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Search Results for " mra "

Targets Recommended: Glucocorticoid Receptor

41

抑制剂 & 化合物

1

天然产物

1

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T0083	Eplerenone Epoxymexrenone,CGP 30083,依普利酮,SC-66110	Glucocorticoid Receptor	Endocrinology/Hormones
	Eplerenone (CGP 30083) 是一种竞争性的、选择性的、具有口服活性的醛固酮 (aldosterone) 拮抗剂，IC50=138 nM。它对孕酮，雄激素，雌激素和糖皮质激素受体的亲和力低，可用于研究高血压和心肌梗死后的心力衰竭。
T18899L	5(6)-TAMRA hydrochloride(98181-63-6 Free base)
	5(6)-TAMRA hydrochloride(98181-63-6 Free base) 含有一种羧酸，可通过羧酸的碳二亚胺活化与伯胺反应。
T9694	Emraclidine CVL-231	AChR	Neuroscience
	Emraclidine (CVL-231) 是一种毒蕈碱 M4 受体阳性变构调节剂，可用于神经系统疾病研究。
T18891L	5-TAMRA chloride(91809-66-4 free base)	Others	Others
	5-TAMRA chloride(91809-66-4 free base) 显示出高效力且活性持续时间短，并且在生理上与孕酮相似。 FGA 的效力大约是黄体酮的 20-25 倍。
TP1711	5-Tamra-DRVYIHP	Others	Others
	5-Tamra-DRVYIHP 是一种含有用寡核苷酸标记的罗丹明衍生物的多肽。
T16982	TAMRA-PEG3-Azide	PROTAC Linker	PROTAC
	TAMRA-PEG3-Azide 是一种 TAMRA 红色荧光染料连接剂，最大激发/发射波长为 553/575 nm。
T18898	5(6)-TAMRA SE 5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯	Others	Others
	5(6)-TAMRA SE (5(6)-Carboxytetramethylrhodamine N-succinimidyl ester) 是荧光染料，能够结合寡聚核苷酸，并用于DNA 测序。
T18905	6-TAMRA 6-羧基四甲基罗丹明,6-Carboxytetramethylrhodamine	Others	Others
	6-TAMRA (6-Carboxytetramethylrhodamine) 常用作制备生物偶联物的荧光团，尤其是用于免疫化学的荧光抗体剂抗生物素蛋白衍生物。
T14054	5-TAMRA-SE 5-羧基四甲基罗丹明琥珀酰亚胺酯,5-Carboxytetramethylrhodamine succinimidyl ester,5-TAMRA-NHS ester	Others	Others
	5-TAMRA-SE 是一种胺反应性荧光剂。它的结合物能够产生一种 pH 不敏感的、明亮的橙红色荧光（Ex/Em~546/579 nm），具有良好的光稳定性。
T18891	5-TAMRA 5-羧基四甲基罗丹明,5-Carboxytetramethylrhodamine	Others	Others
	5-TAMRA (5-Carboxytetramethylrhodamine) 能够产生明亮的、pH 不敏感的橙红色荧光 (λex=546 nm，λem=579 nm)，有良好的光稳定性。
T34783	TAMRA-PEG4-NHS ester
	TAMRA-PEG4-NHS ester is a TAMRA red fluorescent dye derivative containing an NHS ester group which can be used to label the primary amines (-NH2) of proteins, amine-modified oligonucleotides, and other amine-containing molecules.
T67840	5-TAMRA Azide TAMRA Azide, isomer 5	Others	Others
	5-TAMRA Azide (TAMRA Azide, isomer 5) 是一种橙色荧光探针，兼容各种激发源，包括汞弧灯，钨弧灯和氙弧灯，氦氖激光544 nm 线和532 nm 绿激光线。它主要用于检测末端炔标记的生物分子通过铜催化的点击反应(CuAAC)。
T18904	6-TAMRA-SE 6-羧基四甲基罗丹明琥珀酰亚胺酯,6-TAMRA-NHS ester	Others	Others
	6-TAMRA-SE (6-TAMRA-NHS ester) 是一种带有胺反应基的荧光染料，是一种 DNA 自动测序的传统荧光团。
T16983	TAMRA-PEG4-acid	Others	Others
	TAMRA-PEG4-acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T18748	TAMRA-PEG4-methyltetrazine	Others	Others
	TAMRA-PEG4-methyltetrazine is a polyethylene glycol (PEG)-based linker employed for synthesizing proteolysis targeting chimeras (PROTACs)[1].
T61948	MraY-IN-2	Others	Others
	MraY-IN-2 (compound 6) 是有效的细菌转位酶MraY 抑制剂（IC50=4.5 μM），可用于抗菌研究。
TD0066	5(6)-TAMRA [5-(and-6)-Carboxytetramethylrhodamine] Mixed isomers
	5(6)-TAMRA contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. This bright, orange-fluorescent dye produces conjugates with absorption/emission maxima of ~555/580 nm.
T83283	5-TAMRA-Amyloid β-Protein (1-40)
	5-TAMRA-Amyloid β-Protein (1-40)为荧光 (TAMRA) 标记的淀粉样β-蛋白（Amyloid β-Protein）(1-40)片段, 其吸收和发射峰值分别位于Abs/Em=544/572 nm。
T17584	Biotin-PEG4-Dde-TAMRA-PEG3-Azide	Others	Others
	Biotin-PEG4-Dde-TAMRA-PEG3-Azide is a seven-unit polyethylene glycol (PEG) linker that is cleavable and employed in the synthetic production of antibody-drug conjugates (ADCs)[1].
T18749	TAMRA-PEG4-tetrazine	Others	Others
	TAMRA-PEG4-tetrazine is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T15074	DBCO-PEG4-TAMRA	Others	Others
	DBCO-PEG4-TAMRA, contains a DBCO group, is a PEG-based TARMA dye. The TAMRA dye is a dye widely used in oligonucleotide labeling.
T17339	(5,6)TAMRA-PEG3-Azide-PEG3-Desthiobiotin	Others	Others
	(5,6)TAMRA-PEG3-Azide-PEG3-Desthiobiotin is a polyethylene glycol (PEG)-based PROTAC linker utilized for the synthesis of PROTACs.
T74987	TAMRA alkyne, 6-isomer	Others	Others
	TAMRA alkyne, 6-isomer，作为TAMRA的一种连接物，其中TAMRA为发射橙色光的黄蒽类染料，广泛应用于寡核苷酸标记和氨基酸序列分析。此化合物通过引入炔基，实现了与叠氮化合物进行铜催化的点击化学反应的能力。
T78654	MraY-IN-3 hydrochloride	Others	Others
	MraY-IN-1（compound 12a）是一种针对细菌转位酶MraY的有效抑制剂，具有140 μM的IC50值。其对Escherichia coli K12、Bacillus subtilis W23和Pseudomonas fluorescens Pf-5展现出抗菌活性，相应的MIC50为7 µg/mL、12 µg/mL和46 µg/mL。MraY-IN-1适用于抗菌药物的研究领域。
T69315	5-TAMRA Cadaverine	Others	Others
	5-TAMRA cadaverine can used to modify carboxylic acid group in the presence of activators (e.g. EDC, or DCC) or activated esters (e.g. NHS esters) through a stable amide bond.
T18747	TAMRA-PEG3-biotin	Others	Others
	TAMRA-PEG3-biotin is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T16981	TAMRA-Azide-PEG-biotin	Others	Others
	TAMRA-Azide-PEG-biotin is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T18899	5(6)-TAMRA 5(6)-Carboxytetramethylrhodamine,5(6)-羧基四甲基罗丹明	Others	Others
	5(6)-TAMRA (5(6)-Carboxytetramethylrhodamine) 是一种荧光染料分子，广泛地被用作多肽和蛋白质的标记。
T64160	MraY-IN-3	Others	Others
	MraY-IN-3 (12a) 是一种细菌转位酶 MraY 的有效抑制剂 (IC50: 140 μM)。MraY-IN-3 能够作用于 E. coli K12 (MIC: 7 μg/ml)、B. subtilis W23 (MIC: 32 μg/ml)、P. fluorescens Pf-5 (MIC: 46 μg/ml)。
T64172	MraY-IN-1	Others	Others
	MraY-IN-1 (compound 12a) 是细菌转位酶 MraY 的有效抑制剂 (IC50: 140 μM)。MraY-IN-1 对大肠杆菌 K12 (MIC50: 7 μg/ml)、枯草芽孢杆菌 W23 (MIC50: 12 μg/ml) 和荧光假单胞杆菌 Pf-5 (MIC50: 46 μg/ml) 具有抗菌作用。MraY-IN-1 能够用于抗菌的研究。
T70125	Pemrametostat succinate	Others	Others
	Pemrametostat succinate is an orally active, potent and selective inhibitor of protein arginine methyltransferase 5 (PRMT5) that potently inhibits tumor growth in vitro and in vivo in animal models.
T17820	Dde Biotin-PEG4-TAMRA-PEG4 Alkyne	Others	Others
	Dde Biotin-PEG4-TAMRA-PEG4 Alkyne, a PEG-based PROTAC linker, facilitates PROTAC synthesis[1].
T80029	Bak BH3 (72-87), TAMRA-labeled
	BakBH3 (72-87), TAMRA-labeled，是一种具有生物活性的肽类化合物。
T81048	TAMRA hydrazide (6-isomer)
	TAMRA hydrazide (6-isomer) 作为点击化学试剂，特定于与羰基化合物，如醛和酮发生偶联反应。其中，TAMRA 组件作为一种红色荧光团，能与末端炔烃进行反应，实现荧光标记。
T81047	TAMRA-PEG2-Maleimide
	TAMRA-PEG2-Maleimide，一种TAMRA衍生物，含有4个PEG单元。其结构中的maleimide基团能够与硫醇基发生反应，形成共价键。
T81607	Omramotide
	Omramotide是一种免疫制剂，用途为主动免疫（抗肿瘤）。
T16984	TAMRA-PEG4-Alkyne	Others	Others
	TAMRA-PEG4-Alkyne is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T19064	TAMRA-probe 1	Others	Others
	TAMRA-probe 1 is a fluorescent probe for labeling.
T37472	TAMRA-Amyloid-β (1-42) Peptide (trifluoroacetate salt)	Others	Others
	TAMRA-Amyloid-β (1-42) peptide is a fluorescently labeled peptide. Amyloid-β (1-42) (Aβ42) is a neurotoxic 42-residue protein fragment found in amyloid plaques in postmortem cerebral cortex from patients with Alzheimer's disease. Aggregation of Aβ42 results in the formation of neurotoxic fibrils or globular oligomers. TAMRA-Amyloid-β (1-42) peptide is a labeled form of Aβ42 containing carboxytetramethyl rhodamine (TAMRA), which displays excitation/emission maxima of 543/572 nm, respectively.
T2138L	Oxyphencyclimine Oxiphencycliminum,Antulcus,Zamanil,Manir,Caridan,Naridan	Others	Others
	Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.
T8406L	Gadobutrol Monohydrate Gd-DO3A-butrol	Others	Others
	Gadobutrol is a medicinal product used in diagnostic magnetic resonance imaging (MRI) in adults and children. It provides contrast enhancement during cranial, spinal, breast, or other investigations. In the central nervous system, Gadobutrol works by high

化合物

Cat.No: T0083

Synonym: Epoxymexrenone,CGP 30083,依普利酮,SC-66110

Target: Glucocorticoid Receptor

5(6)-TAMRA hydrochloride(98181-63-6 Free base)

Cat.No: T18899L

Cat.No: T9694

Synonym: CVL-231

Target: AChR

5-TAMRA chloride(91809-66-4 free base)

Cat.No: T18891L

Target: Others

5-Tamra-DRVYIHP

Cat.No: TP1711

Target: Others

TAMRA-PEG3-Azide

Cat.No: T16982

Target: PROTAC Linker

Cat.No: T18898

Synonym: 5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯

Target: Others

Cat.No: T18905

Synonym: 6-羧基四甲基罗丹明,6-Carboxytetramethylrhodamine

Target: Others

Cat.No: T14054

Synonym: 5-羧基四甲基罗丹明琥珀酰亚胺酯,5-Carboxytetramethylrhodamine succinimidyl ester,5-TAMRA-NHS ester

Target: Others

Cat.No: T18891

Synonym: 5-羧基四甲基罗丹明,5-Carboxytetramethylrhodamine

Target: Others

TAMRA-PEG4-NHS ester

Cat.No: T34783

Cat.No: T67840

Synonym: TAMRA Azide, isomer 5

Target: Others

Cat.No: T18904

Synonym: 6-羧基四甲基罗丹明琥珀酰亚胺酯,6-TAMRA-NHS ester

Target: Others

TAMRA-PEG4-acid

Cat.No: T16983

Target: Others

TAMRA-PEG4-methyltetrazine

Cat.No: T18748

Target: Others

Cat.No: T61948

Target: Others

5(6)-TAMRA [5-(and-6)-Carboxytetramethylrhodamine] *Mixed isomers*

Cat.No: TD0066

5-TAMRA-Amyloid β-Protein (1-40)

Cat.No: T83283

Biotin-PEG4-Dde-TAMRA-PEG3-Azide

Cat.No: T17584

Target: Others

TAMRA-PEG4-tetrazine

Cat.No: T18749

Target: Others

DBCO-PEG4-TAMRA

Cat.No: T15074

Target: Others

(5,6)TAMRA-PEG3-Azide-PEG3-Desthiobiotin

Cat.No: T17339

Target: Others

TAMRA alkyne, 6-isomer

Cat.No: T74987

Target: Others

MraY-IN-3 hydrochloride

Cat.No: T78654

Target: Others

5-TAMRA Cadaverine

Cat.No: T69315

Target: Others

TAMRA-PEG3-biotin

Cat.No: T18747

Target: Others

TAMRA-Azide-PEG-biotin

Cat.No: T16981

Target: Others

Cat.No: T18899

Synonym: 5(6)-Carboxytetramethylrhodamine,5(6)-羧基四甲基罗丹明

Target: Others

Cat.No: T64160

Target: Others

Cat.No: T64172

Target: Others

Pemrametostat succinate

Cat.No: T70125

Target: Others

Dde Biotin-PEG4-TAMRA-PEG4 Alkyne

Cat.No: T17820

Target: Others

Bak BH3 (72-87), TAMRA-labeled

Cat.No: T80029

TAMRA hydrazide (6-isomer)

Cat.No: T81048

TAMRA-PEG2-Maleimide

Cat.No: T81047

Cat.No: T81607

TAMRA-PEG4-Alkyne

Cat.No: T16984

Target: Others

Cat.No: T19064

Target: Others

TAMRA-Amyloid-β (1-42) Peptide (trifluoroacetate salt)

Cat.No: T37472

Target: Others

Oxyphencyclimine

Cat.No: T2138L

Synonym: Oxiphencycliminum,Antulcus,Zamanil,Manir,Caridan,Naridan

Target: Others

Gadobutrol Monohydrate

Cat.No: T8406L

Synonym: Gd-DO3A-butrol

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T80416	Mram 8	Others	Others
	Mram 8为源自堇菜科植物堇菜中提取的环肽。

天然产物

Cat.No: T80416

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-01117	MRAP Protein, Human, Recombinant (hFc) FALP,FGD2,melanocortin 2 receptor accessory protein,GCCD2,B2...	Human	HEK293 Cells
	MRAP (Melanocortin 2 Receptor Accessory Protein) is a Protein Coding gene. This gene encodes a melanocortin receptor-interacting protein. It belongs to the MRAP family. MRAP, which contains a single transmembrane domain, has a unique structure, an antiparallel homodimer. MRAP is a single transmembrane domain accessory protein and a critical component of the hypothamo pituitary-adrenal axis. MRAP is highly expressed in the adrenal gland and is essential for adrenocorticotropin hormone (ACTH) rece...

重组蛋白

MRAP Protein, Human, Recombinant (hFc)

Cat.No: TMPY-01117

Species: Human

Expression System: HEK293 Cells

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