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Isocarboxazid
很棒产品编号 T4559Cas号 59-63-2
别名 异卡波肼
Isocarboxazid 是不可逆的、非选择性的单胺氧化酶 monoamine oxidase 抑制剂，其在大鼠大脑中测得的 IC50值为4.8 μM。
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Isocarboxazid
很棒 纯度: 99.94%
产品编号 T4559 别名 异卡波肼Cas号 59-63-2
Isocarboxazid 是不可逆的、非选择性的单胺氧化酶 monoamine oxidase 抑制剂，其在大鼠大脑中测得的 IC50值为4.8 μM。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 1 mg | ¥ 239 | 现货 | |
| 2 mg | ¥ 346 | 现货 | |
| 5 mg | ¥ 579 | 现货 | |
| 10 mg | ¥ 849 | 现货 | |
| 25 mg | ¥ 1,420 | 现货 | |
| 50 mg | ¥ 2,090 | 现货 | |
| 100 mg | ¥ 3,150 | 现货 | |
| 500 mg | ¥ 6,990 | 现货 | |
| 1 mL x 10 mM (in DMSO) | ¥ 637 | 现货 |
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纯度:99.94%
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TargetMol 的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。产品介绍
生物活性
化学信息
| 产品描述 | Isocarboxazid has the formula 1-benzyl-2-(5-methyl-3-isoxazolylcarbonyl)hydrazine-isocarboxazid. It is a monoamine oxidase inhibitor.[2] It is used in the treatment of major depression, dysthymic disorder, atypical disorder, panic disorder and the phobic disorders. |
| 靶点活性 | Monoamine oxidase (rat brain):4.8 μM |
| 体外活性 | In vivo studies demonstrated isocarboxazid-driven inhibition of MAO in the brain, heart, and liver. The reduced MAO activity, caused by isocarboxazid, results in an increased concentration of serotonin, epinephrine, norepinephrine, and dopamine in storage sites throughout the central nervous system (CNS) and sympathetic nervous system. The increase of one or more monoamines is the basis for the antidepressant activity of MAO inhibitors like isocarboxazid.[1] |
| 体内活性 | In vitro studies demonstrated isocarboxazid-driven inhibition of MAO in the brain, heart, and liver. The reduced MAO activity, caused by isocarboxazid, results in an increased concentration of serotonin, epinephrine, norepinephrine, and dopamine in storage sites throughout the central nervous system (CNS) and sympathetic nervous system. The increase of one or more monoamines is the basis for the antidepressant activity of MAO inhibitors like isocarboxazid.[1] |
| 别名 | 异卡波肼 |
| 分子量 | 231.25 |
| 分子式 | C12H13N3O2 |
| CAS No. | 59-63-2 |
| Smiles | Cc1cc(no1)C(=O)NNCc1ccccc1 |
| 密度 | 1.206g/cm3 |
储存&溶解度
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| 溶解度信息 | DMSO: 50 mg/mL (216.22 mM)  | |||||||||||||||||||||||||||||||||||
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比如您的给药剂量是 10 mg/kg ，每只动物体重 20 g ，给药体积 100 μL ， 
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