Glycopyrrolate

产品编号 T2387Cas号 596-51-0

别名 格隆溴铵|||Gastrodyn|||Glycopyrronium bromide|||Robinul|||Glycopyrrolate bromide

Glycopyrrolate (Glycopyrrolate bromide) 是一种毒蕈碱拮抗剂，在某些胃肠道疾病中用作解痉剂，并与某些麻醉剂一起减少唾液分泌。

产品编号 T2387别名 格隆溴铵, Gastrodyn, Glycopyrronium bromide, Robinul, Glycopyrrolate bromideCas号 596-51-0

Glycopyrrolate (Glycopyrrolate bromide) 是一种毒蕈碱拮抗剂，在某些胃肠道疾病中用作解痉剂，并与某些麻醉剂一起减少唾液分泌。

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生物活性

产品描述	Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.
体外活性	Glycopyrrolate inhibits EFS-induced contraction of guinea-pig trachea and human airways in a concentration-dependent manner. In competition studies, glycopyrrolate binds human peripheral lung and human airway smooth muscle (HASM) muscarinic receptors with affinities in the nanomolar range (Ki values 0.5–3.6?nM). Glycopyrrolate showed no selectivity in its binding to the M1–M3 receptors. Kinetics studies show that glycopyrrolate dissociates slowly from HASM muscarinic receptors[1].
别名	格隆溴铵, Gastrodyn, Glycopyrronium bromide, Robinul, Glycopyrrolate bromide

化学信息

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

溶解度信息

DMSO: 50 mg/mL (125.52 mM), Sonication is recommended.

H2O: 72 mg/mL (180.8 mM)

Ethanol: 55 mg/mL (138.1 mM)

溶液配制表

DMSO/Ethanol/H2O