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  • 抑制剂&激动剂
    228
    TargetMol | Inhibitors_Agonists
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    9
    TargetMol | Recombinant_Protein
  • 多肽产品
    15
    TargetMol | Peptide_Products
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    3
    TargetMol | PROTAC
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    64
    TargetMol | Natural_Products
1-beta-D-Arabinofuranosyluracil阿糖尿苷,1-β-D-阿糖尿苷,Uracil 1-β-D-arabinofuranoside
T59793083-77-0
1-beta-D-Arabinofuranosyluracil (Uracil 1-β-D-arabinofuranoside) 是一种甲氧基腺苷衍生物,从加勒比海绵 Tectitethya crypta 中分离得到。已经证明其具有多种生物活性,如抗炎活性,缓解疼痛和血管舒张特性。它能够抑制小鼠淋巴瘤细胞的增殖。
  • ¥ 129
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1-(2-Deoxy-2-fluoro-beta-D-arabinofuranosyl)uracil
TNU001469123-94-0
1-(2-Deoxy-2-fluoro-beta-D-arabinofuranosyl)uracil is a Nucleoside, fluoro-modified nucleoside; Arabino-nucleosidde.
  • ¥ 366
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1-{1H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine 2HCl
T50034853680-06-5
1-{1H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine dihydrochloride (1-PPZ-DHC)是一种用作分子结构单元的化合物。它是天然产物哌嗪的类似物,具有广泛的生物活性,包括抗炎、抗肿瘤和抗菌活性,同时还被研究用于治疗神经系统疾病,如阿尔茨海默氏症和帕金森氏症。
  • ¥ 325
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TargetMol | Inhibitor Sale
Kaempferol-3-O-β-D-glucosyl(1-2)rhamnoside
TN6719142451-65-8
Kaempferol-3-O-β-D-glucosyl(1-2)rhamnoside 是一种从阿拉伯茉莉中分离出来的天然产物。
  • ¥ 2350
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D-JNKI-1 acetateD-JNKI-1 acetate(1445179-97-4 Free base),AM-111 acetate
T10937L
D-JNKI-1 acetate (AM-111 acetate) 是一种高效的细胞渗透性 JNK 肽抑制剂。
  • ¥ 1310
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2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv
T34383L144459-71-2In house
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv在Sprague Dawley大鼠上进行测试时显示出高局部抗炎效力和高肺选择性。
  • ¥ 1300
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(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol
TN7029
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol 是一种有用的研究化合物,适用于许多研究应用,包括化学领域和生命科学领域等。
  • ¥ 1050
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1-beta-D-ArabinofuranosylthymineThymine 1-β-D-arabinofuranoside,阿糖胸苷,Spongothymidine
TNU0352605-23-2
1-beta-D-Arabinofuranosylthymine (Thymine 1-β-D-arabinofuranoside) is a purine nucleoside analog. Purine nucleoside analogs have a broad spectrum of antitumor activity, targeting inert lymphoid malignancies and inducing apoptosis.1-beta-D-Arabinofuranosylthymine's anticancer mechanism is dependent on the inhibition of DNA synthesis.1-beta-D-Arabinofuranosylthymine is a purine nucleoside analog.
  • ¥ 743
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3-(2,6-dichlorophenyl)-1-methyl-7-(methylsulfanyl)-1H,2H,3H,4H-pyrimido[4,5-d][1,3]diazin-4-one
T501021799561-19-5
3-(2,6-dichlorophenyl)-1-methyl-7-(methylsulfanyl)-1H,2H,3H,4H-pyrimido[4,5-d][1,3]diazin-4-one 是一种化合物,已被广泛研究用于治疗各种疾病,包括肿瘤、阿尔茨海默症和帕金森病、抗炎药和镇痛剂。
  • ¥ 865
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(25R)-3β,17α-dihydroxy-5α- spirostan-6-one3-O-α-L- rhamnopyranosyl-(1→2)-β- D-glucopyranoside卷丹皂苷
TN7112143051-94-9
(25R)-3β,17α-dihydroxy-5α- spirostan-6-one3-O-α-L- rhamnopyranosyl-(1→2)-β- D-glucopyranoside 是从百合 Lilium brownii var. viridulum 茎中分离得到的天然产物
  • ¥ 780
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1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3,2-d]pyrimidin-2-yl)phenyl)-3-(pyridin-4-yl)urea
T677001144075-47-7In house
1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3,2-d]pyrimidin-2-yl)phenyl)-3-(pyridin-4-yl)urea 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67700,CAS号为 1144075-47-7。
    8-10周
    询价
    Complement factor D-IN-1
    T168981386455-76-0
    Complement factor D-IN-1 is an effective and selective small-molecule reversible factor d inhibitor (IC50s: 0.006 and 0.05 μM in FD Thioesterolytic Fluorescent Assay and a MAC Deposition Assay, respectively).
    • ¥ 3190
    5日内发货
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    TargetMol | Citations 客户已引用
    (-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside(-)-丁香树脂酚-4-O-beta-D-呋喃芹糖基-(1→2)-beta-D-吡喃葡萄糖苷,(-)-Syringaresnol-4-O-beta-D-apiofuranos
    T5S0483136997-64-3
    (-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside ((-)-Syringaresnol-4-O-beta-D-apiofuranos) 是从Albizzia myriophylla 的树皮部分分离得到。
    • ¥ 168
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    TargetMol | Inhibitor Sale
    Genipin 1-β-D-gentiobiosideGenipin 1-β-gentiobioside,Genipin gentiobioside,genipin-1-b-D-gentiobioside,京尼平-1-Β-D-龙胆双糖苷,Genipin 1-gentiobioside,京尼平龙胆双糖苷
    T4S229929307-60-6
    Genipin 1-β-D-gentiobioside 是栀子中丰富和具有生物活性的一种环烯醚萜苷,具有保肝,抗氧化,抗炎和抗血栓形成作用。
    • ¥ 169
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    TargetMol | Inhibitor Sale
    Emodin-1-O-β-D-glucopyranoside大黄素-1-O-Β-D-吡喃葡萄糖苷,大黄素-1-O-β-D-葡萄糖苷,Emodin-1-O-glucoside
    T2S038938840-23-2
    Emodin-1-O-β-D-glucopyranoside (Emodin-1-O-glucoside) 是一种非竞争性细菌神经氨酸酶抑制剂,IC50为 0.85 μM,提取自药用植物虎杖中。
    • ¥ 548
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    TargetMol | Inhibitor Sale
    3-O-α-L-Rhamnopyranosyl-(1→2)-α-L-arabinopyranosyl hederagenin28-O-β-D-xylopyranosyl-(1→6)-β-D-glucopyranosyl ester
    T83345128717-92-0
    3-O-α-L-Rhamnopyranosyl-(1→2)-α-L-arabinopyranosyl hederagenin 28-O-β-D-xylopyranosyl-(1→6)-β-D-glucopyranosyl ester 是一种皂苷化合物,具备抗肿瘤与抗炎特性。
    • 询价
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    Benzyl [5-O-benzoyl-β-D-apiofuranosyl(1→2)]-β-D-glucopyranoside
    TN57411097040-08-8
    Benzyl [5-O-benzoyl-β-D-apiofuranosyl(1→2)]-β-D-glucopyranoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5741,CAS号为 1097040-08-8。
    • ¥ 4040
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    Kaempferol-3-O-α-L-rhamnopyranosyl-(1→6)-β-D-glucopyranosyl-(1→2)-β-D-glucopyranosideKaempferol-3-O-α-L-rhamnopyranosyl-(1->6)-β-D-glucopyranosyl-(1->2)-β-D-glucopyranoside
    TN6460476617-49-9
    Kaempferol-3-O-α-L-rhamnopyranosyl-(1→6)-β-D-glucopyranosyl-(1→2)-β-D-glucopyranoside shows antioxidant activity.
    • ¥ 3420
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    1-(3',5'-dimethoxy)phenyl-2-[4''-O-beta-D-glucopyranosyl (6->1)-O-alpha-L-rhamnopyranosyl]phenylethane
    TN63991338076-61-1
    1-(3',5'-dimethoxy)phenyl-2-[4''-O-β-D-glucopyranosyl (6→1)-O-α-L-rhamnopyranosyl]phenylethane showed cytotoxic activities to Hela and hep2 cell lines.
    • ¥ 2350
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    (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
    T76631103613-84-9
    (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078) 是一种稳定的 Dynorphin A (1-8) 类似物,是 kappa 阿片受体 (KOR) 激动剂。
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    4-Amino-1-(b-D-ribofuranosyl)-7H-pyrrolo[2.3-d]pyrimidine-5-carboxamide
    TNU0272
    Nucleoside Derivatives - 7-Deaza-purine nucleosides; Natural product; inhibitor of protein kinase C 蛋白激酶抑制剂
    • 询价
    5日内发货
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    4,6-Diamino-3-iodo-1-(b-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
    TNU0283908143-13-5
    Nucleoside Derivatives - 8-Aza-7-deaza purine nucleosides, Halo-nucleosides
    • 询价
    5日内发货
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    1-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine
    TNU03872389988-22-9
    Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosides
    • 询价
    5日内发货
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    1-(Piperidin-4-yl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-2(3H)-one
    T66378
    1-(Piperidin-4-yl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-2(3H)-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T66378。
    • 询价
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    1-(((Cyclohexyloxy)carbonyl)oxy)ethyl 2-ethoxy-1-((2'-(1-trityl-1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl)methyl)-1H-benzo[d]imidazole-7-carboxylate
    T65490170791-09-0
    1-(((Cyclohexyloxy)carbonyl)oxy)ethyl 2-ethoxy-1-((2'-(1-trityl-1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl)methyl)-1H-benzo[d]imidazole-7-carboxylate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65490,CAS号为 170791-09-0。
    • 询价
    5日内发货
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    1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine
    TNU03852389988-20-7
    1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside; Amino nucleoside.
    • 询价
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    α-D-Glucose-1-phosphate (sodium salt hydrate)
    T35416150399-99-8
    α-D-Glucose-1-phosphate is an intermediate in glycogen metabolism.1,2It is a precursor in the biosynthesis of UDP-glucose, the glucose donor in glycogen biosynthesis.2α-D-Glucose-1-phosphate can be formed during glycogen breakdownviaphosphorolytic cleavage of glycogen by glycogen phosphorylase.1It can be converted to glucose-6-phosphate by phosphoglucomutase. α-D-Glucose-1-phosphate is combined with CTP by α-D-glucose-1-phosphate cytidylyltransferase to form CDP-glucose in the first step of CDP-D-tyvelose biosynthesis inS. typhi.3Bacterial sucrose phosphorylase converts sucrose and phosphate into D-fructose and α-D-glucose-1-phosphate.4 1.Berg, J.M., Tymoczko, J.L., and Stryer, L.Glycogen breakdown requires the interplay of several enzymesBiochemistry(2002) 2.Berg, J.M., Tymoczko, J.L., and Stryer, L.Glycogen is synthesized and degraded by different pathwaysBiochemistry(2002) 3.Koropatkin, N.M., and Holden, H.M.Molecular structure of ɑ-D-glucose-1-phosphate cytidylyltransferase from Salmonella typhiJ. Biol. Chem.279(42)44023-44029(2004) 4.Goedl, C., Schwarz, A., Minani, A., et al.Recombinant sucrose phosphorylase from Leuconostoc mesenteroides: Characterization, kinetic studies of transglucosylation, and application of immobilised enzyme for production of ɑ-D-glucose 1-phosphateJ. Biotechnol.129(1)77-86(2007)
    • ¥ 875
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    6-Amino-3-iodo-4-methoxy-1-(b-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
    TNU02811997362-11-4
    Nucleoside Derivatives - 7-Deaza-8-aza purine nucleosides; Halo-nucleosides; 6-Modified purine nucleosides
    • 询价
    5日内发货
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    2-(((6-(Difluoromethoxy)-1H-benzo[d]imidazol-2-yl)sulfonyl)methyl)-3,4-dimethoxypyridine 1-oxide
    T67420953787-55-8
    2-(((6-(Difluoromethoxy)-1H-benzo[d]imidazol-2-yl)sulfonyl)methyl)-3,4-dimethoxypyridine 1-oxide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67420,CAS号为 953787-55-8。
    • 询价
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    N4-Benzoyl-1-(6-O-DMTr-2,3-dideoxy-beta-D-erythro-hexopyranosyl)cytosine
    TNU1623145594-00-9
    N4-Benzoyl-1-(6-O-DMTr-2,3-dideoxy-beta-D-erythro-hexopyranosyl)cytosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1623,CAS号为 145594-00-9。
    • 询价
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    N-Acetyl-α-D-glucosamine 1-phosphate disodium
    T7454931281-59-1
    N-acetyl-α-d-glucosamine 1-phosphate disodium (GlcNAc-1-P) 为异位糖磷酸盐,关键中间体于N-糖蛋白生物合成。该化合物同时作为细菌细胞壁组分磷胆酸和鼠胺的代谢前体。
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    6-Amino-4-methoxy-1-(2-deoxy-β-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
    T75185100644-69-7
    6-Amino-4-methoxy-1-(2-deoxy-β-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine 是一种嘧啶核苷类似物,以其广泛的生化功能和抗癌活性著称,其机制涉及DNA合成抑制、RNA合成抑制、抗病毒和免疫调节等多方面。
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    5-Phospho-D-ribose 1-diphosphate (sodium salt hydrate)
    T36973
    5-Phospho-D-ribose 1-diphosphate (PRPP) is a natural intermediate involved in the pentose phosphate pathway leading to purine, pyrimidine, and histidine metabolism. It is also an intermediate in the synthesis of plant hormones, alkaloids, and other secondary metabolites from glucose. Several phosphoribosyltransferases (PRTases) use PRPP as a substrate to add a 5-phosphoribosyl group to another substrate, as in the production of adenosine monophosphate from adenine and PRPP by adenine PRTase. N/A
    • ¥ 1078
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    5-((4-Bromo-2-chlorophenyl)amino)-4-fluoro-1-methyl-1H-benzo[d]imidazole-6-carboxylic acid
    T66323606144-04-1
    5-((4-Bromo-2-chlorophenyl)amino)-4-fluoro-1-methyl-1H-benzo[d]imidazole-6-carboxylic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66323,CAS号为 606144-04-1。
    • 询价
    5日内发货
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    L-Borneol 7-O-[β-D-apiofuranosyl-(1→6)]-β-D-glucopyranosideFT-0775891,Borneol 7-O-[beta-D-apiofuranosyl-(1->6)]-beta-D-glucopyranoside,龙脑 7-O-[Β-D-呋喃芹菜糖基-(1→6)]-Β-D-吡喃葡萄糖苷
    TN144788700-35-0
    Borneol 7-O-[beta-D-apiofuranosyl-(1->6)]-beta-D-glucopyranoside is a natural product from Radix ophiopogonis.
    • ¥ 1520
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    Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside3-O-{2-O-[6-O-(P羟基-反-香豆酰)-葡萄糖基]-鼠李糖基}槲皮素,Quercetin 3-O-beta-(6''-p-coumaroyl)glucopyranosyl(1->2)-alpha-L-rhamnopyranoside
    TN2125143061-65-8
    Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside (Quercetin 3-O-beta-(6''-p-coumaroyl)glucopyranosyl(1->2)-alpha-L-rhamnopyranoside) 是一种从银杏叶中提取出来的化合物。Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside 具有抗氧化的功能。
    • ¥ 894
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    1-b-D-(3-Methoxy naphthalen-2-yl)-2’-deoxyriboside; 1,4-Anhydro-2-deoxy-1-C-(3-methoxy)-naphthalenyl)-D-erythro-pentitol
    TNU16411117893-19-2
    1-b-D-(3-Methoxy naphthalen-2-yl)-2’-deoxyriboside; 1,4-Anhydro-2-deoxy-1-C-(3-methoxy)-naphthalenyl)-D-erythro-pentitol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1641,CAS号为 1117893-19-2。
    • 询价
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    1-(b-D-Xylofuranosyl)-N6-(p-methoxybenzyl)   adenine
    TNU1485
    1-(b-D-Xylofuranosyl)-N6-(p-methoxybenzyl) adenine is a Nucleoside Derivative - Xylo-nucleoside, 6-Modified purine nucleoside.
    • 询价
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    1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one
    TNU08002072145-17-4
    1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one is a Pyridine nucleoside; 2'-C-Methyl nucleoside.
    • 询价
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    5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine
    T644371265884-98-7
    5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64437。
    • 询价
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    1-(b-D-Xylofuranosyl)-N6-(m-trifluoromethyl   benzyl) adenine
    TNU0524
    1-(b-D-Xylofuranosyl)-N6-(m-trifluoromethyl benzyl) adenine is a Nucleoside Derivative - Xylo-nucleoside, 6-Modified purine nucleoside, Fluoro-modified nucleoside.
    • 询价
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    1-thio-β-D-Glucose Tetraacetate
    T3728519879-84-6
    1-thio-β-D-Glucose tetraacetate is a building block.1,2It has been used in the synthesis of aromatic glucosinolates with anti-inflammatory activity, as well as glucosylated poly(pentafluorostyrene) derivatives for coating magnetic iron oxide nanoparticles. 1.Vo, Q.V., Trenerry, C., Rochfort, S., et al.Synthesis and anti-inflammatory activity of aromatic glucosinolatesBioorg. Med. Chem.21(19)5945-5954(2013) 2.Babiuch, K., Wyrwa, R., Wagner, K., et al.Functionalized, biocompatible coating for superparamagnetic nanoparticles by controlled polymerization of a thioglycosidic monomerBiomacromolecules12(3)681-691(2011)
    • ¥ 560
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    Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside麦冬苷元-3-O-Α-L-吡喃鼠李糖基(1→2)-Β-D-吡喃葡萄糖苷,Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside
    T3S1250128502-94-3
    Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside (Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside) 是一种从麦冬根中取得的萜类糖苷,对心血管系统有良好的药理作用。
    • ¥ 1650
    现货
    规格
    数量
    TargetMol | Inhibitor Sale
    1-[(5E)-3-O-[(Bis-di-isopropyl   amino)(2-cyanoethoxy) phosphino]-5,6-dideoxy-6-(diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hex-5-enofuranosyl]-5-methyluracil
    TNU12891345562-47-1
    1-[(5E)-3-O-[(Bis-di-isopropyl amino)(2-cyanoethoxy) phosphino]-5,6-dideoxy-6-(diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hex-5-enofuranosyl]-5-methyluracil is a Nucleoside Phosphoramidite; Nucleoside Derivative - Phosphorus-containing nucleotide; 5'-Modified nucleoside.
    • 询价
    5日内发货
    规格
    数量
    1-[6-Phosphono-2-O-methyl-β-D-ribo-hexofuranosyl]uracil
    TNU10122095417-68-6
    1-[6-Phosphono-2-O-methyl-β-D-ribo-hexofuranosyl]uracil is a Nucleoside Derivative - Phosphorus-containing nucleotide; 2'-Modified nucleoside; 5'-Modified nucleoside; 2'-Modified nucleoside.
    • 询价
    5日内发货
    规格
    数量
    1-(b-D-Xylofuranosyl)-2-thiouracil
    TNU03712305416-17-3
    Nucleoside Derivatives - Xylo-nucleosides, Thio-nucleosides
    • 询价
    5日内发货
    规格
    数量
    1,4-Dihydroxy-2-carbomethoxy-3-prenylnaphthalene-1-O-β-D-glucopyranoside1,4-Dihydroxy-2-carbomethoxy-3-prenylnaphthalene-1-O-beta-glucopyranoside
    TN11691415729-43-9
    1,4-Dihydroxy-2-carbomethoxy-3-prenylnaphthalene-1-O-beta-glucopyranoside may have DNA topoisomerases I and II inhibitory activity and cytotoxicity.
    • ¥ 2100
    期货
    规格
    数量
    2,4,6-Trichlorol-3-methyl-5-methoxy-phenol 1-O-β-d-glucopyranosyl-(1 → 6)-β-d-glucopyranoside
    T389291447969-66-5
    2,4,6-Trichlorol-3-methyl-5-methoxy-phenol 1-O-β-d-glucopyranosyl-(1 → 6)-β-d-glucopyranoside is a chlorophenyl glycoside that is commonly found in the bulbs of Lilium brownie var. viridulum. This compound has been observed to exhibit a weak inhibition of NO production in LPS-stimulated RAW 264.7 cells.
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    数量