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F-15599 是一种高度选择性的 G 蛋白偏向 5-HT1A 受体激动剂,Ki 值为 3.4 nM。
F-15599 是一种高度选择性的 G 蛋白偏向 5-HT1A 受体激动剂,Ki 值为 3.4 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 959 | 现货 | |
5 mg | ¥ 1,880 | 现货 | |
10 mg | ¥ 2,860 | 现货 | |
25 mg | ¥ 4,650 | 现货 | |
50 mg | ¥ 6,480 | 现货 | |
100 mg | ¥ 8,760 | 现货 | |
200 mg | ¥ 11,800 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 1,980 | 现货 |
产品描述 | F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM). |
靶点活性 | 5-HT1A:3.4 nM(ki) |
体内活性 | F-15599 exerted very potent (ID50 = 0.095 and 0.0059 mg/kg, respectively) anti-aggressive effects in male WTG rats. At 4.5-fold higher dose ranges, the anti-aggressive effects were accompanied by concomitant motor inactivity and/or reduction of social engagement. Pretreatment with WAY-100635 counteracted the behavioural effects of both agonists[1]. |
动物实验 | F-15599 agonists were acutely administered intraperitoneally in aggressive resident male WTG rats confronting an intruder[1]. |
分子量 | 394.85 |
分子式 | C19H21ClF2N4O |
CAS No. | 635323-95-4 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 22.5 mg/mL (56.98 mM) | ||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||
DMSO
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