride (Periactin hydrochloride) 是一种 5-HT2A 受体拮抗剂,具有抗抑郁和抗血清素作用。它具有抗血小板活性,可用于血栓栓塞性疾病的研究。 | |||
T2335 |
Ebastine
Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Ebastine (Kestine) 是一种可口服的组胺 H1 受体拮抗剂,用于过敏性鼻炎的症状和慢性特发性荨麻疹的研究。 | |||
T0147 |
Clemastine fumarate
HS-592 (fumarate),富马酸氯马斯汀,Meclastine fumarate,Meclastine (fumarate) |
Autophagy; Histamine Receptor | Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Clemastine fumarate (Meclastine (fumarate)) 是一种合成乙醇胺,具有抗胆碱能、镇静和组胺 H1 拮抗作用。 | |||
T0205 |
Brompheniramine maleate
Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。 | |||
T3609 |
Dioxopromethazine
Prothanon,Dioxoprothazine,盐酸二氧丙嗪 |
Others | Others |
Dioxopromethazine (Dioxoprothazine) 是一种口服具有活性的抗组胺药,能够抑制哮喘症状。 | |||
T21014 |
Thonzylamine hydrochloride
Resistab,Thonzylamine HCl,Novohetramin,Neohetramine hydrochloride,Anahist |
AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Thonzylamine hydrochloride (Resistab) 是一种抗胆碱能和抗组胺药,用作止痒药。 | |||
T25875 |
Noberastine
R64947,T25875,R-64947,R 64947 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Noberastine (R 64947) 是一种新型组胺 H1拮抗剂,具有强效和特异性的外周抗组胺活性。 | |||
T7477 |
Antazoline
|
Others | Others |
Antazoline 具有抗组胺和抗胆碱能作用。它用于治疗各种心律失常。 | |||
T1470 |
Fexofenadine hydrochloride
Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) 是一种抗组胺药,用于治疗过敏性鼻炎、血管性水肿和慢性荨麻疹。 | |||
T0174 |
Cyproheptadine hydrochloride sesquihydrate
Peritol,盐酸赛庚啶半水合物,Periactin hydrochloride,Cyproheptadine hydrochloride,赛庚啶盐酸盐 |
5-HT Receptor; Histone Methyltransferase; Histamine Receptor | Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cyproheptadine hydrochloride sesquihydrate (Peritol) 是一种抗组胺剂,也是血清素和组胺2拮抗剂。 | |||
T7564 |
Chlorphenoxamine
Contristamine,氯苯沙明 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Chlorphenoxamine (Contristamine) 是一种抗组胺药和抗胆碱能药,用作止痒药和抗帕金森病药。 | |||
T68150 |
Talastine
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Talastine 是一种抗组胺化合物,可诱发过敏性皮疹。 | |||
T31488 |
Dimethindene
Dimetindeno,Z 2001,Dimetindene,二甲茚定,Z-2001,Z2001 |
Potassium Channel; Endogenous Metabolite; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Dimethindene (Dimetindeno) 是 H1受体的选择性拮抗剂,阻断 K+电流。Dimethindene 表现出抗组胺和抗胆碱作用。 | |||
T4526 |
Piperoxan hydrochloride
dl-Piperoxan hydrochloride,盐酸哌罗克生,Benodaine hydrochloride |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Piperoxan hydrochloride (Benodaine hydrochloride) 是第一代抗组胺剂,是一种 α2肾上腺素受体拮抗剂。 | |||
T29096L |
Vapitadine
R 129160 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Vapitadine 是一种非镇静性抗组胺化合物,可缓解特应性皮炎引起的瘙痒。 | |||
T6562 |
Latrepirdine dihydrochloride
Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin |
Beta Amyloid; 5-HT Receptor; Adrenergic Receptor; GluR; Autophagy; Histamine Receptor | Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) 是一种具有口服活性和神经活性的多种药物靶点的拮抗剂,可刺激淀粉样前体蛋白分解代谢和 β-淀粉样蛋白分泌。 | |||
T1170 |
Olopatadine hydrochloride
盐酸奥洛他定,Olopatadine HCl,KW4679,ALO4943A |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Olopatadine hydrochloride (ALO4943A) 是一种抗组胺药,具有稳定肥大细胞的特性,用作治疗过敏性结膜炎的滴眼液。 | |||
T4563 |
Thonzylamine
neohetramine,松齐拉敏 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂,具有抗组胺和抗过敏特性,可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。 | |||
T4250 |
Bilastine
比拉斯汀,Bilaxten |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Bilastine (Bilaxten) 是新型抗组胺药,对H1组胺受体具有高度选择性,起效快,作用时间长的特性,可用于变应性鼻结膜炎和荨麻疹。 | |||
T0785 |
Dexchlorpheniramine Maleate
S-(+)-Chlorpheniramine maleate salt,右泛醇,马来酸右氯苯那敏 |
Dopamine Receptor; 5-HT Receptor; Norepinephrine; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Dexchlorpheniramine Maleate (S-(+)-Chlorpheniramine maleate salt) 是一种具有抗胆碱能特性的抗组胺药,用于治疗花粉热或荨麻疹等过敏性疾病。 | |||
T0113 |
Mebhydrolin napadisylate
Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,美海屈林萘二磺酸盐,Omeril,Diazoline |
5-HT Receptor; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mebhydrolin napadisylate (Incidal) 是一种抗组胺药,用于缓解组胺释放引起的过敏症状,如鼻过敏和过敏性皮肤病。 | |||
T21419 |
Diphenhydramine
苯海拉明,Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Diphenhydramine (Syntedril) 是第一代具有抗胆碱能作用的H1 受体拮抗剂,它能透过血脑屏障。 | |||
T0092 |
Antazoline hydrochloride
盐酸安他唑啉,Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Antazoline hydrochloride (Phenazoline hydrochloride) 是一种抗组胺药,可与组胺H1受体结合,阻断内源性组胺的作用。它也具有抗胆碱能特性,可缓解鼻塞,也可用作眼药水。 | |||
T0059 |
Diphenylpyraline hydrochloride
盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。 | |||
T21390 |
Fexofenadine
Carboxyterfenadine,Telfast,非索非那定,MDL 16.455,Allegra |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Fexofenadine (Carboxyterfenadine) 是一种抗组胺药物,用于治疗过敏症状,如鼻塞、花粉热和荨麻疹。与第一代抗组胺药相比,它通过血脑屏障并引起镇静的能力较差。 | |||
T21428 |
Mianserin
Lantanon,Lumin,Norval,Lerivon,Depnon |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mianserin 是H1受体反向激动剂,是四环抗抑郁药(TeCA)治疗家族中的一种精神活性化合物,具有抗抑郁、抗焦虑、止吐、促氧、催眠和抗组胺作用,可作为去甲肾上腺素和特定的血清素联合用药能治疗抑郁症。 | |||
T0445L |
Promethazine hydrochloride
盐酸异丙嗪,Promethazine HCl,Phenergan |
Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Promethazine hydrochloride (Promethazine HCl) 是抗组胺药物,是 H1 受体的强拮抗剂和 mACh 受体的中度拮抗剂,对 5-HT2A、5-HT2C、D2 和 α1-肾上腺素能受体具有中等亲和力。 | |||
T9084 |
Cetirizine Impurity B dihydrochloride
De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride,西替利嗪杂质B二盐酸盐,西替利嗪杂质04 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) 是 Cetirizine dihydrochloride 的杂质。Cetirizine 是一种抗组胺剂,是口服有活力的、特异性 H1受体拮抗剂。它能够抑制过敏反应期间嗜酸性粒细胞趋化,可以标记抗过敏特性。 | |||
T19839 |
Oxatomide
Oxatomida |
P2X Receptor; Calcium Channel; 5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Oxatomide (Oxatomida) 是一种有效且具有口服活性的双重 H1 组胺受体 和 P2X7 受体双重拮抗剂,具有抗组胺和抗过敏活性。Oxatomide 可用于阻断人 P2X7 受体中 ATP 诱导的电流 ,IC50 为 0.95 μM。Oxatomide 对 ATP 诱导的 Ca2+ 内流具有抑制作用,IC50 值为 0.43 μM。Oxatomide 对 5-羟色胺具有抑制作用。Oxatomide可用于治疗免疫系统疾病和研究超敏反应。 | |||
T40652 |
Meclizine
Meclozine |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Meclizine (Meclozine) (Meclozine)具有抗组胺作用,可可逆地抑制组胺与H1受体的相互作用。Meclizine 是哌嗪类H1拮抗剂的一个成员。Meclizine 是一种有效的抗运动病剂。Meclizine 可通过血脑屏障。Meclizine 是小鼠组成型雄烷受体(CAR)的激动剂配体,也是人CAR 的反向激动剂。Meclizine 可用于polyQ 毒性疾病的研究,如亨廷顿病。 | |||
T27836 |
Linadryl hydrochloride
A 446,A446,A-446 |
Others | Others |
Linadryl hydrochloride may have antihistamine activity. | |||
T11180 |
Embramine
|
Others | Others |
Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine. | |||
T0059L |
Diphenylpyraline
Difenilpiralina,AN 1041,AN1041,Dayfen,AN-1041,二苯拉林 |
Others | Others |
Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine. | |||
T25320 |
Diafen NN
NSC3410,NSC 3410,NSC-3410 |
Others | Others |
Diafen NN is an antihistamine agent. | |||
T36949 |
Niaprazine
|
5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Niaprazine 是有效的组胺 H1 受体拮抗剂,具有抗组胺和抗血清素活性。Niaprazine 在睡眠障碍方面有研究的价值。 | |||
T34152 |
Propiomazine Hydrochloride
PL043501,Largon |
Others | Others |
Propiomazine Hydrochloride is an antihistamine that blocks H1 receptors. | |||
T25033 |
Alcaftadine carboxylic acid
|
Others | Others |
Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis. | |||
T24851 |
Talastine HCl
HL-2186,Talastine hydrochloride,HL2186,Ahanon,HL 2186 |
Others | Others |
Talastine is an antihistamine drug. | |||
T25413 |
Fenethazine
RP 3015,Lisergan,Phenetazine,RP-3015,Ethysene |
Others | Others |
Fenethazine is an effective antihistamine used as an antiallergic drug. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7521 |
Azaphen
Pipofezin hydrochloride,阿扎吩,Pipofezine hydrochloride,Azafen |
5-HT Receptor; Serotonin Transporter | GPCR/G Protein; Neuroscience |
Azaphen (Pipofezin hydrochloride) 是一种 5-羟色胺重吸收抑制剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10280 |
Alimemazine D6
Trimeprazine D6 |
Others | Others |
Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine. | |||
T19233 |
Cetirizine D4 dihydrochloride
Cetirizine D4 dihydrochloride (1219803-84-5 free base) |
Others | Others |
Cetirizine D4 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | |||
T10770 |
Cetirizine D8
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | |||
T10769 |
Cetirizine D4
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | |||
T19234 |
Cetirizine D8 dihydrochloride
盐酸西替利嗪 D8 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | |||
T10816 |
Cinnarizine D8
|
Others | Others |
Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker. | |||
TMIJ-0259 |
Bilastine-d6
|
||
Bilastine-d6 是 Bilastine 的氘代化合物。Bilastine 的 CAS 号为 202189-78-4。Bilastine是新型抗组胺药,对H1组胺受体具有高度选择性,起效快,作用时间长的特性,可用于变应性鼻结膜炎和荨麻疹。 | |||
TMIJ-0260 |
Bilastine-d4
|
||
Bilastine-d4 是 Bilastine 的氘代化合物。Bilastine 的 CAS 号为 202189-78-4。Bilastine是新型抗组胺药,对H1组胺受体具有高度选择性,起效快,作用时间长的特性,可用于变应性鼻结膜炎和荨麻疹。 | |||
TMID-0188 |
Mianserin-d3
|
||
Mianserin-d3 是 Mianserin 的氘代化合物。Mianserin 的 CAS 号为 24219-97-4。Mianserin是H1受体反向激动剂,是四环抗抑郁药(TeCA)治疗家族中的一种精神活性化合物,具有抗抑郁、抗焦虑、止吐、促氧、催眠和抗组胺作用,可作为去甲肾上腺素和特定的血清素联合用药能治疗抑郁症。 |