首页 工具
登录
购物车

搜索结果

Search Results for " antidepressants "
Targets Recommended: MAO Monoamine Oxidase

11

抑制剂 & 化合物

2

天然产物

3

化合物库

2

同位素标记化合物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name
L9860 抗抑郁症化合物库

1163 compounds
1163 种与抑郁症相关的化合物,可以用于高通量和高内涵筛选
L2800 5-羟色胺分子库

268 compounds
268 种生物活性小分子化合物,用于高通量、高内涵筛选;
L5100 含氟化合物库

574 compounds
574 个含氟化合物的独特集合,可用于高通量筛选和高内涵筛选;

化合物库

抗抑郁症化合物库
Cat.No: L9860
Compounds: 1163
5-羟色胺分子库
Cat.No: L2800
Compounds: 268
含氟化合物库
Cat.No: L5100
Compounds: 574
Cat. No. Product Name Target Signaling Pathways
T0084 Moclobemide

吗氯贝胺,Ro111163

MAO; Monoamine Oxidase Metabolism; Neuroscience
Moclobemide (Ro111163) 是可逆的、可透过血脑屏障的单胺氧化酶 (MAO-A) 抑制剂,能够抑制 hMAO-A (IC50=6.061 μM)。它上调慢性应激小鼠海马祖细胞的增殖。
T0172 Maprotiline hydrochloride

Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil

5-HT Receptor; Adrenergic Receptor; AChR; Norepinephrine; Autophagy; Histamine Receptor Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Maprotiline hydrochloride (Psymion) 是一种桥环四环类抗抑郁药,是去甲肾上腺素重吸收抑制剂。
T0450L Fluoxetine hydrochloride

Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140

5-HT Receptor; Serotonin Transporter; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Fluoxetine hydrochloride (Lilly110140) 是一种高度特异性血清素摄取抑制剂。它被用作抗抑郁药,并且通常比传统的抗抑郁药具有更可接受的副作用特征。
T0943 Carbamazepine

卡马西平,NSC 169864

Mitophagy; Sodium Channel; Autophagy Autophagy; Membrane transporter/Ion channel
Carbamazepine (NSC-169864) 是与三环抗抑郁药化学相关的三环化合物,具有抗惊厥和镇痛特性。它通过减少多突触反应和阻断强直后增强发挥其抗惊厥活性。 它通常用于治疗与三叉神经痛相关的疼痛。
T25047 Alfetamine

alpha-allyl-phenethylamine

Others Others
Alfetamine is a chemical compound of the phenethylamine family. It is similar to imipramine and amitriptyline, two tricyclic antidepressants.
T31604 Edivoxetine

LY-2216684,LY 2216684,LY2216684

Others Others
Edivoxetine( LY2216684) is a selective norepinephrine reuptake inhibitor being developed as a treatment for attention deficit hyperactivity disorder (ADHD) and antidepressants.
T23628 AD-2646

AD2646

Others Others
AD-2646 is a new quinoline derivative. It also has similar pharmacological properties to tricyclic antidepressants.
T37307 Nordoxepin hydrochloride

Others Others
Doxepin is a tricyclic antidepressant. Desmethyldoxepin is the primary metabolite of doxepin, produced by metabolism at the liver. The metabolism of tricyclic antidepressants, including doxepin, is affected by a variety of factors, including age, genetics, and drug-drug interactions.
T68327 Dexnafenodone Free Base

Others Others
Dexnafenodone Free Base is a potent inhibitor of noradrenaline, and to a lesser degree of serotonin reuptake, induced changes in the pattern of sleep which are comparable to those of non‐sedating tricyclic antidepressants.
T69943 Citalopram oxalate

Others Others
Citalopram oxalate is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol uptake in alcoholics and is used in depressed patients who also suffer from tardive dyskinesia in preference to tricyclic antidepressants, which aggravate this condition.
T60265 NV-5138 hydrochloride

Others Others
NV-5138 hydrochloride 是一种亮氨酸类似物,是一个具有选择性和口服活性的脑内的mTORC1的激动剂,可与 Sestrin2 结合。NV-5138 hydrochloride 可用于抗抑郁的研究。

化合物

Moclobemide
Cat.No: T0084
Synonym: 吗氯贝胺,Ro111163
Target: MAO, Monoamine Oxidase
Maprotiline hydrochloride
Cat.No: T0172
Synonym: Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil
Target: 5-HT Receptor, Adrenergic Receptor, AChR, Norepinephrine, Autophagy, Histamine Receptor
Fluoxetine hydrochloride
Cat.No: T0450L
Synonym: Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140
Target: 5-HT Receptor, Serotonin Transporter, Autophagy
Carbamazepine
Cat.No: T0943
Synonym: 卡马西平,NSC 169864
Target: Mitophagy, Sodium Channel, Autophagy
Alfetamine
Cat.No: T25047
Synonym: alpha-allyl-phenethylamine
Target: Others
Edivoxetine
Cat.No: T31604
Synonym: LY-2216684,LY 2216684,LY2216684
Target: Others
AD-2646
Cat.No: T23628
Synonym: AD2646
Target: Others
Nordoxepin hydrochloride
Cat.No: T37307
Synonym:
Target: Others
Dexnafenodone Free Base
Cat.No: T68327
Synonym:
Target: Others
Citalopram oxalate
Cat.No: T69943
Synonym:
Target: Others
NV-5138 hydrochloride
Cat.No: T60265
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1045 Trimipramine maleate

Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐

Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂,对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。

天然产物

Trimipramine maleate
Cat.No: T1045
Synonym: Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐
Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Cat. No. Product Name Target Signaling Pathways
TMID-0207 Maprotiline-d5 Hydrochloride

Maprotiline-d5 Hydrochloride 是 Maprotiline Hydrochloride 的氘代化合物。Maprotiline Hydrochloride 的 CAS 号为 10347-81-6。Maprotiline hydrochloride 是一种桥环四环类抗抑郁药,是去甲肾上腺素重吸收抑制剂。
TMIJ-0044 Carbamazepine-d10

Carbamazepine-d10 是 Carbamazepine 的氘代化合物。Carbamazepine 的 CAS 号为 298-46-4。Carbamazepine是与三环抗抑郁药化学相关的三环化合物,具有抗惊厥和镇痛特性。它通过减少多突触反应和阻断强直后增强发挥其抗惊厥活性。 它通常用于治疗与三叉神经痛相关的疼痛。

同位素标记化合物

Maprotiline-d5 Hydrochloride
Cat.No: TMID-0207
Synonym:
Target:
Carbamazepine-d10
Cat.No: TMIJ-0044
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼