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kdm5c70

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  • 抑制剂&激动剂
    97
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    6
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    2
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    TargetMol | Natural_Products
Quilseconazole Formic acid(1340593-70-5 Free base)Quilseconazole Formic acid(1340593-70-5 Free base)
T16704L In house
Quilseconazole Formic acid 是真菌 Cyp51 的选择性抑制剂,对新型隐球菌和格特隐球菌具有有效活性。
  • ¥ 1530
现货
规格
数量
TargetMol | Inhibitor Sale
C3a 70-77 2TFA(63555-63-5(free base))Complement 3a (70-77)
T7497L
C3a 70-77 2TFA(63555-63-5(free base)) (Complement 3a (70-77)) 是对应于 C3a 的 COOH 末端的八肽。
  • ¥ 479
现货
规格
数量
TargetMol | Inhibitor Sale
5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE5-乙基-4,5,6,7-四氢-噻唑并[5,4-C]吡啶-2-胺
T891217899-49-9
5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE 靶向 PLK1。
  • ¥ 281
现货
规格
数量
TargetMol | Inhibitor Sale
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide
T9944246238-55-1In house
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide抑制多药耐药蛋白(MRP1)。
  • ¥ 774
现货
规格
数量
TargetMol | Inhibitor Sale
KDM5-C70
T156481596348-32-1
KDM5-C70 是 KDM5-C49 的乙酯衍生物,是一种有效的细胞渗透性泛 KDM5 组蛋白去甲基化酶抑制剂。它在骨髓瘤细胞中具有抗增殖作用,可诱导全基因组 H3K4me3 水平升高。
  • ¥ 245
现货
规格
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TargetMol | Citations 客户已引用
5’-O-Benzoyl-2’-O,4’-C-methyleneuridine
TNU1577293751-31-2
5'-O-Benzoyl-2'-O,4'-C-methyleneuridine is a Nucleoside Derivative - LNA related nucleoside; Protected nucleoside with NH2/OH open.
  • 询价
5日内发货
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5’-O-Benzoyl-3’-O-(4-methoxybenzoyl)-2’-O,4’-C-methyleneuridine
TNU1249
5'-O-Benzoyl-3'-O-(4-methoxybenzoyl)-2'-O,4'-C-methyleneuridine is a Nucleoside Derivative - LNA-related nucleoside.
  • 询价
5日内发货
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5’(R)-C-Methyl-N6-methyladenosine
TNU0409
Nucleoside Derivatives - 5’-Modified nucleosides; 6-Modified purine nucleosides; N-Methylated nucleosides
  • 询价
5日内发货
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5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride
T66095720720-96-7
5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66095,CAS号为 720720-96-7。
  • 询价
5日内发货
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5’(R)-C-Methyl-5-fluorouridine
T75079
5’(R)-C-Methyl-5-fluorouridine 是尿嘧啶核苷类似物,具有潜在抗癫痫能力。该类似物用于研究抗惊厥和抗焦虑活性,进而开发新型降压药物。
  • 询价
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5-Hydroxymethyl-2’-C-methyluridine
TNU03322305415-92-1
Nucleoside Derivatives - 2’-Modified nucleosides, 5-Modified pyrimidine nucleosides
  • 询价
5日内发货
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2’-C-methyl-5-fluorouriddine
TNU013823643-38-1
Nucleosides and Reagents - Fluoro-modified nucleoside; 2’-C-methyl nucleoside; ; 5-Modified pyrimidine nucleoside
  • 询价
5日内发货
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1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one
TNU08002072145-17-4
1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one is a Pyridine nucleoside; 2'-C-Methyl nucleoside.
  • 询价
5日内发货
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5’(R)-C-Methylguanosine
TNU026185421-89-2
5'(R)-C-Methylguanosine is a Nucleoside Derivative - 5'-Modified nucleoside.
  • 询价
5日内发货
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2’-C-Methyl-5-methyluridine
TNU0144119410-84-3
2'-C-Methyl-5-methyluridine is a 2'-C-Methyl nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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Rev 2’-O-MOE-C(Bz)-5’-amidite; N4-Benzoyl-3'-O-(4,4’-dimethoxy trityl)-2'-O-(2-methoxyethyl)cytidine-5’-CED phosphoramidite
TNU1531
Rev 2’-O-MOE-C(Bz)-5’-amidite; N4-Benzoyl-3'-O-(4,4’-dimethoxy trityl)-2'-O-(2-methoxyethyl)cytidine-5’-CED phosphoramidite 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU1531。
  • 询价
5日内发货
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Dichloro[1,3-bis(2,4,6-trimethylphenyl)-2-imidazolidinylidene][[5-[(dimethylamino)sulfonyl]-2-(1-methylethoxy-O)phenyl]methylene-C]ruthenium(II)
T66135918870-76-5
Dichloro[1,3-bis(2,4,6-trimethylphenyl)-2-imidazolidinylidene][[5-[(dimethylamino)sulfonyl]-2-(1-methylethoxy-O)phenyl]methylene-C]ruthenium(II) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T66135。
  • 询价
5日内发货
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2-Bromo-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine
FL0118143150-92-9
2-Bromo-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine 是一种片段分子,在生命科学相关研究中具有广泛的应用。
  • ¥ 285
现货
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5’(R)-C-Methyluridine
TNU021372159-54-7
5'(R)-C-Methyluridine is a Nucleoside Derivative - 5'-Modified nucleoside.
  • 询价
5日内发货
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2’,3’,5’-Tri-O-benzoyl-2’-C-methyl-5-methyluridine
TNU0836957535-53-4
2',3',5'-Tri-O-benzoyl-2'-C-methyl-5-methyluridine is a 2'-C-Methyl nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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N-Trityl-N4-benzoyl-morpholino-C-5’-O-phosphoramidite
TNU1469
N-Trityl-N4-benzoyl-morpholino-C-5'-O-phosphoramidite is a Nucleoside Derivative - Morpholino nucleoside; Phosphoramidite.
  • 询价
5日内发货
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5-O-Benzoyl-1,2,3-tri-O-acetyl-4-C-fluoromethyl-D-ribofuranose
TNU1197
5-O-Benzoyl-1,2,3-tri-O-acetyl-4-C-fluoromethyl-D-ribofuranose is a Carbohydrate Derivative.
  • 询价
5日内发货
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5’(R)-C-Methyl-5-methyluridine
TNU0215129745-35-3
Nucleoside Derivatives - 5’-Modified nucleosides, 5-Modified pyrimidine nucleosides
  • 询价
5日内发货
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5-O-Benzoyl-1,2,3-tri-O-acetyl-4-C-methyl-D-ribofuranose
TNU1196503543-44-0
5-O-Benzoyl-1,2,3-tri-O-acetyl-4-C-methyl-D-ribofuranose is a Carbohydrate Derivative.
  • 询价
5日内发货
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tert-Butyl 4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate
T663741280210-79-8
tert-Butyl 4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66374,CAS号为 1280210-79-8。
  • 询价
5日内发货
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2’-C-Methyl-5-methoxyuridine
TNU01452072145-45-8
2'-C-Methyl-5-methoxyuridine is a 2'-C-Methyl nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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Rev 2’-O-MOE-C(Bz)-5’-amidite
T75206
Rev 2’-O-MOE-C(Bz)-5’-amidite 是一种具有广泛抗肿瘤活性的嘌呤核苷类似物,主要针对惰性淋巴系统恶性肿瘤。其抗癌机制包括抑制 DNA 合成和诱导细胞凋亡 (apoptosis)。
  • 询价
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5’-O-Benzoyl-3’-O-(4-methoxybenzyl)-2’-O,4’-C-methyleneuridine
T75186
5’-O-Benzoyl-3’-O-(4-methoxybenzyl)-2’-O,4’-C-methyleneuridine 是一种具有广泛抗肿瘤活性的嘌呤核苷类似物,主要针对惰性淋巴系统的恶性肿瘤。其作用机制主要通过抑制 DNA 合成和诱导细胞凋亡 (apoptosis) 实现。
  • 询价
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5-Chloro-3-phenylbenzo[c]isoxazole
T66589719-64-2
5-Chloro-3-phenylbenzo[c]isoxazole 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66589,CAS号为 719-64-2。
  • 询价
5日内发货
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5-Iodo-2’-C-methyl uridine
TNU00931203461-96-4
5-Iodo-2'-C-methyl uridine is a 2'-C-Methyl nucleoside; Halo-nucleoside.
  • 询价
5日内发货
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5-O-Benzoyl-4-C-hydroxymethyl-2,3-O-isopropylidene-1-O-methyl-beta-D-ribofuranose
TNU1195327614-69-7
5-O-Benzoyl-4-C-hydroxymethyl-2,3-O-isopropylidene-1-O-methyl-beta-D-ribofuranose is a Carbohydrate Derivative.
  • 询价
5日内发货
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5’(R)-C-Methyl-3-deazauridine
TNU02602305415-82-9
Nucleoside Derivatives - 5’-Modified nucleosides; 3-Deazauridines
  • 询价
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2’,3’,5’-Tri-O-benzoyl-2’-C-methyl-5-methoxyuridine
TNU08372072145-79-8
2',3',5'-Tri-O-benzoyl-2'-C-methyl-5-methoxyuridine is a 2'-C-Methyl nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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5-Methyl-2’-O,4’-C-methylenecytidine
TNU0414847650-87-7
5-Methyl-2'-O,4'-C-methylenecytidine is a Nucleoside Derivative - LNA-related nucleoside.
  • ¥ 138
5日内发货
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2’,3’,5’-Tri-O-(t-butyldimethylsilyl)-4’-C-hydroxymethyl uridine
TNU0949232588-97-5
Nucleoside Derivative –4’-Modified nucleosides; Protected nucleosides with NH2 OH group
  • 询价
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3’-beta-C-Methyl-5-methyluridine
TNU0380934002-35-4
3'-beta-C-Methyl-5-methyluridine is a Nucleoside Derivative - 3'-Modified nucleoside.
  • 询价
5日内发货
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7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine
T355341032570-74-3
7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine is a building block.1It has been used in the synthesis of PI3K inhibitors. 1.Scott, W.J., Hentemann, M.F., Rowley, R.B., et al.Discovery and SAR of novel 2,3-dihydroimidazo[1,2-c]quinazoline PI3K inhibitors: Identification of copanlisib (BAY 80-6946)ChemMedChem.11(14)1517-1530(2016)
  • ¥ 560
35日内发货
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4’-C-Methyl-5-methylcytidine
TNU0402764644-12-4
4'-C-Methyl-5-methylcytidine is a Nucleoside Derivative - 4'-Modified nucleoside.
  • 询价
5日内发货
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5-Fluoro-4’-C-methyluridine
TNU0400660845-69-2
5-Fluoro-4'-C-methyluridine is a Nucleoside Derivative - 4'-Modified nucleoside; Fluoro-modified nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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2’-beta-C-Ethynyl-5-methyluridine
TNU1500
2'-beta-C-Ethynyl-5-methyluridine is a Nucleoside Derivative - 2'-Modified nucleoside.
  • 询价
5日内发货
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5-Amino-2-(2-furanyl)-7H-pyrazolo[4,3-e][1,2,4]   triazolo[1,5-c] pyrimidine
TNU1219162401-16-3
Scaffolds and Templates; Heterocyclic Compounds - Fused polyheterocycles
  • 询价
5日内发货
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5-Fluoro-3’-beta-C-methyluridine
TNU1489
5-Fluoro-3'-beta-C-methyluridine is a Nucleoside Derivative - 3'-Modified nucleoside, 5-Modified pyrimidine nucleoside, Fluoro-modified nucleoside.
  • 询价
5日内发货
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1-(2,3,5-Tribenzoyl-2-C-b-methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one
TNU07992072145-38-9
1-(2,3,5-Tribenzoyl-2-C-b-methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one is a Pyridine nucleoside; 2'-C-Methyl nucleoside.
  • 询价
5日内发货
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3’-Deoxy-3’-a-C-methyl-5-fluorouridine
TNU022137731-67-2
3'-Deoxy-3'-a-C-methyl-5-fluorouridine is a Nucleoside Derivative - 3'-Modified nucleoside, 5-Modified pyrimidine nucleoside, Fluoro-modified nucleoside.
  • 询价
5日内发货
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Cathepsin C-IN-5
T624942825567-97-1
CathepsinC-IN-5 (compound SF38) 为一高效、选择性、口服活性的组织蛋白酶 C (Cat C) 抑制剂,其针对Cat C、Cat L、Cat S、Cat B、Cat K 的IC50s 分别为 59.9 nM、4.26 µM、>5 µM、>5 µM、>5 µM。该化合物能够抑制骨髓和血液中的Cat C活性,降低中性粒细胞丝氨酸蛋白酶(NSP)的激活,并展现抗炎活性。
  • ¥ 8620
10-14周
规格
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6-(2-O-Methyl-beta-D-ribofuranosyl)-3-(2-oxo-propyl)-6H-imidazo[1,2-c]pyrimidin-5-one
TNU00052095417-54-0
Nucleoside Derivatives - 2’-Modified nucleosides; Scaffolds and Templates;Bi-Tricyclic nucleosides
  • 询价
5日内发货
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2’,3’,5’-Tri-O-benzoyl-2’-C-methyl-5-fluorouriddine
TNU08292072145-49-2
2',3',5'-Tri-O-benzoyl-2'-C-methyl-5-fluorouriddine is a Fluoro-modified nucleoside; 2'-C-methyl nucleoside; 5-Modified pyrimidine nucleoside.
  • 询价
5日内发货
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3’-beta-C-Ethynyl-5-methyluridine
TNU0481180300-52-1
Nucleoside Derivatives - 3’-Modified purine nucleosides
  • 询价
5日内发货
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