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Targets Recommended: Antibacterial Antibiotic Autophagy

88

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0510 Sulfaguanidine

Sulfaguine,Guanicil,磺胺脒

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfaguanidine (Guanicil) 是一种具有口服活性的磺胺类抗菌剂和抗生素。它可用于肠道感染,例如细菌性痢疾的研究。
T7533 Taurolidine

Apoptosis; Others; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Others
Taurolidine 是一种广谱抗菌剂,用于预防中心静脉导管相关感染。它具有抗真菌和抗肿瘤作用。
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T6385 Amoxicillin Sodium

阿莫西林钠,Clavulanate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin Sodium (Clavulanate) 是一种有广谱抗菌活性,口服吸收好的抗生素。它能抑制细胞壁中多肽的生物合成,可抑制细胞生长。
T0921 Sulfabenzamide

Sultrin,N-Sulfanilylbenzamide,苯甲酰磺胺

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfabenzamide (N-Sulfanilylbenzamide) 是一种磺胺类抗菌剂,可单独使用或与磺胺噻唑和磺胺乙酰胺一起用作阴道内的局部抗菌制剂。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T1177 Sulfaquinoxaline

磺胺喹恶啉,Avicocid,磺胺喹噁啉,Sulphaquinoxaline,Sulfabenzpyrazine

Others; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Others
Sulfaquinoxaline (Sulfabenzpyrazine) 是一种兽用抗菌剂,对革兰氏阴性菌和革兰氏阳性菌均有活性。它能用于预防球虫病和细菌感染。
TP1444 Magainin 2

蛙皮素 2

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Magainin 2是从非洲爪蟾皮肤中分离得到的一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌显示出抗生素活性,对原生动物也有活性。它通过优先与细菌膜中丰富的阴离子磷脂相互作用而发挥细胞毒性作用。
T1434 Clarithromycin

A-56268,克拉霉素

P450; ribosome; MRP; Antibacterial; Antibiotic; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology
Clarithromycin (A-56268) 具有广谱的抗菌活性。它抑制 CYP3A4催化的三唑仑 α-羟基化,IC50(Ki) 值为 56 (43) μM。它抑制 HERG 钾电流。它可削弱连接 hERG1 和 PI3K 的信号通路影响自噬流 。
T19717 Cyclo-L-Trp-L-Trp

Antifungal Microbiology/Virology
Cyclo-L-Trp-L-Trp 是一种广谱抗真菌剂。它还诱导组蛋白的高度乙酰化。
T4989 Fosfomycin Tromethamine

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T0917 Sulfaquinoxaline sodium salt

SQ-Na,磺胺喹恶啉钠盐,Sulfaquinoxaline sodium,磺胺喹啉钠

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Sulfaquinoxaline sodium salt (SQ-Na) 是一种兽用广谱抗菌剂,有抗革兰氏阴性菌和革兰氏阳性菌活性。Sulfaquinoxaline 能用于预防球虫病和细菌感染。
T1000L Chlorhexidine diacetate

醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras

CAT; Antibacterial; Antibiotic; Antifection Microbiology/Virology; oxidation-reduction
Chlorhexidine diacetate (Bactigras) 是一种双胍类杀菌剂,能快速消灭革兰氏阳性菌和革兰氏阴性菌。它也用作漱口水以防止口腔菌斑。
T20702 Ormetoprim

Ro5-9754,奥美普林,Ro 5-9754,Ro-5-9754

Antibiotic Microbiology/Virology
Ormetoprim (Ro 5-9754) 是一种兽用抗菌剂,通常用于水产养殖和家禽行业,可以预防疾病在淡水水产养殖中的传播,促进家畜的生长。
T3125 Amikacin sulfate

Amikacin Sulfate Salt,阿米卡霉素硫酸,硫酸阿米卡星

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Amikacin sulfate 是一种氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它抑制大多数革兰氏阴性细菌,还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T1233 Oxolinic acid

Emyrenil,Nidantin,NSC 110364,恶喹酸,Dioxacin,Urinox

Dopamine Receptor; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology; Neuroscience
Oxolinic acid (Nidantin) 是一种抗生素,对革兰氏阴性菌和革兰氏阳性菌均有效,可研究急性和慢性尿路感染。它是一种 DNA/RNA 合成抑制剂,也是一种多巴胺摄取抑制剂,能刺激小鼠的活跃过度。
T7865 Danofloxacin

达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine

Others; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
T0195 Secnidazole

RP-14539,PM-185184,塞克硝唑

Antibiotic; Parasite Microbiology/Virology
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。
T7419 Sutezolid

PNU-100480,U-100480,PF-02341272

Antibacterial; Antibiotic Microbiology/Virology
Sutezolid (U-100480) 是一种具有口服活性恶唑烷酮抗菌剂,通过抑制细菌蛋白质合成发挥作用。它有抗分枝杆菌活性,可研究耐药结核病。
T3131 Fosfomycin calcium

Phosphomycin calcium salt,Fosmicin,磷霉素钙

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T1005L Amoxicillin trihydrate

Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。
T0331 Moxifloxacin hydrochloride

盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
T6382 Amikacin disulfate

硫酸阿米卡星,Pierami,阿米卡星硫酸盐,BAY-416651 sulfate,BB-K8,Amikacin sulfate

Antibacterial; Antibiotic Microbiology/Virology
Amikacin disulfate (BAY-416651 sulfate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它对大多数革兰氏阴性细菌都有效。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T6383 Amikacin hydrate

阿米卡星水合物,BAY416651 hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Amikacin hydrate (BAY416651 hydrate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T1733 Ciprofloxacin EP IMpurity A

Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A

Antibiotic Microbiology/Virology
Ciprofloxacin EP IMpurity A (Fluoroquinolonic Acid) 是一种抗生素和抗菌剂。
T30785 Cefacetrile

Cefacetrilum,Cefacetrilo,Celospor,Cephacetrile,Cefacetril

Antibiotic Microbiology/Virology
Cefacetrile (Cephacetrile) 是一种广谱的头孢类抗生素,具有抗菌活性,可用于研究革兰氏菌感染,作用与头孢噻吩作用。
T6349L Sitafloxacin

DU-6859A,Sitafloxacin anhydrous,DU 6859,DU6859,DU-6859,DU 6859A,DU6859A

Antibiotic Microbiology/Virology
Sitafloxacin (Sitafloxacin anhydrous) 是一种具有口服活性的氟喹诺酮类抗生素,具有广谱的抗菌活性。Sitafloxacin 可用于研究呼吸道感染和尿路感染。
T30787 Cefetamet sodium

Ro 15-8074/001,Ro15-8074/001,Ro-15-8074/001

Antibiotic Microbiology/Virology
Cefetamet sodium (Ro 15-8074/001) 是一种可口服的头孢类抗生素,具有抗菌活性,可用于研究肝硬化和肺部感染。
T20022 Cephalexin monohydrate

Cephalexin hydrate,Cephacillin hydrate,Cefalexin hydrate

Antibiotic Microbiology/Virology
Cephalexin monohydrate (Cephalexin hydrate) 是一种可口服的半合成头孢菌素类抗生素,具有显著的抗菌活性, 通过靶向青霉素结合蛋白 (PBPs)抑制细菌增殖。
TP1763L Magainin 1 acetate

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Magainin 1 acetate 是一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌表现出抗生素活性。
T1400L Demeclocycline

Ledermycin,Bioterciclin,Deteclo,Declostatin,Deganol

Antibacterial Microbiology/Virology
Demeclocycline (Declostatin) 是一种四环素类抗生素,产自金霉素链霉菌(Streptomyces aureofaciens)菌株。Demeclocycline 具有抗菌活性,能抑制血管加压素对肾小管的作用,从而导致利尿。Demeclocycline 可用诱导尿崩症和急性肾衰竭。
T36020 Florfenicol amine hydrochloride

Antibiotic Microbiology/Virology
Florfenicol amine hydrochloride 是一种人工合成的兽用抗生素,具有抗菌活性。Florfenicol amine hydrochloride 在水产养殖业和牧业养殖业中应用广泛,可以用来研究巴氏杆菌、爱德华氏菌、大肠杆菌和沙门氏杆菌引起的疾病。
T74821 Nemonoxacin

TG-873870

Antibacterial Microbiology/Virology
Nemonoxacin (TG-873870) 是一种可口服的非氟化喹诺酮类抗生素,具有广谱的抗菌活性,抑制葡萄球菌、链球菌和肠球菌、淋病奈瑟菌和流感嗜血杆菌均。Nemonoxacin 可用于研究细菌感染和社区获得性肺炎。
T14922 Cefodizime

Antibacterial; Antibiotic Microbiology/Virology
Cefodizime 是一种新型头孢菌素抗生素,具有广泛的生物活性。Cefodizime 对肾脏没有毒性且具有良好的耐受性和免疫调节活性,具有抗菌活性,可用于研究呼吸系统和泌尿系统的严重感染。
T1101 Minocycline hydrochloride

Minocycline HCl,盐酸米诺环素,美满霉素

HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Minocycline hydrochloride (Minocycline HCl) 属于四环素类抗生素,具有出色的吸收和组织渗透性。Minocycline hydrochloride 是一种广谱的抗菌剂,可用于多种细菌感染以及痤疮的治疗。
T25085 Amythiamicin B

Others Others
Amythiamicin B is a novel antimicrobial antibiotic.
T1070L Cefmetazole

Sodium, Cefmetazole,Cefmetazolum,Cefmetazolo

Others Others
Cefmetazole is a second-generation semi-synthetic β-lactam cephalosporin antibiotic with antimicrobial activity.
T25037 Aldecalmycin

Others Others
Aldecalmycin is a new antimicrobial antibiotic isolated from Streptomyces.
T26455 A 83016F

A-83016F,A83016F

Others Others
A 83016F, an antibiotic from an actinomycete designated A83016, exhibits weak antimicrobial activity.
T26479 A32390A

A-32390A,A 32390A

Others Others
A32390A, an antibiotic inhibitor, shows antimicrobial activity against gram-positive bacteria and fungi.
T16382 Oleandomycin

Others Others
Oleandomycin is similar to Erythromycin has antimicrobial activity. Oleandomycin is a macrolide antibiotic structurally closely related to Erythromycin.
T70429 TP-6076

Others Others
TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A. baumannii.
T28046 Mirosamicin

A 11725 II,Antibiotic AR 5-2

Others Others
Mirosamicin is a macrolide antibiotic, it has antimicrobial effect against gram-positive bacteria, some gram-negative bacteria and mycoplasma.
T31104 CS 461

CS461,CS-461

Others Others
CS 461 is a cephalosporin antibiotic that has shown effective antimicrobial activity against a variety of bacteria in vitro and in vivo.
T1466L Difloxacin HCl

Others Others
Difloxacin 是第二代合成的氟喹诺酮抗菌抗生素。
T39683 Human β-defensin-3

Human β-defensin-3,HβD-3

Human β-defensin-3 (HβD-3) is an antibiotic antimicrobial peptide synthesized by epithelial cells. It exhibits potent antimicrobial properties and mitigates inflammatory cytokine responses. HβD-3 efficiently targets various microorganisms, displaying IC90 values ranging from 6 to 25 μg/ml.
T37350 TBI-223

Others Others
TBI-223 is an orally bioavailable oxazolidinone antibiotic with antimicrobial properties. It exhibits potent activity against Mycobacterium tuberculosis (Mtb)[1][2].
T85067 Berkeleylactone E

Others Others
Berkeleylactone E为一种大环内酯类抗生素。
T83042 Antimicrobial agent-26

Others Others
Antimicrobial agent-26?是一款降低抗生素耐药性的高效抗菌化合物。
T80304 Aurein 5.2

Antibiotic Microbiology/Virology
Aurein 5.2是一种具有抗菌活性的抗生素肽类化合物。

化合物

Sulfaguanidine
Cat.No: T0510
Synonym: Sulfaguine,Guanicil,磺胺脒
Target: Antibacterial, Antibiotic, Autophagy
Taurolidine
Cat.No: T7533
Synonym:
Target: Apoptosis, Others, Antibacterial, Antibiotic
Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
Amoxicillin Sodium
Cat.No: T6385
Synonym: 阿莫西林钠,Clavulanate
Target: Antibacterial, Antibiotic
Sulfabenzamide
Cat.No: T0921
Synonym: Sultrin,N-Sulfanilylbenzamide,苯甲酰磺胺
Target: Antibacterial, Antibiotic, Autophagy
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Sulfaquinoxaline
Cat.No: T1177
Synonym: 磺胺喹恶啉,Avicocid,磺胺喹噁啉,Sulphaquinoxaline,Sulfabenzpyrazine
Target: Others, Antibacterial, Antibiotic, Parasite
Magainin 2
Cat.No: TP1444
Synonym: 蛙皮素 2
Target: Antibacterial, Antibiotic, Antifungal
Clarithromycin
Cat.No: T1434
Synonym: A-56268,克拉霉素
Target: P450, ribosome, MRP, Antibacterial, Antibiotic, Autophagy
Cyclo-L-Trp-L-Trp
Cat.No: T19717
Synonym:
Target: Antifungal
Fosfomycin Tromethamine
Cat.No: T4989
Synonym:
Target: Antibacterial, Antibiotic
Sulfaquinoxaline sodium salt
Cat.No: T0917
Synonym: SQ-Na,磺胺喹恶啉钠盐,Sulfaquinoxaline sodium,磺胺喹啉钠
Target: Antibacterial, Antibiotic, Parasite
Chlorhexidine diacetate
Cat.No: T1000L
Synonym: 醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras
Target: CAT, Antibacterial, Antibiotic, Antifection
Ormetoprim
Cat.No: T20702
Synonym: Ro5-9754,奥美普林,Ro 5-9754,Ro-5-9754
Target: Antibiotic
Amikacin sulfate
Cat.No: T3125
Synonym: Amikacin Sulfate Salt,阿米卡霉素硫酸,硫酸阿米卡星
Target: ribosome, Antibacterial, Antibiotic
Oxolinic acid
Cat.No: T1233
Synonym: Emyrenil,Nidantin,NSC 110364,恶喹酸,Dioxacin,Urinox
Target: Dopamine Receptor, DNA/RNA Synthesis, Antibacterial, Antibiotic
Danofloxacin
Cat.No: T7865
Synonym: 达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine
Target: Others, DNA/RNA Synthesis, Antibacterial, Antibiotic
Secnidazole
Cat.No: T0195
Synonym: RP-14539,PM-185184,塞克硝唑
Target: Antibiotic, Parasite
Sutezolid
Cat.No: T7419
Synonym: PNU-100480,U-100480,PF-02341272
Target: Antibacterial, Antibiotic
Fosfomycin calcium
Cat.No: T3131
Synonym: Phosphomycin calcium salt,Fosmicin,磷霉素钙
Target: Antibacterial, Antibiotic
Amoxicillin trihydrate
Cat.No: T1005L
Synonym: Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate
Target: Antibacterial, Antibiotic
Moxifloxacin hydrochloride
Cat.No: T0331
Synonym: 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl
Target: Topoisomerase, Antibacterial, Antibiotic
Amikacin disulfate
Cat.No: T6382
Synonym: 硫酸阿米卡星,Pierami,阿米卡星硫酸盐,BAY-416651 sulfate,BB-K8,Amikacin sulfate
Target: Antibacterial, Antibiotic
Amikacin hydrate
Cat.No: T6383
Synonym: 阿米卡星水合物,BAY416651 hydrate
Target: Others, Antibacterial, Antibiotic
Ciprofloxacin EP IMpurity A
Cat.No: T1733
Synonym: Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A
Target: Antibiotic
Cefacetrile
Cat.No: T30785
Synonym: Cefacetrilum,Cefacetrilo,Celospor,Cephacetrile,Cefacetril
Target: Antibiotic
Sitafloxacin
Cat.No: T6349L
Synonym: DU-6859A,Sitafloxacin anhydrous,DU 6859,DU6859,DU-6859,DU 6859A,DU6859A
Target: Antibiotic
Cefetamet sodium
Cat.No: T30787
Synonym: Ro 15-8074/001,Ro15-8074/001,Ro-15-8074/001
Target: Antibiotic
Cephalexin monohydrate
Cat.No: T20022
Synonym: Cephalexin hydrate,Cephacillin hydrate,Cefalexin hydrate
Target: Antibiotic
Magainin 1 acetate
Cat.No: TP1763L
Synonym:
Target: Antibacterial, Antibiotic, Antifungal
Demeclocycline
Cat.No: T1400L
Synonym: Ledermycin,Bioterciclin,Deteclo,Declostatin,Deganol
Target: Antibacterial
Florfenicol amine hydrochloride
Cat.No: T36020
Synonym:
Target: Antibiotic
Nemonoxacin
Cat.No: T74821
Synonym: TG-873870
Target: Antibacterial
Cefodizime
Cat.No: T14922
Synonym:
Target: Antibacterial, Antibiotic
Minocycline hydrochloride
Cat.No: T1101
Synonym: Minocycline HCl,盐酸米诺环素,美满霉素
Target: HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Amythiamicin B
Cat.No: T25085
Synonym:
Target: Others
Cefmetazole
Cat.No: T1070L
Synonym: Sodium, Cefmetazole,Cefmetazolum,Cefmetazolo
Target: Others
Aldecalmycin
Cat.No: T25037
Synonym:
Target: Others
A 83016F
Cat.No: T26455
Synonym: A-83016F,A83016F
Target: Others
A32390A
Cat.No: T26479
Synonym: A-32390A,A 32390A
Target: Others
Oleandomycin
Cat.No: T16382
Synonym:
Target: Others
TP-6076
Cat.No: T70429
Synonym:
Target: Others
Mirosamicin
Cat.No: T28046
Synonym: A 11725 II,Antibiotic AR 5-2
Target: Others
CS 461
Cat.No: T31104
Synonym: CS461,CS-461
Target: Others
Difloxacin HCl
Cat.No: T1466L
Synonym:
Target: Others
Human β-defensin-3
Cat.No: T39683
Synonym: Human β-defensin-3,HβD-3
Target:
TBI-223
Cat.No: T37350
Synonym:
Target: Others
Berkeleylactone E
Cat.No: T85067
Synonym:
Target: Others
Antimicrobial agent-26
Cat.No: T83042
Synonym:
Target: Others
Aurein 5.2
Cat.No: T80304
Synonym:
Target: Antibiotic
Cat. No. Product Name Target Signaling Pathways
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
T1032 Erythromycin

红霉素,E-Mycin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。
T6995 Ochromycinone

STA 21,STA21,STA-21

Antibacterial; STAT JAK/STAT signaling; Microbiology/Virology; Stem Cells
Ochromycinone (STA 21) 是一种天然抗生素,也是一种 STAT3抑制剂。它可抑制 STAT3DNA 结合活性,STAT3二聚化。它具有抗癌和抗菌活性。
T22308 Dimboa

2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布

Others; Antibacterial; Antibiotic; Antifungal Microbiology/Virology; Others
Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) 是抗生素,是禾本科植物化学防御系统的一部分。 它对许多已研究的细菌和真菌菌株具有生长抑制特性。它表现出强大的自由基清除活性和较弱的铁 (III) 离子还原活性和有抗氧化活性。
T0146 Tioconazole

UK-20349,Vagistat,噻康唑

Antibiotic; Antifection; Antifungal Microbiology/Virology
Tioconazole (Vagistat) 是一种广谱性的抗真菌咪唑衍生物。它抑制几种皮肤真菌和几种酵母菌的 MIC50分别小于 3.12 mg/L 和 9 mg/L。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
T1153 Trimethoprim

NIH 204,BW 56-72,甲氧苄啶,NSC-106568

DHFR; DNA/RNA Synthesis; Antifolate; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Trimethoprim (NSC-106568) 是抑菌抗生素,也是具有口服活性的二氢叶酸还原酶抑制剂。它对多种革兰氏阳性和革兰氏阴性需氧细菌具有活性,可用于尿路感染,肺孢子菌肺炎和志贺氏菌病的研究。
T15717 Lasalocid

Lasalocid-A,Antibiotic X-537A,Ionophore X-537A

Antibacterial Microbiology/Virology
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。
T6402 Azomycin

2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin

Antibacterial; Antibiotic Microbiology/Virology
Azomycin (Ro 05-9129) 是一种可抑制有氧革兰氏阳性菌和革兰氏阴性菌的生长的抗生素。
T7148 JOSAMYCIN

EN-141,交沙霉素

Antibacterial; Antibiotic Microbiology/Virology
Josamycin (EN-141) 是一种大环内酯类抗生素,对多种病原体有抗菌活性。它对核糖体的解离常数Kd 为 5.5 nM。
T10278 Alamethicin

Antibacterial Microbiology/Virology
Alamethicin 是从 Trichoderma viride 中分离得到的一种通道形成抗生素肽,具有潜在的抗菌活性,抑制甲烷生成并促进生物电化学系统中的乙酰生成。
T4136 Lapachol

Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin

Others; Influenza Virus; Antibacterial; Parasite; Antifungal Microbiology/Virology; Others
Lapachol (CI75490) 是从Tabebuia avellanedae 中分离得到的一种萘醌。它具有具有抗菌、抗炎、镇痛、抗肿瘤和抗生素特性。
T28764 SF2312

SF-2312,SF 2312

Glucokinase; Antibacterial Metabolism; Microbiology/Virology
SF2312 是一种由放线菌微孢子菌产生的天然膦酸盐抗生素,是高效的糖酵解酶烯醇化酶抑制剂。SF2312 具有抗菌活性,可抑制细菌生长,对革兰氏阴性和革兰氏阴性菌均具有抑制作用。SF2312 抑制人重组 ENO1 和 ENO2。
T0950 Neomycin sulfate

Framycin sulfate,硫酸新霉素

Phospholipase; ribosome; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Neomycin sulfate (Framycin sulfate) 是一种广谱的氨基糖苷类抗生素。Neomycin sulfate 可以阻断细菌蛋白质的合成以发挥抗菌活性。Neomycin sulfate 常用于筛选具有 Neo 抗性基因的原核和真核细胞。
T8641 Vancomycin

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Vancomycin 是一种糖肽类抗生素,可以通过改变细胞膜的渗透性并选择性地抑制核糖核酸的合成以发挥抗菌活性。Vancomycin 可以用于治疗所有抗生素均无效的严重感染。
T20779 Kitasamycin tartrate

Leucomycin tartrate

Others Others
Kitasamycin tartrate, a macrolide antibiotic produced by Streptomyces kitasatoensis, has a wide spectrum of antimicrobial activity.
T75443 Tomaymycin

Others Others
Tomaymycin 是一种抗肿瘤抗生素。Tomaymycin 对革兰氏阳性菌具有抗菌活性。
TN7553 Dihydroaeruginoic Acid

CGP 52547

Others Others
Dihydroaeruginoic acid, an antibiotic sourced originally from P. fluorescens, exhibits antimicrobial efficacy in disc assays against diverse pathogens, including R. solani, P. ultimum, B. cinerea, S. rolfsii, C. gloeosporioides, F. oxysporum, and S. tritici fungi, along with B. subtilis, E. herbicola, and S. albus bacteria, at a concentration of 200 μg/disc.
T38241 2-Aminoimidazole

Others Others
2-Aminoimidazole is a potent antibiofilm agent and adjuvant to antimicrobial treatments, which effectively disrupts bacterial self-protection mechanisms by inhibiting biofilm formation and genetically-encoded antibiotic resistance traits. Additionally, 2-Aminoimidazole acts as a weak noncompetitive inhibitor of human arginase I, with a Ki value of 3.6 mM[1][2][3].
T11233 Erythromycin thiocyanate

Antibacterial Microbiology/Virology
Erythromycin thiocyanate acts by binding to bacterial 50S ribosomal subunits and inhibits RNA-dependent protein synthesis by blockage of transpeptidation and/or translocation reactions, without affecting synthesis of nucleic acid .Erythromycin thiocyanate
T75753 Magainin 1 TFA

Others Others
Magainin 1 TFA (Magainin I TFA) 是从 Xenopus laevis 皮肤中分离出的一种抗菌和两亲性肽。Magainin 1 TFA 对多种革兰氏阴性和革兰氏阳性细菌均表现出抗生素活性。
T73673 Thiomarinol A

Others Others
Thiomarinol A (4-Hydroxythiomarinol C) 是一种有效的抗生素。Thiomarinol A 是二硫代吡咯酮和海藻酸的混合物。Thiomarinol A 显示出抗菌活性。Thiomarinol A 以剂量依赖性方式抑制 MRSA IleRS,Kiapp 值为 19 nM。
T35741 Gliovirin

Others Others
Gliovirin is a fungal metabolite that has been found inT. harzianumand has fungicidal, antimicrobial and anti-inflammatory activities.1It is active against the plant pathogenic fungusP. ultimum(MIC = 60 ng/ml) and the parasiteT. brucei brucei(IC50= 90 ng/ml), but has no effect on the plant pathogenic fungiR. solani,P. omnivorum,T. basicola,R. arrhizus, andV. dahliaeor the bacteriaB. thuringiensis,P. fluorescens, andX. malvacearumwhen used at concentrations up to 1,000 ng/ml.2,3Gliovirin decrease...

天然产物

Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
Erythromycin
Cat.No: T1032
Synonym: 红霉素,E-Mycin
Target: ribosome, Antibacterial, Antibiotic
Ochromycinone
Cat.No: T6995
Synonym: STA 21,STA21,STA-21
Target: Antibacterial, STAT
Dimboa
Cat.No: T22308
Synonym: 2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布
Target: Others, Antibacterial, Antibiotic, Antifungal
Tioconazole
Cat.No: T0146
Synonym: UK-20349,Vagistat,噻康唑
Target: Antibiotic, Antifection, Antifungal
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Trimethoprim
Cat.No: T1153
Synonym: NIH 204,BW 56-72,甲氧苄啶,NSC-106568
Target: DHFR, DNA/RNA Synthesis, Antifolate, Antibacterial, Antibiotic
Lasalocid
Cat.No: T15717
Synonym: Lasalocid-A,Antibiotic X-537A,Ionophore X-537A
Target: Antibacterial
Azomycin
Cat.No: T6402
Synonym: 2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin
Target: Antibacterial, Antibiotic
JOSAMYCIN
Cat.No: T7148
Synonym: EN-141,交沙霉素
Target: Antibacterial, Antibiotic
Alamethicin
Cat.No: T10278
Synonym:
Target: Antibacterial
Lapachol
Cat.No: T4136
Synonym: Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin
Target: Others, Influenza Virus, Antibacterial, Parasite, Antifungal
SF2312
Cat.No: T28764
Synonym: SF-2312,SF 2312
Target: Glucokinase, Antibacterial
Neomycin sulfate
Cat.No: T0950
Synonym: Framycin sulfate,硫酸新霉素
Target: Phospholipase, ribosome, Antibacterial, Antibiotic
Vancomycin
Cat.No: T8641
Synonym:
Target: Antibacterial, Antibiotic, Autophagy
Kitasamycin tartrate
Cat.No: T20779
Synonym: Leucomycin tartrate
Target: Others
Tomaymycin
Cat.No: T75443
Synonym:
Target: Others
Dihydroaeruginoic Acid
Cat.No: TN7553
Synonym: CGP 52547
Target: Others
2-Aminoimidazole
Cat.No: T38241
Synonym:
Target: Others
Erythromycin thiocyanate
Cat.No: T11233
Synonym:
Target: Antibacterial
Magainin 1 TFA
Cat.No: T75753
Synonym:
Target: Others
Thiomarinol A
Cat.No: T73673
Synonym:
Target: Others
Gliovirin
Cat.No: T35741
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-00672 Azurocidin/CAP37 Protein, Human, Recombinant (His)

AZU,NAZC,azurocidin 1,hHBP,AZAMP,HUMAZUR,CAP37,HBP,AZU1

Human HEK293 Cells
Azurocidin (AZU1), also known as heparin-binding protein (HBP) or cationic antimicrobial protein 37 (CAP37), is an azurophil granule antibiotic protein, with monocyte chemotactic and antibacterial activity. The Azurophil granules, specialized lysosomes of the neutrophil, contain at least 10 proteins implicated in the killing of microorganisms. Azurocidin is a member of the serine protease family that includes Cathepsin G, neutrophil elastase (NE), and proteinase 3 (PR3), however, Azurocidin is n...

重组蛋白

Azurocidin/CAP37 Protein, Human, Recombinant (His)
Cat.No: TMPY-00672
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
T10306 Amoxicillin D4

Amoxycillin D4

Others Others
Amoxicillin D4 (Amoxycillin D4) is a deuterium-labeled Amoxicillin. Amoxicillin is an antibiotic with broad-spectrum antimicrobial activity.
TMIJ-0158 Sitafloxacin-d4

Sitafloxacin-d4 是 Sitafloxacin 的氘代化合物。Sitafloxacin 的 CAS 号为 127254-12-0。Sitafloxacin (Sitafloxacin anhydrous) 是一种具有口服活性的氟喹诺酮类抗生素,具有广谱的抗菌活性。Sitafloxacin 可用于研究呼吸道感染和尿路感染。

同位素标记化合物

Amoxicillin D4
Cat.No: T10306
Synonym: Amoxycillin D4
Target: Others
Sitafloxacin-d4
Cat.No: TMIJ-0158
Synonym:
Target:
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