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Selpercatinib (LOXO-292) 是 RET 激酶抑制剂,抑制 RET (WT)、RET (V804M) 、RET (G810R)的 IC50分别为 14.0 nM、24.1 nM、530.7 nM,具有抗肿瘤活性。
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Selpercatinib (LOXO-292) 是 RET 激酶抑制剂,抑制 RET (WT)、RET (V804M) 、RET (G810R)的 IC50分别为 14.0 nM、24.1 nM、530.7 nM,具有抗肿瘤活性。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 313 | 现货 | |
5 mg | ¥ 472 | 现货 | |
10 mg | ¥ 823 | 现货 | |
25 mg | ¥ 1,490 | 现货 | |
50 mg | ¥ 2,390 | 现货 | |
100 mg | ¥ 3,820 | 现货 | |
200 mg | ¥ 5,450 | 现货 | |
500 mg | ¥ 8,190 | 现货 |
产品描述 | Selpercatinib (LOXO-292) is a tyrosine kinase inhibitor with antineoplastic properties(IC50 of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M) , and RET (G810R), respectively) |
靶点活性 | RET (V804M):24.1 nM , RET (G810R):530.7 nM, RET (WT):14.0 nM |
别名 | LOXO-292 |
分子量 | 525.6 |
分子式 | C29H31N7O3 |
CAS No. | 2152628-33-4 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
溶解度信息 | DMSO: 5.26 mg/mL (10 mM), Sonication is recommended. | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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