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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 416 | 现货 | |
5 mg | ¥ 1,130 | 现货 | |
10 mg | ¥ 1,920 | 现货 | |
25 mg | ¥ 3,250 | 现货 | |
50 mg | ¥ 4,750 | 现货 | |
100 mg | ¥ 6,780 | 现货 |
产品描述 | 2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide (GDC046), a potent lead analog, has good kinase selectivity, physicochemical properties and pharmacokinetic profile. |
靶点活性 | TYK2:4.8 nM (Ki), JAK1:0.7 nM (Ki), JAK2:0.7 nM (Ki), JAK3:0.4 nM (Ki) |
别名 | GDC046 |
分子量 | 350.2 |
分子式 | C16H13Cl2N3O2 |
CAS No. | 1258292-64-6 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
溶解度信息 | DMSO: 3.33 mg/mL (9.52 mM) | |||||||||||||||
溶液配制表 | ||||||||||||||||
DMSO
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