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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22367 |
Methylprednisolone succinate
Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate,甲基泼尼松龙琥珀酸酯 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Methylprednisolone succinate (Methylprednisolone hemisuccinate) 是合成的糖皮质激素,常用作抗炎剂。 | |||
T0294 |
6α-Methylprednisolone 21-hemisuccinate sodium salt
Asmacortone,Methylprodnisolone Sodium Succinate,甲强龙琥珀酸钠,Metypresol,Methylprednisolone sodium succinate,Corticel,6-Methylprednisolone succinate sodium |
Glucocorticoid Receptor; Glucagon Receptor | Endocrinology/Hormones; GPCR/G Protein |
6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone) 是一种糖皮质激素,是一种有效的抗炎剂,半衰期比 Prednisolone 长。 | |||
T1171L |
Methylprednisolone Aceponate
MPA,SH 440,SH-440,SH440,Advantan,醋丙甲泼尼龙 |
Others | Others |
Methylprednisolone Aceponate (SH 440) 是一种非卤化皮质类固醇,是一种有效的抗炎剂。 | |||
T21338 |
Methylprednisolone Acetate
Depo-Medrate,Depometicort,Depo-Medrin,Depo-medrol,Depomedrone,Lemod |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Methylprednisolone Acetate(Depo-Medrate) 具有抑制氧自由基的能力,可用于治疗急性脊髓损伤。 | |||
T9047 |
Fluprednisolone
NSC-47439,NSC 47439,氟泼尼龙,NSC47439 |
Others | Others |
Fluprednisolone (NSC-47439) 是一种合成糖皮质激素,具有抗炎特性。 | |||
T37763 |
BTD
|
Others | Others |
Selective TRPC5 activator (EC50 = 1.4 μM in a calcium influx assay, 1.3 μM in whole cell patch clamp assay). Displays >14.5-fold selectivity for TRPC5 over other TRP channels (EC50 = 20.6 μM for TRPM8). Also activates TRPC1:5 and TRPC4:5 heteromers. Beckmann et al (2017) A benzothiadiazine derivative and methylprednisolone are novel and selective activators of transient receptor potential canonical 5 (TRPC5) channels. Cell Calcium. 66 10 PMID:28807145 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMID-0146 |
Methylprednisolone-d7
|
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Methylprednisolone-d7 是 Methylprednisolone 的氘代化合物。Methylprednisolone 的 CAS 号为 83-43-2。Methylprednisolone 是一种具有类似抗炎作用的强的松龙衍生物。它是皮质类固醇,可作用于糖皮质激素受体。它通过激活ACE2并降低 IL-6 水平来改善严重的COVID-19。 | |||
TMID-0145 |
Methylprednisolone-d2
|
||
Methylprednisolone-d2 是 Methylprednisolone 的氘代化合物。Methylprednisolone 的 CAS 号为 83-43-2。Methylprednisolone 是一种具有类似抗炎作用的强的松龙衍生物。它是皮质类固醇,可作用于糖皮质激素受体。它通过激活ACE2并降低 IL-6 水平来改善严重的COVID-19。 |