4
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0272 |
Nilutamide
尼鲁米特,RU23908 |
Androgen Receptor | Endocrinology/Hormones |
Nilutamide (RU23908) 是一种非甾体抗雄激素药物,有用于转移性前列腺癌的潜力。 | |||
T15507 |
Hycanthone
Etrenol(mesylate),Win 249-33,海恩酮 |
DNA/RNA Synthesis; Topoisomerase; Parasite | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Hycanthone (Etrenol(mesylate)) 是 Lucanthone 的生物活性代谢产物,是一种抗血吸虫病药。它是一个噻吨酮类 DNA 嵌入剂,可抑制 RNA 合成以及 DNA 拓扑异构酶 I 和 II。它通过直接蛋白质结合来抑制核酸生物合成并抑制嘌呤内切核酸酶1,KD 为 10 nM。 | |||
T28555 |
Ro 13-3978
Ro-13-3978,Ro-133978,Ro13-3978,Ro133978 |
Others | Others |
RO13-3978 is a broad-spectrum antischistosomal. Ro 13-3978 has excellent antischistosomal properties in vivo. | |||
T28079 |
MMV665852
MMV-665852,MMV 665852 |
Others | Others |
MMV665852, an antischistosomal agent, has been shown to inhibit worm viability in vitro and reduce worm burden in S. mansoni-infected mice. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3254 |
PHYTOL
植醇,trans-Phytol,(E)-Phytol |
Antibacterial; PPAR; Parasite | DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
PHYTOL (trans-Phytol) 是一种从叶绿素中提取的二萜醇,广泛应用于食品添加剂和医药领域,具有很好的抗血吸虫特性。它具有抗伤害、抗氧化、抗炎、抗过敏等作用。它对结核分枝杆菌和金黄色葡萄球菌具有抗菌活性。 | |||
TN1190 |
14,15 β-Dihydroxyklaineanone
14,15beta-Dihydroxyklaineanone |
Parasite | Microbiology/Virology |
14,15 β-Dihydroxyklaineanone(14,15beta-Dihydroxyklaineanone)从 Eurycoma longifolia 中分离得到的苦味素类化合物,具有抗肿瘤促进、抗血吸虫和杀疟原虫活性。 |