Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6759L |
AP-III-a4 hydrochloride (1177827-73-4 free base)
ENOblock hydrochloride,AP-III-a4 hydrochloride |
Others | Others |
AP-III-a4 hydrochloride (ENOblock hydrochloride) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo. IC50 value: 0.576 uM [1] | |||
T6759 |
AP-III-a4
ENOblock |
Glucokinase | Metabolism |
AP-III-a4 (ENOblock) 是第一个非底物类似物,可直接与烯醇酶结合,IC50=0.576 uM,可阻碍体内癌细胞转移。 |