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lesogaberan

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  • 抑制剂&激动剂
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    TargetMol | Inhibitors_Agonists
Lesogaberan
AZD-3355
T15737344413-67-8
Lesogaberan is an effective and selective GABAB receptor agonist (EC50: 8.6 nM for human recombinant GABAB receptors). For rat brain GABAB and GABAA receptors, the binding affinity (Kis) is 5.1 nM and 1.4 μM, respectively.
  • ¥ 10600
6-8周
规格
数量
Lesogaberan napadisylate
AZD-3355 napadisylate
T40572477956-38-0
Lesogaberan (AZD-3355) napadisylate is a potent and selective agonist of GABA B receptors, with an EC 50 of 8.6 nM for human recombinant GABA B receptors. It demonstrates an affinity (Ki) of 5.1 nM for rat GABA B receptors and 1.4 μM for GABA A receptors, as determined by its displacement of [3H]GABA binding in brain membranes. Notably, Lesogaberan napadisylate exerts a peripheral mode of action, inhibiting transient lower esophageal sphincter relaxation.
  • ¥ 10600
6-8周
规格
数量
Lesogaberan hydrochloride
AZD-3355 hydrochloride
T72215
Lesogaberan (AZD-3355) hydrochloride 是一种有效的选择性 GABAB 受体激动剂,对人重组 GABAB 受体的 EC50为 8.6 nM。通过脑膜中 [3H]GABA 结合位移测量,Lesogaberan hydrochloride 对大鼠 GABAB 和 GABAA 受体的亲和力 (Kis):分别为 5.1 nM 和 1.4 μM。Lesogaberan hydrochloride 通过外周作用模式抑制短暂的食管下括约肌松弛。
  • ¥ 3330
期货
规格
数量
AZD-3355
T68662805251-29-0
AZD-3355, also known as Lesogaberan, is a GABA(B)-receptor agonist reflux inhibitor.
  • ¥ 10600
6-8周
规格
数量