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Hydroxyfasudil (Hydroxy-Fasudil) 是一种ROCK 抑制剂,对ROCK1和ROCK2的IC50分别为 0.73 和 0.72 μM。
Hydroxyfasudil (Hydroxy-Fasudil) 是一种ROCK 抑制剂,对ROCK1和ROCK2的IC50分别为 0.73 和 0.72 μM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 285 | 现货 | |
2 mg | ¥ 383 | 现货 | |
5 mg | ¥ 579 | 现货 | |
10 mg | ¥ 832 | 现货 | |
25 mg | ¥ 1,620 | 现货 | |
50 mg | ¥ 2,590 | 现货 | |
100 mg | ¥ 3,830 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 637 | 现货 |
产品描述 | Hydroxyfasudil (Hydroxy-Fasudil) is a ROCK inhibitor(IC50s of 0.73 and 0.72 μM for ROCK1 and ROCK2, respectively). |
靶点活性 | PKA:37 μM, ROCK2:0.72 μM, ROCK1:0.73 μM |
别名 | Hydroxy-Fasudil, 羟基法舒地尔, HA-1100 |
分子量 | 307.37 |
分子式 | C14H17N3O3S |
CAS No. | 105628-72-6 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 31 mg/mL (100.86 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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