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TargetMol产品目录中 "

(rac)rotigotine hydrochloride

"的结果
  • 抑制剂&激动剂
    16
    TargetMol | Inhibitors_Agonists
  • 同位素
    7
    TargetMol | Isotope_Products
(Rac)-Rotigotine hydrochloride
T12676102120-99-0
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
  • ¥ 258
5日内发货
规格
数量
rac-7-hydroxy Propranolol (hydrochloride)
T3623176275-67-7
rac-7-hydroxy Propranolol (hydrochloride) is a ring-hydroxylated isomer and metabolite of propranolol that is an antagonist at β-adrenergic receptors (0.95 potency relative to propranolol). It also demonstrates potent vasodilator activity (0.20 potency relative to propranolol; pA2 = 7.58).
  • ¥ 4810
35日内发货
规格
数量
rac-Desethyl Oxybutynin (hydrochloride)
T3780181039-77-2
rac-Desethyl oxybutynin is an active metabolite of the muscarinic acetylcholine receptor (mAChR) antagonist oxybutynin .1,2,3rac-Desethyl oxybutynin is formed from oxybutynin by the cytochrome P450 (CYP) isoform CYP3A4.2It binds to mAChRs in isolated rat bladder, submaxillary gland, heart, and colon with Kivalues of 5.38, 3.12, 16, and 5.59 nM, respectively.rac-Desethyl oxybutynin (0.4 and 0.8 mg/kg) reduces micturition pressure in rats.3
  • ¥ 1380
35日内发货
规格
数量
rac Desmethyl Citalopram Hydrochloride
T6785197743-99-2
rac Desmethyl Citalopram Hydrochloride 是一种5-羟色胺摄取抑制剂,IC50值为0.013μM。
  • ¥ 937
现货
规格
数量
Rotigotine HydrochlorideRotigotine (Hydrochloride),N 0923,N-0924,Rotigotine HCl,罗替戈汀盐酸盐,盐酸罗替戈汀,N-0923
T21446125572-93-2
Rotigotine Hydrochloride (N-0924) 是多巴胺受体激动剂,是5-HT1A 受体的部分激动剂,以及α2B-肾上腺素受体的拮抗剂,具有抗帕金森病活性。
  • ¥ 138
现货
规格
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rac threo-Dihydro Bupropion-d9 Hydrochloride
TMIH-0475
rac threo-Dihydro Bupropion-d9 Hydrochloride 是 rac threo-Dihydro Bupropion Hydrochloride 的氘代化合物。rac threo-Dihydro Bupropion Hydrochloride 的 CAS 号为 1396889-62-5。
  • ¥ 4800
5日内发货
规格
数量
(Rac)-IBT6A hydrochloride
T739421807619-60-8
(Rac)-IBT6A hydrochloride 是 IBT6A hydrochloride 的消旋体。IBT6A 是 Ibrutinib 的一种杂质。IBT6A 可用于合成 IBT6A-Ibrutinib 二聚体和 IBT6A 加合物。Ibrutinib 是一种不可逆的选择性 Btk 抑制剂,IC50为 0.5 nM。
  • 询价
规格
数量
Rotigotine D7 HydrochlorideN-0923 D7 Hydrochloride
T12760
Rotigotine D7 Hydrochloride is the deuterium labeled Rotigotine(N-0923), which is an agonist of dopamine D2 and D3 receptor.
  • 询价
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rac NorMetanephrine-d3 Hydrochloride
TMIH-04741085333-97-6
rac NorMetanephrine-d3 Hydrochloride 是 rac NorMetanephrine Hydrochloride 的氘代化合物。
  • ¥ 2880
5日内发货
规格
数量
rac-Paroxetine-d4 Hydrochloride
TMID-00421217683-35-6
rac-Paroxetine-d4 Hydrochloride 是 rac-Paroxetine Hydrochloride 的氘代化合物。rac-Paroxetine Hydrochloride 的 CAS 号为 78246-49-8。Paroxetine hydrochloride 是一种血清素摄取抑制剂,能抑制 GRK2 活性,IC50值为 14 μM。它可研究抑郁症。
  • ¥ 8250
5日内发货
规格
数量
rac Atomoxetine-d5 Hydrochloride托莫西汀-d5 盐酸盐
TMID-02021398065-95-6
rac Atomoxetine-d5 Hydrochloride 是 rac Atomoxetine Hydrochloride 的氘代化合物。rac Atomoxetine Hydrochloride 的 CAS 号为 82857-40-7。
  • 询价
35日内发货
规格
数量
(Rac)-Atomoxetine D7 hydrochloride(Rac)-LY 139603 D7,(Rac)-Tomoxetine D7 hydrochloride
T12657
(Rac)-Atomoxetine D7 hydrochloride is a deuterium labeled (Rac)-Atomoxetine hydrochloride. (Rac)-Atomoxetine hydrochloride is a racemic form of Atomoxetine hydrochloride.
  • ¥ 3200
5日内发货
规格
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(Rac)-IBT6A hydrochloride (1412418-47-3 free base)(Rac)-IBT6A hydrochloride
T10625L
(Rac)-IBT6A hydrochloride is a racemate of IBT6A. IBT6A is an impurity of Ibrutinib. IBT6A can be used in the synthesis of IBT6A Ibrutinib dimer and IBT6A adduct. Ibrutinib is a Btk inhibitor (IC50: 0.5 nM).
  • 询价
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rac Metanephrine-d3 Hydrochloride Salt
TMIH-04731215507-88-2
rac Metanephrine-d3 Hydrochloride Salt 是 rac Metanephrine Hydrochloride Salt 的氘代化合物。
  • ¥ 2630
5日内发货
规格
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(Rac)-5-Hydroxymethyl Tolterodine hydrochloride(Rac)-5-Hydroxymethyl Tolterodine hydrochloride,(Rac)-PNU-200577hydrochloride,(Rac)-Desfesoterodine hydrochloride
T40161250214-40-5
(Rac)-5-Hydroxymethyl Tolterodine hydrochloride, also known as (Rac)-Desfesoterodine hydrochloride, is an active metabolite of Tolterodine that functions as a mAChR antagonist. It exhibits significant affinity (K i values) for M1, M2, M3, M4, and M5 receptors, with values of 2.3 nM, 2 nM, 2.5 nM, 2.8 nM, and 2.9 nM, respectively. This compound is commonly employed in research related to overactive bladder conditions.
  • ¥ 1150
5日内发货
规格
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(Rac)-CP-601927 hydrochloride
T39833230615-01-7
(Rac)-CP-601927 hydrochloride is the racemate form of CP-601927, which is a nicotinic acetylcholine receptor (nAChR) agonist. It exhibits Ki values of 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively.
  • ¥ 2120
5日内发货
规格
数量